Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(41 products)
- Aminopeptidase(67 products)
- CETP(18 products)
- Carbonic Anhydrase(178 products)
- Casein Kinase(130 products)
- DHFR(33 products)
- Decarboxylase(4 products)
- Dehydrogenase(271 products)
- FAAH(64 products)
- FXR(58 products)
- Factor Xa(80 products)
- Fatty Acid Synthase(33 products)
- Ferroptosis(215 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(54 products)
- HIF/HIF Prolyl-Hydroxylase(142 products)
- HMG-CoA Reductase(33 products)
- Hydroxylase(30 products)
- IDO(82 products)
- LDL(8 products)
- Lipase(98 products)
- Lipid(58 products)
- Lipoxygenase(124 products)
- MAO(87 products)
- MPO(2 products)
- NAMPT(36 products)
- P450(6 products)
- PAI-1(25 products)
- PDE(166 products)
- PED(1 products)
- PKM(15 products)
- PPAR(164 products)
- Phospholipase(82 products)
- ROR(42 products)
- Retinoid Receptor(29 products)
- SGK(11 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(42 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
Show 34 more subcategories
Found 8626 products of "Metabolism"
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ML404
CAS:<p>ML404 is the mitochondrial permeability transition pore inhibitor.</p>Formula:C17H13ClN2O3Purity:98%Color and Shape:SolidMolecular weight:328.75AVX-001
CAS:<p>AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.</p>Formula:C21H29F3OSColor and Shape:SolidMolecular weight:386.51IDH-C227
CAS:<p>IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.</p>Formula:C30H31FN4O2Color and Shape:SolidMolecular weight:498.59Enpp-1-IN-10
CAS:<p>Enpp-1-IN-10 inhibits ENPP1 with 3.866 μM Ki, useful in cancer research.</p>Formula:C13H12N6OSColor and Shape:SolidMolecular weight:300.34CDK2-IN-11
CAS:<p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>Formula:C18H14ClN7O2SColor and Shape:SolidMolecular weight:427.87UK-500001
CAS:<p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>Formula:C26H24F3N3O4Purity:98%Color and Shape:SolidMolecular weight:499.48MR 16728 hydrochloride
CAS:<p>stimulates the release of acetylcholine from synaptosomes</p>Formula:C23H37ClN2OPurity:98%Color and Shape:SolidMolecular weight:393.01FTase-IN-1
CAS:<p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>Formula:C23H16N2O2SColor and Shape:SolidMolecular weight:384.45DSHN
CAS:<p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>Formula:C15H17NO5SPurity:98%Color and Shape:SolidMolecular weight:323.36ML387
CAS:<p>ML387 is an inhibitor of human NAD(+)- dependent 15- hydroxyprostaglandin dehydrogenase.</p>Formula:C20H21N3O2Purity:98%Color and Shape:SolidMolecular weight:335.4GSK360A
CAS:<p>GSK360A is a novel prolyl hydroxylase (PHD) domain-containing enzyme inhibitor.</p>Formula:C17H17FN2O5Purity:98%Color and Shape:SolidMolecular weight:348.33DNS-8254
CAS:<p>DNS-8254: Potent, selective PDE2 inhibitor, enhances memory (IC50=8 nM), effective in rat memory tests.</p>Formula:C18H15BrF3N5OPurity:98%Color and Shape:SolidMolecular weight:454.24LY367385
CAS:<p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>Formula:C10H11NO4Purity:98%Color and Shape:SolidMolecular weight:209.2BRD6897
CAS:BRD6897 is a mitochondrial content inducer that increases the cellular content of mitochondria.Formula:C25H21N3O2S2Purity:97.74%Color and Shape:SolidMolecular weight:459.58ONO-6126
CAS:<p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>Formula:C20H27N3O4Purity:98%Color and Shape:SolidMolecular weight:373.45Semotiadil recemate fumarate
CAS:Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.Formula:C33H36N2O10SPurity:98%Color and Shape:SolidMolecular weight:652.71MMG-0358
CAS:<p>MMG-0358 is a novel potent IDO1 inhibitor, showing low cytotoxicity and higher selectivity for IDO1 over TDO enzyme.</p>Formula:C8H6ClN3OColor and Shape:SolidMolecular weight:195.61SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Formula:C30H27Cl2N3O4Color and Shape:SolidMolecular weight:564.46PKM2 activator 3
CAS:<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Formula:C15H11ClF2N2O3SColor and Shape:SolidMolecular weight:372.77ALRT 1550
CAS:<p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>Formula:C23H32O2Color and Shape:SolidMolecular weight:340.5LB42908
CAS:<p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>Formula:C32H31N5O3Color and Shape:SolidMolecular weight:533.62FCE 28654
CAS:<p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>Formula:C25H35N2O7PColor and Shape:SolidMolecular weight:506.53N-Oleoyl Leucine
CAS:<p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>Formula:C24H45NO3Purity:98.25%Color and Shape:SolidMolecular weight:395.62L 669262
CAS:<p>L 669262 is a potent inhibitor of HMG-CoA reductase.</p>Formula:C25H36O6Color and Shape:SolidMolecular weight:432.55LH65.3
CAS:<p>LH65.3 is an inhibitor of S. typhimurium infection on the activity of DUSP3, DUSP11, and DUSP27.</p>Formula:C21H20N2O5SPurity:98%Color and Shape:SolidMolecular weight:412.46MEDS433
CAS:<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Formula:C20H11F4N3O2Color and Shape:SolidMolecular weight:401.31ARN19874
CAS:<p>ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].</p>Formula:C19H14N4O4SPurity:98%Color and Shape:SolidMolecular weight:394.4Benserazide
CAS:<p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>Formula:C10H15N3O5Color and Shape:SolidMolecular weight:257.24Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Formula:C15H20O3Color and Shape:SolidMolecular weight:248.32Rosuvastatin lactone
CAS:<p>Tilavonemab (ABBV-8E12) is a monoclonal antibody that binds to the N-terminus of the human microtubule-associated protein tau.</p>Formula:C22H26FN3O5SColor and Shape:SolidMolecular weight:463.52PDE2/PDE10-IN-1
CAS:<p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>Formula:C15H10ClN5Purity:98%Color and Shape:SolidMolecular weight:295.73DNJNAc
CAS:<p>DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.</p>Formula:C8H16N2O4Purity:98.65% - 99.37%Color and Shape:SolidMolecular weight:204.22IHMT-PI3Kδ-372
CAS:<p>IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.</p>Formula:C26H23F2N7O2Purity:99.77%Color and Shape:SolidMolecular weight:503.5Ciraparantag
CAS:<p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>Formula:C22H48N12O2Purity:98%Color and Shape:SolidMolecular weight:512.7Glucokinase activator 1
CAS:Glucokinase activator 1 is a liver-directed glucokinase activator (EC50: 34 nM).Formula:C27H20F2N2O7S2Purity:98%Color and Shape:SolidMolecular weight:586.58Adenosine 5'-phosphosulfate (sodium salt)
CAS:<p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>Formula:C10H12N5Na2O10PSColor and Shape:SolidMolecular weight:471.24SHP504
CAS:<p>SHP504 is an inhibitor of SHP2 phosphatase and acts on SHP21-525 (IC50: 21 μM).</p>Formula:C23H15ClN4O4Color and Shape:SolidMolecular weight:446.84Pancreatic lipase/Carboxylesterase 1-IN-1
CAS:<p>Compound 39 is a dual inhibitor of PL (IC50: 2.13 μM) and hCES1A (IC50: 0.055 μM).</p>Formula:C30H44O4Color and Shape:SolidMolecular weight:468.67ML218
CAS:ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.Formula:C19H26Cl2N2OPurity:99.2% - 99.45%Color and Shape:SolidMolecular weight:369.33Quetiapine sulfoxide
CAS:<p>Quetiapine sulfoxide: Main metabolite of Quetiapine, a 5-HT agonist & dopamine antagonist antipsychotic.</p>Formula:C21H25N3O3SPurity:98%Color and Shape:Pale Yellow SolidMolecular weight:399.51Pulixin
CAS:<p>Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).</p>Formula:C14H11NO4Color and Shape:SolidMolecular weight:257.24HZ52
CAS:<p>HZ52: Potent reversible 5-LO inhibitor; IC50 0.7 μM; blocks LTs in human leukocytes.</p>Formula:C24H26ClN3O2SColor and Shape:SolidMolecular weight:456ATX inhibitor 20
CAS:<p>ATX inhibitor 20 is a potent inhibitor of ATX (IC50: 2.3 nM).</p>Formula:C31H34FN5O3Color and Shape:SolidMolecular weight:543.63Ro 41-0960
CAS:<p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>Formula:C13H8FNO5Purity:98%Color and Shape:SolidMolecular weight:277.2Glyoxalase I inhibitor
CAS:<p>Glyoxalase I inhibitor, a candidate for anticancer agents, is a potent Glyoxalase I (GLO1) inhibitor.</p>Formula:C21H30BrClN4O8SPurity:98%Color and Shape:SolidMolecular weight:613.91IHVR-11029
CAS:<p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>Formula:C18H27F2NO5Color and Shape:SolidMolecular weight:375.41Argininic acid
CAS:<p>Argininic acid is an α-amino acid used in the biosynthesis of proteins.</p>Formula:C6H13N3O3Purity:98%Color and Shape:SolidMolecular weight:175.19Atreleuton
CAS:<p>Atreleuton (ABT-761), reversible oral 5-LO inhibitor, selectively blocks leukotriene formation.</p>Formula:C16H15FN2O2SPurity:98%Color and Shape:SolidMolecular weight:318.37Manninotrionate
CAS:<p>Manninotrionate, an antitumor agent, linked to BSA; rabbit antiserum made, doesn't agglutinate Ehrlich tumor cells with alpha-D-galactosyl groups.</p>Formula:C18H32KO17Purity:98%Color and Shape:SolidMolecular weight:559.5354,5,6,7-Tetrabromobenzimidazole
CAS:<p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>Formula:C7H2Br4N2Color and Shape:SolidMolecular weight:433.72hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Formula:C12H12N4O5S2Color and Shape:SolidMolecular weight:356.38103D5R
CAS:<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4Utibapril
CAS:Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.Formula:C22H31N3O5SPurity:98%Color and Shape:SolidMolecular weight:449.564-Acetylsimvastatin
CAS:<p>4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).</p>Formula:C27H40O6Purity:98%Color and Shape:SolidMolecular weight:460.6LY 269415
CAS:<p>LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis.</p>Formula:C19H28N2O2SColor and Shape:SolidMolecular weight:348.5Mesopram
CAS:<p>PDE4 inhibitor, orally active</p>Formula:C14H19NO4Purity:98%Color and Shape:SolidMolecular weight:265.3Cgp 8065
CAS:<p>Cgp 8065 is a filaricidal compound, a dithiocarbamate-derivative of amoscanate.</p>Formula:C16H15N3O4S2Color and Shape:SolidMolecular weight:377.44XY101
CAS:<p>XY101 is a selective, metabolically stable and orally available agonist of RORγ inverse(IC50 of 30 nM and a Kd of 380 nM).</p>Formula:C25H20F7NO4SPurity:99.83%Color and Shape:SolidMolecular weight:563.48Prolyl Endopeptidase Inhibitor 1
CAS:Prolyl Endopeptidase Inhibitor 1 is a potent inhibitor of prolyl endopeptidase (PEP; PE)(Ki : 15 nM) , has anti-amnesic effect.Formula:C15H24N2O4Purity:98%Color and Shape:SolidMolecular weight:296.36IHVR-19029
CAS:<p>IHVR-19029: ER α-glucosidases I/II inhibitor, IC50 0.48μM; halts Ebola, Dengue, Rift Valley fever virus replication.</p>Formula:C23H45N3O5Color and Shape:SolidMolecular weight:443.62SHP836
CAS:<p>SHP836 is an inhibitor of SHP2 allosteric (IC50: 12 μM for the full-length SHP2).</p>Formula:C16H19Cl2N5Purity:98%Color and Shape:SolidMolecular weight:352.26ROR Modulator I
CAS:<p>ROR Modulator I is the first potent inverse agonist of the retinoid-related orphan receptor. It also has dual selectivity for RORβ and RORγt.</p>Formula:C26H20Cl2N2O4S2Purity:98%Color and Shape:SolidMolecular weight:559.48L 30
CAS:<p>L 30 is a blocker of the sodium channel.</p>Formula:C15H24N2OPurity:98%Color and Shape:SolidMolecular weight:248.3611β-HSD1-IN-10
CAS:<p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>Formula:C16H10F3NO2Color and Shape:SolidMolecular weight:305.25Pitstop1
CAS:<p>Clathrin-IN-1 selectively inhibits clathrin, potentially blocking virus entry and modulating cell signals.</p>Formula:C19H14N2NaO5SPurity:98%Color and Shape:SolidMolecular weight:405.38Quinalizarin
CAS:Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.Formula:C14H8O6Purity:98%Color and Shape:SolidMolecular weight:272.21RORγt inverse agonist 28
CAS:<p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>Formula:C23H18Cl2F3NO5SColor and Shape:SolidMolecular weight:548.36SHP844
CAS:<p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>Formula:C29H24ClN5O6Color and Shape:SolidMolecular weight:573.98hCAIX-IN-10
CAS:<p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>Formula:C28H21N3O3SColor and Shape:SolidMolecular weight:479.55FR-221647
CAS:<p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>Formula:C14H17N3O2Color and Shape:SolidMolecular weight:259.3CAY10761
CAS:<p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).</p>Formula:C7H8N4O2S2Color and Shape:SolidMolecular weight:244.29Dapaconazole
CAS:<p>Dapaconazole is used as a drug candidate for antifungals.</p>Formula:C19H15Cl2F3N2OColor and Shape:SolidMolecular weight:415.244-Desmethyl Istradefylline
CAS:<p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>Formula:C19H22N4O4Purity:98%Color and Shape:SolidMolecular weight:370.40SDZ-MKS 492
CAS:SDZ-MKS 492 is a selective type III isozyme cyclic nucleotide phosphodiesterase inhibitor.Formula:C20H27N5O6Purity:98%Color and Shape:SolidMolecular weight:433.46Acetaldophosphamide
CAS:<p>Acetaldophosphamide is a novel stable aldophosphamide analog.</p>Formula:C11H21Cl2N2O6PColor and Shape:SolidMolecular weight:379.177-Biopterin
CAS:<p>7-Biopterin, a 7-substituted pterin, forms non-enzymatically and elevates in urine of hyperphenylalaninemics with PCBD mutations.</p>Formula:C9H11N5O3Color and Shape:SolidMolecular weight:237.22Transketolase-IN-2
CAS:<p>Transketolase-IN-2, potent herbicidal agent, inhibits weeds like Digitaria sanguinalis and Amaranthus retroflexus.</p>Formula:C18H9F3N2O3SColor and Shape:SolidMolecular weight:390.34Dibefurin
CAS:<p>Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.</p>Formula:C18H16O8Color and Shape:SolidMolecular weight:360.31OL-135
CAS:<p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>Formula:C21H22N2O2Color and Shape:SolidMolecular weight:334.41Enpp-1-IN-9
CAS:<p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>Formula:C17H24N4O5SColor and Shape:SolidMolecular weight:396.46CP-532623
CAS:<p>CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.</p>Formula:C27H27F9N2O3Purity:98%Color and Shape:SolidMolecular weight:598.5Soluble epoxide hydrolase inhibitor
CAS:<p>Soluble epoxide hydrolase inhibitor is a soluble epoxide hydrolase inhibitor (human soluble epoxide hydrolase (h-sEH) with pIC50 of 8.4).</p>Formula:C18H12F5N5O3Purity:98%Color and Shape:SolidMolecular weight:441.31EN40
CAS:<p>EN40, as a covalent ligand, is a selective inhibitor of aldehyde dehydrogenase 3A1 (IC50: 2 uM).</p>Formula:C13H15NO2Color and Shape:SolidMolecular weight:217.26Clofenamide
CAS:<p>Clofenamide is a low-ceiling sulfonamide diuretic.</p>Formula:C6H7ClN2O4S2Color and Shape:SolidMolecular weight:270.71Y-29794 oxalate
CAS:<p>Inhibitor of prolyl endopeptidase</p>Formula:C25H36N2O5S2Purity:98%Color and Shape:SolidMolecular weight:508.69Glutamamide
CAS:<p>Glutamamide is an anticancer drug.</p>Formula:C5H11N3O2Purity:98%Color and Shape:SolidMolecular weight:145.16POP-IN-2
CAS:<p>Compound 7k (POP-IN-2) is a potent POP inhibitor with Ki of 6 nM, useful in neurodegenerative and cancer studies.</p>Formula:C24H33BN2O5Color and Shape:SolidMolecular weight:440.34Vilazodone carboxylic acid
CAS:<p>Vilazodone carboxylic acid is a vilazodone metabolite observed in both urine and plasma.</p>Formula:C26H26N4O3Purity:98%Color and Shape:SolidMolecular weight:442.51hCAIX/XII-IN-6
<p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>Formula:C26H23N3O6S4Color and Shape:SolidMolecular weight:601.74Telotristat besilate
CAS:<p>Telotristat besilate is an inhibitor of tryptophan hydroxylase.</p>Formula:C31H28ClF3N6O6SPurity:98%Color and Shape:SolidMolecular weight:705.11IDO1/TDO-IN-3
CAS:<p>IDO1/TDO-IN-3 inhibits IDO1 (IC50: 0.005 μM) and TDO (IC50: 0.004 μM) with strong anti-tumor activity and low toxicity.</p>Formula:C16H6ClF2N3O2Color and Shape:SolidMolecular weight:345.69YCT529 free acid
CAS:<p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>Formula:C29H25NO3Color and Shape:SolidMolecular weight:435.51SHP2-IN-13
CAS:<p>SHP2-IN-13 is an orally active, highly selective allosteric inhibitor targeting the SHP2 “tunnel site,” exhibiting an IC50 of 83.0 nM.</p>Formula:C16H21N7OColor and Shape:SolidMolecular weight:327.38Fadrozole HCl hydrate
CAS:<p>Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.</p>Formula:C14H13N3ClHH2OPurity:98%Color and Shape:SolidMolecular weight:268.74Izumerogant
CAS:<p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>Formula:C22H18ClF4N5O2Color and Shape:SolidMolecular weight:495.86M8891
CAS:M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.Formula:C20H17F2N3O3Color and Shape:SolidMolecular weight:385.36Trandolaprilate hydrate
CAS:<p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>Formula:C22H32N2O6Color and Shape:SolidMolecular weight:420.5RORγt Inverse agonist 8
CAS:<p>RORγt Inverse agonist 8 is a potent, selective, orally bioavailable RORγt inverse agonist(human RORγt-LBD with an IC50 of 19 nM).</p>Formula:C26H33N7O2Purity:98%Color and Shape:SolidMolecular weight:475.59ASP3662
CAS:<p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>Formula:C19H16ClF3N4O2Color and Shape:SolidMolecular weight:424.8Palmostatin B
CAS:<p>Palmostatin B is a modulator of Ras-signaling that acts by targeting acyl protein thioesterase 1 (APT1) and 2 (APT2) in cells.</p>Formula:C23H36O4Purity:98%Color and Shape:SolidMolecular weight:376.53
