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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8625 products of "Metabolism"

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  • Ethyl phenylglyoxylate

    CAS:
    <p>Ethyl phenylglyoxylate (AI3 10033) is a simultaneous inhibitor and substrate of chicken liver carboxylesterase.</p>
    Formula:C10H10O3
    Purity:98.46%
    Color and Shape:Yellow Liquid
    Molecular weight:178.18
  • Z-Arg(Z)2-OH

    CAS:
    <p>Z-Arg(Z)2-OH can be used in the assay to screen proteolytic activities in mite homogenates.</p>
    Formula:C30H32N4O8
    Purity:99.1400%
    Color and Shape:Solid
    Molecular weight:576.6
  • ent-Tadalafil

    CAS:
    <p>ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS).</p>
    Formula:C22H19N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.4
  • Sodium lauroyl glutamate

    CAS:
    <p>Sodium lauroyl glutamate (Acylglutamate LS-11) is an amino acid detergent and increases the solubility of long-chain alkyl gallates such as alkyl gallates.</p>
    Formula:C17H30NNaO5
    Purity:97.13%
    Color and Shape:Solid
    Molecular weight:351.41
  • Bitertanol

    CAS:
    <p>Bitertanol (KWG 0599) is a triazole fungicide. Bitertanol inhibits demethylation, disrupts membrane function, and prevents sterol synthesis.</p>
    Formula:C20H23N3O2
    Purity:99.88%
    Color and Shape:Clear Browm Clear Liquid
    Molecular weight:337.42
  • Transketolase-IN-3

    CAS:
    <p>Transketolase-IN-3: potent TK inhibitor with herbicidal effects on DS and AR, useful for herbicide research.</p>
    Formula:C20H9ClF3NO3
    Color and Shape:Solid
    Molecular weight:403.74
  • sEH inhibitor-17

    CAS:
    <p>sEH inhibitor-17 (compound 4f) is an orally active soluble epoxide hydrolase (sEH) inhibitor with an IC50 value of 2.94 nM. This compound exhibits anti-inflammatory properties.</p>
    Formula:C18H21F3N2O4S
    Color and Shape:Solid
    Molecular weight:418.43
  • 3-O-Methyltolcapone

    CAS:
    <p>3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.</p>
    Formula:C15H13NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:287.27
  • GS-566500

    CAS:
    <p>GS-566500 is a compound of Sofosbuvir metabolite.</p>
    Formula:C13H19FN3O9P
    Color and Shape:Solid
    Molecular weight:411.28
  • DC-6-14

    CAS:
    <p>DC-6-14 is a cationic lipid known for its gene transfection activity, commonly utilized in the synthesis of liposomes.</p>
    Formula:C37H73ClN2O5
    Color and Shape:Solid
    Molecular weight:661.44
  • Flurtamone

    CAS:
    <p>Flurtamone is an agricultural chemical. Flurtamone mainly used as an herbicide.</p>
    Formula:C18H14F3NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.30
  • Leucylarginine

    CAS:
    <p>Leucylarginine hinders antinociception induced by L-arginine.</p>
    Formula:C12H25N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:287.36
  • Dihydro Dutasteride

    CAS:
    <p>Dihydro Dutasteride is a metabolite of Dutasteride. Dutasteride is an effective inhibitor of five α-reductase isozymes.</p>
    Formula:C27H32F6N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:530.55
  • Acetaminophen mercapturate

    CAS:
    <p>Paracetamol Mercapturate is a metabolite of Acetaminophen. It can also be used in the biological study of urinary antihypertensive drugs.</p>
    Formula:C13H16N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.34
  • ARN-6039

    CAS:
    <p>ARN-6039 is an oral RORγ inverse agonist for Autoimmune Neuroinflammation, active in HEK 293 cells and CD4+T cells.</p>
    Formula:C21H21F3N2O3
    Color and Shape:Solid
    Molecular weight:406.40
  • Thevetin A

    CAS:
    <p>Thevetin A is a useful organic compound for research related to life sciences. The catalog number is T124930 and the CAS number is 37933-66-7.</p>
    Formula:C42H64O19
    Color and Shape:Solid
    Molecular weight:872.955
  • Dimepiperate

    CAS:
    <p>Dimepiperate is an agent of biochemical.</p>
    Formula:C15H21NOS
    Color and Shape:Solid
    Molecular weight:263.40
  • PD 113413

    CAS:
    <p>PD 113413 is a metabolite of quinapril, an angiotensin-converting enzyme inhibitor for the treatment of hypertension and congestive heart failure.</p>
    Formula:C23H24N2O4
    Color and Shape:Solid
    Molecular weight:392.45
  • PPM1A-IN-1

    CAS:
    <p>PPM1A-IN-1 (Compound IV-4) is an inhibitor of the PP2C Ser/Thr protein phosphatase Mg2+/Mn2+-dependent 1A. It exhibits antibacterial activity against Mycobacterium tuberculosis.</p>
    Formula:C16H15BrFNO2
    Color and Shape:Solid
    Molecular weight:352.2
  • Trimosulfa

    CAS:
    <p>Trimosulfa is a combination of trimethoprim and sulfamethoxazole, an antibiotic combination. Sulfamethoxazole inhibits dihydropteroate synthase, while trimethoprim inhibits dihydrofolate reductase (dihydrofolate reductase), making it effective for mild to moderate bacterial infections against many Gram-negative and Gram-positive bacteria.</p>
    Formula:C24H29N7O6S
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:543.6
  • 1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine

    CAS:
    <p>1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.</p>
    Formula:C44H84NO8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:786.11
  • PNU-200579

    CAS:
    <p>PNU-200579 is a bio-active chemical.</p>
    Formula:C22H29NO3
    Color and Shape:Solid
    Molecular weight:355.47
  • 1,2-Dipalmitoyl-sn-glycerol 3-phosphate

    CAS:
    <p>1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.</p>
    Formula:C35H69O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:648.89
  • Prasugrel chloride impurity

    CAS:
    <p>Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.</p>
    Formula:C20H21ClFNO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.9
  • Proadifen

    CAS:
    <p>Proadifen is a non-selective cytochrome P450 enzymes inhibitor, preventing some types of drug metabolism.</p>
    Formula:C23H31NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.5
  • MDI-2268

    CAS:
    <p>MDI-2268, an inhibitor of plasma kallikrein inhibitor 1 (PAI-1), exhibits strong antithrombotic properties. It plays a role in regulating blood coagulation by promoting fibrinolysis and is applicable in research related to deep vein thrombosis.</p>
    Formula:C10H10F3N3O3
    Color and Shape:Solid
    Molecular weight:277.20
  • (+)-Xylariamide A

    CAS:
    <p>(+)-Xylariamide A is a probe used for mycobacterial and fungal carbonic anhydrase.</p>
    Formula:C14H14ClNO6
    Color and Shape:Solid
    Molecular weight:327.72
  • Difluoro atorvastatin

    CAS:
    <p>Difluoro atorvastatin: an atorvastatin impurity reducing blood lipids, inhibits SV-SMC proliferation/invasion (IC50: 0.39/2.39 μM).</p>
    Formula:C33H34F2N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:576.63
  • Buthidazole

    CAS:
    <p>Buthidazole is a herbicide for selective weed control in corn.</p>
    Formula:C10H16N4O2S
    Color and Shape:Solid
    Molecular weight:256.33
  • Nicodan Percutan

    CAS:
    <p>Nicodan Percutan (Propylnicotinat) is the propyl ester form of niacin, which is found in various animal and plant tissues to form the coenzymes NAD and NADP.</p>
    Formula:C9H11NO2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:165.19
  • Desmethylnortriptyline

    CAS:
    <p>Desmethylnortriptyline, a tricyclic antidepressant metabolite of nortriptyline and amitriptyline, treats depression.</p>
    Formula:C18H19N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.35
  • Chol-5-en-24-al-3β-ol

    CAS:
    <p>Chol-5-en-24-al-3β-ol is a steroid compound.</p>
    Formula:C24H38O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.56
  • Milvexian

    CAS:
    <p>Milvexian (BMS-986177) is an oral antithrombotic, reversibly inhibiting human/rabbit FXIa with K i of 0.11/0.38 nM.</p>
    Formula:C28H23Cl2F2N9O2
    Color and Shape:Solid
    Molecular weight:626.45
  • PTC-510 TFA salt

    CAS:
    <p>PTC-510 TFA salt inhibits hypoxia-induced VEGF expression.</p>
    Formula:C26H26BrN3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:524.48
  • Betrixaban

    CAS:
    <p>Betrixaban is a non-VKORC1 anticoagulant targeting factor Xa, with low hERG affinity, used to prevent VTE in adults with mobility issues.</p>
    Formula:C23H22ClN5O3
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:451.91
  • Tolrestat

    CAS:
    <p>Tolrestat (AY-27773) is a potent inhibitor of aldose reductase (IC50 = 35 nM).</p>
    Formula:C16H14F3NO3S
    Purity:98.89% - >99.99%
    Color and Shape:Solid
    Molecular weight:357.35
  • L-m-Tyrosine

    CAS:
    <p>L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.</p>
    Formula:C9H11NO3
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:181.19
  • 4-POBN

    CAS:
    <p>4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).</p>
    Formula:C7H9N3O
    Purity:99.60%
    Color and Shape:White Crystalline Powder
    Molecular weight:151.17
  • Tesaglitazar

    CAS:
    <p>Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα</p>
    Formula:C20H24O7S
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:408.47
  • PCI-27483

    CAS:
    <p>PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.</p>
    Formula:C26H24N6O9S
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:596.57
  • Calcipotriol monohydrate

    CAS:
    <p>Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.</p>
    Formula:C27H42O4
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:430.62
  • BIBB 515

    CAS:
    <p>BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.</p>
    Formula:C22H21ClN2O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:380.87
  • PF-05175157

    CAS:
    <p>PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,</p>
    Formula:C23H27N5O2
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:405.49
  • 3-Phenylbutyric acid

    CAS:
    <p>3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.</p>
    Formula:C10H12O2
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:164.2
  • E3330

    CAS:
    <p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>
    Formula:C21H30O6
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:378.46
  • 1-Decanesulfonic acid

    CAS:
    <p>1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.</p>
    Formula:C10H22O3S
    Color and Shape:Solid
    Molecular weight:222.35
  • BAY 59-9435

    CAS:
    <p>HSL-IN-2 is a selective inhibitor of Hormone Sensitive Lipase (HSL; IC50: 0.023 μM).</p>
    Formula:C14H22N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.34
  • S32826 disodium

    CAS:
    <p>autotaxin inhibitor</p>
    Formula:C21H36NNa2O4P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.47
  • SCH-351591

    CAS:
    <p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>
    Formula:C17H10Cl2F3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.18
  • Nebicapone

    CAS:
    <p>Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.</p>
    Formula:C14H11NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.24
  • CAY10487

    CAS:
    <p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>
    Formula:C13H15NO5
    Color and Shape:Solid
    Molecular weight:265.26
  • Clofenamide

    CAS:
    <p>Clofenamide is a low-ceiling sulfonamide diuretic.</p>
    Formula:C6H7ClN2O4S2
    Color and Shape:Solid
    Molecular weight:270.71
  • LG 101506

    CAS:
    <p>RXR modulator</p>
    Formula:C25H34F2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.53
  • OMDM-2

    CAS:
    <p>OMDM-2 is a metabolically stable and selective inhibitor of anandamide cellular uptake (ACU), exhibiting a Ki value of 3.0 μM in RBL-2H3 cells.</p>
    Formula:C27H45NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.65
  • Spiraprilat

    CAS:
    <p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>
    Formula:C20H26N2O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.56
  • hCA I-IN-1

    CAS:
    <p>hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).</p>
    Formula:C27H23N5O4S
    Color and Shape:Solid
    Molecular weight:513.57
  • ALDH1A1-IN-3

    CAS:
    <p>ALDH1A1-IN-3 selectively inhibits ALDH1A1, enhances HepG2 glucose consumption for metabolic research.</p>
    Formula:C31H36F3N5O4
    Color and Shape:Solid
    Molecular weight:599.64
  • 2'-O-Methyladenosine

    CAS:
    <p>2'-O-Methyladenosine, a methylated adenine residue is found in the urine of normals and adenosine deaminase deficient patients.</p>
    Formula:C11H15N5O4
    Purity:99.89%
    Color and Shape:White Solid
    Molecular weight:281.27
  • 93-O17O

    CAS:
    <p>93-O17O is a cationic lipidoid used in lipid nanoparticles for spleen-targeted delivery and genome editing in mice.</p>
    Formula:C44H83N3O6
    Color and Shape:Solid
    Molecular weight:750.15
  • Isospaglumate sodium

    CAS:
    <p>Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.</p>
    Formula:C11H16N2NaO8
    Color and Shape:Solid
    Molecular weight:327.245
  • (Rac)-RK-682

    CAS:
    <p>(Rac)-RK-682 racemate; inhibits PTP-1B, LMW-PTP, CDC-25B with IC50s: 8.6, 12.4, 0.7 µM respectively.</p>
    Formula:C21H36O5
    Color and Shape:Solid
    Molecular weight:368.51
  • OSMI-3

    CAS:
    <p>OSMI-3 is a potent and cell-permeable inhibitor of O-GlcNAc transferase (OGT) for the study of cancer and cardiovascular disease.</p>
    Formula:C32H35N3O9S2
    Purity:99.03% - 99.08%
    Color and Shape:Solid
    Molecular weight:669.77
  • NCT-506

    CAS:
    <p>NCT-506 is an orally bioavailable inhibitors of aldehyde dehydrogenase 1A1 (ALDH1A1) (IC50 of 7 nM).</p>
    Formula:C25H23FN4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:478.54
  • α-Glucosidase-IN-2

    CAS:
    <p>α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an</p>
    Formula:C17H11N3O2S2
    Color and Shape:Solid
    Molecular weight:353.42
  • JNJ-42314415

    CAS:
    <p>JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.</p>
    Formula:C19H23N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.42
  • LY 221068

    CAS:
    <p>LY 221068 is a potent antioxidant with anti-inflammatory activity.</p>
    Formula:C20H30N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.53
  • hCAIX/XII-IN-2

    CAS:
    <p>Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); &gt;10,000 nM (hCAI/II).</p>
    Formula:C19H14N2O4
    Color and Shape:Solid
    Molecular weight:334.33
  • ARN19874

    CAS:
    <p>ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].</p>
    Formula:C19H14N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.4
  • DO-264

    CAS:
    <p>DO-264 is an inhibitor of autohydrolase structural domain 12 (ABHD12) and an inhibitor of cellular LysoPS degradation that enhances LPS-induced phagocytosis.</p>
    Formula:C23H20Cl2F3N5O2S
    Purity:97.72% - 99.95%
    Color and Shape:Solid
    Molecular weight:558.4
  • TC-E 5005

    CAS:
    <p>PDE10A inhibitor</p>
    Formula:C15H18N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:270.33
  • MAGLi 432

    CAS:
    <p>MAGLi 432: Potent MAGL inhibitor, selective and reversible. IC50: 4.2 nM (human), 3.1 nM (mouse). Useful for neurological disorder research.</p>
    Formula:C22H24BrClN2O2
    Color and Shape:Solid
    Molecular weight:463.8
  • p-Valerylphenol

    CAS:
    p-Valerylphenol (NSC-49186) can be used to synthesize acylphenoxyacetic acid compounds.
    Formula:C11H14O2
    Purity:99.87%
    Color and Shape:White To Light Beige Powder
    Molecular weight:178.23
  • M8891

    CAS:
    <p>M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial &amp; tumor cell growth, antiangiogenic &amp; antitumor.</p>
    Formula:C20H17F2N3O3
    Color and Shape:Solid
    Molecular weight:385.36
  • GW844520

    CAS:
    <p>GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.</p>
    Formula:C20H15ClF3NO3
    Color and Shape:Solid
    Molecular weight:409.79
  • PF-06471553

    CAS:
    <p>PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).</p>
    Formula:C23H25N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:467.54
  • Oosponol

    CAS:
    <p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>
    Formula:C11H8O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:220.18
  • Propaquizafop

    CAS:
    <p>Propaquizafop, a phenoxyisopropionic acid derivative, is used as a herbicide.</p>
    Formula:C22H22ClN3O5
    Purity:98%
    Color and Shape:Colourless-To-Brown Crystals
    Molecular weight:443.88
  • α-Glucosidase-IN-3

    CAS:
    <p>α-Glucosidase-IN-3 is an oleanolic acid oxime ester derivative targeting α-glucosidase and α-amylase with an IC50 value of 0.35 μM for α-glucosidase.</p>
    Formula:C39H53NO4
    Color and Shape:Solid
    Molecular weight:599.84
  • Acetylhydrolase-IN-1

    CAS:
    <p>Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).</p>
    Formula:C23H48NO7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.6
  • T-1095A

    CAS:
    <p>T-1095A, a T-1095 metabolite, inhibits SGLTs, lowers blood glucose, improves glucose intolerance in mice, and prevents neuropathy in diabetic rats.</p>
    Formula:C24H26O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.46
  • M77976

    CAS:
    <p>M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.</p>
    Formula:C17H16N2O3
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:296.32
  • Crilvastatin

    CAS:
    <p>Crilvastatin (PMD 387) is an HMGCR inhibitor with cholesterol-lowering activity that inhibits cholesterol uptake in rats with hereditary hypercholesterolemia.</p>
    Formula:C14H23NO3
    Purity:98.69% - 99.54%
    Color and Shape:Solid
    Molecular weight:253.34
  • Tanogitran

    CAS:
    <p>Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.</p>
    Formula:C25H31N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.56
  • KT109

    CAS:
    <p>KT109 is a DAGLβ inhibitor (IC50=42nM), lessens LPS allodynia in mice without tolerance, and has no major side effects.</p>
    Formula:C27H26N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.52
  • SGK1-IN-2

    CAS:
    <p>SGK1-IN-2 (14h) is a selective inhibitor of SGK1 (serum and glucocorticoid regulated kinase 1)(with an IC50 of 5 nM at 10 μM ATP concentration).</p>
    Formula:C17H12Cl2N6O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.29
  • CDK2-IN-11

    CAS:
    <p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>
    Formula:C18H14ClN7O2S
    Color and Shape:Solid
    Molecular weight:427.87
  • Benserazide

    CAS:
    <p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>
    Formula:C10H15N3O5
    Color and Shape:Solid
    Molecular weight:257.24
  • Leniquinsin

    CAS:
    <p>Leniquinsin is an antihypertensive compound. It is a phosphodiesterase inhibitor and a potent vasodilator.</p>
    Formula:C20H20N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.38
  • Aldophosphamide

    CAS:
    <p>Aldophosphamide possesses apoptotic antitumor activity.</p>
    Formula:C7H15Cl2N2O3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.09
  • AK-106

    CAS:
    <p>AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.</p>
    Formula:C26H25N3O3
    Color and Shape:Solid
    Molecular weight:427.49
  • Glutamamide

    CAS:
    <p>Glutamamide is an anticancer drug.</p>
    Formula:C5H11N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:145.16
  • IDO1/TDO-IN-2

    CAS:
    <p>IDO1/TDO-IN-2: IDO1/TDO inhibitor; IC50s: IDO1, 0.1μM; TDO, 0.07μM; potential for cancer research.</p>
    Formula:C16H9N3O2
    Color and Shape:Solid
    Molecular weight:275.26
  • α-Amylase/α-Glucosidase-IN-1

    CAS:
    <p>α-Amylase/α-Glucosidase-IN-1 (compound 33) is an effective inhibitor of α-amylase/α-glucosidase with IC 50 s of 2.01, 2.09 μM for α-amylase and α-glucosidase,</p>
    Formula:C11H9N5
    Color and Shape:Solid
    Molecular weight:211.22
  • L-Xylulose

    CAS:
    <p>L-Xylulose: a rare sugar, key in metabolism, α-glucosidase inhibitor, lowers glucose, precursor to antiviral drug components.</p>
    Formula:C5H10O5
    Color and Shape:Solid
    Molecular weight:150.13
  • LAZABEMIDE

    CAS:
    <p>Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and &gt; 100 μM for MAO-B and MAO-A respectively).</p>
    Formula:C8H10ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:199.64
  • LCL521 dihydrochloride

    CAS:
    <p>LCL521 dihydrochloride is a dual inhibitor of ACDase and ASMase, modulating sphingolipid metabolism with potential in cancer and metabolic research.</p>
    Formula:C31H54Cl2N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.69
  • Acetyltrialanine

    CAS:
    <p>Acetyltrialanine is a dipeptide compound that binds at two sites on the Tb+3-pancreatic elastase complex and can be used as a nitrogen source.</p>
    Formula:C11H19N3O5
    Purity:99.53%
    Color and Shape:White Powder
    Molecular weight:273.29
  • BNS

    CAS:
    <p>BNS is a potent, prolyl-hydroxylase 2 (PHD2)-selective inhibitor.</p>
    Formula:C18H16N2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.46
  • CGS 35601

    CAS:
    <p>CGS 35601 is a single molecule inhibitor of triple vasopeptidase.</p>
    Formula:C23H31N3O4S
    Color and Shape:Solid
    Molecular weight:445.57
  • hCAIX/XII-IN-3

    CAS:
    <p>Compound 6q inhibits hCAIX/CAXII; K i : hCAI &gt;10000 nM, hCAII &gt;10000 nM, hCAIX 66.2 nM, hCAXII 4.4 nM.</p>
    Formula:C20H13F3N2O4
    Color and Shape:Solid
    Molecular weight:402.32
  • hCAII-IN-2

    CAS:
    <p>hCAII-IN-2 inhibits human carbonic anhydrases I, II, IX, XII with Ki values of 261.4, 3.8, 19.6, 45.2 nM respectively.</p>
    Formula:C25H18ClN5O4S
    Color and Shape:Solid
    Molecular weight:519.96
  • UKI-1

    CAS:
    <p>UKI-1 is a urokinase-type plasminogen activator system synthetic inhibitor.</p>
    Formula:C32H47N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:613.81
  • Genz-669178

    CAS:
    <p>Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).</p>
    Formula:C17H14N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.38
  • Dacisteine

    CAS:
    <p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>
    Formula:C7H11NO4S
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:205.23
  • IM176OUT05

    CAS:
    <p>IM176OUT05 activates stem cell metabolism with hair regrowth-promoting effects.</p>
    Formula:C11H17N5
    Color and Shape:Solid
    Molecular weight:219.29
  • L 656224

    CAS:
    <p>L 656224 is a 5-LO inhibitor.</p>
    Formula:C20H21ClO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.83
  • Fenleuton

    CAS:
    <p>Fenleuton is a 5-lipoxygenase inhibitor.</p>
    Formula:C17H15FN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:314.31
  • RP 73163 Racemate

    CAS:
    <p>RP 73163 Racemate is the racemate of RP 73163. RP 73163 is a potent inhibitor of ACAT, shows cholesterol lowering activity.</p>
    Formula:C25H28N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.58
  • Dimethyl-bisphenol A

    CAS:
    <p>DMBPA inhibits HIF-1α, promotes its degradation by detaching Hsp90, and reduces Vegfa mRNA expression.</p>
    Formula:C17H20O2
    Color and Shape:Solid
    Molecular weight:256.34
  • GKA-22

    CAS:
    <p>GKA-22 is a human glucokinase allosteric activator in the absence of glucose.</p>
    Formula:C22H22N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.49
  • HCAIX-IN-2

    CAS:
    <p>HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).</p>
    Formula:C19H16N8O4S
    Color and Shape:Solid
    Molecular weight:452.45
  • RORγt inverse agonist 30

    CAS:
    <p>RORγt inverse agonist 30 (Compound 1) is a potent RORγt inverse agonist (IC50: 46 nM).</p>
    Formula:C24H31N3O3S
    Color and Shape:Solid
    Molecular weight:441.59
  • Desfluoro-atorvastatin

    CAS:
    <p>Desfluoro-atorvastatin is an impurity of atorvastatin, an oral HMG-CoA reductase inhibitor that lowers blood lipids.</p>
    Formula:C33H36N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.65
  • KM04416

    CAS:
    <p>KM04416 is a GPD2 inhibitor that inhibits LUAD progression by modulating immune cell infiltration.</p>
    Formula:C12H11NO3S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:249.29
  • Mevalonic acid

    CAS:
    <p>Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.</p>
    Formula:C6H12O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:148.16
  • XEN103

    CAS:
    <p>XEN103 is a potent and selective Stearoyl-CoA Desaturase-1 inhibitor.</p>
    Formula:C22H23F4N5O2
    Color and Shape:Solid
    Molecular weight:465.44
  • γ-Methylleucine

    CAS:
    <p>Gamma-Methylleucine (2-Amino-3-tert-butylpropionic acid) is an auxiliary for copper-catalyzed asymmetric Michael reactions.</p>
    Formula:C7H15NO2
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:145.2
  • FKGK11

    CAS:
    <p>FKGK11 is a potent inhibitor of GVIA iPLA2.</p>
    Formula:C13H13F5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.23
  • Piragliatin

    CAS:
    <p>Piragliatin (RO4389620) activates glucokinase, boosts insulin, and lowers glucose in type 2 diabetes.</p>
    Formula:C19H20ClN3O4S
    Color and Shape:Solid
    Molecular weight:421.9
  • Seviteronel racemate

    CAS:
    <p>Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase.</p>
    Formula:C18H17F4N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.34
  • Saterinone hydrochloride

    CAS:
    <p>Saterinone hydrochloride is an inhibitor of phosphodiesterase III (PDE III).</p>
    Formula:C27H31ClN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.01
  • Amastatin

    CAS:
    <p>Amastatin is a non-toxic inhibitor of aminopeptidase A and leucine aminopeptidase, and its Ki for aminopeptidase A is 1 μM .</p>
    Formula:C21H38N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.55
  • JTV-519

    CAS:
    <p>K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by</p>
    Formula:C25H33ClN2O2S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:461.06
  • Seviteronel R enantiomer

    CAS:
    <p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>
    Formula:C18H17F4N3O3
    Purity:97.97% - >99.99%
    Color and Shape:Solid
    Molecular weight:399.34
  • ARL-67156 trisodium salt hydrate

    CAS:
    <p>ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.</p>
    Formula:C15H24Br2N5O12P3
    Color and Shape:Solid
    Molecular weight:719.11
  • (Rac)-Etavopivat

    CAS:
    <p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>
    Formula:C22H23N3O6S
    Color and Shape:Solid
    Molecular weight:457.5
  • Darexaban glucuronide

    CAS:
    <p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>
    Formula:C33H38N4O10
    Color and Shape:Solid
    Molecular weight:650.68
  • CDK2-IN-12

    CAS:
    <p>CDK2-IN-12 (10b), potent CDK2 inhibitor, IC50: 11.6 μM; inhibits hCA I/II/IX/XII, KI: 3534/638.4/44.3/48.8 nM; anti-cancer properties.</p>
    Formula:C20H17N9O2S
    Color and Shape:Solid
    Molecular weight:447.47
  • GS 389

    CAS:
    <p>GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.</p>
    Formula:C19H23NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:313.39
  • SAR629

    CAS:
    <p>SAR-629 is an MGL inhibitor or 2-AG degradation inhibitor.</p>
    Formula:C20H19F2N5O
    Color and Shape:Solid
    Molecular weight:383.39
  • Fexarine

    CAS:
    <p>Fexarine is a potent, selective agonist of farnesoid X receptor.</p>
    Formula:C31H31NO5
    Color and Shape:Solid
    Molecular weight:497.58
  • PDE-9 inhibitor

    CAS:
    <p>PDE-9 inhibitor is used for treatment neurodegenerative diseases.</p>
    Formula:C22H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.48
  • Arcapillin

    CAS:
    <p>Arcapillin, an anticancer agent, induces apoptosis mediated at least in part by the ERS pathway and inhibits hepatoma tumor growth.</p>
    Formula:C18H16O8
    Color and Shape:Solid
    Molecular weight:360.31
  • hCAIX-IN-11

    CAS:
    <p>hCAIX-IN-11 inhibits carbonic anhydrases IX &amp; XII with Ki of 32.7 nM &amp; 623.5 nM, respectively.</p>
    Formula:C21H15ClN4O3
    Color and Shape:Solid
    Molecular weight:406.82
  • L-Canaline

    CAS:
    <p>L-Canaline is a nonprotein amino acid with IC50 of 297 nM against malaria, anticancer properties, and blocks ornithine aminotransferase.</p>
    Formula:C4H10N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:134.13
  • Otamixaban

    CAS:
    <p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>
    Formula:C25H26N4O4
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:446.5
  • FASN-IN-5

    CAS:
    <p>FASN-IN-5 is a FASN inhibitor, useful for studying cancer and metabolic diseases.</p>
    Formula:C29H26N4O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:462.54
  • ATX inhibitor 19

    CAS:
    <p>ATX inhibitor 19 is a potent inhibitor of ATX (IC50: 156 nM).</p>
    Formula:C28H33ClN6O2S
    Color and Shape:Solid
    Molecular weight:553.12
  • PKR activator 1

    CAS:
    <p>PKR activator 1 is a potent activator of pyruvate kinase-R (PKR).</p>
    Formula:C16H14N8OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.47
  • Fodipir

    CAS:
    <p>Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cell</p>
    Formula:C22H32N4O14P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:638.46
  • Carbazomycin B

    CAS:
    <p>Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).</p>
    Formula:C15H15NO2
    Color and Shape:Solid
    Molecular weight:241.29
  • Anticancer agent 70

    CAS:
    <p>Compound 21 is a powerful anticancer agent with cytotoxicity against various cancers, causing cell cycle arrest and affecting p53/p21 levels and mitochondria.</p>
    Formula:C13H9Cl2N3O2S
    Color and Shape:Solid
    Molecular weight:342.2
  • Asp-AMS

    CAS:
    <p>Asp-AMS is a strong competitive inhibitor of the mitochondrial enzyme and also an aspartyl-tRNA synthetase inhibitor.</p>
    Formula:C14H19N7O9S
    Color and Shape:Solid
    Molecular weight:461.41
  • PDE1-IN-3

    CAS:
    <p>PDE1-IN-3 is a selective inhibitor of human phosphodiesterase 1 (PDE1).</p>
    Formula:C18H24N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.41
  • Enpp-1-IN-6

    CAS:
    <p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>
    Formula:C22H28N4O5S
    Color and Shape:Solid
    Molecular weight:460.55
  • PDE10-IN-5

    CAS:
    <p>PDE10-IN-5 is a phosphodiesterase 10 (PDE 10) inhibitor that can be used to study certain central nervous system disorders.</p>
    Formula:C26H19F3N4O
    Color and Shape:Solid
    Molecular weight:460.45
  • ML-262

    CAS:
    <p>ML-262 is an effective inhibitor of hepatic lipid droplet formation and is used in studies of non-alcoholic fatty liver disease.</p>
    Formula:C27H32N2O4S
    Color and Shape:Solid
    Molecular weight:480.62
  • Phortress free base

    CAS:
    <p>Phortress free base is a P450 CYP1A1-activated antitumor prodrug with antitumor activity.</p>
    Formula:C20H23FN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.49
  • LY 56110

    CAS:
    <p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>
    Formula:C17H12Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.2
  • hCAI/II-IN-1

    CAS:
    <p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>
    Formula:C18H29N5O3S3
    Color and Shape:Solid
    Molecular weight:459.65
  • LEI-106

    CAS:
    <p>LEI-106 is an effective dual inhibitor of DAGL-α and ABHD6, with Ki values of 0.7 and 0.8 μM respectively, for obesity and metabolic syndrome research.</p>
    Formula:C26H27NO6S
    Color and Shape:Solid
    Molecular weight:481.56
  • Phenylthiazolylthiourea

    CAS:
    <p>Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.</p>
    Formula:C10H9N3S2
    Color and Shape:Solid
    Molecular weight:235.33
  • LY367385

    CAS:
    <p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>
    Formula:C10H11NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.2
  • SHP2 inhibitor LY6

    CAS:
    <p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>
    Formula:C30H27Cl2N3O4
    Color and Shape:Solid
    Molecular weight:564.46
  • PKM2 activator 3

    CAS:
    <p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>
    Formula:C15H11ClF2N2O3S
    Color and Shape:Solid
    Molecular weight:372.77
  • Afegostat

    CAS:
    <p>Afegostat is a pharmacological chaperone that specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum with high affinity.</p>
    Formula:C6H13NO3
    Purity:98%
    Color and Shape:Yellow Low-Melting Solid
    Molecular weight:147.17
  • Epiroprim

    CAS:
    <p>Epiroprim (Ro11-8958) is a selective dihydrofolate reductase (DHFR) inhibitor with antibacterial activity, inhibiting Staphylococcus and Streptococcus.</p>
    Formula:C19H23N5O2
    Purity:99.68% - >99.99%
    Color and Shape:Solid
    Molecular weight:353.42
  • LB42908

    CAS:
    <p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>
    Formula:C32H31N5O3
    Color and Shape:Solid
    Molecular weight:533.62
  • N-Oleoyl Leucine

    CAS:
    <p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>
    Formula:C24H45NO3
    Purity:98.25%
    Color and Shape:Solid
    Molecular weight:395.62
  • MEDS433

    CAS:
    <p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>
    Formula:C20H11F4N3O2
    Color and Shape:Solid
    Molecular weight:401.31
  • KT185

    CAS:
    KT185 is an orally-bioavailable and brain-penetrant ABHD6 inhibitor (IC50: 0.21 nM in Neuro2A cells).
    Formula:C32H33N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.64
  • Loxoprofenol-SRS

    CAS:
    <p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>
    Formula:C15H20O3
    Color and Shape:Solid
    Molecular weight:248.32
  • SR1555 HCl

    CAS:
    <p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>
    Formula:C22H22F6N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.41
  • IDO-IN-4

    CAS:
    <p>IDO-IN-4 is an indoleamine 2,3-dioxygenase 1 (IDO-1) inhibitor.</p>
    Formula:C26H35N3O3
    Color and Shape:Solid
    Molecular weight:437.57
  • Ambuphylline

    CAS:
    <p>Ambuphylline (Bufylline) is a theophylline derivative and bronchodilator for asthma and lung disease research.</p>
    Formula:C11H19N5O3
    Color and Shape:Solid
    Molecular weight:269.305
  • Talarozole (R enantiomer)

    CAS:
    <p>Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.</p>
    Formula:C21H23N5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.51
  • Quetiapine sulfoxide

    CAS:
    <p>Quetiapine sulfoxide: Main metabolite of Quetiapine, a 5-HT agonist &amp; dopamine antagonist antipsychotic.</p>
    Formula:C21H25N3O3S
    Purity:98%
    Color and Shape:Pale Yellow Solid
    Molecular weight:399.51
  • GlcN-6-P Synthase-IN-1

    CAS:
    <p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase &amp; CYP3A4. Has antimicrobial activity and CNS penetration.'</p>
    Formula:C20H21N7S
    Color and Shape:Solid
    Molecular weight:391.49
  • PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Formula:C17H19Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.27
  • hDHODH-IN-11

    CAS:
    <p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>
    Formula:C24H23N3O3
    Color and Shape:Solid
    Molecular weight:401.46
  • Rev 5975

    CAS:
    <p>Rev 5975 is a non-sulfhydryl ACE-inhibitor.</p>
    Formula:C24H30N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.51
  • Nampt activator-3

    CAS:
    <p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37
  • 14-dehydro Zymostenol

    CAS:
    <p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>
    Formula:C27H44O
    Color and Shape:Solid
    Molecular weight:384.64
  • hCAI/II-IN-2

    CAS:
    <p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>
    Formula:C12H12N4O5S2
    Color and Shape:Solid
    Molecular weight:356.38
  • 103D5R

    CAS:
    <p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>
    Formula:C20H21N3O2
    Color and Shape:Solid
    Molecular weight:335.4
  • AVX-001

    CAS:
    <p>AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.</p>
    Formula:C21H29F3OS
    Color and Shape:Solid
    Molecular weight:386.51
  • S07-2010

    CAS:
    <p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>
    Formula:C19H21N3O3S
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:371.45
  • ONO-6126

    CAS:
    <p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>
    Formula:C20H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.45
  • IQA

    CAS:
    <p>IQA is a casein kinase 2 (CK2) inhibitor.</p>
    Formula:C17H12N2O3
    Color and Shape:Solid
    Molecular weight:292.29
  • 11β-HSD1-IN-10

    CAS:
    <p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>
    Formula:C16H10F3NO2
    Color and Shape:Solid
    Molecular weight:305.25
  • FR-221647

    CAS:
    <p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>
    Formula:C14H17N3O2
    Color and Shape:Solid
    Molecular weight:259.3
  • CAY10761

    CAS:
    <p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-&lt;0.125 mM).</p>
    Formula:C7H8N4O2S2
    Color and Shape:Solid
    Molecular weight:244.29
  • IHMT-PI3Kδ-372

    CAS:
    <p>IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.</p>
    Formula:C26H23F2N7O2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:503.5
  • Ciraparantag

    CAS:
    <p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>
    Formula:C22H48N12O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:512.7
  • Sp-cAMPS

    CAS:
    <p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>
    Formula:C10H12N5O5PS
    Color and Shape:Solid
    Molecular weight:345.27
  • hCAI/II-IN-3

    CAS:
    <p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>
    Formula:C16H18N4O4S2
    Color and Shape:Solid
    Molecular weight:394.47
  • Kurasoin B

    CAS:
    <p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>
    Formula:C18H17NO2
    Color and Shape:Solid
    Molecular weight:279.33
  • YCT529 free acid

    CAS:
    <p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>
    Formula:C29H25NO3
    Color and Shape:Solid
    Molecular weight:435.51
  • Glyoxalase I inhibitor

    CAS:
    <p>Glyoxalase I inhibitor, a candidate for anticancer agents, is a potent Glyoxalase I (GLO1) inhibitor.</p>
    Formula:C21H30BrClN4O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:613.91
  • Izumerogant

    CAS:
    <p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>
    Formula:C22H18ClF4N5O2
    Color and Shape:Solid
    Molecular weight:495.86
  • Trandolaprilate hydrate

    CAS:
    <p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>
    Formula:C22H32N2O6
    Color and Shape:Solid
    Molecular weight:420.5
  • Argininic acid

    CAS:
    <p>Argininic acid is an α-amino acid used in the biosynthesis of proteins.</p>
    Formula:C6H13N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:175.19
  • ASP3662

    CAS:
    <p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>
    Formula:C19H16ClF3N4O2
    Color and Shape:Solid
    Molecular weight:424.8
  • TM-1

    CAS:
    <p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>
    Formula:C26H32N2O6
    Color and Shape:Solid
    Molecular weight:468.54
  • Atreleuton

    CAS:
    <p>Atreleuton (ABT-761), reversible oral 5-LO inhibitor, selectively blocks leukotriene formation.</p>
    Formula:C16H15FN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.37
  • 4,5,6,7-Tetrabromobenzimidazole

    CAS:
    <p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>
    Formula:C7H2Br4N2
    Color and Shape:Solid
    Molecular weight:433.72
  • CAY10486

    CAS:
    <p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>
    Formula:C19H19NO4
    Color and Shape:Solid
    Molecular weight:325.36
  • Valibose

    CAS:
    <p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>
    Formula:C10H21NO6
    Color and Shape:Solid
    Molecular weight:251.28
  • (R)-Irsenontrine

    CAS:
    <p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>
    Formula:C22H22N4O3
    Color and Shape:Solid
    Molecular weight:390.44
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81