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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8626 products of "Metabolism"

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  • Sodium lauroyl glutamate

    CAS:
    <p>Sodium lauroyl glutamate (Acylglutamate LS-11) is an amino acid detergent and increases the solubility of long-chain alkyl gallates such as alkyl gallates.</p>
    Formula:C17H30NNaO5
    Purity:97.13%
    Color and Shape:Solid
    Molecular weight:351.41
  • (+)-Xylariamide A

    CAS:
    <p>(+)-Xylariamide A is a probe used for mycobacterial and fungal carbonic anhydrase.</p>
    Formula:C14H14ClNO6
    Color and Shape:Solid
    Molecular weight:327.72
  • Proadifen

    CAS:
    <p>Proadifen is a non-selective cytochrome P450 enzymes inhibitor, preventing some types of drug metabolism.</p>
    Formula:C23H31NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.5
  • Fmoc-Asp(OtBu)-Thr(psi(Me,Me)pro)-OH

    CAS:
    <p>Fmoc-Asp(OtBu)-Thr(psi(Me,Me)pro)-OH is a dipeptide.</p>
    Formula:C30H36N2O8
    Color and Shape:Solid
    Molecular weight:552.62
  • PD 113413

    CAS:
    <p>PD 113413 is a metabolite of quinapril, an angiotensin-converting enzyme inhibitor for the treatment of hypertension and congestive heart failure.</p>
    Formula:C23H24N2O4
    Color and Shape:Solid
    Molecular weight:392.45
  • 2-Hydroxy-3′-O-methyladenosine

    CAS:
    <p>2-Hydroxy-3′-O-methyladenosine serves as a synthetic intermediate in the study of ischemic heart disease, cerebrovascular disease, kidney disease, inflammatory allergies, and more. Derived from 2-Hydroxy-3′-O-methyladenosine, 2-phenylamino-N6,2-O-dimethyladenosine acts as an adenosine deaminase inhibitor with a Ki of 13 nM.</p>
    Formula:C11H15N5O5
    Color and Shape:Solid
    Molecular weight:297.27
  • PAT-494

    CAS:
    <p>PAT-494 is an inhibitor of type II Autotaxin.</p>
    Formula:C20H16FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.36
  • Nicodan Percutan

    CAS:
    <p>Nicodan Percutan (Propylnicotinat) is the propyl ester form of niacin, which is found in various animal and plant tissues to form the coenzymes NAD and NADP.</p>
    Formula:C9H11NO2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:165.19
  • Prasugrel chloride impurity

    CAS:
    <p>Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.</p>
    Formula:C20H21ClFNO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.9
  • Trimosulfa

    CAS:
    <p>Trimosulfa is a combination of trimethoprim and sulfamethoxazole, an antibiotic combination. Sulfamethoxazole inhibits dihydropteroate synthase, while trimethoprim inhibits dihydrofolate reductase (dihydrofolate reductase), making it effective for mild to moderate bacterial infections against many Gram-negative and Gram-positive bacteria.</p>
    Formula:C24H29N7O6S
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:543.6
  • Difluoro atorvastatin

    CAS:
    <p>Difluoro atorvastatin: an atorvastatin impurity reducing blood lipids, inhibits SV-SMC proliferation/invasion (IC50: 0.39/2.39 μM).</p>
    Formula:C33H34F2N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:576.63
  • JZP-MA-11

    CAS:
    <p>"JZP-MA-11 is a PET ligand that selectively targets ABHD6, inhibits with 126 nM IC50, and crosses the BBB for preclinical brain studies."</p>
    Formula:C15H17FN4O2S
    Color and Shape:Solid
    Molecular weight:336.38
  • GPAT-IN-1

    CAS:
    <p>GPAT-IN-1 is a glycerol 3-phosphate acyltransferase (GPAT) inhibitor, which can be used to study obesity and diabetes.</p>
    Formula:C21H26ClNO4S
    Purity:99.60% - 99.60%
    Color and Shape:Solid
    Molecular weight:423.95
  • DC-6-14

    CAS:
    <p>DC-6-14 is a cationic lipid known for its gene transfection activity, commonly utilized in the synthesis of liposomes.</p>
    Formula:C37H73ClN2O5
    Color and Shape:Solid
    Molecular weight:661.44
  • Flurtamone

    CAS:
    <p>Flurtamone is an agricultural chemical. Flurtamone mainly used as an herbicide.</p>
    Formula:C18H14F3NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.30
  • RPR132595A

    CAS:
    RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).
    Formula:C28H30N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.56
  • Acetaminophen mercapturate

    CAS:
    <p>Paracetamol Mercapturate is a metabolite of Acetaminophen. It can also be used in the biological study of urinary antihypertensive drugs.</p>
    Formula:C13H16N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.34
  • MDI-2268

    CAS:
    <p>MDI-2268, an inhibitor of plasma kallikrein inhibitor 1 (PAI-1), exhibits strong antithrombotic properties. It plays a role in regulating blood coagulation by promoting fibrinolysis and is applicable in research related to deep vein thrombosis.</p>
    Formula:C10H10F3N3O3
    Color and Shape:Solid
    Molecular weight:277.20
  • Ethyl phenylglyoxylate

    CAS:
    <p>Ethyl phenylglyoxylate (AI3 10033) is a simultaneous inhibitor and substrate of chicken liver carboxylesterase.</p>
    Formula:C10H10O3
    Purity:98.46%
    Color and Shape:Yellow Liquid
    Molecular weight:178.18
  • HSL-IN-5

    CAS:
    <p>HSL-IN-5 (Example 21) is a hormone-sensitive lipase (HSL) inhibitor with an IC₅₀ value of 0.2 μM, suitable for diabetes research.</p>
    Formula:C18H23F3N2O4
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:388.38
  • Milvexian

    CAS:
    <p>Milvexian (BMS-986177) is an oral antithrombotic, reversibly inhibiting human/rabbit FXIa with K i of 0.11/0.38 nM.</p>
    Formula:C28H23Cl2F2N9O2
    Color and Shape:Solid
    Molecular weight:626.45
  • Thevetin A

    CAS:
    <p>Thevetin A is a useful organic compound for research related to life sciences. The catalog number is T124930 and the CAS number is 37933-66-7.</p>
    Formula:C42H64O19
    Color and Shape:Solid
    Molecular weight:872.955
  • Bitertanol

    CAS:
    <p>Bitertanol (KWG 0599) is a triazole fungicide. Bitertanol inhibits demethylation, disrupts membrane function, and prevents sterol synthesis.</p>
    Formula:C20H23N3O2
    Purity:99.88%
    Color and Shape:Clear Browm Clear Liquid
    Molecular weight:337.42
  • PPM1A-IN-1

    CAS:
    <p>PPM1A-IN-1 (Compound IV-4) is an inhibitor of the PP2C Ser/Thr protein phosphatase Mg2+/Mn2+-dependent 1A. It exhibits antibacterial activity against Mycobacterium tuberculosis.</p>
    Formula:C16H15BrFNO2
    Color and Shape:Solid
    Molecular weight:352.2
  • 3-O-Methyltolcapone

    CAS:
    <p>3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.</p>
    Formula:C15H13NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:287.27
  • sEH inhibitor-17

    CAS:
    <p>sEH inhibitor-17 (compound 4f) is an orally active soluble epoxide hydrolase (sEH) inhibitor with an IC50 value of 2.94 nM. This compound exhibits anti-inflammatory properties.</p>
    Formula:C18H21F3N2O4S
    Color and Shape:Solid
    Molecular weight:418.43
  • BAY-721973

    CAS:
    <p>BAY-721973 is a bio-active chemical.</p>
    Formula:C21H16ClF3N4O4
    Color and Shape:Solid
    Molecular weight:480.82
  • Dimepiperate

    CAS:
    <p>Dimepiperate is an agent of biochemical.</p>
    Formula:C15H21NOS
    Color and Shape:Solid
    Molecular weight:263.40
  • Buthidazole

    CAS:
    <p>Buthidazole is a herbicide for selective weed control in corn.</p>
    Formula:C10H16N4O2S
    Color and Shape:Solid
    Molecular weight:256.33
  • FAAH-IN-8

    CAS:
    <p>FAAH-IN-8 (compound 11) is a competitive inhibitor of FAAH with an IC50 of 6.7 nM and a Ki of 5 nM. It exhibits high blood-brain permeability and a significant antioxidant profile without neurotoxicity [1].</p>
    Formula:C18H14N4O
    Color and Shape:Solid
    Molecular weight:302.33
  • SHP2-IN-29

    CAS:
    <p>SHP2-IN-29 (Compound 3), a potent inhibitor of SHP2, exhibits an IC 50 of 0.18 μM. Additionally, this compound demonstrates inhibitory activity against PTP1B and TCPTP, with IC 50 values of 4.27 μM and 4.74 μM, respectively.</p>
    Formula:C16H20O4
    Color and Shape:Solid
    Molecular weight:276.33
  • AKU-005

    CAS:
    <p>AKU-005 is a dual inhibitor of FAAH and MAGL, exhibiting IC50 values of 63 nM and 389 nM against rat and human FAAH, respectively. This compound has potential for researching trigeminal nociceptive hypersensitivity.</p>
    Formula:C20H21N5O
    Color and Shape:Solid
    Molecular weight:347.41
  • H-Arg-Lys-OH

    CAS:
    <p>H-Arg-Lys-OH is a dipeptide formed from L-lysine residues and L-arginyl.</p>
    Formula:C12H26N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.37
  • Atorvastatin acetonide

    CAS:
    <p>Atorvastatin acetonide, an impurity in Atorvastatin, lowers blood lipids; from patent WO2011131605A1.</p>
    Formula:C36H39FN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:598.7
  • 8-Azaadenine

    CAS:
    <p>8-Azaadenine (NSC-32797) is an inhibitor of xanthine oxidase with IC50 of 0.54 μM and Ki of 0.66 μM.</p>
    Formula:C4H4N6
    Purity:99.68%
    Color and Shape:White Powder
    Molecular weight:136.11
  • Nitrophenide

    CAS:
    Nitrophenide, a 3,3'-Dinitrodiphenyl disulfide, blocks M1PDH in the mannitol cycle, serving as an anticoccidial.
    Formula:C12H8N2O4S2
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:308.33
  • Transketolase-IN-3

    CAS:
    <p>Transketolase-IN-3: potent TK inhibitor with herbicidal effects on DS and AR, useful for herbicide research.</p>
    Formula:C20H9ClF3NO3
    Color and Shape:Solid
    Molecular weight:403.74
  • PNU-200579

    CAS:
    <p>PNU-200579 is a bio-active chemical.</p>
    Formula:C22H29NO3
    Color and Shape:Solid
    Molecular weight:355.47
  • 1-Decanesulfonic acid

    CAS:
    <p>1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.</p>
    Formula:C10H22O3S
    Color and Shape:Solid
    Molecular weight:222.35
  • Tolrestat

    CAS:
    <p>Tolrestat (AY-27773) is a potent inhibitor of aldose reductase (IC50 = 35 nM).</p>
    Formula:C16H14F3NO3S
    Purity:98.89% - >99.99%
    Color and Shape:Solid
    Molecular weight:357.35
  • Tesaglitazar

    CAS:
    <p>Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα</p>
    Formula:C20H24O7S
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:408.47
  • BIBB 515

    CAS:
    <p>BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.</p>
    Formula:C22H21ClN2O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:380.87
  • E3330

    CAS:
    <p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>
    Formula:C21H30O6
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:378.46
  • PCI-27483

    CAS:
    <p>PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.</p>
    Formula:C26H24N6O9S
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:596.57
  • L-m-Tyrosine

    CAS:
    <p>L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.</p>
    Formula:C9H11NO3
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:181.19
  • PF-05175157

    CAS:
    <p>PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,</p>
    Formula:C23H27N5O2
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:405.49
  • Calcipotriol monohydrate

    CAS:
    <p>Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.</p>
    Formula:C27H42O4
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:430.62
  • 3-Phenylbutyric acid

    CAS:
    <p>3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.</p>
    Formula:C10H12O2
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:164.2
  • 4-POBN

    CAS:
    <p>4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).</p>
    Formula:C7H9N3O
    Purity:99.60%
    Color and Shape:White Crystalline Powder
    Molecular weight:151.17
  • BKIDC-1553

    CAS:
    <p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>
    Formula:C22H23N5O2
    Color and Shape:Solid
    Molecular weight:389.45
  • TK-642

    CAS:
    <p>TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.</p>
    Formula:C17H20ClN7S
    Color and Shape:Solid
    Molecular weight:389.91
  • AMP-Deoxynojirimycin

    CAS:
    <p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>
    Formula:C22H39NO5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:397.55
  • JNJ-42165279 dihydrochloride

    CAS:
    <p>JNJ-42165279 (dihydrochloride) is an FAAH inhibitor with IC50 values of 70 nM for hFAAH and 313 nM for rFAAH, respectively [1].</p>
    Formula:C18H19Cl3F2N4O3
    Color and Shape:Solid
    Molecular weight:483.72
  • Phosphodiesterase-IN-1

    CAS:
    <p>Phosphodiesterase-IN-1 (Compound 7), a phosphodiesterase (PDE) inhibitor, exhibits anti-Plasmodium and antiproliferative activities. It effectively inhibits P. falciparum (strain 3D7) with an IC 50 value of 0.64 μM [1].</p>
    Formula:C15H15FN4O
    Color and Shape:Solid
    Molecular weight:286.3
  • Epostane

    CAS:
    <p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>
    Formula:C22H31NO3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:357.49
  • Riboflavine phosphate

    CAS:
    <p>Riboflavine phosphate (Flavin mononucleotide) is a derivative of Riboflavin.</p>
    Formula:C17H21N4O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.34
  • N-(α-Linolenoyl) Tyrosine

    CAS:
    <p>Certain chronic neurologic disorders, such as Parkinson's disease, are caused by an insufficiency of the neurotransmitter dopamine secondary to the degeneration</p>
    Formula:C27H39NO4
    Color and Shape:Solid
    Molecular weight:441.6
  • HFI-437

    CAS:
    <p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>
    Formula:C23H20N2O5
    Color and Shape:Solid
    Molecular weight:404.42
  • 2-TEDC

    CAS:
    <p>2-TEDC: Potent LOX inhibitor, blocks 5-LOX, 12-LOX, 15-LOX (IC50: 0.09, 0.013, 0.5 μM); aids atherosclerosis research.</p>
    Formula:C16H13NO4S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:315.34
  • Roxyl-9

    CAS:
    <p>Roxyl-9 is an inhibitor of IDO1 (Indoleamine 2,3-dioxygenase 1) [1].</p>
    Formula:C18H13N3O2
    Color and Shape:Solid
    Molecular weight:303.31
  • SAHO

    CAS:
    <p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>
    Formula:C14H20N6O6S
    Color and Shape:Solid
    Molecular weight:400.41
  • JNJ-42314415

    CAS:
    <p>JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.</p>
    Formula:C19H23N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.42
  • BMP-22

    CAS:
    <p>BMP-22 selectively inhibits autotaxin (IC50=170 nM), blocks LPA production and MM1 cell invasion, and reduces lung metastases in mice at 0.5 mg/kg/day.</p>
    Formula:C22H39O3P
    Color and Shape:Solid
    Molecular weight:382.52
  • Clethodim

    CAS:
    <p>Clethodim is a selective herbicide inhibiting acetyl-CoA carboxylase, effective on grasses with low environmental persistence and moderate toxicity to wildlife.</p>
    Formula:C17H26ClNO3S
    Purity:99.99%
    Color and Shape:Light Yellow Liquid
    Molecular weight:359.91
  • α-Glucosidase-IN-6

    CAS:
    <p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>
    Formula:C24H17ClF3NO3S
    Color and Shape:Solid
    Molecular weight:491.91
  • Glyoxalase I inhibitor 4

    CAS:
    <p>Glyoxalase I inhibitor 4 is a potent inhibitor of glyoxalase I (GLO1) (Ki: 10 nM).</p>
    Formula:C17H21IN4O8S
    Color and Shape:Solid
    Molecular weight:568.34
  • Enpp-1-IN-17

    CAS:
    <p>Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and &gt;1 μM for ATP</p>
    Formula:C18H24N4O2
    Color and Shape:Solid
    Molecular weight:328.41
  • BRD9500

    CAS:
    <p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>
    Formula:C15H18FN3O2
    Color and Shape:Solid
    Molecular weight:291.32
  • JZP-MA-13


    <p>JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.</p>
    Formula:C14H15FN4O3S
    Color and Shape:Solid
    Molecular weight:338.36
  • Flutolanil

    CAS:
    <p>Flutolanil: a fungicide targeting R. solani in rice, toxic to zebrafish.</p>
    Formula:C17H16F3NO2
    Color and Shape:Solid
    Molecular weight:323.31
  • BI-4924

    CAS:
    BI-4924 is a PHGDH inhibitor that disrupts serine biosynthesis by intracellular trapping and can be used to study metabolic disorders.
    Formula:C21H20Cl2N2O6S
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:499.36
  • Lp-PLA2-IN-4

    CAS:
    <p>Lp-PLA2-IN-4, a potent inhibitor of Lp-PLA2/PAF-AH, may target Alzheimer's, atherosclerosis. (WO2021228159A1, Compound 38)</p>
    Formula:C23H18F5N3O4
    Color and Shape:Solid
    Molecular weight:495.4
  • GGsTop

    CAS:
    <p>GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.</p>
    Formula:C13H18NO7P
    Purity:98.96%
    Color and Shape:Solid
    Molecular weight:331.26
  • IDO-IN-11

    CAS:
    <p>IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).</p>
    Formula:C19H23BrFN7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:544.4
  • IACS-8968 R-enantiomer

    CAS:
    <p>IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Formula:C17H18F3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.35
  • FC11409B

    CAS:
    <p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>
    Formula:C29H23BF4N2O3S
    Color and Shape:Solid
    Molecular weight:566.38
  • LY 113174

    CAS:
    <p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>
    Formula:C17H10Cl2N2
    Color and Shape:Solid
    Molecular weight:313.18
  • 3-Oxo-hop-22(29)-ene

    CAS:
    <p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>
    Formula:C30H48O
    Color and Shape:Solid
    Molecular weight:424.7
  • LEO 39652

    CAS:
    <p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>
    Formula:C23H23N3O5
    Color and Shape:Solid
    Molecular weight:421.45
  • α-Glucosidase-IN-2

    CAS:
    <p>α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an</p>
    Formula:C17H11N3O2S2
    Color and Shape:Solid
    Molecular weight:353.42
  • BMS-351

    CAS:
    <p>BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.</p>
    Formula:C15H12F3N3
    Color and Shape:Solid
    Molecular weight:291.27
  • hCAIX/XII-IN-4

    CAS:
    <p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and &gt;10000 nM (CAI/CAII).</p>
    Formula:C20H16N2O5
    Color and Shape:Solid
    Molecular weight:364.35
  • Carbonic anhydrase inhibitor 11

    CAS:
    <p>Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.</p>
    Formula:C19H15F3N4O3S2
    Color and Shape:Solid
    Molecular weight:468.47
  • PTP1B-IN-15

    CAS:
    <p>PTP1B-IN-15 is a potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor that has shown research potential in type II diabetes and obesity.</p>
    Formula:C19H17Br2NO5S
    Color and Shape:Solid
    Molecular weight:531.22
  • (S)-Bromoenol lactone

    CAS:
    <p>(S)-BEL, a chiral inhibitor of iPLA2β, blocks vasopressin-induced arachidonate release in A10 cells; IC50 = 2μM.</p>
    Formula:C16H13BrO2
    Color and Shape:Solid
    Molecular weight:317.18
  • Glycogen phosphorylase-IN-1

    CAS:
    <p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>
    Formula:C17H15ClF2N4O4
    Purity:97.98% - 98.15%
    Color and Shape:Solid
    Molecular weight:412.78
  • sEH inhibitor-3

    CAS:
    <p>sEH inhibitor-3 is an orally available, selective and potent inhibitor of sEH for cancer research.</p>
    Formula:C19H23F4N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.4
  • Senazodan hydrochloride

    CAS:
    <p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>
    Formula:C15H15ClN4O
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:302.76
  • ICI 211965

    CAS:
    <p>ICI 211965 is a selective and orally potent of 5-Lipoxygenase (5-LPO).</p>
    Formula:C24H23NO2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.51
  • SCH-42354

    CAS:
    <p>SCH-42354: potent oral NEP inhibitor, activates ANP &amp; leu-enkephalin, has anti-hypertensive properties, IC50s of 8.3 &amp; 10.0 nM.</p>
    Formula:C16H23NO3S2
    Color and Shape:Solid
    Molecular weight:341.49
  • BI-135585

    CAS:
    <p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>
    Formula:C28H32N2O4
    Purity:99.45% - 99.57%
    Color and Shape:Solid
    Molecular weight:460.57
  • FXR agonist 4


    <p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>
    Formula:C21H28ClN3O
    Color and Shape:Solid
    Molecular weight:373.92
  • 6-Hydroxyluteolin

    CAS:
    <p>6-Hydroxyluteolin, a flavonoid compound extracted from Salvia amarissima Ortega, inhibits aldose reductase (AR) and has antimicrobial activity.</p>
    Formula:C15H10O7
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:302.24
  • IDO-IN-14

    CAS:
    <p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>
    Formula:C23H23ClN4O2
    Color and Shape:Solid
    Molecular weight:422.91
  • AMG-7980

    CAS:
    <p>AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.</p>
    Formula:C19H22N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.4
  • MitoTEMPO hydrate

    CAS:
    <p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>
    Formula:C29H35N2O2P·Cl·H2O
    Color and Shape:Solid
    Molecular weight:528.04
  • Quinethazone

    CAS:
    <p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>
    Formula:C10H12ClN3O3S
    Color and Shape:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)
    Molecular weight:289.74
  • HS79

    CAS:
    <p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>
    Formula:C19H22N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.47
  • Hydroxychlorodenafil

    CAS:
    <p>Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>
    Formula:C19H23ClN4O3
    Color and Shape:Solid
    Molecular weight:390.86
  • Lp-PLA2-IN-3

    CAS:
    <p>Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.</p>
    Formula:C20H13ClF3N3O3S
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:467.85