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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8595 products of "Metabolism"

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  • Butaperazine maleate

    CAS:
    <p>Butaperazine maleate, a phenothiazine derivative, is an antipsychotic.</p>
    Formula:C32H39N3O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:641.73
  • PF-4191834

    CAS:
    <p>PF-4191834: Non-iron, non-redox 5-LOX inhibitor, IC50 = 229 nM, 300x selective over 12/15-LOX, inactive on COX enzymes.</p>
    Formula:C22H23N3O2S
    Purity:99.83% - 99.98%
    Color and Shape:Solid
    Molecular weight:393.5
  • Nampt-IN-9

    CAS:
    <p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>
    Formula:C26H33N3O4
    Color and Shape:Solid
    Molecular weight:451.56
  • SU 10603

    CAS:
    <p>SU 10603 is a specific inhibitor of 17α-hydroxylase (also known as CYP17A1 and P450c17) used to study steroid hormone synthesis.</p>
    Formula:C15H12ClNO
    Purity:99.93% - 99.96%
    Color and Shape:Solid
    Molecular weight:257.72
  • Autotaxin-IN-1

    CAS:
    <p>Autotaxin-IN-1: strong inhibitor for osteoarthritis pain; IC50=2.2 nM; good PK and PK/PD.</p>
    Formula:C21H23N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.45
  • CD 2314

    CAS:
    <p>CD2314 is a potent and subtype-selective RARβ receptor agonist with a Kd of 195 nM in S91 melanoma cells [1].</p>
    Formula:C23H24O2S
    Color and Shape:Solid
    Molecular weight:364.5
  • ABL127

    CAS:
    <p>ABL127 inhibits PME-1 with IC50s of 6.4 nM in HEK293T cells and 4.2 nM in MDA-MB-231 cells.</p>
    Formula:C17H20N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.35
  • Zofenoprilat arginine

    CAS:
    <p>Zofenoprilat arginine is an antihypertensive.</p>
    Formula:C21H33N5O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:499.65
  • WAY-213613

    CAS:
    <p>WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.</p>
    Formula:C16H13BrF2N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.19
  • Besigliptin Tosylate

    CAS:
    <p>Besigliptin Tosylate, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>
    Formula:C25H36FN5O5S
    Color and Shape:Solid
    Molecular weight:537.65
  • A 924

    CAS:
    <p>A 924 is an amino acid derivative with antineoplastic activity.</p>
    Formula:C30H57N7O11
    Color and Shape:Solid
    Molecular weight:691.81
  • Renytoline

    CAS:
    <p>Renytoline is a new anti-inflammatory of arthritis.</p>
    Formula:C21H16N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.37
  • ST-1892

    CAS:
    <p>ST-1892 is a soluble partial FXR agonist.</p>
    Formula:C16H12N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.28
  • Brofaromine

    CAS:
    Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).
    Formula:C14H16BrNO2
    Color and Shape:Solid
    Molecular weight:310.19
  • Lith-O-Asp

    CAS:
    <p>Lith-O-Asp is a sialytransferase (ST) inhibitor,(IC50s:12-37 μM).</p>
    Formula:C28H45NO6
    Color and Shape:Solid
    Molecular weight:491.66
  • Anticancer agent 70

    CAS:
    <p>Compound 21 is a powerful anticancer agent with cytotoxicity against various cancers, causing cell cycle arrest and affecting p53/p21 levels and mitochondria.</p>
    Formula:C13H9Cl2N3O2S
    Color and Shape:Solid
    Molecular weight:342.2
  • KM04416

    CAS:
    <p>KM04416 is a GPD2 inhibitor that inhibits LUAD progression by modulating immune cell infiltration.</p>
    Formula:C12H11NO3S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:249.29
  • HS80

    CAS:
    <p>HS-80, a Fasnall enantiomer, selectively inhibits FASN, blocking lipid synthesis (IC50: 7.13 μM).</p>
    Formula:C19H22N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.47
  • NE21650

    CAS:
    <p>NE21650, a bisphosphonate, inhibits isopentenyl diphosphate isomerase and farnesyl diphosphate synthase.</p>
    Formula:C8H13NO7P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.14
  • PDE1-IN-3

    CAS:
    <p>PDE1-IN-3 is a selective inhibitor of human phosphodiesterase 1 (PDE1).</p>
    Formula:C18H24N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.41
  • Brocresine

    CAS:
    <p>Brocresine is an aromatic L-amino acid decarboxylase inhibitor. It has both a peripheral and central action.</p>
    Formula:C7H8BrNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:218.05
  • KB 5666

    CAS:
    <p>KB 5666, a quinazoline derivative, is a lipid peroxidation inhibitor. It protects the brain from both cellular and functional consequences of ischemia.</p>
    Formula:C24H32N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.54
  • PF04471141 HCl

    CAS:
    <p>PF-04471141 is an effective and selective inhibitor of the calcium-activated phosphodiesterase PDE1 (IC50 = 35 nM).</p>
    Formula:C16H24ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.83
  • Enpp-1-IN-6

    CAS:
    <p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>
    Formula:C22H28N4O5S
    Color and Shape:Solid
    Molecular weight:460.55
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Formula:C24H35ClN2O5
    Color and Shape:Solid
    Molecular weight:467
  • VP3.15

    CAS:
    <p>VP3.15 is an orally bioavailable and CNS-penetrant dual inhibitor of phosphodiesterase (PDE)7- GSK3 (IC50s: 1.59 μM and 0.88 μM for PDE7 and GSK-3).</p>
    Formula:C20H22N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.48
  • Quinaprilat

    CAS:
    <p>Quinaprilat inhibits angiotensin converting enzyme.</p>
    Formula:C23H26N2O5
    Purity:98%
    Color and Shape:Crystalline Solid
    Molecular weight:410.46
  • Fadrozole HCl hydrate

    CAS:
    <p>Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.</p>
    Formula:C14H13N3ClHH2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.74
  • KT185

    CAS:
    <p>KT185 is an orally-bioavailable and brain-penetrant ABHD6 inhibitor (IC50: 0.21 nM in Neuro2A cells).</p>
    Formula:C32H33N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.64
  • TM6008

    CAS:
    <p>TM6008 is an inhibitor of prolyl hydroxylase that protects against cell death after hypoxia.</p>
    Formula:C21H17N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.39
  • ML368

    CAS:
    <p>ML368 is a selective inhibitor of CYP3A4.</p>
    Formula:C26H18N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.46
  • IDH-C227

    CAS:
    <p>IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.</p>
    Formula:C30H31FN4O2
    Color and Shape:Solid
    Molecular weight:498.59
  • UK-500001

    CAS:
    <p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>
    Formula:C26H24F3N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:499.48
  • 2-Hydroxy atorvastatin calcium salt

    CAS:
    <p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>
    Formula:C33H34FN2O60·5Ca
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:593.68
  • VU0155056

    CAS:
    <p>VU0155056 is a dual PLD1/2 inhibitor with IC50 &lt; 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>
    Formula:C25H26N4O2
    Purity:98.6% - 99.15%
    Color and Shape:Solid
    Molecular weight:414.5
  • JTV-519

    CAS:
    <p>K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by</p>
    Formula:C25H33ClN2O2S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:461.06
  • LYPLAL1-IN-1

    CAS:
    <p>LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.</p>
    Formula:C29H29N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.59
  • Gallopamil hydrochloride

    CAS:
    <p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>
    Formula:C28H41ClN2O5
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:521.09
  • MP-10 succinate

    CAS:
    <p>MP-10 succinate is a potent and specific inhibitor of PDE10A.</p>
    Formula:C29H26N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.54
  • NSC117079

    CAS:
    <p>NSC117079 is a novel PHLPP1/2 (Pleckstrin homology domain and leucine rich repeat protein phosphatase) inhibitor that activates neuronal AKT .</p>
    Formula:C20H15N3O7S2
    Purity:98.11%
    Color and Shape:Solid
    Molecular weight:473.48
  • Semotiadil recemate fumarate

    CAS:
    <p>Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.</p>
    Formula:C33H36N2O10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:652.71
  • SHP2 inhibitor LY6

    CAS:
    <p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>
    Formula:C30H27Cl2N3O4
    Color and Shape:Solid
    Molecular weight:564.46
  • PKM2 activator 3

    CAS:
    <p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>
    Formula:C15H11ClF2N2O3S
    Color and Shape:Solid
    Molecular weight:372.77
  • Desfluoro-atorvastatin

    CAS:
    <p>Desfluoro-atorvastatin is an impurity of atorvastatin, an oral HMG-CoA reductase inhibitor that lowers blood lipids.</p>
    Formula:C33H36N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.65
  • Arfolitixorin

    CAS:
    <p>Arfolitixorin is an antifolate modulator.</p>
    Formula:C20H23N7O6
    Color and Shape:Solid
    Molecular weight:457.44
  • (R)-Bromoenol lactone

    CAS:
    <p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>
    Formula:C16H13BrO2
    Color and Shape:Solid
    Molecular weight:317.18
  • Migoprotafib

    CAS:
    <p>Migoprotafib (GDC-1971) is a potent and highly selective SHP2 (Src Homology-2 Domain-Containing Phosphatase 2) inhibitor for advanced solid tumours.</p>
    Formula:C25H26N8O
    Color and Shape:Solid
    Molecular weight:454.53
  • LB42908

    CAS:
    <p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>
    Formula:C32H31N5O3
    Color and Shape:Solid
    Molecular weight:533.62
  • ONO-6126

    CAS:
    <p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>
    Formula:C20H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.45
  • N-Oleoyl Leucine

    CAS:
    <p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>
    Formula:C24H45NO3
    Purity:98.25%
    Color and Shape:Solid
    Molecular weight:395.62
  • Pemetrexed tromethamine

    CAS:
    <p>Pemetrexed tromethamine is a chemotherapy drug used for pleural mesothelioma and non-small cell lung cancer.</p>
    Formula:C20H21N5O6·2C4H11NO3·2H2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:705.72
  • MEDS433

    CAS:
    <p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>
    Formula:C20H11F4N3O2
    Color and Shape:Solid
    Molecular weight:401.31
  • Lu AF58801

    CAS:
    <p>Lu AF58801 is a brain penetrant positive allosteric and selective modulator of alpha-7 nicotinic acetylcholine receptors.</p>
    Formula:C20H23NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:325.4
  • Disulfamide

    CAS:
    <p>Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.</p>
    Formula:C7H9ClN2O4S2
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:284.74
  • Afegostat D-Tartrate

    CAS:
    <p>Afegostat D-Tartrate: pharmacological chaperone, reversibly binds acid-β-glucosidase in ER with high affinity.</p>
    Formula:C10H19NO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.26
  • Loxoprofenol-SRS

    CAS:
    <p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>
    Formula:C15H20O3
    Color and Shape:Solid
    Molecular weight:248.32
  • VDM 11

    CAS:
    <p>anandamide transport inhibitor</p>
    Formula:C27H39NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.6
  • Entacapone sodium salt

    CAS:
    <p>Entacapone sodium salt, a potent peripheral COMT inhibitor (IC50=151 nM), hinders α-syn/β-amyloid aggregation and protects PC12 cells.</p>
    Formula:C14H15N3NaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.28
  • DNJNAc

    CAS:
    <p>DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.</p>
    Formula:C8H16N2O4
    Purity:98.65% - 99.37%
    Color and Shape:Solid
    Molecular weight:204.22
  • Razaxaban hydrochloride

    CAS:
    <p>Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.</p>
    Formula:C24H21ClF4N8O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:564.92
  • L-5-BromoTryptophan

    CAS:
    <p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>
    Formula:C11H11BrN2O2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:283.12
  • BMS270394

    CAS:
    <p>BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.</p>
    Formula:C23H26FNO4
    Color and Shape:Solid
    Molecular weight:399.46
  • CID-7309015

    CAS:
    <p>CID-7309015 inhibits TDP1, slows malaria parasite death, disrupts ABHD5/perilipin-1 interaction, affects ROR gamma activity, and targets HCV.</p>
    Formula:C21H18O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.36
  • CFG920

    CAS:
    <p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>
    Formula:C14H13ClN4O
    Color and Shape:Solid
    Molecular weight:288.73
  • Quetiapine sulfoxide

    CAS:
    <p>Quetiapine sulfoxide: Main metabolite of Quetiapine, a 5-HT agonist &amp; dopamine antagonist antipsychotic.</p>
    Formula:C21H25N3O3S
    Purity:98%
    Color and Shape:Pale Yellow Solid
    Molecular weight:399.51
  • GlcN-6-P Synthase-IN-1

    CAS:
    <p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase &amp; CYP3A4. Has antimicrobial activity and CNS penetration.'</p>
    Formula:C20H21N7S
    Color and Shape:Solid
    Molecular weight:391.49
  • PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Formula:C17H19Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.27
  • hDHODH-IN-11

    CAS:
    <p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>
    Formula:C24H23N3O3
    Color and Shape:Solid
    Molecular weight:401.46
  • Nampt activator-3

    CAS:
    <p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37
  • MRL-871

    CAS:
    <p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>
    Formula:C22H12ClF3N2O3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:444.79
  • GK470

    CAS:
    <p>GK470 is a group IVA cytosolic phospholipase A2 inhibitor.</p>
    Formula:C21H27NO4S
    Color and Shape:Solid
    Molecular weight:389.51
  • (Z)-Pitavastatin calcium

    CAS:
    <p>(Z)-Pitavastatin calcium is the Z-Isomer of Pitavastatin hemicacium. Pitavastatin calcium is a potent of hydroxymethylglutaryl-CoA (HMG-CoA) reductase.</p>
    Formula:C50H50CaF2N2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:885.031
  • Acetyl-CoA Carboxylase-IN-1

    CAS:
    <p>Acetyl-CoA Carboxylase-IN-1 (ACC-IN-1) is a potent acetyl-CoA carboxylase (ACC) inhibitor with antibacterial activity, used in metabolic disease research.</p>
    Formula:C13H9Br2N5
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:395.05
  • PF-07208254

    CAS:
    <p>PF-07208254, a potent BDK inhibitor, enhances cardiometabolic endpoints in mice [1].</p>
    Formula:C7H2ClFO2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.67
  • Paranyline hydrochloride

    CAS:
    <p>Paranyline hydrochloride has anti-inflammatory activity.</p>
    Formula:C21H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.83
  • IMB-XMA0038

    CAS:
    <p>IMB-XMA0038 is a Mycobacterium tuberculosis aspartate semialdehyde dehydrogenase inhibitor with antimicrobial activity for use in tuberculosis research.</p>
    Formula:C11H10N4O6
    Purity:98.94% - 99.96%
    Color and Shape:Solid
    Molecular weight:294.22
  • hCAI/II-IN-2

    CAS:
    <p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>
    Formula:C12H12N4O5S2
    Color and Shape:Solid
    Molecular weight:356.38
  • 10-Nitrooleic acid

    CAS:
    <p>CXA-10, an endogenous NFA, modulates Nrf2, NF-κB, and boosts caveolin-1 levels.</p>
    Formula:C18H33NO4
    Color and Shape:Solid
    Molecular weight:327.46
  • Xanthine oxidase-IN-7

    CAS:
    <p>Xanthine oxidase-IN-7: Potent oral XO inhibitor (IC50=0.36μM), lowers serum uric acid, promising for hyperuricemia/gout research.</p>
    Formula:C16H14N4O2
    Color and Shape:Solid
    Molecular weight:294.31
  • Senazodan

    CAS:
    <p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>
    Formula:C15H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.3
  • MAO-IN-1

    CAS:
    <p>MAO-IN-1 is a potent monoamine oxidase B (MAO B) inhibitor (IC50: 20 nM) for the study of neurologically related diseases.</p>
    Formula:C17H19ClO4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:322.78
  • L-693612 HCl

    CAS:
    <p>L-693612 HCl is an inhibitor of carbonic anhydrase.</p>
    Formula:C14H25ClN2O5S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.01
  • UCM 765

    CAS:
    <p>UCM 765 is a partial agonist of melatonin MT(2) receptor.</p>
    Formula:C17H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.35
  • GOAT-IN-1

    CAS:
    <p>GOAT-IN-1 blocks GOAT, potentially treating diabetes, hyperlipidemia, and various brain disorders.</p>
    Formula:C18H13ClF3NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.81
  • Rociverine

    CAS:
    <p>Rociverine is an anticholinergic compound used as a smooth muscle relaxant.</p>
    Formula:C20H37NO3
    Color and Shape:Solid
    Molecular weight:339.51
  • HIF-IN-33

    CAS:
    <p>HIF-IN-33 is an inhibitor of HIF pathway.</p>
    Formula:C21H17F3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.38
  • VEC6

    CAS:
    <p>VEC6 is a VEZF1–DNA interaction inhibitor that recapitulates RhoB loss in ischaemic retinopathy.</p>
    Formula:C14H20N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.34
  • BCM-599

    CAS:
    <p>BCM-599 is a HBV capsid assembly inhibitor. BCM-599 showed IC50 of 0.88 μM and CC50 of 144 μM in HepG2.2.15 cells.</p>
    Formula:C14H10Cl2FN3O2
    Color and Shape:Solid
    Molecular weight:342.15
  • CX08005

    CAS:
    <p>CX08005 inhibits PTP1B, cuts liver fat, and improves microcirculation in NAFLD.</p>
    Formula:C28H39NO4
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:453.61
  • SCD1 Inhibitor

    CAS:
    <p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>
    Formula:C21H20F3N3O3
    Color and Shape:Solid
    Molecular weight:419.4
  • RORγt inverse agonist 28

    CAS:
    <p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>
    Formula:C23H18Cl2F3NO5S
    Color and Shape:Solid
    Molecular weight:548.36
  • SHP844

    CAS:
    <p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>
    Formula:C29H24ClN5O6
    Color and Shape:Solid
    Molecular weight:573.98
  • hCAIX-IN-10

    CAS:
    <p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>
    Formula:C28H21N3O3S
    Color and Shape:Solid
    Molecular weight:479.55
  • BMS-593214

    CAS:
    <p>BMS-593214 is an inhibitor of active site-directed factor VIIa and a non-competitive inhibitor of the VIIa-activated substrate FX.</p>
    Formula:C31H27N3O4
    Purity:96.63% - 98.04%
    Color and Shape:Solid
    Molecular weight:505.56
  • N-Monoacetylcystine

    CAS:
    <p>N-Monoacetylcystine is a paracetamol poisoning antidote. It is used in the treatment of influenza A virus pandemic.</p>
    Formula:C8H14N2O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.34
  • TES-991

    CAS:
    <p>TES-991 is a potent and selective inhibitor of human α Amino-β-carboxymuconate-ε-semialdehyde Decarboxylase (ACMSD)(IC50 of 3 nM).</p>
    Formula:C17H11N7OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.45
  • Bucricaine

    CAS:
    <p>Bucricaine is an anesthetic drug.</p>
    Formula:C17H22N2
    Color and Shape:Solid
    Molecular weight:254.37
  • SPK-601

    CAS:
    <p>SPK-601 is an inhibitor of phosphatidylcholine-specific phospholipase C.</p>
    Formula:C11H16KOS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.47
  • BBMP

    CAS:
    <p>BBMP is an inhibitor of mitochondrial permeability transition pore.</p>
    Formula:C12H11BrN2O3S
    Color and Shape:Solid
    Molecular weight:343.2
  • D5D-IN-326

    CAS:
    <p>D5D-IN-326: oral delta-5 desaturase inhibitor; IC50=72 nM (rat), 22 nM (human); no impact on D6D/D9D; lowers insulin resistance and body weight in obese mice.</p>
    Formula:C17H11F8N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.27
  • IDO-IN-3

    CAS:
    <p>IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).</p>
    Formula:C11H12BrFN6O2
    Color and Shape:Solid
    Molecular weight:359.15
  • Sp-cAMPS

    CAS:
    <p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>
    Formula:C10H12N5O5PS
    Color and Shape:Solid
    Molecular weight:345.27
  • FKGK11

    CAS:
    <p>FKGK11 is a potent inhibitor of GVIA iPLA2.</p>
    Formula:C13H13F5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.23
  • hCAI/II-IN-3

    CAS:
    <p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>
    Formula:C16H18N4O4S2
    Color and Shape:Solid
    Molecular weight:394.47
  • BIA 3-335

    CAS:
    <p>BIA 3-335, an inhibition of catechol-O-methyltransferase, could have applications for Parkinson's Disease.</p>
    Formula:C20H22Cl2F3N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:512.31
  • PDE7 inhibitor S14

    CAS:
    <p>PDE7 inhibitor S14 is a cell-permeable PDE7 inhibitor that acts by targeting the cyclic adenosine monophosphate (cAMP)/cAMP-response element-binding protein (</p>
    Formula:C14H10N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:254.31
  • Dehydro-ZINC39395747

    CAS:
    <p>Dehydro-ZINC39395747 enhances NO in cells and inhibits cytochrome b5 reductase 3 (IC50: 9.14μM, Kd: 1.11μM).</p>
    Formula:C12H9N3O2S2
    Color and Shape:Solid
    Molecular weight:291.35
  • A-1293201

    CAS:
    <p>A-1293201 is a potent and selective NAMPT inhibitor.</p>
    Formula:C21H23N3O3
    Color and Shape:Solid
    Molecular weight:365.43
  • Kurasoin B

    CAS:
    <p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>
    Formula:C18H17NO2
    Color and Shape:Solid
    Molecular weight:279.33
  • Rovazolac

    CAS:
    <p>Rovazolac (ALX-101) is a liver x receptor (LXR) modulator used in the study of immune system disorders and atopic dermatitis.</p>
    Formula:C21H19F3N2O4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:452.45
  • BMS 961

    CAS:
    <p>BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).</p>
    Formula:C23H26FNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.46
  • YCT529 free acid

    CAS:
    <p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>
    Formula:C29H25NO3
    Color and Shape:Solid
    Molecular weight:435.51
  • CR4056

    CAS:
    <p>CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of</p>
    Formula:C17H12N4
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:272.3
  • SLC26A3-IN-3

    CAS:
    <p>SLC26A3-IN-3 (compound 4az), a potent SLC26A3 inhibitor with an IC50 of 40 nM, is utilized for constipation and cystic fibrosis research [1].</p>
    Formula:C20H17IO5
    Color and Shape:Solid
    Molecular weight:464.25
  • Izumerogant

    CAS:
    <p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>
    Formula:C22H18ClF4N5O2
    Color and Shape:Solid
    Molecular weight:495.86
  • Clinolamide

    CAS:
    <p>Clinolamide is an antilipidemic agent.</p>
    Formula:C24H43NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.6
  • Trandolaprilate hydrate

    CAS:
    <p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>
    Formula:C22H32N2O6
    Color and Shape:Solid
    Molecular weight:420.5
  • ASP3662

    CAS:
    <p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>
    Formula:C19H16ClF3N4O2
    Color and Shape:Solid
    Molecular weight:424.8
  • AF267

    CAS:
    <p>AF267 is a M1 muscarinic agonist that works by restoring cognitive impairments.</p>
    Formula:C10H18N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:214.33
  • DY3002

    CAS:
    <p>DY3002 is a novel, selective and potent EGFR Inhibitor, it overcomes T790M-Mediated Resistance in Non-Small Cell Lung Cancer.</p>
    Formula:C24H25ClN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.95
  • Pteropterin monohydrate

    CAS:
    <p>Pteropterin monohydrate is an antineoplastic agent.</p>
    Formula:C29H35N9O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:717.64
  • ALDH1A1-IN-2

    CAS:
    <p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>
    Formula:C25H23ClN4O3S
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:494.99
  • PF-04822163

    CAS:
    <p>PF-04822163 is a potent inhibitor of PDE1 with IC50 value of 0.0024 μM.</p>
    Formula:C19H17ClN2O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:340.8
  • ZINC05626394

    CAS:
    <p>ZINC05626394 is a Cytochrome b5 reductase 3 inhibitor that acts by increasing NO bioavailability.</p>
    Formula:C11H10N2OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:250.34
  • CAY10762

    CAS:
    <p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>
    Formula:C15H13NOS
    Color and Shape:Solid
    Molecular weight:255.33
  • Naftidrofuryl

    CAS:
    <p>Naftidrofuryl treats peripheral and cerebral vascular issues, boosts cell oxidation, and relaxes muscles.</p>
    Formula:C24H33NO3
    Color and Shape:Solid
    Molecular weight:383.52
  • CYP3A4-IN-3

    CAS:
    <p>CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.</p>
    Formula:C34H39N3O3S
    Color and Shape:Solid
    Molecular weight:569.76
  • Cholesteryl behenate

    CAS:
    <p>Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.</p>
    Formula:C49H88O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:709.22
  • GNF362

    CAS:
    <p>GNF362 is an ITPKB inhibitor that inhibits Itpka and Itpkc and reverses the migratory stimulatory effect of ITPKA overexpression.</p>
    Formula:C22H21F3N6
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:426.44
  • IDO1-IN-21

    CAS:
    <p>IDO1-IN-21 (compound 10m), with an IC50 of 0.64 μM, acts as an IDO1 inhibitor and has demonstrated efficacy in suppressing tumor growth in murine models [1].</p>
    Formula:C21H19F2N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.45
  • OHM1

    CAS:
    <p>OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53</p>
    Formula:C24H42N6O5
    Color and Shape:Solid
    Molecular weight:494.63
  • LASSBio-1366

    CAS:
    <p>LASSBio-1366 is an agonist of adenosine A2a receptor that acts by attenuating the progression of monocrotaline-induced pulmonary hypertension.</p>
    Formula:C19H22N2O5
    Color and Shape:Solid
    Molecular weight:358.39
  • LY 186126

    CAS:
    <p>LY 186126 is a potent cGI-PDE inhibitor with reversible, high affinity (Ka = 6 nM) binding to a single class of SaR binding sites.</p>
    Formula:C16H19N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.34
  • PMPMEase-IN L-23

    CAS:
    <p>PMPMEase-IN L-23 is a novel prenylated methylated protein methylesterase inhibitor.</p>
    Formula:C12H21FO2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.42
  • AGI-14100

    CAS:
    <p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>
    Formula:C29H22ClF4N5O3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:599.96
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • SCD1 inhibitor-1

    CAS:
    SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).
    Formula:C21H23N3NaO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • hCAXII-IN-2

    CAS:
    <p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>
    Formula:C21H18ClN3O4
    Color and Shape:Solid
    Molecular weight:411.84
  • Teglicar

    CAS:
    <p>Teglicar is a selective and reversible liver isoform of carnitine palmitoyl-transferase 1 (L-CPT1) inhibitor.</p>
    Formula:C22H45N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.61
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Formula:C20H21N3O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.4
  • α-Glucosidase-IN-16

    CAS:
    <p>α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM.</p>
    Formula:C22H18FNS
    Color and Shape:Solid
    Molecular weight:347.45
  • Cefetrizole

    CAS:
    <p>Ceftezole is an α-Glucosidase inhibitor (IC50: 2.1 μM; Ki: 0.578 μM).</p>
    Formula:C16H15N5O4S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:437.52
  • Kojibiose

    CAS:
    <p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>
    Formula:C12H22O11
    Purity:99.933%
    Color and Shape:Solid
    Molecular weight:342.3
  • Icomucret

    CAS:
    <p>Icomucret can be used for the Treatment of Dry Eye.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47
  • ALDH3A1-IN-2

    CAS:
    <p>ALDH3A1-IN-2 is a potent inhibitor targeting ALDH3A1 (IC50=1.29µM), potentially useful in cancer research.</p>
    Formula:C11H14N2O3
    Color and Shape:Solid
    Molecular weight:222.24
  • Dopropidil

    CAS:
    <p>Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.</p>
    Formula:C20H35NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.5
  • 4,6-O-Ethylidene-α-D-glucose

    CAS:
    <p>4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucose</p>
    Formula:C8H14O6
    Color and Shape:Solid
    Molecular weight:206.19
  • SA57

    CAS:
    <p>SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).</p>
    Formula:C17H23ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.83
  • URB532

    CAS:
    <p>URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Formula:C18H21NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.36
  • NSC-84096

    CAS:
    <p>NSC-84096 is an endopeptidase activity inhibitor of botulinum neurotoxin type A light chain (rBoNT/A-LC).</p>
    Formula:C25H19N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.44
  • Fluindione

    CAS:
    <p>Fluindione is a hematologic drug.</p>
    Formula:C15H9FO2
    Color and Shape:Solid
    Molecular weight:240.23
  • ISQ-1 HCl

    CAS:
    <p>ISQ-1 HCl is an isoquinolinone (IKur) blocker with possible atrial arrhythmia activity.</p>
    Formula:C20H23ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.86
  • Glyoxalase I inhibitor 2

    CAS:
    <p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>
    Formula:C24H23N3O4S
    Color and Shape:Solid
    Molecular weight:449.52
  • FSG67

    CAS:
    <p>FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].</p>
    Formula:C16H25NO4S
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:327.44
  • BAY 73-6691

    CAS:
    <p>BAY 73-6691 is an inhibitor of brain penetrant PDE9A.</p>
    Formula:C15H12ClF3N4O
    Color and Shape:Solid
    Molecular weight:356.73
  • α-2,3-sialyltransferase-IN-1

    CAS:
    <p>α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).</p>
    Formula:C28H45NO6
    Purity:98% - 98%
    Color and Shape:Solid
    Molecular weight:491.66
  • SQ-24,798

    CAS:
    <p>SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).</p>
    Formula:C7H15N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:205.28
  • UK-371804 HCl

    CAS:
    <p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>
    Formula:C14H17Cl2N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.29
  • iGP-5

    CAS:
    <p>iGP-5 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>
    Formula:C21H17N3O3
    Color and Shape:Solid
    Molecular weight:359.38
  • Oncrasin-72

    CAS:
    Oncrasin-72 is an analog of oncrasin-1. It has antitumor activity mediated by JNK activation and STAT3 inhibition.
    Formula:C16H14ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:271.74
  • JNJ-40413269

    CAS:
    <p>JNJ-40413269 inhibits FAAH, engages central targets, and is effective in rat neuropathic pain.</p>
    Formula:C19H15ClF3N3O
    Color and Shape:Solid
    Molecular weight:393.79
  • Antitumor agent-87

    CAS:
    <p>Antitumor agent-87: potent, high CYP1A1 affinity (Ki 0.23µM), antiproliferative, arrests G2/M cell cycle.</p>
    Formula:C22H28N2O6S
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:448.53
  • THR-0921

    CAS:
    <p>THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study cardiovascular and metabolic diseases.</p>
    Formula:C28H25NO7S
    Purity:100% - 99.83%
    Color and Shape:Solid
    Molecular weight:519.57
  • ML202

    CAS:
    <p>ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.</p>
    Formula:C18H17N3O3S2
    Color and Shape:Solid
    Molecular weight:387.48
  • OH-Ubenimex

    CAS:
    <p>OH-Ubenimex is an orally active aminopeptidase inhibitor that has an immunomodulating action.</p>
    Formula:C16H24N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.37
  • SQ 28853

    CAS:
    <p>SQ 28853 is an inhibitor of ACE with diuretic properties.</p>
    Formula:C19H25ClN4NaO6S3
    Color and Shape:Solid
    Molecular weight:560.05
  • Aminopeptidase-IN-1

    CAS:
    <p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>
    Formula:C18H16N2O6
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:356.33
  • Albaconazole

    CAS:
    <p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>
    Formula:C20H16ClF2N5O2
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:431.82
  • GNE-3500

    CAS:
    <p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>
    Formula:C24H30FN3O3S
    Color and Shape:Solid
    Molecular weight:459.58
  • DHODH-IN-17

    CAS:
    <p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>
    Formula:C12H9ClN2O2
    Purity:99.41% - 99.52%
    Color and Shape:Solid
    Molecular weight:248.67
  • YM-75466

    CAS:
    <p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>
    Formula:C28H35N5O8S2
    Color and Shape:Solid
    Molecular weight:633.74
  • Palmostatin B

    CAS:
    <p>Palmostatin B is a modulator of Ras-signaling that acts by targeting acyl protein thioesterase 1 (APT1) and 2 (APT2) in cells.</p>
    Formula:C23H36O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.53
  • IDO-IN-16

    CAS:
    <p>IDO-IN-16 (compound 5) is an IDO inhibitor (IC50: 36 nM).</p>
    Formula:C22H21F3N4O
    Color and Shape:Solid
    Molecular weight:414.42
  • MJN228

    CAS:
    <p>MJN228 is a NUCB1 inhibitor that blocks AEA-DA probe labeling of endogenous NUCB1 in Neuro2a cells and can be used to study metabolic disorders.</p>
    Formula:C20H20N4O3
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:364.4
  • ARI-3531

    CAS:
    <p>ARI-3531 is a selective prolyl endopeptidase inhibitor.</p>
    Formula:C15H22BN3O4
    Color and Shape:Solid
    Molecular weight:319.16
  • WES-1

    CAS:
    <p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>
    Formula:C20H20N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.46
  • Ipenoxazone

    CAS:
    <p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>
    Formula:C22H34N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.52
  • (Rac)-3′-Hydroxy simvastatin

    CAS:
    <p>(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.</p>
    Formula:C25H38O6
    Color and Shape:Solid
    Molecular weight:434.57
  • Hexazinone

    CAS:
    <p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>
    Formula:C12H20N4O2
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:252.31
  • PC945

    CAS:
    <p>PC945 (Opelconazole) is an antifungal compound that inhibits CYP51A/CYP51B and can be used to study fungal infections of the lungs.</p>
    Formula:C38H37F3N6O3
    Purity:98.89% - 99.37%
    Color and Shape:Solid
    Molecular weight:682.73
  • 5-LOX-IN-1

    CAS:
    <p>5-LOX-IN-1 is a 5-Lipoxygenase (5-LOX) inhibitor (IC50: 2.3 μM).5-LOX-IN-1 can be used for cancer research.</p>
    Formula:C20H18N2O2S
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:350.43
  • GAC0003A4

    CAS:
    <p>GAC0003A4 is an LXR inverse agonist with antitumor activity for the study of advanced pancreatic cancer and other recalcitrant malignancies.</p>
    Formula:C20H24N2O3
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:340.42
  • hCAI/II-IN-6

    CAS:
    <p>hCAI/II-IN-6 is a selective and orally active inhibitor of human carbonic anhydrase (CA).</p>
    Formula:C19H24N4O3S
    Purity:97.07%
    Color and Shape:Solid
    Molecular weight:388.48
  • JNJ-42226314

    CAS:
    <p>JNJ-42226314 is a MAGL inhibitor with anti-injury effects and has shown efficacy in neuropathic pain and inflammatory pain models.</p>
    Formula:C26H24FN5O2S
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:489.56
  • CM037

    CAS:
    <p>CM037 (A-37) is a selective ALDH1A1 (acetaldehyde dehydrogenase 1A1) inhibitor (IC50; 4.6 µM) with antitumor activity and may be used in studies to eliminate</p>
    Formula:C21H25N3O3S2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:431.57
  • Didesethyl chloroquine

    CAS:
    <p>Didesethyl chloroquine, a chloroquine metabolite, is an effective myocardial inhibitor and antimalarial.</p>
    Formula:C14H18ClN3
    Purity:98.11%
    Color and Shape:Solid
    Molecular weight:263.77
  • UCM05

    CAS:
    <p>UCM05 is a potent FASN and FtsZ inhibitor active against HER2+ breast cancer and B. subtilis (MIC 100 μM), but not E. coli.</p>
    Formula:C24H16O10
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:464.38
  • KT182

    CAS:
    <p>KT182 is a selective and  potent inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells.</p>
    Formula:C27H26N4O2
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:438.52
  • Tiapamil hydrochloride

    CAS:
    <p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>
    Formula:C26H38ClNO8S2
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:592.16
  • MFI8

    CAS:
    <p>MFI8 is a compound that regulates mitochondrial fission and can be used to study aging.</p>
    Formula:C16H18ClNO
    Purity:99.08% - 99.78%
    Color and Shape:Solid
    Molecular weight:275.77
  • Vatanidipine

    CAS:
    <p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>
    Formula:C41H42N4O6
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:686.8
  • BMS 753

    CAS:
    <p>BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).</p>
    Formula:C21H21NO4
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:351.4
  • KRH102140

    CAS:
    <p>KRH102140 is a PHD2 activator that reduces angiogenesis by inhibiting HIF-1alpha, used in cardiovascular disease research.</p>
    Formula:C25H24FNO
    Purity:98.31% - 99.61%
    Color and Shape:Solid
    Molecular weight:373.46
  • JNJ-DGAT2-A

    CAS:
    <p>JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.</p>
    Formula:C24H16BrFN4O2S
    Purity:98.3%
    Color and Shape:Solid
    Molecular weight:523.38
  • Utreloxastat

    CAS:
    <p>Utreloxastat (PTC857) is a novel 15-lipoxygenase inhibitor that can be used to study amyotrophic lateral sclerosis<br>.</p>
    Formula:C18H28O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:276.41
  • PKUMDL-LC-101-D04

    CAS:
    <p>PKUMDL-LC-101-D04 enhances GPX4, curbs iron death, boosts enzyme activity 150% at 20 μM, effective in wild-type MEF, reduces lipid peroxide toxicity.</p>
    Formula:C14H23ClN4O2S2
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:378.94
  • NG-497

    CAS:
    <p>NG-497, a selective inhibitor of human ATGL, blocks lipolysis in adipocytes and aids cancer research.</p>
    Formula:C18H21NO4
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:315.36
  • 4-Hydroxymephenytoin

    CAS:
    <p>4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.</p>
    Formula:C12H14N2O3
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:234.25
  • NecroX-5

    CAS:
    <p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>
    Formula:C27H39N3O9S3
    Purity:99.944%
    Color and Shape:Solid
    Molecular weight:645.81
  • Fenoverine

    CAS:
    <p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>
    Formula:C26H25N3O3S
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:459.56