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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8626 products of "Metabolism"

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  • Anticancer agent 70

    CAS:
    <p>Compound 21 is a powerful anticancer agent with cytotoxicity against various cancers, causing cell cycle arrest and affecting p53/p21 levels and mitochondria.</p>
    Formula:C13H9Cl2N3O2S
    Color and Shape:Solid
    Molecular weight:342.2
  • PGMI-004A

    CAS:
    <p>PGMI-004A is an effective inhibitor of phosphoglycerate mutase 1 (IC50: 13.1 μM).</p>
    Formula:C21H12F3NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.38
  • Rev 6207

    CAS:
    <p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>
    Formula:C21H31N3O5
    Color and Shape:Solid
    Molecular weight:405.49
  • PGAM1-IN-1

    CAS:
    <p>PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].</p>
    Formula:C19H11ClFNO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.81
  • MIPS1455

    CAS:
    <p>MIPS1455 is a photoactivatable allosteric M1 muscarinic acetylcholine receptor ligand.</p>
    Formula:C24H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.4
  • Eprozinol dihydrochloride

    CAS:
    <p>Eprozinol dihydrochloride has anti-bronchoconstrictive activity.</p>
    Formula:C22H31ClN2O2
    Color and Shape:Solid
    Molecular weight:390.95
  • Arabinose 1,5-diphosphate

    CAS:
    <p>Arabinose 1,5-diphosphate is a bisphosphatase inhibitor.</p>
    Formula:C5H12O11P2
    Color and Shape:Solid
    Molecular weight:310.09
  • AJS1669

    CAS:
    <p>AJS1669, an activator of muscle glycogen synthase, improves glucose metabolism and reduces body fat mass in mice.</p>
    Formula:C26H21F2NO6S
    Color and Shape:Solid
    Molecular weight:513.51
  • Cholesteryl Palmitoleate

    CAS:
    <p>Cholesteryl palmitoleate, a cholesterol ester, exhibits elevated plasma levels in ApoE-/- mice following exposure to cigarette smoke and in pediatric patients diagnosed with biliary atresia. It serves as a standard for identifying cholesterol esters in human meibomian gland secretions.</p>
    Formula:C43H74O2
    Color and Shape:Solid
    Molecular weight:623.1
  • Albifylline

    CAS:
    <p>Albifylline: a xanthine derivative, anti-asthmatic, reduces leukocyte adhesion, enhances liver microcirculation post-hemorrhagic shock.</p>
    Formula:C13H20N4O3
    Color and Shape:Solid
    Molecular weight:280.32
  • AHR-activator-1023

    CAS:
    <p>AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.</p>
    Formula:C14H8Cl2N2O
    Color and Shape:Solid
    Molecular weight:291.13
  • AHR-15010

    CAS:
    <p>AHR-15010 is a novel anti-arthritic agent.</p>
    Formula:C10H16N2O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.37
  • K103 Hydrochloride

    CAS:
    <p>K103 Hydrochloride, an inhibitor of peptidoglycan synthesis, targets the lipid II precursor.</p>
    Formula:C19H22Cl2N2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.36
  • MK-0952

    CAS:
    <p>MK-0952 treats memory loss and cognitive issues; it's a potent, selective PDE4 inhibitor with restricted blood activity.</p>
    Formula:C28H22FN3O4
    Color and Shape:Solid
    Molecular weight:483.49
  • 2-Methyldecanenitrile

    CAS:
    <p>2-Methyldecanenitrile, intense peach scent with lactone notes, stable in all pH, effective at low concentration.</p>
    Formula:C11H21N
    Purity:98%
    Color and Shape:Colourless Liquid Liquid
    Molecular weight:167.29
  • AZD8329

    CAS:
    <p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>
    Formula:C25H31N3O3
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:421.53
  • GSK 264220A

    CAS:
    <p>endothelial lipase and lipoprotein lipase inhibitor</p>
    Formula:C17H21N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.43
  • Levophencynonate HCl

    CAS:
    <p>Levophencynonate HCl is a muscarinic receptor antagonist.</p>
    Formula:C22H32ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.95
  • Z-321

    CAS:
    <p>Z-321 is an inhibitor of prolyl endopeptidase.</p>
    Formula:C19H24N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.47
  • DU717

    CAS:
    <p>DU717 is an antihypertensive agent.</p>
    Formula:C12H15ClN4O2S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:314.79
  • 3-Oxo-hop-22(29)-ene

    CAS:
    <p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>
    Formula:C30H48O
    Color and Shape:Solid
    Molecular weight:424.7
  • LEO 39652

    CAS:
    <p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>
    Formula:C23H23N3O5
    Color and Shape:Solid
    Molecular weight:421.45
  • CGP-28014

    CAS:
    <p>CGP-28014 inhibits COMT, boosts renal dopamine &amp; DOPAC excretion, lowers HVA, no effect on renal sodium.</p>
    Formula:C12H19N3O
    Color and Shape:Solid
    Molecular weight:221.3
  • ME-143

    CAS:
    <p>ME-143, a 2nd-gen NADH oxidase inhibitor, blocks WNT/β-catenin pathway, active against various cancers in vitro/vivo.</p>
    Formula:C21H18O4
    Color and Shape:Solid
    Molecular weight:334.37
  • AMPD2 inhibitor 2


    <p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>
    Formula:C26H27F2N3O3
    Color and Shape:Solid
    Molecular weight:467.51
  • 11β-HSD1-IN-9

    CAS:
    <p>11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.</p>
    Formula:C13H9F3N2O
    Color and Shape:Solid
    Molecular weight:266.22
  • CL 242817

    CAS:
    <p>CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).</p>
    Formula:C18H21NO5S
    Color and Shape:Solid
    Molecular weight:363.43
  • Nampt-IN-7

    CAS:
    <p>Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).</p>
    Formula:C20H21N5O3
    Color and Shape:Solid
    Molecular weight:379.41
  • DGAT1-IN-3

    CAS:
    <p>DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.</p>
    Formula:C20H19F3N4O3
    Color and Shape:Solid
    Molecular weight:420.39
  • 14(S)-HDHA

    CAS:
    <p>DHA is an ω-3 important for development and therapy for inflammation and cancer; its derivative, 14(S)-HDHA, aids in reducing inflammation.</p>
    Formula:C22H32O3
    Color and Shape:Solid
    Molecular weight:344.49
  • Camylofin Hydrochloride

    CAS:
    <p>Camylofin HCl is an antispasmodic used in labor treatment and is also used to deliver drug therapy for ulcerative colinitis.</p>
    Formula:C19H33ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.94
  • 8-CSC

    CAS:
    <p>8-CSC: hMAO-B inhibitor (Ki: 235 nM, baboon liver) &amp; A2A receptor affinity (Ki: 36 nM, rat brain).</p>
    Formula:C16H15ClN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.77
  • Risotilide

    CAS:
    <p>Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.</p>
    Formula:C15H27N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.52
  • F-1394

    CAS:
    <p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>
    Formula:C33H61N3O6
    Color and Shape:Solid
    Molecular weight:595.85
  • NC1153

    CAS:
    <p>NC1153 blocks IL-2/JAK3/STAT5a/b, aids allograft survival, reduces toxicities.</p>
    Formula:C18H38Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:369.42
  • MAO-B Inhibitor 58

    CAS:
    <p>MAO-B inhibitor 58 is an effective, selective, and reversible inhibitor of monoamine oxidase B.</p>
    Formula:C14H9Cl2N3
    Color and Shape:Solid
    Molecular weight:290.15
  • KCN1

    CAS:
    <p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>
    Formula:C26H27NO5S
    Color and Shape:Solid
    Molecular weight:465.56
  • RORγt modulator 2

    CAS:
    <p>RORγt modulator 2 is a modulator of retinol-related orphan receptor γt (RORyt) (IC50&lt;50 nM) and can be used in the study of RORγt-mediated diseases such as pain</p>
    Formula:C28H29ClN2O4S
    Color and Shape:Solid
    Molecular weight:525.06
  • Muristerone A

    CAS:
    <p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>
    Formula:C27H44O8
    Color and Shape:Solid
    Molecular weight:496.63
  • CK2-IN-6

    CAS:
    <p>CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.</p>
    Formula:C19H16ClN7O2
    Color and Shape:Solid
    Molecular weight:409.83
  • IDO1-IN-17

    CAS:
    <p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>
    Formula:C28H32BrClFN5O2
    Color and Shape:Solid
    Molecular weight:604.94
  • Carbonic anhydrase inhibitor 13

    CAS:
    <p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>
    Formula:C17H15N5O3S2
    Color and Shape:Solid
    Molecular weight:401.46
  • hCAIX-IN-6

    CAS:
    <p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>
    Formula:C18H12N2O4S
    Color and Shape:Solid
    Molecular weight:352.36
  • MSPG

    CAS:
    <p>mGlu receptor antagonist</p>
    Formula:C9H11NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:245.25
  • α-Glucosidase-IN-10

    CAS:
    <p>α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.</p>
    Formula:C21H15BrN4O2S
    Color and Shape:Solid
    Molecular weight:467.34
  • S 12340

    CAS:
    <p>S 12340 is a potent inhibitor of the oxidative modification of low-density lipoprotein.</p>
    Formula:C24H38N2O3S
    Color and Shape:Solid
    Molecular weight:434.64
  • UCM 765

    CAS:
    <p>UCM 765 is a partial agonist of melatonin MT(2) receptor.</p>
    Formula:C17H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.35
  • TUPS

    CAS:
    <p>TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.</p>
    Formula:C14H18F3N3O4S
    Color and Shape:Solid
    Molecular weight:381.37
  • AX 048

    CAS:
    <p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>
    Formula:C22H41NO4
    Color and Shape:Solid
    Molecular weight:383.57
  • Oxagrelate

    CAS:
    <p>Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.</p>
    Formula:C14H16N2O4
    Color and Shape:Solid
    Molecular weight:276.29
  • PDE5-IN-4

    CAS:
    <p>PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,</p>
    Formula:C21H27N5O5S
    Color and Shape:Solid
    Molecular weight:461.53
  • Boc-Glu(OBzl)-OSu

    CAS:
    <p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>
    Formula:C21H26N2O8
    Color and Shape:Solid
    Molecular weight:434.44
  • α-Amylase/α-Glucosidase-IN-2

    CAS:
    <p>α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM</p>
    Formula:C22H16ClN5
    Color and Shape:Solid
    Molecular weight:385.85
  • IDO1-IN-15

    CAS:
    <p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>
    Formula:C13H14BrFN6O3
    Color and Shape:Solid
    Molecular weight:401.19
  • CL67

    CAS:
    <p>CL67 is a hypoxia-inducible factor pathway inhibitor. It acts by binding to a G-quadruplex higher-order structure in the HIF promoter sequence in vitro.</p>
    Formula:C38H42N10O2
    Color and Shape:Solid
    Molecular weight:670.81
  • hCAIX-IN-14

    CAS:
    <p>hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .</p>
    Formula:C11H17ClN6O2S
    Color and Shape:Solid
    Molecular weight:332.81
  • ATX inhibitor 8

    CAS:
    <p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>
    Formula:C28H26N10O
    Color and Shape:Solid
    Molecular weight:518.57
  • FAAH-IN-7


    <p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>
    Formula:C26H29N3O4
    Color and Shape:Solid
    Molecular weight:447.53
  • Enpp-1-IN-8

    CAS:
    <p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>
    Formula:C19H26N6O4S
    Color and Shape:Solid
    Molecular weight:434.51
  • Risarestat

    CAS:
    <p>Risarestat (CT-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (TR) antagonist for the treatment of hypoglycemia.</p>
    Formula:C16H21NO4S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:323.41
  • Rentiapril racemate

    CAS:
    <p>Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.</p>
    Formula:C13H15NO4S2
    Purity:98.96% - >99.99%
    Color and Shape:Solid
    Molecular weight:313.39
  • MDK-4823

    CAS:
    <p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>
    Formula:C28H36N4O
    Color and Shape:Solid
    Molecular weight:444.61
  • NBD-125

    CAS:
    <p>NBD-125 (B-12) is a berberine analogue. NBD-125 is an RXRα activator. The IC50 value of NBD-125 in KM12C cell is 31.10 μM [1].</p>
    Formula:C19H18ClNO2
    Color and Shape:Solid
    Molecular weight:327.81
  • p-Synephrine

    CAS:
    <p>p-Synephrine is a natural product for research related to life sciences. The catalog number is T8265 and the CAS number is 614-35-7.</p>
    Formula:C9H13NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:167.21
  • Nampt-IN-9

    CAS:
    <p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>
    Formula:C26H33N3O4
    Color and Shape:Solid
    Molecular weight:451.56
  • Delapril

    CAS:
    <p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>
    Formula:C26H32N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • Metyltetraprole

    CAS:
    <p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>
    Formula:C19H17ClN6O2
    Color and Shape:Solid
    Molecular weight:396.83
  • α-Glucosidase-IN-9

    CAS:
    <p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>
    Formula:C19H12N4OS
    Color and Shape:Solid
    Molecular weight:344.39
  • GNX-865

    CAS:
    <p>GNX-865 is an inhibitor of mitochondrial permeability transition pore (mtPTP).</p>
    Formula:C16H14ClNO3
    Color and Shape:Solid
    Molecular weight:303.74
  • TM6008

    CAS:
    <p>TM6008 is an inhibitor of prolyl hydroxylase that protects against cell death after hypoxia.</p>
    Formula:C21H17N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.39
  • (Rac)-3′-Hydroxy simvastatin

    CAS:
    <p>(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.</p>
    Formula:C25H38O6
    Color and Shape:Solid
    Molecular weight:434.57
  • YM-75466

    CAS:
    <p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>
    Formula:C28H35N5O8S2
    Color and Shape:Solid
    Molecular weight:633.74
  • LTV-1

    CAS:
    <p>LTV-1 has the potential for autoimmunity treatment. LTV-1 is a potent lymphoid tyrosine phosphatase (LYP) inhibitor in T cells with an IC50 of 508 nM.</p>
    Formula:C26H20N2O5S
    Color and Shape:Solid
    Molecular weight:472.51
  • GNE-3500

    CAS:
    <p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>
    Formula:C24H30FN3O3S
    Color and Shape:Solid
    Molecular weight:459.58
  • hCAIX-IN-7

    CAS:
    <p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: &gt;10000 nM).</p>
    Formula:C18H12FNO3
    Color and Shape:Solid
    Molecular weight:309.29
  • DMPAC-Chol

    CAS:
    <p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>
    Formula:C33H58N2O2
    Color and Shape:Solid
    Molecular weight:514.83
  • Glyoxalase I inhibitor 2

    CAS:
    <p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>
    Formula:C24H23N3O4S
    Color and Shape:Solid
    Molecular weight:449.52
  • Fluindione

    CAS:
    <p>Fluindione is a hematologic drug.</p>
    Formula:C15H9FO2
    Color and Shape:Solid
    Molecular weight:240.23
  • Senazodan

    CAS:
    <p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>
    Formula:C15H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.3
  • URB532

    CAS:
    <p>URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Formula:C18H21NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.36
  • AN3199

    CAS:
    <p>AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.</p>
    Formula:C17H18BNO5
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:327.14
  • SCD1 inhibitor-1

    CAS:
    SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).
    Formula:C21H23N3NaO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • Inolitazone dihydrochloride

    CAS:
    <p>Inolitazone dihydrochloride is an effective, high-affinity PPARγ agonist; its biological activity is dependent on PPARγ (IC50:0.8 nM) to inhibit cell growth.</p>
    Formula:C27H28Cl2N4O4S
    Color and Shape:Solid
    Molecular weight:575.51
  • Kojibiose

    CAS:
    <p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>
    Formula:C12H22O11
    Purity:99.933%
    Color and Shape:Solid
    Molecular weight:342.3
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • Cholesteryl behenate

    CAS:
    <p>Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.</p>
    Formula:C49H88O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:709.22
  • PSB-1410

    CAS:
    <p>PSB-1410 is a selective and highly efficient monoamine oxidase B (MAO-B) inhibitor, which can be used in research on neurological diseases.</p>
    Formula:C15H10Cl2N2O
    Purity:98.69%
    Color and Shape:Solid
    Molecular weight:305.16
  • CYP3A4-IN-3

    CAS:
    <p>CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.</p>
    Formula:C34H39N3O3S
    Color and Shape:Solid
    Molecular weight:569.76
  • α-Glucosidase-IN-4

    CAS:
    <p>α-Glucosidase-IN-4 is a potent α-glucosidase inhibitor with antihypertensive and hypoglycemic activity.</p>
    Formula:C19H14O4
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:306.31
  • BI 689648

    CAS:
    <p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>
    Formula:C16H18N4O2
    Color and Shape:Solid
    Molecular weight:298.34
  • Quazodine

    CAS:
    <p>Quazodine is a phosphodiesterase inhibitor.</p>
    Formula:C12H14N2O2
    Color and Shape:Solid
    Molecular weight:218.25
  • EP6

    CAS:
    <p>EP6 blocks 5-LO, key in the AA cascade, reducing leukotrienes to curb inflammation and allergies.</p>
    Formula:C24H30N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:390.52
  • Abiraterone metabolite 1

    CAS:
    <p>Abiraterone metabolite 1, a derivative of abiraterone, inhibits CYP17A1, halts androgen formation, aiding in prostate cancer treatment.</p>
    Formula:C24H33NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.52
  • hCAII-IN-1

    CAS:
    <p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>
    Formula:C21H21BrN6O4S
    Color and Shape:Solid
    Molecular weight:533.4
  • ALRT 1550

    CAS:
    <p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>
    Formula:C23H32O2
    Color and Shape:Solid
    Molecular weight:340.5
  • Endothelial lipase inhibitor-1

    CAS:
    <p>Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.</p>
    Formula:C22H22N4O4
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:406.43
  • Deltasonamide 2

    CAS:
    <p>Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>
    Formula:C30H39ClN6O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:647.25
  • 7-Ketolithocholic acid

    CAS:
    <p>7-Ketolithocholic acid absorbs and reduces endogenous bile acid and cholesterol secretion.</p>
    Formula:C24H38O4
    Purity:98.68% - 99.9%
    Color and Shape:White - Almost White Solid Powder
    Molecular weight:390.56
  • TM6089

    CAS:
    <p>TM6089 is an inhibitor of Prolyl Hydroxylase that stimulates HIF activity without iron chelation, induces angiogenesis, and protects organ against ischemia.</p>
    Formula:C13H14N4O3S
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:306.34
  • hCAIX-IN-10

    CAS:
    <p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>
    Formula:C28H21N3O3S
    Color and Shape:Solid
    Molecular weight:479.55
  • SHP844

    CAS:
    <p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>
    Formula:C29H24ClN5O6
    Color and Shape:Solid
    Molecular weight:573.98
  • Angiogenesis agent 1

    CAS:
    <p>Compound C-31, a salidroside-based glycoside, activates HIF-1α and may aid in diabetic limb ischemia studies.</p>
    Formula:C20H24O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.4
  • RORγt inverse agonist 28

    CAS:
    <p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>
    Formula:C23H18Cl2F3NO5S
    Color and Shape:Solid
    Molecular weight:548.36
  • ASM-IN-1

    CAS:
    <p>ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.</p>
    Formula:C16H12BrN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:390.19
  • HZ52

    CAS:
    <p>HZ52: Potent reversible 5-LO inhibitor; IC50 0.7 μM; blocks LTs in human leukocytes.</p>
    Formula:C24H26ClN3O2S
    Color and Shape:Solid
    Molecular weight:456
  • ATX inhibitor 20

    CAS:
    <p>ATX inhibitor 20 is a potent inhibitor of ATX (IC50: 2.3 nM).</p>
    Formula:C31H34FN5O3
    Color and Shape:Solid
    Molecular weight:543.63
  • Endothall

    CAS:
    <p>Endothall is an effective protein phosphatase 2A (PP2A) inhibitor, exerting inhibitory effects on both PP2A and PP1, with IC50 values of 90 nM and 5 µM,</p>
    Formula:C8H10O5
    Purity:98.92% - ≥98%
    Color and Shape:Cyrstalline White Solid The Monohydrate Is In The Form Of Colorless Crystals Non Corrosive Used As A Selective Herbicide
    Molecular weight:186.16
  • AVE5688

    CAS:
    <p>AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa).</p>
    Formula:C16H8ClF5N2O5
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:438.69
  • GK187

    CAS:
    <p>GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.</p>
    Formula:C14H15F5O2
    Color and Shape:Solid
    Molecular weight:310.26
  • Leniquinsin

    CAS:
    <p>Leniquinsin is an antihypertensive compound. It is a phosphodiesterase inhibitor and a potent vasodilator.</p>
    Formula:C20H20N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.38
  • 1E7-03

    CAS:
    <p>1E7-03 is an inhibitor of HIV-1 transcription, by targeting host Protein Phosphatase-1 (PP1).</p>
    Formula:C28H29N3O6
    Color and Shape:Solid
    Molecular weight:503.55
  • Oosponol

    CAS:
    <p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>
    Formula:C11H8O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:220.18
  • Lucerastat

    CAS:
    <p>Lucerastat(NBDGJ) is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.</p>
    Formula:C10H21NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:219.28
  • 2-TEDC

    CAS:
    <p>2-TEDC: Potent LOX inhibitor, blocks 5-LOX, 12-LOX, 15-LOX (IC50: 0.09, 0.013, 0.5 μM); aids atherosclerosis research.</p>
    Formula:C16H13NO4S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:315.34
  • Clethodim

    CAS:
    <p>Clethodim is a selective herbicide inhibiting acetyl-CoA carboxylase, effective on grasses with low environmental persistence and moderate toxicity to wildlife.</p>
    Formula:C17H26ClNO3S
    Purity:99.99%
    Color and Shape:Light Yellow Liquid
    Molecular weight:359.91
  • Oleyl Anilide

    CAS:
    <p>"Oleyl analide (OA) inhibits ACAT (IC50 26 μM), linked to toxic oil syndrome (TOS) with eosinophilia, T-cell activation, and high IL-4, IL-2R, IL-5."</p>
    Formula:C24H39NO
    Color and Shape:Solid
    Molecular weight:357.57
  • GGsTop

    CAS:
    <p>GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.</p>
    Formula:C13H18NO7P
    Purity:98.96%
    Color and Shape:Solid
    Molecular weight:331.26
  • Senazodan hydrochloride

    CAS:
    <p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>
    Formula:C15H15ClN4O
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:302.76
  • BKIDC-1553

    CAS:
    <p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>
    Formula:C22H23N5O2
    Color and Shape:Solid
    Molecular weight:389.45
  • GSK376501A

    CAS:
    <p>GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.</p>
    Formula:C32H37NO6
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:531.64
  • AMP-Deoxynojirimycin

    CAS:
    <p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>
    Formula:C22H39NO5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:397.55
  • Epostane

    CAS:
    <p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>
    Formula:C22H31NO3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:357.49
  • ATX inhibitor 5

    CAS:
    <p>ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.</p>
    Formula:C22H18ClF3N6O
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:474.87
  • Quinapril-d5

    CAS:
    <p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>
    Formula:C25H25D5N2O5
    Color and Shape:Solid
    Molecular weight:443.55
  • TF-S14

    CAS:
    <p>TF-S14 is an inverse agonist of RORγt. It functions by binding to RORγt and inhibiting its activity, leading to a reduction in Th17 cell-associated cytokine production, including IL-17A, IL-21, and IL-22. TF-S14 is applicable in research related to autoimmune diseases and allogeneic transplant rejection.</p>
    Formula:C22H27N3O2S
    Color and Shape:Solid
    Molecular weight:397.53
  • SAHO

    CAS:
    <p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>
    Formula:C14H20N6O6S
    Color and Shape:Solid
    Molecular weight:400.41
  • JNJ-42314415

    CAS:
    <p>JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.</p>
    Formula:C19H23N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.42
  • TA-7552

    CAS:
    <p>TA-7552 is a potent agent of cholesterol-lowering.</p>
    Formula:C25H26O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.47
  • BMP-22

    CAS:
    <p>BMP-22 selectively inhibits autotaxin (IC50=170 nM), blocks LPA production and MM1 cell invasion, and reduces lung metastases in mice at 0.5 mg/kg/day.</p>
    Formula:C22H39O3P
    Color and Shape:Solid
    Molecular weight:382.52
  • BFE-37

    CAS:
    <p>BFE-37 is a partial agonist of beta-adrenergic.</p>
    Formula:C16H23NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.36
  • PMPMEase-IN L-28

    CAS:
    <p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>
    Formula:C17H29FO2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.54
  • L 662583

    CAS:
    <p>L 662583 is a topical inhibitor of carbonic anhydrase.</p>
    Formula:C13H17ClN2O5S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.93
  • Cedefingol

    CAS:
    <p>Cedefingol is an antineoplastic agent.</p>
    Formula:C20H41NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:343.54
  • Pirbuterol hydrochloride

    CAS:
    <p>Pirbuterol hydrochloride is a bronchodilator.</p>
    Formula:C12H21ClN2O3
    Color and Shape:Solid
    Molecular weight:276.76
  • Pegnivacogin

    CAS:
    <p>Pegnivacogin is a coagulation factor IXa RNA aptamer inhibitor.</p>
    Formula:C20H40N3O11P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.52
  • D-4418

    CAS:
    <p>D-4418, a PDE4 inhibitor in development, targets asthma and COPD as an anti-inflammatory treatment.</p>
    Formula:C16H11Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.18
  • L-651392

    CAS:
    <p>L-651392 is an inhibitor of leukotriene.</p>
    Formula:C14H10BrNO3S
    Color and Shape:Solid
    Molecular weight:352.2
  • MMV-667492

    CAS:
    <p>MMV-667492 is an effective inhibitor of Ezrin.</p>
    Formula:C17H19N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:313.35
  • MLS000536924

    CAS:
    <p>MLS000536924 is a potent and selective competitive human epithelial 15-lipoxygenase-2 inhibitor.</p>
    Formula:C16H15N3S
    Color and Shape:Solid
    Molecular weight:281.38
  • Lysine Orotate

    CAS:
    <p>Lysine Orotate blocks Herpes virus replication, effective against HSV-1, HSV-2, CMV, EBV, and Varicella.</p>
    Formula:C11H18N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.28
  • PG-9 maleate

    CAS:
    <p>Increases release of acetylcholine</p>
    Formula:C21H26BrNO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.34
  • OH-Ubenimex

    CAS:
    <p>OH-Ubenimex is an orally active aminopeptidase inhibitor that has an immunomodulating action.</p>
    Formula:C16H24N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.37
  • α-RA-F

    CAS:
    <p>Alpha-RA-F increases collagen, lowers MMPs in human fibroblasts, non-toxic.</p>
    Formula:C16H16N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:300.31
  • myomiR-IN-1

    CAS:
    <p>myomiR-IN-1 inhibits myoD translation in C2C12 cells, doesn't affect myoD mRNA, and reduces differentiation markers.</p>
    Formula:C33H27NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:533.57
  • 2-Iodoestradiol

    CAS:
    <p>2-Iodoestradiol is an effective human sex hormone-binding globulin (SHBG) ligand.</p>
    Formula:C18H23IO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.28
  • OMS-824

    CAS:
    <p>OMS-824 is a phosphodiesterase-10 inhibitor that slows or stops the hydrolysis of cAMP and cGMP.</p>
    Formula:C21H21BrN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.32
  • PF-05387252

    CAS:
    <p>PF-05387252 is an effective and selective inhibitor of the IRAK4.</p>
    Formula:C25H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.51
  • Mixanpril

    CAS:
    <p>Mixanpril is an RB 105 lipophilic prodrug.</p>
    Formula:C21H23NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.48
  • Statine

    CAS:
    <p>Statine is a protease inhibitor that is active against pepsin and other acid proteases.</p>
    Formula:C8H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:175.23
  • TRC210258

    CAS:
    <p>TRC210258 is a TGR5 agonist that acts by decreasing glycemic and dyslipidemic cardiovascular risk in animal models of diabesity.</p>
    Formula:C20H14ClFN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.8
  • JNJ-DGAT1-A

    CAS:
    <p>JNJ-DGAT1-A is a DGAT1-selective inhibitor.</p>
    Formula:C31H35Cl2N5O3
    Color and Shape:Solid
    Molecular weight:596.55
  • WAY127093B racemate

    CAS:
    <p>WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.</p>
    Formula:C23H28N4O4
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:424.49
  • IDO inhibitor 1

    CAS:
    <p>IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 &lt;100 nM).with potential immunomodulating and antineoplastic activities.</p>
    Formula:C11H13BrFN7O4S
    Purity:99.805%
    Color and Shape:Solid
    Molecular weight:438.23
  • PF 04671536 hydrochloride

    CAS:
    <p>Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.</p>
    Formula:C14H19ClN8OS
    Color and Shape:Solid
    Molecular weight:382.87
  • Imazodan hydrochloride

    CAS:
    <p>Imazodan hydrochloride (CI-914 HCl) is a potent and selective type III phosphodiesterase inhibitor used in the treatment of chronic congestive heart failure.</p>
    Formula:C13H13ClN4O
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:276.72
  • Mesopram

    CAS:
    <p>PDE4 inhibitor, orally active</p>
    Formula:C14H19NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:265.3
  • TAK 21d

    CAS:
    <p>Potent FAAH inhibitor</p>
    Formula:C19H17F2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:397.38
  • Nafenopin

    CAS:
    <p>Nafenopin is a peroxisome proliferator, it is used to promote liver tumors and has been used as an antihyperlipoproteinemic agent.</p>
    Formula:C20H22O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.39
  • PF-05388169

    CAS:
    <p>PF-05388169 is an effective and selective inhibitor of IRAK4.</p>
    Formula:C22H21N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.42
  • Glyoxalase I inhibitor 4

    CAS:
    <p>Glyoxalase I inhibitor 4 is a potent inhibitor of glyoxalase I (GLO1) (Ki: 10 nM).</p>
    Formula:C17H21IN4O8S
    Color and Shape:Solid
    Molecular weight:568.34
  • CM026

    CAS:
    <p>CM026 inhibits ALDH1A1 selectively, binds to its aldehyde pocket uncompetitively.</p>
    Formula:C22H30N6O4
    Color and Shape:Solid
    Molecular weight:442.51
  • ABT-418

    CAS:
    <p>ABT-418, a nicotinic acetylcholine receptor (nAchR) agonist, is used potentially for the treatment of attention deficit disorder.</p>
    Formula:C9H14N2O
    Color and Shape:Solid
    Molecular weight:166.22
  • Nampt activator-3

    CAS:
    <p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37
  • hDHODH-IN-11

    CAS:
    <p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>
    Formula:C24H23N3O3
    Color and Shape:Solid
    Molecular weight:401.46
  • Safrazine Hydrochloride

    CAS:
    <p>Safrazine Hydrochloride is a monoamine oxidase inhibitor (MOI) that is irreversible.</p>
    Formula:C11H17ClN2O2
    Color and Shape:Solid
    Molecular weight:244.718
  • PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Formula:C17H19Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.27
  • TPN729

    CAS:
    <p>TPN729, a PDE5 inhibitor, has an IC50 of 2.28 nM, used to research erectile dysfunction.</p>
    Formula:C25H36N6O4S
    Color and Shape:Solid
    Molecular weight:516.66
  • (R)-MLN-4760

    CAS:
    <p>(R)-MLN-4760, the R-enantiomer of MLN-4760, functions as an ACE2 inhibitor and exhibits a half maximal inhibitory concentration (IC50) of 8.4 μM, identifying it</p>
    Formula:C19H23Cl2N3O4
    Color and Shape:Solid
    Molecular weight:428.31
  • MDK-0738

    CAS:
    <p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>
    Formula:C15H16O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.29
  • hCAI/II-IN-1

    CAS:
    <p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>
    Formula:C18H29N5O3S3
    Color and Shape:Solid
    Molecular weight:459.65
  • hCAI/II-IN-5

    CAS:
    <p>hCAI/II-IN-5 inhibits human carbonic anhydrase I &amp; II, α-Glycosidase, and AChE, for diabetes, heart failure, Alzheimer's, ulcers, epilepsy research.</p>
    Formula:C21H18Cl2N8O4S2
    Color and Shape:Solid
    Molecular weight:581.45
  • Carbazomycin B

    CAS:
    <p>Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).</p>
    Formula:C15H15NO2
    Color and Shape:Solid
    Molecular weight:241.29
  • Fodipir

    CAS:
    <p>Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cell</p>
    Formula:C22H32N4O14P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:638.46
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Formula:C20H21N3O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.4
  • 4&prime;-Deoxyphlorizin

    CAS:
    <p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>
    Formula:C21H24O9
    Color and Shape:Solid
    Molecular weight:420.41
  • Pemetrexed tromethamine

    CAS:
    <p>Pemetrexed tromethamine is a chemotherapy drug used for pleural mesothelioma and non-small cell lung cancer.</p>
    Formula:C20H21N5O6·2C4H11NO3·2H2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:705.72
  • Arfolitixorin

    CAS:
    <p>Arfolitixorin is an antifolate modulator.</p>
    Formula:C20H23N7O6
    Color and Shape:Solid
    Molecular weight:457.44
  • Diniprofylline

    CAS:
    <p>Diniprofylline, a phosphodiesterase inhibitor, has been used as a peripheral nervous system agent, a bronchodilator agent, and an anti-asthamtic agent.</p>
    Formula:C22H20N6O6
    Color and Shape:Solid
    Molecular weight:464.43
  • Gcase activator 3

    CAS:
    <p>Gcase activator 3 is a glucocerebrosidase (GCase) activator that enhances GBA1 mutant fibroblast lysosomal GCase activity.</p>
    Formula:C23H20N4O2
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:384.43
  • NPD-001

    CAS:
    <p>NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).</p>
    Formula:C33H40N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:584.71
  • CD 2314

    CAS:
    <p>CD2314 is a potent and subtype-selective RARβ receptor agonist with a Kd of 195 nM in S91 melanoma cells [1].</p>
    Formula:C23H24O2S
    Color and Shape:Solid
    Molecular weight:364.5
  • Darexaban glucuronide

    CAS:
    <p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>
    Formula:C33H38N4O10
    Color and Shape:Solid
    Molecular weight:650.68
  • ZSET-845

    CAS:
    <p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>
    Formula:C21H18N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:314.38
  • Dibefurin

    CAS:
    <p>Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.</p>
    Formula:C18H16O8
    Color and Shape:Solid
    Molecular weight:360.31
  • YZ9

    CAS:
    <p>Y29 is a potent PFKFB3 inhibitor with an IC50 of 0.183 µM, and acts as a competitive inhibitor against Fru-6-P with a Ki of 0.094 µM[1].</p>
    Formula:C12H10O5
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:234.2
  • Enpp-1-IN-9

    CAS:
    <p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>
    Formula:C17H24N4O5S
    Color and Shape:Solid
    Molecular weight:396.46
  • PD0176078

    CAS:
    <p>PD0176078 () is a newly blocker of N-type Calcium channel.</p>
    Formula:C23H30F2N2O
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:388.49
  • PPARα-MO-1

    CAS:
    <p>PPARα-MO-1 is a potent modulator of PPARα.</p>
    Formula:C27H37NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.59
  • Glucokinase activator 3

    CAS:
    <p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>
    Formula:C26H33N2O9PS2
    Color and Shape:Solid
    Molecular weight:612.65
  • α-Glucosidase-IN-8

    CAS:
    <p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>
    Formula:C19H20FN3O2
    Color and Shape:Solid
    Molecular weight:341.38
  • Riboflavine phosphate

    CAS:
    <p>Riboflavine phosphate (Flavin mononucleotide) is a derivative of Riboflavin.</p>
    Formula:C17H21N4O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.34
  • ML368

    CAS:
    <p>ML368 is a selective inhibitor of CYP3A4.</p>
    Formula:C26H18N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.46
  • ACC1/2-IN-1

    CAS:
    <p>ACC1/2-IN-1 is a potent inhibitor of ACC1/2 and acts on ACC1 (IC50: 98.06 nM) and ACC2 (IC50: 29.43 nM). ACC1/2-IN-1 can be used in cancer research.</p>
    Formula:C34H32N4O4
    Color and Shape:Solid
    Molecular weight:560.64
  • 7β,27-dihydroxy Cholesterol

    CAS:
    <p>7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt.</p>
    Formula:C27H46O3
    Color and Shape:Solid
    Molecular weight:418.65
  • N-(α-Linolenoyl) Tyrosine

    CAS:
    <p>Certain chronic neurologic disorders, such as Parkinson's disease, are caused by an insufficiency of the neurotransmitter dopamine secondary to the degeneration</p>
    Formula:C27H39NO4
    Color and Shape:Solid
    Molecular weight:441.6
  • FAAH-IN-5

    CAS:
    <p>FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.</p>
    Formula:C21H19N3O6S
    Color and Shape:Solid
    Molecular weight:441.46
  • IDH2R140Q-IN-1

    CAS:
    <p>IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.</p>
    Formula:C22H20F6N6
    Color and Shape:Solid
    Molecular weight:482.42
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Formula:C24H35ClN2O5
    Color and Shape:Solid
    Molecular weight:467
  • HIF-1/2α-IN-2

    CAS:
    <p>HIF-1/2α-IN-2 is a potent inhibitor of HIF-1/2α, which effectively reduces the levels of HIF-1/2α.</p>
    Formula:C16H11FN4O2S
    Color and Shape:Solid
    Molecular weight:342.35
  • OMDM-3

    CAS:
    <p>OMDM-3 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 16.6 μM).</p>
    Formula:C29H43NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.66