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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Urocortin (rat) acetate
    Targetmol
    + Info

    Urocortin (rat) acetate

    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Purity:97.76%
    Color and Shape:Soild

    Ref: TM-TP1020L

  • Indacaterol maleate
    Targetmol
    + Info

    Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:508.56

    Ref: TM-T1239

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purity:98.55%
    Color and Shape:Yellowish White Crystalline Powder
    Molecular weight:431.55

    Ref: TM-T0081

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79

    Ref: TM-T1519L

  • 2-Bromo-6-methoxynaphthalene
    Targetmol
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    2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Formula:C11H9BrO
    Purity:98.51%
    Color and Shape:White To Off-White Powder
    Molecular weight:237.09

    Ref: TM-T0663

  • Amiselimod hydrochloride
    Targetmol
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    Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Formula:C19H31ClF3NO3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:413.9

    Ref: TM-T10305

  • Prucalopride
    Targetmol
    + Info

    Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Formula:C18H26ClN3O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:367.87

    Ref: TM-T2542

  • Clonidine hydrochloride
    Targetmol
    + Info

    Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purity:99.16% - 99.86%
    Color and Shape:Solid
    Molecular weight:266.55

    Ref: TM-T1247

  • Methyldopa
    Targetmol
    + Info

    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Formula:C10H13NO4
    Purity:98.95% - 99.86%
    Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Molecular weight:211.21

    Ref: TM-T0505

  • CYM 50769
    Targetmol
    + Info

    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purity:98% - 99.08%
    Color and Shape:Solid
    Molecular weight:416.86

    Ref: TM-T22702

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:231.65

    Ref: TM-T77565

  • Fluvoxamine maleate
    Targetmol
    + Info

    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Formula:C19H25F3N2O6
    Purity:99.92% - 99.94%
    Color and Shape:White Crystalline Powder
    Molecular weight:434.41

    Ref: TM-T1077

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43

    Ref: TM-T1211

  • PF429242 dihydrochloride
    Targetmol
    + Info

    PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Formula:C25H37Cl2N3O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:482.49

    Ref: TM-T12437

  • Roxatidine Acetate hydrochloride
    Targetmol
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9

    Ref: TM-T0157

  • Naftopidil
    Targetmol
    + Info

    Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Formula:C24H28N2O3
    Purity:99.60% - 99.97%
    Color and Shape:White Crystalline Powder
    Molecular weight:392.49

    Ref: TM-T0696

  • NF-56-EJ40 hydrochloride
    Targetmol
    + Info

    NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Formula:C27H31Cl2N3O3
    Purity:99.33%
    Color and Shape:Soild
    Molecular weight:516.46

    Ref: TM-T12216L

  • Fluoxetine
    Targetmol
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    Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Formula:C17H18F3NO
    Purity:99.07% - 99.28%
    Color and Shape:Solid
    Molecular weight:309.33

    Ref: TM-T0450

  • Aripiprazole
    Targetmol
    + Info

    Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39

    Ref: TM-T1566

  • Fluoxetine hydrochloride
    Targetmol
    + Info

    Fluoxetine hydrochloride

    CAS:
    Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.
    Formula:C17H19ClF3NO
    Purity:99.6% - 99.98%
    Color and Shape:White To Off-White Crystalline Solid White To Off-White Powder
    Molecular weight:345.787

    Ref: TM-T0450L