GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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L-765314
CAS:L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.Formula:C27H34N6O5Purity:99.73%Color and Shape:SolidMolecular weight:522.6TG6-10-1
CAS:TG6-10-1 is an EP2 antagonist.Formula:C23H23F3N2O4Purity:99.66% - ≥95%Color and Shape:SolidMolecular weight:448.43F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formula:C19H21ClF2N4OPurity:98.72%Color and Shape:SolidMolecular weight:394.85Ref: TM-T7281
1mg49.00€5mg92.00€10mg152.00€25mg295.00€50mg477.00€100mg715.00€200mg982.00€1mL*10mM (DMSO)104.00€Dolasetron
CAS:Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formula:C19H20N2O3Purity:99.84% - 99.86%Color and Shape:White PowderMolecular weight:324.375-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formula:C4H6N2O3Purity:99.99%Color and Shape:SolidMolecular weight:130.1ESI-09
CAS:ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Formula:C16H15ClN4O2Purity:97.24% - 99.57%Color and Shape:SolidMolecular weight:330.77Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purity:>99.99%Color and Shape:SolidMolecular weight:1672.92(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4Dimemorfan phosphate
CAS:Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.Formula:C18H25N·H3O4PPurity:99.65%Color and Shape:SolidMolecular weight:353.4Takeda103A
CAS:Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.Formula:C24H23F2N7OPurity:97.17%Color and Shape:SolidMolecular weight:463.48Ref: TM-T24850
1mg85.00€2mg105.00€5mg164.00€10mg258.00€25mg424.00€50mg562.00€100mg787.00€200mg1,035.00€1mL*10mM (DMSO)187.00€CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28TCS-OX2-29
CAS:TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formula:C23H31N3O3Purity:99.81%Color and Shape:SolidMolecular weight:397.51Ref: TM-T4965
1mg35.00€5mg70.00€10mg96.00€25mg156.00€50mg215.00€100mg303.00€200mg449.00€1mL*10mM (DMSO)77.00€CCG-50014
CAS:CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.Formula:C16H13FN2O2SPurity:98.53%Color and Shape:SolidMolecular weight:316.35Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formula:C11H6O4Purity:99.97%Color and Shape:SolidMolecular weight:202.16Dazoxiben
CAS:Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase
Formula:C12H13ClN2O3Purity:99.99%Color and Shape:SolidMolecular weight:268.7TRAP-6
CAS:TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).Formula:C34H56N10O9Purity:>99.99%Color and Shape:SolidMolecular weight:748.87Ref: TM-T7625
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg274.00€50mg411.00€100mg550.00€200mg785.00€1mL*10mM (DMSO)126.00€Netupitant
CAS:Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).Formula:C30H32F6N4OPurity:99.43%Color and Shape:SolidMolecular weight:578.59Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purity:97.35%Color and Shape:SolidMolecular weight:1260.24β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptorFormula:C164H271N51O50S3Purity:99.35%Color and Shape:SolidMolecular weight:3853.46Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Formula:C40H42ClN5O7Purity:97.94% - 98.4%Color and Shape:SolidMolecular weight:740.24BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.
Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonistFormula:C37H48F6N8O11Purity:98.54%Color and Shape:SolidMolecular weight:894.81Ref: TM-T7740
1mg48.00€2mg60.00€5mg86.00€10mg138.00€25mg274.00€50mg411.00€100mg607.00€1mL*10mM (DMSO)170.00€RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formula:C25H28ClN3O2Purity:99.74%Color and Shape:SolidMolecular weight:437.96Acrivastine
CAS:Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Formula:C22H24N2O2Purity:99.73% - >99.99%Color and Shape:SolidMolecular weight:348.44Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formula:C32H39NO4Purity:99.35%Color and Shape:White To Off-White SolidMolecular weight:501.66Mebhydrolin
CAS:Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Exo-1
CAS:Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormula:C15H12FNO3Purity:99.45%Color and Shape:SolidMolecular weight:273.26Ref: TM-T9200
5mg52.00€10mg78.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€500mg642.00€1mL*10mM (DMSO)65.00€Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Vazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purity:98.93%Color and Shape:SolidMolecular weight:675.3Ref: TM-T8682
1mg107.00€5mg227.00€10mg334.00€25mg565.00€50mg805.00€100mg1,111.00€1mL*10mM (DMSO)329.00€Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Formula:C17H21NOPurity:98.07%Color and Shape:SolidMolecular weight:255.35SB 242084
CAS:SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formula:C21H19ClN4O2Purity:99.75% - ≥98%Color and Shape:SolidMolecular weight:394.85AnaMorelin hydrochloride
CAS:AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formula:C31H43ClN6O3Purity:99.18% - ≥98%Color and Shape:SolidMolecular weight:583.16Ref: TM-T7225
1mg35.00€2mg50.00€5mg73.00€10mg96.00€25mg145.00€50mg177.00€100mg235.00€1mL*10mM (DMSO)95.00€5-Iodotubercidin
CAS:5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.
Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15Zuclopenthixol
CAS:Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.Formula:C22H25ClN2OSPurity:98.9% - 99.82%Color and Shape:SolidMolecular weight:400.96CS 2100
CAS:CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.
Formula:C25H23N3O4SPurity:99.19%Color and Shape:SolidMolecular weight:461.53PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.881-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formula:C149H234N40O47SPurity:98% - 99.65%Color and Shape:SolidMolecular weight:3369.76LUN42518 HCl 47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.Formula:C17H20ClN3OPurity:99.96%Color and Shape:SolidMolecular weight:317.81Ref: TM-T8738
1mg62.00€5mg125.00€10mg180.00€25mg298.00€50mg419.00€100mg567.00€200mg752.00€1mL*10mM (DMSO)123.00€Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formula:C50H68F2N6O4·C4H6O6Purity:99.24% - 99.98%Color and Shape:SolidMolecular weight:1005.2BAY 41-2272
CAS:BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.Formula:C20H17FN6Purity:99.54%Color and Shape:SolidMolecular weight:360.39Gadolinium chloride
CAS:Gadolinium chloride is a calcium-sensing receptor (CaSR) agonistFormula:Cl3GdPurity:98%Color and Shape:White Crystalline SolidMolecular weight:263.61RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.
Formula:C17H16FN3Purity:99.32%Color and Shape:SolidMolecular weight:281.331-Oleoyl lysophosphatidic acid sodium
CAS:1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formula:C21H40O7P·NaPurity:98.75% - 99.24%Color and Shape:SolidMolecular weight:458.51Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.68%Color and Shape:SolidMolecular weight:545.51Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formula:C10H17N3SPurity:99.78%Color and Shape:SolidMolecular weight:211.33Atogepant
CAS:Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formula:C29H23F6N5O3Purity:99.66%Color and Shape:SolidMolecular weight:603.52Ref: TM-T26682
1mg147.00€5mg250.00€10mg313.00€25mg620.00€50mg1,108.00€100mg1,611.00€200mg2,178.00€1mL*10mM (DMSO)334.00€Benzylthiouracil
CAS:Benzylthiouracil (6-Benzyl-2-thiouracil) induces ANCA-associated glomerulonephritis in Graves' disease patients and is used to study hyperthyroidism.Formula:C11H10N2OSPurity:99.65%Color and Shape:SolidMolecular weight:218.28S1RA
CAS:S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formula:C20H23N3O2Purity:99.45%Color and Shape:SolidMolecular weight:337.42Maropitant citrate
CAS:Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.Formula:C38H50N2O9Purity:98.91%Color and Shape:SolidMolecular weight:678.81Bucindolol
CAS:Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.Formula:C22H25N3O2Purity:99.9%Color and Shape:SolidMolecular weight:363.45Fenoterol hydrobromide
CAS:Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formula:C17H22BrNO4Purity:99.88%Color and Shape:SolidMolecular weight:384.27BMS-986278
CAS:BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,
Formula:C22H31N5O5Purity:99.86%Color and Shape:SolidMolecular weight:445.51(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purity:99.75%Color and Shape:SolidMolecular weight:265.35SID 7969543
CAS:SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formula:C24H24N2O7Purity:98.94%Color and Shape:SolidMolecular weight:452.46Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purity:99.41% - >99.99%Color and Shape:SolidMolecular weight:517.66Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formula:C16H22ClN3O2Purity:98.97% - 99.09%Color and Shape:SolidMolecular weight:323.82Ref: TM-T38507
1mg93.00€2mg124.00€5mg200.00€10mg359.00€25mg692.00€50mg945.00€100mg1,279.00€200mg1,701.00€Levocetirizine Dihydrochloride
CAS:Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.
Formula:C21H27Cl3N2O3Purity:99.89%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:461.81Medetomidine
CAS:Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formula:C13H16N2Purity:99.88%Color and Shape:SolidMolecular weight:200.28Ref: TM-T21492
2mg38.00€5mg57.00€10mg77.00€25mg128.00€50mg193.00€100mg290.00€200mg447.00€1mL*10mM (DMSO)62.00€Fenoprofen
CAS:Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formula:C15H14O3Purity:98.4%Color and Shape:SolidMolecular weight:242.27Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46AF-710B
CAS:AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.Formula:C20H27N3OSPurity:98.62% - 99.89%Color and Shape:SolidMolecular weight:357.51Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurity:98.05% - 98.07%Color and Shape:SolidMolecular weight:261.36Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purity:97.11%Color and Shape:SolidMolecular weight:333.47INCB 3284
CAS:INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formula:C26H31F3N4O4Purity:97.81% - 99.42%Color and Shape:SolidMolecular weight:520.54CP-105696
CAS:CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.Formula:C28H28O4Purity:99.78%Color and Shape:SolidMolecular weight:428.52CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formula:C25H41NO2Purity:98.78%Color and Shape:SolidMolecular weight:387.6WIN 51,708
CAS:WIN 51,708 is an antagonist of neurokinin-1 receptor.Formula:C29H33N3OPurity:99%Color and Shape:SolidMolecular weight:439.59(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purity:99.37%Color and Shape:SolidMolecular weight:265.35UCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formula:C19H20N2O2Purity:98.88%Color and Shape:SolidMolecular weight:308.37Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurity:99.04% - 99.88%Color and Shape:SolidMolecular weight:315.47Alfuzosin
CAS:Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formula:C19H27N5O4Purity:99.64%Color and Shape:White Crystaline PowderMolecular weight:389.45Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formula:C15H19N5Purity:99.74%Color and Shape:SolidMolecular weight:269.35Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purity:99.94%Color and Shape:SolidMolecular weight:383.49Ref: TM-TQ0315
2mg34.00€5mg50.00€10mg80.00€25mg130.00€50mg178.00€100mg284.00€200mg408.00€1mL*10mM (DMSO)55.00€Canagliflozin hemihydrate
CAS:Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.Formula:C48H52F2O11S2Purity:99.42% - 99.96%Color and Shape:SolidMolecular weight:907.05KB-5492 free base
CAS:KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formula:C23H30N2O6Purity:97.10% - 97.94%Color and Shape:SolidMolecular weight:430.49Ref: TM-T62396
2mg39.00€5mg58.00€10mg82.00€25mg119.00€50mg168.00€100mg249.00€500mg613.00€1mL*10mM (DMSO)64.00€Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formula:(C6H14N2O2)x·xHBrColor and Shape:SolidMolecular weight:227.102Atipamezole
CAS:Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formula:C14H16N2Purity:99.88%Color and Shape:Off-White To Light Yellow Crystal PowderMolecular weight:212.29GAT211
CAS:GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.Formula:C22H18N2O2Purity:99.7%Color and Shape:SolidMolecular weight:342.39Ref: TM-T27405
1mg34.00€5mg66.00€10mg90.00€25mg148.00€50mg210.00€100mg310.00€500mg750.00€1mL*10mM (DMSO)73.00€Trabodenoson
CAS:Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Ref: TM-T34914
1mg40.00€5mg89.00€10mg116.00€25mg187.00€50mg285.00€100mg411.00€200mg577.00€1mL*10mM (DMSO)88.00€Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formula:C20H20ClNO4Purity:99.79%Color and Shape:SolidMolecular weight:373.8WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purity:99.96%Color and Shape:White SolidMolecular weight:538.645Ref: TM-T3453
2mg46.00€5mg66.00€10mg95.00€25mg159.00€50mg226.00€100mg334.00€500mg807.00€1mL*10mM (DMSO)79.00€Protein deglycase DJ-1 against-1
CAS:Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formula:C24H23N3O4Purity:97.23%Color and Shape:SolidMolecular weight:417.46GRK6-IN-2
CAS:GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.
Formula:C21H21FN6Purity:98.94%Color and Shape:SolidMolecular weight:376.43A2ti-1
CAS:A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.Formula:C20H22N4O2SPurity:99.86%Color and Shape:SolidMolecular weight:382.48Ref: TM-T36432
1mg94.00€5mg200.00€10mg313.00€25mg620.00€50mg982.00€100mg1,341.00€500mg2,682.00€1mL*10mM (DMSO)286.00€S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formula:C19H34O3Purity:97.05% - 98.55%Color and Shape:SolidMolecular weight:310.47Ozanimod hydrochloride
CAS:Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formula:C23H25ClN4O3Purity:99.81%Color and Shape:SolidMolecular weight:440.92Ref: TM-T62552
1mg47.00€5mg92.00€10mg137.00€25mg268.00€50mg432.00€100mg620.00€200mg875.00€1mL*10mM (DMSO)101.00€L-368,899 hydrochloride
CAS:L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formula:C26H43ClN4O5S2Purity:99.59%Color and Shape:SolidMolecular weight:591.23Ref: TM-T11794
2mg105.00€5mg147.00€10mg230.00€25mg439.00€50mg685.00€100mg964.00€1mL*10mM (DMSO)200.00€SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purity:98.78% - 99.86%Color and Shape:SolidMolecular weight:428.41Ref: TM-T37816
1mg35.00€5mg75.00€10mg114.00€25mg260.00€50mg485.00€100mgTo inquire1mL*10mM (DMSO)84.00€Clopidogrel thiolactone
CAS:Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.Formula:C16H16ClNO3SPurity:98.79%Color and Shape:SolidMolecular weight:337.82Ref: TM-T5501
1mg96.00€5mg205.00€10mg326.00€25mg557.00€50mg803.00€100mg1,063.00€200mg1,459.00€1mL*10mM (DMSO)227.00€5-LOX inhibitor
CAS:5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) is an itraconazole impurity, a LOX-5 inhibitor.Formula:C22H27N5O2Purity:98.01%Color and Shape:SolidMolecular weight:393.48LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94Opipramol
CAS:Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.Formula:C23H29N3OPurity:99.84% - 99.98%Color and Shape:SolidMolecular weight:363.5Nebentan potassium
CAS:Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.Formula:C24H20KN5O5SPurity:99.05%Color and Shape:SolidMolecular weight:529.61Ref: TM-T36008
1mg52.00€2mg77.00€5mg111.00€10mg177.00€25mg313.00€50mg502.00€100mg680.00€200mg888.00€1mL*10mM (DMSO)133.00€ACT-462206
CAS:ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formula:C20H24N2O4SPurity:99.45%Color and Shape:SolidMolecular weight:388.48Ref: TM-T26559
1mg44.00€5mg93.00€10mg137.00€25mg279.00€50mg445.00€100mg707.00€500mg1,415.00€1mL*10mM (DMSO)93.00€Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formula:C20H21FN2OPurity:99.78% - 99.89%Color and Shape:SolidMolecular weight:324.39CGP 20712 A
CAS:CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formula:C24H29F3N4O8SPurity:99.37%Color and Shape:SolidMolecular weight:590.57Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3
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