Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(42 products)
- Aminopeptidase(76 products)
- CETP(20 products)
- Carbonic Anhydrase(196 products)
- Casein Kinase(139 products)
- DHFR(30 products)
- Decarboxylase(4 products)
- Dehydrogenase(302 products)
- FAAH(64 products)
- FXR(62 products)
- Factor Xa(87 products)
- Fatty Acid Synthase(37 products)
- Ferroptosis(227 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(56 products)
- HIF/HIF Prolyl-Hydroxylase(146 products)
- HMG-CoA Reductase(34 products)
- Hydroxylase(36 products)
- IDO(84 products)
- LDL(7 products)
- Lipase(107 products)
- Lipid(62 products)
- Lipoxygenase(133 products)
- MAO(85 products)
- MPO(2 products)
- NAMPT(40 products)
- P450(6 products)
- PAI-1(26 products)
- PDE(169 products)
- PED(1 products)
- PKM(17 products)
- PPAR(170 products)
- Phospholipase(85 products)
- ROR(47 products)
- Retinoid Receptor(18 products)
- SGK(10 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(43 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
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Found 9188 products of "Metabolism"
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p-Valerylphenol
CAS:p-Valerylphenol (NSC-49186) can be used to synthesize acylphenoxyacetic acid compounds.Formula:C11H14O2Purity:99.87%Color and Shape:White To Light Beige PowderMolecular weight:178.23Propaquizafop
CAS:Propaquizafop, a phenoxyisopropionic acid derivative, is used as a herbicide.Formula:C22H22ClN3O5Purity:98%Color and Shape:Colourless-To-Brown CrystalsMolecular weight:443.88Acetylhydrolase-IN-1
CAS:Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).Formula:C23H48NO7PPurity:98%Color and Shape:SolidMolecular weight:481.6Lp-PLA2-IN-3
CAS:Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.Formula:C20H13ClF3N3O3SPurity:99.84%Color and Shape:SolidMolecular weight:467.85Ref: TM-T11874
1mg90.00€2mg132.00€5mg215.00€1mL*10mM (DMSO)220.00€10mg340.00€25mg565.00€50mg797.00€100mg1,063.00€500mg2,142.00€Hydroxychlorodenafil
CAS:Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.Formula:C19H23ClN4O3Color and Shape:SolidMolecular weight:390.86HS79
CAS:HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.Formula:C19H22N4SPurity:98%Color and Shape:SolidMolecular weight:338.47PDE5-IN-4
CAS:PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,Formula:C21H27N5O5SColor and Shape:SolidMolecular weight:461.53M77976
CAS:M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.Formula:C17H16N2O3Purity:99.92%Color and Shape:SolidMolecular weight:296.32Oxagrelate
CAS:Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.Formula:C14H16N2O4Color and Shape:SolidMolecular weight:276.29Andolast
CAS:Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.Formula:C15H11N9OColor and Shape:SolidMolecular weight:333.31sEH inhibitor-14
CAS:sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with anFormula:C16H12F3N3O4Color and Shape:SoildMolecular weight:367.28SGK1-IN-2
CAS:SGK1-IN-2 (14h) is a selective inhibitor of SGK1 (serum and glucocorticoid regulated kinase 1)(with an IC50 of 5 nM at 10 μM ATP concentration).Formula:C17H12Cl2N6O2SPurity:98%Color and Shape:SolidMolecular weight:435.29MitoTEMPO hydrate
CAS:MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.Formula:C29H35N2O2P·Cl·H2OColor and Shape:SolidMolecular weight:528.04Enpp-1-IN-5
CAS:Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.Formula:C17H26N6O4SColor and Shape:SolidMolecular weight:410.49Benserazide
CAS:Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.Formula:C10H15N3O5Color and Shape:SolidMolecular weight:257.24mIDH1-IN-1
CAS:mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).Formula:C25H27N3O5Color and Shape:SolidMolecular weight:449.5UK-414,495
CAS:UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.Formula:C16H25N3O3SColor and Shape:SolidMolecular weight:339.45AMG-7980
CAS:AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.Formula:C19H22N4O2Purity:98%Color and Shape:SolidMolecular weight:338.4Glucokinase activator 3
CAS:Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.Formula:C26H33N2O9PS2Color and Shape:SolidMolecular weight:612.65α-Glucosidase-IN-8
CAS:α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].Formula:C19H20FN3O2Color and Shape:SolidMolecular weight:341.38Eggmanone
CAS:EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.Formula:C20H20N2O2S3Color and Shape:SolidMolecular weight:416.58hCAIX-IN-6
CAS:6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.Formula:C18H12N2O4SColor and Shape:SolidMolecular weight:352.36Carbonic anhydrase inhibitor 13
CAS:Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).Formula:C17H15N5O3S2Color and Shape:SolidMolecular weight:401.46IDO1-IN-17
CAS:IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .Formula:C28H32BrClFN5O2Color and Shape:SolidMolecular weight:604.94FAAH-IN-5
CAS:FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.Formula:C21H19N3O6SColor and Shape:SolidMolecular weight:441.46IDH2R140Q-IN-1
CAS:IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.Formula:C22H20F6N6Color and Shape:SolidMolecular weight:482.42Glutamamide
CAS:Glutamamide is an anticancer drug.Formula:C5H11N3O2Purity:98%Color and Shape:SolidMolecular weight:145.16PKR activator 2
CAS:PKR activator 2 is a potent activator of pyruvate kinase-R (PKR).Formula:C18H16N8OSPurity:98%Color and Shape:SolidMolecular weight:392.44CK2-IN-6
CAS:CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.Formula:C19H16ClN7O2Color and Shape:SolidMolecular weight:409.83RORγt modulator 2
CAS:RORγt modulator 2 is a modulator of retinol-related orphan receptor γt (RORyt) (IC50<50 nM) and can be used in the study of RORγt-mediated diseases such as painFormula:C28H29ClN2O4SColor and Shape:SolidMolecular weight:525.06KCN1
CAS:KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.Formula:C26H27NO5SColor and Shape:SolidMolecular weight:465.56F-1394
CAS:F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.Formula:C33H61N3O6Color and Shape:SolidMolecular weight:595.85SCH-42354
CAS:SCH-42354: potent oral NEP inhibitor, activates ANP & leu-enkephalin, has anti-hypertensive properties, IC50s of 8.3 & 10.0 nM.Formula:C16H23NO3S2Color and Shape:SolidMolecular weight:341.49ICI 211965
CAS:ICI 211965 is a selective and orally potent of 5-Lipoxygenase (5-LPO).Formula:C24H23NO2SPurity:98%Color and Shape:SolidMolecular weight:389.51LCL521 dihydrochloride
CAS:LCL521 dihydrochloride is a dual inhibitor of ACDase and ASMase, modulating sphingolipid metabolism with potential in cancer and metabolic research.Formula:C31H54Cl2N4O7Purity:98%Color and Shape:SolidMolecular weight:665.6914(S)-HDHA
CAS:DHA is an ω-3 important for development and therapy for inflammation and cancer; its derivative, 14(S)-HDHA, aids in reducing inflammation.Formula:C22H32O3Color and Shape:SolidMolecular weight:344.49CGS 35601
CAS:CGS 35601 is a single molecule inhibitor of triple vasopeptidase.Formula:C23H31N3O4SColor and Shape:SolidMolecular weight:445.57hCAIX/XII-IN-3
CAS:Compound 6q inhibits hCAIX/CAXII; K i : hCAI >10000 nM, hCAII >10000 nM, hCAIX 66.2 nM, hCAXII 4.4 nM.Formula:C20H13F3N2O4Color and Shape:SolidMolecular weight:402.3211β-HSD1-IN-6
CAS:11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).Formula:C21H19ClN4OColor and Shape:SolidMolecular weight:378.86(±)-γ-Tocopherol
CAS:(±)-γ-Tocopherol is a form of vitamin E with antioxidant and anti-inflammatory properties.Formula:C28H48O2Color and Shape:SolidMolecular weight:416.68Genz-669178
CAS:Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).Formula:C17H14N4OSPurity:98%Color and Shape:SolidMolecular weight:322.38CL 242817
CAS:CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).Formula:C18H21NO5SColor and Shape:SolidMolecular weight:363.4311β-HSD1-IN-9
CAS:11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.Formula:C13H9F3N2OColor and Shape:SolidMolecular weight:266.22BMS-351
CAS:BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.Formula:C15H12F3N3Color and Shape:SolidMolecular weight:291.27RP 73163 Racemate
CAS:RP 73163 Racemate is the racemate of RP 73163. RP 73163 is a potent inhibitor of ACAT, shows cholesterol lowering activity.Formula:C25H28N4OSPurity:98%Color and Shape:SolidMolecular weight:432.58Glucocerebrosidase-IN-1
CAS:Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.Formula:C13H27NO3Color and Shape:SolidMolecular weight:245.36AMPD2 inhibitor 2
AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.Formula:C26H27F2N3O3Color and Shape:SolidMolecular weight:467.51MDPD
CAS:MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.Formula:C21H19N3O3Color and Shape:SolidMolecular weight:361.39Lombricine
CAS:Lombricine, as a phosphodiester of 2-guanidinoethanol and D-serine in structure, is a phosphagen that is unique to earthworms.Formula:C6H15N4O6PColor and Shape:SolidMolecular weight:270.18Antiproliferative agent-10
Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.Formula:C35H36Cl2N7PRuColor and Shape:SolidMolecular weight:757.66XEN103
CAS:XEN103 is a potent and selective Stearoyl-CoA Desaturase-1 inhibitor.Formula:C22H23F4N5O2Color and Shape:SolidMolecular weight:465.44Saterinone hydrochloride
CAS:Saterinone hydrochloride is an inhibitor of phosphodiesterase III (PDE III).Formula:C27H31ClN4O4Purity:98%Color and Shape:SolidMolecular weight:511.01hCA I-IN-2
CAS:hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).Formula:C26H20BrN5O3SColor and Shape:SolidMolecular weight:562.44RORγt modulator 3
CAS:RORγt modulator 3 is a modulator of retinol-related orphan receptor γt (RORγt) and can be used to study RORγt-mediated diseases such as pain, COPD, inflammationFormula:C25H25ClFN3O4SColor and Shape:SolidMolecular weight:518Zidovudine glucuronide
CAS:Zidovudine glucuronide: an NRTI antiretroviral for HIV/AIDS treatment; blocks HIV reverse transcriptase, stops viral DNA formation.Formula:C16H21N5O10Color and Shape:SolidMolecular weight:443.37Amastatin
CAS:Amastatin is a non-toxic inhibitor of aminopeptidase A and leucine aminopeptidase, and its Ki for aminopeptidase A is 1 μM .Formula:C21H38N4O8Purity:98%Color and Shape:SolidMolecular weight:474.55BI-L 357
CAS:BI-L 357, a prodrug of BL-L 226, is a selective, orally active inhibitor of 5-lipoxygenase.Formula:C18H18O4SColor and Shape:SolidMolecular weight:330.4CDK2-IN-12
CAS:CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.Formula:C20H17N9O2SColor and Shape:SolidMolecular weight:447.47PF-04279405
CAS:PF-04279405 is a potent and selective glucokinase activator.Formula:C25H25FN4O4Color and Shape:SolidMolecular weight:464.49PDE-9 inhibitor
CAS:PDE-9 inhibitor is used for treatment neurodegenerative diseases.Formula:C22H27N5O2Purity:98%Color and Shape:SolidMolecular weight:393.48JZP-MA-13
JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.Formula:C14H15FN4O3SColor and Shape:SolidMolecular weight:338.36BRD9500
CAS:BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.Formula:C15H18FN3O2Color and Shape:SolidMolecular weight:291.32Anti-hyperglycemic agent-1
CAS:Anti-hyperglycemic agent 1 is a potent inhibitor of alpha-glucosidase (IC50: 0.53 μM). anti-Hyperglycemic agent 1 can be used to study diabetes.Formula:C20H15BrN2O3Color and Shape:SolidMolecular weight:411.25Glyoxalase I inhibitor 7
CAS:Glyoxalase I inhibitor 7 (Compound 6) is a potent inhibitor of glyoxalase I (Glo-I) with an IC50 of 3.65 μM. It exhibits potential as an anticancer agent [1].Formula:C17H16N4O3SColor and Shape:SolidMolecular weight:356.4BTX161
CAS:BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.Formula:C15H16N2O3Color and Shape:SolidMolecular weight:272.3ATX inhibitor 19
CAS:ATX inhibitor 19 is a potent inhibitor of ATX (IC50: 156 nM).Formula:C28H33ClN6O2SColor and Shape:SolidMolecular weight:553.12JTP 103237
CAS:JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.Formula:C24H29F3N6OColor and Shape:SolidMolecular weight:474.52SHP2-IN-5
CAS:SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cellFormula:C12H8O6Color and Shape:SolidMolecular weight:248.19Asp-AMS
CAS:Asp-AMS is a strong competitive inhibitor of the mitochondrial enzyme and also an aspartyl-tRNA synthetase inhibitor.Formula:C14H19N7O9SColor and Shape:SolidMolecular weight:461.41HFI-437
CAS:HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].Formula:C23H20N2O5Color and Shape:SolidMolecular weight:404.42PDE10-IN-5
CAS:PDE10-IN-5 is a phosphodiesterase 10 (PDE 10) inhibitor that can be used to study certain central nervous system disorders.Formula:C26H19F3N4OColor and Shape:SolidMolecular weight:460.45FABP4/5-IN-5
CAS:FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].Formula:C23H14ClF2NO4SColor and Shape:SolidMolecular weight:473.88RO6806051
CAS:RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.Formula:C21H19ClN6Color and Shape:SolidMolecular weight:390.87Methazolamide-d6
CAS:Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.Formula:C5H2D6N4O3S2Color and Shape:SolidMolecular weight:242.31Phortress free base
CAS:Phortress free base is a P450 CYP1A1-activated antitumor prodrug with antitumor activity.Formula:C20H23FN4OSPurity:98%Color and Shape:SolidMolecular weight:386.49Quinapril-d5
CAS:Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.Formula:C25H25D5N2O5Color and Shape:SolidMolecular weight:443.55PX20606
CAS:PX20606 is an orally active farnesoid X receptor (FXR) agonist, demonstrating EC50 values of 220 nM (mFXR) and 50 nM (hFXR) in Gal4-FXR assays. It induces the expression of the tumor suppressor gene NDRG2 and inhibits tumor growth and metastasis in a mouse HCC model. Additionally, PX20606 exhibits hepatoprotective properties.
Formula:C29H22Cl3NO4Color and Shape:SolidMolecular weight:554.85ATX inhibitor 5
CAS:ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.Formula:C22H18ClF3N6OPurity:99.73%Color and Shape:SolidMolecular weight:474.87Ref: TM-T10409
1mg46.00€5mg94.00€1mL*10mM (DMSO)96.00€10mg149.00€25mg245.00€50mg338.00€100mg460.00€200mg622.00€T-82
CAS:T-82 is an acetylcholinesterase inhibitor that may ameliorate the impairment of memory induced by acetylcholinergic dysfunction.Formula:C31H36ClN3O5SColor and Shape:SolidMolecular weight:598.15Xanthine oxidase-IN-5
CAS:Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.Formula:C18H16FN3O3Color and Shape:SolidMolecular weight:341.34Afegostat
CAS:Afegostat is a pharmacological chaperone that specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum with high affinity.Formula:C6H13NO3Purity:98%Color and Shape:Yellow Low-Melting SolidMolecular weight:147.17ICI 153110
CAS:ICI 153110: Oral phosphodiesterase inhibitor for treating congestive heart failure, has inotropic, vasodilator effects.Formula:C11H11N3OPurity:98%Color and Shape:SolidMolecular weight:201.22KT185
CAS:KT185 is an orally-bioavailable and brain-penetrant ABHD6 inhibitor (IC50: 0.21 nM in Neuro2A cells).Formula:C32H33N5O2Purity:98%Color and Shape:SolidMolecular weight:519.64Ambuphylline
CAS:Ambuphylline (Bufylline) is a theophylline derivative and bronchodilator for asthma and lung disease research.Formula:C11H19N5O3Color and Shape:SolidMolecular weight:269.305TK-642
CAS:TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.Formula:C17H20ClN7SColor and Shape:SolidMolecular weight:389.91BKIDC-1553
CAS:BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45Talarozole (R enantiomer)
CAS:Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.Formula:C21H23N5SPurity:98%Color and Shape:SolidMolecular weight:377.51Rev 5975
CAS:Rev 5975 is a non-sulfhydryl ACE-inhibitor.Formula:C24H30N2O5Purity:98%Color and Shape:SolidMolecular weight:426.51hCAIX-IN-8
CAS:hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.Formula:C19H16N4O6Color and Shape:SolidMolecular weight:396.35PRRSV/CD163-IN-1
CAS:PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.Formula:C25H24FN5O5S2Color and Shape:SolidMolecular weight:557.62Xanthine oxidase-IN-4
CAS:Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.Formula:C15H13N5O2Color and Shape:SolidMolecular weight:295.3PDE4-IN-11
CAS:PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.Formula:C21H19FN2O2Color and Shape:SolidMolecular weight:350.39AVX-001
CAS:AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.Formula:C21H29F3OSColor and Shape:SolidMolecular weight:386.51Clethodim
CAS:Clethodim is a selective herbicide inhibiting acetyl-CoA carboxylase, effective on grasses with low environmental persistence and moderate toxicity to wildlife.Formula:C17H26ClNO3SPurity:99.99%Color and Shape:Light Yellow LiquidMolecular weight:359.91BI-4924
CAS:BI-4924 is a PHGDH inhibitor that disrupts serine biosynthesis by intracellular trapping and can be used to study metabolic disorders.Formula:C21H20Cl2N2O6SPurity:99.55%Color and Shape:SolidMolecular weight:499.36IDO-IN-11
CAS:IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).Formula:C19H23BrFN7O4SPurity:98%Color and Shape:SolidMolecular weight:544.4Glycogen phosphorylase-IN-1
CAS:Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.Formula:C17H15ClF2N4O4Purity:97.98% - 98.15%Color and Shape:SolidMolecular weight:412.78Senazodan hydrochloride
CAS:Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.Formula:C15H15ClN4OPurity:99.93%Color and Shape:SolidMolecular weight:302.76ENPP1 inhibitor 43
CAS:ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.Formula:C16H18N6O3SColor and Shape:SolidMolecular weight:374.42IHMT-PI3Kδ-372
CAS:IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.Formula:C26H23F2N7O2Purity:99.77%Color and Shape:SolidMolecular weight:503.5
