GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formula:C118H190N36O30S2Purity:96.86%Color and Shape:SolidMolecular weight:2657.12Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formula:C15H20Cl2N2O3Purity:99.17%Color and Shape:SolidMolecular weight:347.24SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Ref: TM-T6979
1mg40.00€2mg51.00€5mg85.00€10mg125.00€25mg225.00€50mg364.00€100mg582.00€1mL*10mM (DMSO)86.00€Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg38.00€2mg50.00€5mg84.00€10mg118.00€25mg220.00€50mg403.00€100mg582.00€500mg1,198.00€1mL*10mM (DMSO)120.00€JNJ-7777120
CAS:JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formula:C14H16ClN3OPurity:99.83% - 99.96%Color and Shape:SolidMolecular weight:277.75CGP71683 hydrochloride
CAS:CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formula:C26H30ClN5O2SPurity:99.92%Color and Shape:SolidMolecular weight:512.07Bevantolol hydrochloride
CAS:Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formula:C20H28ClNO4Purity:99.49%Color and Shape:SolidMolecular weight:381.9Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formula:C28H29F2N3OPurity:99.63% - >99.99%Color and Shape:SolidMolecular weight:461.55RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formula:C25H27N3O3Purity:98.64% - 99.62%Color and Shape:SolidMolecular weight:417.5Idazoxan hydrochloride
CAS:Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.Formula:C11H12N2O2·HClPurity:99.42% - 99.84%Color and Shape:SolidMolecular weight:240.69Ref: TM-T0115
2mg35.00€5mg52.00€10mg78.00€25mg133.00€50mg187.00€100mg281.00€200mg416.00€1mL*10mM (DMSO)50.00€Ivabradine hydrochloride
CAS:Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formula:C27H37ClN2O5Purity:99% - 99.73%Color and Shape:SolidMolecular weight:505.05Tripelennamine citrate
CAS:Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.Formula:C22H29N3O7Color and Shape:SolidMolecular weight:447.488Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19HPI 1
CAS:HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formula:C27H29NO6Purity:97.6%Color and Shape:SolidMolecular weight:463.52Ref: TM-T22089
1mg47.00€2mg60.00€5mg92.00€10mg135.00€25mg217.00€50mg324.00€100mg472.00€500mg1,026.00€1mL*10mM (DMSO)107.00€Chlorphenesin
CAS:Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.Formula:C9H11ClO3Purity:99.59%Color and Shape:SolidMolecular weight:202.63N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Ref: TM-T5158
2mg34.00€5mg48.00€10mg79.00€25mg152.00€50mg235.00€100mg344.00€200mg490.00€1mL*10mM (DMSO)58.00€SBI-115
CAS:SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5Formula:C14H13ClN2O4SPurity:99.53% - 99.78%Color and Shape:SolidMolecular weight:340.78AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formula:C11H9Cl2N3O3SPurity:99.80% - >99.99%Color and Shape:SolidMolecular weight:334.18Ref: TM-T4300
1mg34.00€5mg66.00€10mg105.00€25mg217.00€50mg334.00€100mg502.00€500mg1,063.00€1mL*10mM (DMSO)73.00€C-021
CAS:C 021 dihydrochloride is a potent CCR4 antagonist.Formula:C27H41N5O2Purity:99.74% - 99.90%Color and Shape:SolidMolecular weight:467.65Ref: TM-T21870
1mg51.00€2mg71.00€5mg96.00€10mg153.00€25mg303.00€50mg469.00€100mg655.00€1mL*10mM (DMSO)96.00€AC-55541
CAS:AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29Taladegib
CAS:Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formula:C26H24F4N6OPurity:98.75% - >99.99%Color and Shape:SolidMolecular weight:512.5Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Sevoflurane
CAS:Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formula:C4H3F7OPurity:98%Color and Shape:Less Oil Colorless OilMolecular weight:200.05Ref: TM-T22425
2mg39.00€5mg54.00€10mg75.00€25mg110.00€50mg158.00€100mg226.00€200mg339.00€1mL*10mM (DMSO)56.00€ML-SI3
CAS:CCG-143140 is a GLP-1 receptor inverse agonists.Formula:C23H31N3O3SPurity:99.75%Color and Shape:SolidMolecular weight:429.58PGS-IN-1
CAS:PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formula:C19H26O3Purity:99.39%Color and Shape:SolidMolecular weight:302.41Ref: TM-T10098
1mg52.00€5mg97.00€10mg170.00€25mg369.00€50mg540.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)110.00€BMS-813160
CAS:BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formula:C25H40N8O2Purity:99.66% - 99.79%Color and Shape:SolidMolecular weight:484.64Ref: TM-T4584
1mg63.00€5mg137.00€10mg187.00€25mg341.00€50mg567.00€100mg810.00€500mg1,644.00€1mL*10mM (DMSO)145.00€HhAntag
CAS:HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activityFormula:C24H23ClN4O3Purity:95.73%Color and Shape:SolidMolecular weight:450.92Maraviroc
CAS:Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formula:C29H41F2N5OPurity:97.13% - 99.59%Color and Shape:Brown SolidMolecular weight:513.67Ref: TM-T6016
5mg51.00€10mg95.00€25mg160.00€50mg273.00€100mg492.00€200mg633.00€500mg998.00€1mL*10mM (DMSO)59.00€Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formula:C41H52N4O4SPurity:97.87%Color and Shape:SolidMolecular weight:696.94Ref: TM-TQ0297
1mg63.00€2mg90.00€5mg133.00€10mg212.00€25mg423.00€50mg550.00€100mg715.00€200mg964.00€1mL*10mM (DMSO)200.00€SAG
CAS:SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.
Formula:C28H28ClN3OSPurity:97.37% - 98.88%Color and Shape:SolidMolecular weight:490.06Ciliobrevin A
CAS:Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formula:C17H9Cl2N3O2Purity:98.54% - 99.57%Color and Shape:SolidMolecular weight:358.18Ref: TM-T3156
2mg42.00€5mg59.00€10mg85.00€25mg168.00€50mg235.00€100mg331.00€200mg492.00€1mL*10mM (DMSO)69.00€SANT-1
CAS:SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formula:C23H27N5Purity:99.93% - >99.99%Color and Shape:SolidMolecular weight:373.49Vercirnon
CAS:Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formula:C22H21ClN2O4SPurity:99.23%Color and Shape:SolidMolecular weight:444.93Ref: TM-T17225
1mg105.00€5mg259.00€10mg406.00€25mg680.00€50mg938.00€100mg1,301.00€500mg2,593.00€1mL*10mM (DMSO)363.00€SAG hydrochloride (912545-86-9(free base))
CAS:SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.Formula:C28H29Cl2N3OSPurity:99.19% - 99.97%Color and Shape:SolidMolecular weight:526.52Ref: TM-T4211
1mg49.00€2mg65.00€5mg90.00€10mg114.00€25mg222.00€50mg334.00€100mg502.00€200mg717.00€1mL*10mM (DMSO)105.00€R243
CAS:R243 is CCR8 signaling and chemotaxis inhibitor.Formula:C21H27NO4Purity:99.03%Color and Shape:SolidMolecular weight:357.44Ref: TM-T24700
1mg40.00€2mg52.00€5mg80.00€10mg117.00€25mg207.00€50mg333.00€100mg495.00€1mL*10mM (DMSO)90.00€Sonidegib
CAS:Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.Formula:C26H26F3N3O3Purity:98% - 99.97%Color and Shape:SolidMolecular weight:485.5Salmeterol Xinafoate
CAS:Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formula:C36H45NO7Purity:98% - 98.24%Color and Shape:White SolidMolecular weight:603.75MRT-81
CAS:MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formula:C31H29N3O5SPurity:99.72%Color and Shape:SolidMolecular weight:555.64Ref: TM-T9532
1mg48.00€5mg97.00€10mg145.00€25mg255.00€50mg368.00€100mg505.00€200mg692.00€1mL*10mM (DMSO)116.00€VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34Treprostinil
CAS:Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).Formula:C23H34O5Purity:99.29%Color and Shape:SolidMolecular weight:390.51Ref: TM-T5150
1mg34.00€5mg71.00€10mg108.00€25mg221.00€50mg355.00€100mg533.00€200mg755.00€1mL*10mM (DMSO)60.00€Asapiprant
CAS:Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.Formula:C24H27N3O7SPurity:99.64%Color and Shape:SolidMolecular weight:501.55Ref: TM-T5386
1mg40.00€5mg97.00€10mg156.00€25mg284.00€50mg449.00€100mg730.00€200mg938.00€1mL*10mM (DMSO)105.00€Nelociguat
CAS:Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:C19H17FN8O2Purity:99.19%Color and Shape:SolidMolecular weight:408.39Neurokinin A
CAS:Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formula:C50H80N14O14SPurity:>99.99%Color and Shape:White To Off-White Lyophilized SolidMolecular weight:1133.32Siponimod hemifumarate
CAS:Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.Formula:C62H74F6N4O10Color and Shape:SolidMolecular weight:1149.282Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
Formula:C52H77N13O13Purity:99.93%Color and Shape:SolidMolecular weight:1092.27I-191
CAS:I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formula:C23H26FN5O2Purity:99.8%Color and Shape:SolidMolecular weight:423.48Ticagrelor metabolite M5
CAS:Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.Formula:C14H22N6O4SPurity:99.35%Color and Shape:SolidMolecular weight:370.43Gastrin I (human) acetate
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (Formula:C99H128N20O33SPurity:98.84%Color and Shape:SolidMolecular weight:2158.25AR-M 1896 Acetate
AR-M 1896 Acetate is the selective agonist of GalR2.Formula:C56H85N13O16Purity:99.76%Color and Shape:SolidMolecular weight:1196.35Ref: TM-T21646L
1mg537.00€2mg727.00€5mg1,064.00€10mg1,454.00€25mg2,147.00€50mg2,822.00€1mL*10mM (DMSO)2,213.00€AM966
CAS:AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.Formula:C27H23ClN2O5Purity:98.06% - 99.79%Color and Shape:SolidMolecular weight:490.93Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.Formula:C38H60F6N8O10SPurity:99%Color and Shape:SolidMolecular weight:934.992-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09Motilin (26-47), human, porcine
CAS:Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formula:C120H188N34O35SPurity:98%Color and Shape:SolidMolecular weight:2699.07Ref: TM-TP1425
1mg111.00€5mg334.00€10mg504.00€25mg745.00€50mg999.00€100mg1,341.00€200mg1,773.00€500µg86.00€LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purity:98.36%Color and Shape:SolidMolecular weight:473.93Ref: TM-T7303
2mg34.00€5mg66.00€10mg99.00€25mg205.00€50mg334.00€100mg522.00€200mg743.00€1mL*10mM (DMSO)70.00€Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formula:C18H18ClN3OPurity:99.88%Color and Shape:Pale Yellowish Crystals From Petroleum Ether SolidMolecular weight:327.81GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formula:C149H226N40O45Purity:99.85%Color and Shape:White PowderMolecular weight:3297.63ACTH (1-17) acetate
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).Formula:C97H149N29O25SPurity:98.53%Color and Shape:SolidMolecular weight:2153.47Pergolide
CAS:Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormula:C19H26N2SPurity:99.95%Color and Shape:SolidMolecular weight:314.49Ref: TM-T21340
2mg37.00€5mg54.00€10mg77.00€25mg110.00€50mg164.00€100mg237.00€200mg350.00€1mL*10mM (DMSO)60.00€Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.88RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.
Formula:C17H16FN3Purity:99.32%Color and Shape:SolidMolecular weight:281.33Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formula:C24H25FN4O2Purity:99.33%Color and Shape:SolidMolecular weight:420.48Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formula:C20H25ClN2OSPurity:99.17%Color and Shape:SolidMolecular weight:376.94Pasireotide Acetate
CAS:The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Formula:C60H70N10O11Purity:98.64% - 99.92%Color and Shape:SolidMolecular weight:1107.26Ref: TM-TP2207
1mg90.00€2mg138.00€5mg236.00€10mg409.00€25mg745.00€50mg1,189.00€100mg1,684.00€200mg2,268.00€Ozanimod
CAS:Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formula:C23H24N4O3Purity:98.68% - 99.58%Color and Shape:SolidMolecular weight:404.46Ref: TM-T6923
1mg46.00€5mg90.00€10mg137.00€25mg268.00€50mg430.00€100mg622.00€200mg879.00€500mg1,305.00€1mL*10mM (DMSO)90.00€ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.Formula:C77H123N25O19S2Purity:97.2%Color and Shape:SolidMolecular weight:1767.09Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formula:C25H28ClN3O2Purity:99.74%Color and Shape:SolidMolecular weight:437.96Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurity:97.62%Color and Shape:SolidMolecular weight:370.28Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83CYM2503
CAS:CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.
Formula:C45H55N5O7Purity:97.04%Color and Shape:SolidMolecular weight:777.95Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.Formula:C63H93N15O20SPurity:98.11%Color and Shape:SolidMolecular weight:1412.57HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purity:99.51%Color and Shape:SolidMolecular weight:614.57Netupitant
CAS:Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).Formula:C30H32F6N4OPurity:99.43%Color and Shape:SolidMolecular weight:578.59Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
2mg35.00€5mg51.00€10mg88.00€25mg120.00€50mg170.00€100mg250.00€200mg373.00€1mL*10mM (DMSO)57.00€Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.95% - 99.13%Color and Shape:SolidMolecular weight:269.73Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formula:C11H6O4Purity:99.97%Color and Shape:SolidMolecular weight:202.16Cinacalcet hydrochloride
CAS:Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-Formula:C22H23ClF3NPurity:99.96% - >99.99%Color and Shape:Off-White To Tan SolidMolecular weight:393.87Ref: TM-T2406
10mg50.00€25mg70.00€50mg88.00€100mg144.00€200mg185.00€500mg309.00€1mL*10mM (DMSO)52.00€BAY 41-8543
CAS:BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).
Formula:C21H21FN8OPurity:99.86%Color and Shape:SolidMolecular weight:420.44TCS-OX2-29
CAS:TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formula:C23H31N3O3Purity:99.81%Color and Shape:SolidMolecular weight:397.51Ref: TM-T4965
1mg35.00€5mg70.00€10mg96.00€25mg156.00€50mg215.00€100mg303.00€200mg449.00€1mL*10mM (DMSO)77.00€Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.Formula:C63H104N22O17SPurity:98.33%Color and Shape:SolidMolecular weight:1473.72β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurity:99.64%Color and Shape:SolidMolecular weight:2720.97L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFormula:C18H20Cl2N4Purity:97.36%Color and Shape:SolidMolecular weight:363.28Ref: TM-T11799
5mg40.00€10mg65.00€25mg111.00€50mg178.00€100mg259.00€200mg374.00€1mL*10mM (DMSO)34.00€Vericiguat
CAS:Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.
Formula:C19H16F2N8O2Purity:98.86% - 99.93%Color and Shape:SolidMolecular weight:426.38Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purity:>99.99%Color and Shape:SolidMolecular weight:1672.92Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Formula:C24H32ClNO6Purity:99.73%Color and Shape:Colorless LiquidMolecular weight:465.97Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:C19H26ClNOSPurity:99.53% - 99.56%Color and Shape:Almost White To White Crystalline PowderMolecular weight:351.93Bombesin acetate(31362-50-2 free base)
CAS:Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).Formula:C73H114N24O20SPurity:98.44%Color and Shape:SolidMolecular weight:1679.92FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formula:C41H61F3N10O10Purity:99.32%Color and Shape:SolidMolecular weight:910.99Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg50.00€10mg73.00€25mg138.00€50mg241.00€100mg358.00€200mg523.00€500mg822.00€1mL*10mM (DMSO)52.00€Blarcamesine hydrochloride
CAS:Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).Formula:C19H24ClNOPurity:99.57% - 99.9%Color and Shape:SolidMolecular weight:317.85Ref: TM-T4111
1mg35.00€2mg48.00€5mg70.00€10mg104.00€25mg207.00€50mg359.00€100mg588.00€200mg833.00€1mL*10mM (DMSO)78.00€Pranlukast hemihydrate
CAS:Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.Formula:C27H23N5O40·5H2OPurity:99.28%Color and Shape:SolidMolecular weight:490.52carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formula:C52H75N13O13S2Purity:99.86%Color and Shape:SolidMolecular weight:1154.37Fipamezole HCl
CAS:Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.Formula:C14H16ClFN2Color and Shape:SolidMolecular weight:266.74Urapidil
CAS:Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formula:C20H29N5O3Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:387.48
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