Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(41 products)
- Aminopeptidase(67 products)
- CETP(18 products)
- Carbonic Anhydrase(178 products)
- Casein Kinase(130 products)
- DHFR(33 products)
- Decarboxylase(4 products)
- Dehydrogenase(271 products)
- FAAH(64 products)
- FXR(58 products)
- Factor Xa(80 products)
- Fatty Acid Synthase(33 products)
- Ferroptosis(215 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(54 products)
- HIF/HIF Prolyl-Hydroxylase(142 products)
- HMG-CoA Reductase(33 products)
- Hydroxylase(30 products)
- IDO(82 products)
- LDL(8 products)
- Lipase(98 products)
- Lipid(58 products)
- Lipoxygenase(124 products)
- MAO(87 products)
- MPO(2 products)
- NAMPT(36 products)
- P450(6 products)
- PAI-1(25 products)
- PDE(166 products)
- PED(1 products)
- PKM(15 products)
- PPAR(164 products)
- Phospholipase(82 products)
- ROR(42 products)
- Retinoid Receptor(29 products)
- SGK(11 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(42 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
Show 34 more subcategories
Found 8626 products of "Metabolism"
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GOT1 inhibitor-1
CAS:<p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>Formula:C19H19ClN4OPurity:99.70%Color and Shape:SolidMolecular weight:354.83SR3335
CAS:<p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>Formula:C13H9F6NO3S2Purity:99.77%Color and Shape:SolidMolecular weight:405.34AZ876
CAS:<p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>Formula:C24H29N3O3SPurity:99.86%Color and Shape:SolidMolecular weight:439.57SR8278
CAS:<p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>Formula:C18H19NO3S2Purity:99.44% - 99.73%Color and Shape:SolidMolecular weight:361.48BRL-50481
CAS:<p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>Formula:C9H12N2O4SPurity:99.66%Color and Shape:SolidMolecular weight:244.27Toloxatone
CAS:<p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>Formula:C11H13NO3Purity:98.58%Color and Shape:SolidMolecular weight:207.23Obafistat
CAS:<p>Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.</p>Formula:C15H16FN5O3SPurity:99.71%Color and Shape:SolidMolecular weight:365.38BI-187004
CAS:<p>BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.</p>Formula:C21H18N4OPurity:98.63%Color and Shape:SolidMolecular weight:342.39U-104
CAS:<p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>Formula:C13H12FN3O3SPurity:98.76% - 99.88%Color and Shape:SolidMolecular weight:309.32Gonadorelin Acetate (33515-09-2 free base)
CAS:<p>Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) is hypothalamic neuropeptide which plays a key role in the control of</p>Formula:C59H83N17O17Purity:99.42% - 99.46%Color and Shape:White Or Off-White PowderMolecular weight:1302.39AUDA
CAS:<p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>Formula:C23H40N2O3Purity:99.50%Color and Shape:SolidMolecular weight:392.58p-Fluoro-L-phenylalanine
CAS:<p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>Formula:C9H10FNO2Purity:99.63%Color and Shape:White To Off-White PowderMolecular weight:183.18BW-A 78U
CAS:<p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>Formula:C13H12FN5Purity:99.45%Color and Shape:SolidMolecular weight:257.27GSK805
CAS:<p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>Formula:C23H18Cl2F3NO4SPurity:98% - ≥95%Color and Shape:SolidMolecular weight:532.362-Bromo-4'-hydroxyacetophenone
CAS:<p>2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).</p>Formula:C8H7BrO2Purity:98.64%Color and Shape:Clear Colorless To Light Yellow LiquidMolecular weight:215.04Telaglenastat
CAS:<p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>Formula:C26H24F3N7O3SPurity:97.57% - 99.89%Color and Shape:SolidMolecular weight:571.57Pargyline
CAS:<p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>Formula:C11H13NPurity:95.64% - 97.21%Color and Shape:SolidMolecular weight:159.23PfDHODH-IN-2
CAS:<p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>Formula:C13H12ClNO3SPurity:98.9%Color and Shape:SolidMolecular weight:297.76Pentamidine isethionate
CAS:<p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>Formula:C23H36N4O10S2Purity:98% - 99.83%Color and Shape:Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)Molecular weight:592.68FG-2216
CAS:<p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>Formula:C12H9ClN2O4Purity:97.1% - >99.99%Color and Shape:SolidMolecular weight:280.66JZL 184
CAS:<p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>Formula:C27H24N2O9Purity:97.56% - 99.31%Color and Shape:SolidMolecular weight:520.49RGX-104
CAS:<p>RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)</p>Formula:C34H33ClF3NO3Purity:98.79% - 99.53%Color and Shape:SolidMolecular weight:596.08KPT9274
CAS:KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.Formula:C35H29F3N4O3Purity:99.75% - 99.93%Color and Shape:SolidMolecular weight:610.62LOX-IN-3 dihydrochloride
CAS:<p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>Formula:C13H15Cl2FN2O2SPurity:99.96%Color and Shape:SolidMolecular weight:353.24Cobicistat
CAS:<p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>Formula:C40H53N7O5S2Purity:97.36% - 99.62%Color and Shape:SolidMolecular weight:776.02Glycerol 3-phosphate biscyclohexylammonium salt
CAS:<p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>Formula:C15H35N2O6PPurity:99.94%Color and Shape:SolidMolecular weight:370.42ARM1
CAS:<p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>Formula:C16H14N2SPurity:99.36%Color and Shape:SolidMolecular weight:266.36(±)-Amiflamine
CAS:<p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>Formula:C12H20N2Purity:97.24%Color and Shape:SolidMolecular weight:192.3Cecropin P1, porcine acetate
<p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>Formula:C149H257N45O45Purity:95.4% - 98%Color and Shape:SolidMolecular weight:3398.91Bempedoic acid
CAS:<p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>Formula:C19H36O5Purity:99.85% - 99.94%Color and Shape:SolidMolecular weight:344.49Efonidipine hydrochloride monoethanolate
CAS:<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formula:C36H45ClN3O8PPurity:>99.99%Color and Shape:SolidMolecular weight:714.181-Ethynylpyrene
CAS:<p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>Formula:C18H10Purity:98.48%Color and Shape:SolidMolecular weight:226.27Suvecaltamide
CAS:Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.Formula:C20H23F3N2O2Purity:99.29% - 99.70%Color and Shape:SolidMolecular weight:380.4Diflubenzuron
CAS:<p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>Formula:C14H9ClF2N2O2Purity:99.58% - 99.96%Color and Shape:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective InsecticideMolecular weight:310.68GSK1016790A
CAS:<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formula:C28H32Cl2N4O6S2Purity:97.37% - 99.38%Color and Shape:SolidMolecular weight:655.61DHBP dibromide
CAS:<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formula:C24H38Br2N2Purity:99.73%Color and Shape:Yellow To Yellow-Green Powder Or FlakesMolecular weight:514.38(Rac)-LB-100
CAS:<p>LB-100, a novel Protein Phosphatase 2A (PP2A) inhibitor, sensitizes malignant meningioma cells to the therapeutic effects of radiation</p>Formula:C13H20N2O4Purity:97.11% - 99.77%Color and Shape:SolidMolecular weight:268.31Pep 2-8 ammonium salt(1541011-97-5 free base)
<p>Pep 2-8 ammonium salt inhibits PCSK9-LDL receptor binding (IC50 = 0.8 μM), boosting LDL uptake in HepG2 cells.</p>Formula:C83H113N17O24Purity:95.76% - 99.87%Color and Shape:SolidMolecular weight:1732.912,5-Di-tert-butylhydroquinone
CAS:<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formula:C14H22O2Purity:97.11%Color and Shape:PelletslargecrystalsMolecular weight:222.32kb NB 142-70
CAS:<p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>Formula:C11H9NO2S2Purity:98.15% - ≥95%Color and Shape:SolidMolecular weight:251.32AGN 193109
CAS:<p>AGN 193109, a retinoid analog, is a potent and specific antagonist of RARs (Kds: 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ).</p>Formula:C28H24O2Purity:99.87% - 99.89%Color and Shape:SolidMolecular weight:392.49D-Valine
CAS:<p>D-Valine (H-D-Val-OH) is the enantiomer of L-Valine.</p>Formula:C5H11NO2Purity:99.93%Color and Shape:White CrystalsMolecular weight:117.15GSK2033
CAS:<p>GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).</p>Formula:C29H28F3NO5S2Purity:99.70%Color and Shape:SolidMolecular weight:591.66Efonidipine
CAS:Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Formula:C34H38N3O7PPurity:98.35% - 99.47%Color and Shape:SolidMolecular weight:631.66IDO5L
CAS:<p>IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).</p>Formula:C9H7ClFN5O2Purity:99.49% - 99.75%Color and Shape:SolidMolecular weight:271.64Tedizolid
CAS:<p>Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of</p>Formula:C17H15FN6O3Purity:96.97% - 99.89%Color and Shape:SolidMolecular weight:370.34Pimecrolimus
CAS:<p>Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.</p>Formula:C43H68ClNO11Purity:99.53% - 99.87%Color and Shape:White Crystalline PowderMolecular weight:810.45SI-113
CAS:<p>SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.</p>Formula:C23H24N6OPurity:98.93%Color and Shape:SolidMolecular weight:400.48BAY-876
CAS:<p>BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.</p>Formula:C24H16F4N6O2Purity:98.61% - 99.78%Color and Shape:SolidMolecular weight:496.42Benzenesulfonamide
CAS:<p>Benzenesulfonamide (Benzosulfonamide) ia an inhibitor of carbonic anhydrases.</p>Formula:C6H7NO2SPurity:99.42% - 99.99%Color and Shape:White Crystalline PowderMolecular weight:157.19
