GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43Icatibant Acetate
CAS:<p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>Formula:C61H93N19O15SPurity:99.68%Color and Shape:SolidMolecular weight:1364.57MK-2894 sodium salt
CAS:MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.Formula:C25H22F3NNaO3SPurity:98%Color and Shape:SolidMolecular weight:496.5Terazosin
CAS:Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.Formula:C19H25N5O4Color and Shape:SolidMolecular weight:387.43Melanotan I
CAS:Melanotan I is a non-specific melanocortin receptor (MCR) agonist, an α-melanocyte-stimulating hormone (α-MSH) analog, which is injected subcutaneously toFormula:C78H111N21O19Purity:>99.99%Color and Shape:SolidMolecular weight:1646.85Bosentan
CAS:<p>Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.</p>Formula:C27H29N5O6SPurity:99.74% - 99.84%Color and Shape:Pale Yellow To Off-White SolidMolecular weight:551.614Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92Frovatriptan Succinate
CAS:Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.Formula:C18H25N3O6Color and Shape:SolidMolecular weight:379.41PNU-282987
CAS:PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).Formula:C14H18Cl2N2OPurity:99% - >99.99%Color and Shape:SolidMolecular weight:301.21Triprolidine
CAS:Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formula:C19H22N2Color and Shape:SolidMolecular weight:278.39Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32Pramlintide acetate(151126-32-8 free base)
CAS:<p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>Formula:C173H271N51O55S2Purity:>99.99%Color and Shape:SolidMolecular weight:4009SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formula:C46H60F3N13O12SPurity:98.49%Color and Shape:SolidMolecular weight:1076.124F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49PAR-4 Agonist Peptide, amide TFA
CAS:PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.Formula:C36H49F3N8O9Purity:99.72%Color and Shape:SolidMolecular weight:794.82Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.Formula:C42H69N13O12Purity:98.37%Color and Shape:SolidMolecular weight:948.08Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:904.02PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Formula:C26H32O4Purity:98.53%Color and Shape:SolidMolecular weight:408.53Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formula:C99H163N27O34Purity:99.25%Color and Shape:SolidMolecular weight:2275.51ACTH 11-24 acetate(4237-93-8 free base)
CAS:ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.Formula:C79H138N24O18Purity:>99.99%Color and Shape:SolidMolecular weight:1712.12CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purity:98.24%Color and Shape:SolidMolecular weight:3140.5BAR501
CAS:BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formula:C26H46O3Purity:99.29% - 99.68%Color and Shape:SolidMolecular weight:406.64AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formula:C21H24ClF2NOPurity:99.89%Color and Shape:SolidMolecular weight:379.87AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:98.87%Color and Shape:SolidMolecular weight:478.47CP 376395
CAS:CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.Formula:C21H30N2OPurity:99.86% - 99.94%Color and Shape:SolidMolecular weight:326.48TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Formula:C23H23F3N2O4Purity:99.66% - ≥95%Color and Shape:SolidMolecular weight:448.43Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.Formula:C54H81N15O14Purity:99.01%Color and Shape:SolidMolecular weight:1164.31Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurity:99.26% - 99.62%Color and Shape:White SolidMolecular weight:285.77Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purity:99.39%Color and Shape:SolidMolecular weight:386.4Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.Formula:C37H62N10O11Purity:98.1800%Color and Shape:SolidMolecular weight:822.95Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Formula:C18H25N·H3O4PPurity:99.65%Color and Shape:SolidMolecular weight:353.4Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purity:99.83% - 99.97%Color and Shape:SolidMolecular weight:403.52Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formula:C32H39NO4Purity:99.35%Color and Shape:White To Off-White SolidMolecular weight:501.66Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Exo-1
CAS:Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormula:C15H12FNO3Purity:99.45%Color and Shape:SolidMolecular weight:273.26Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Naftopidil dihydrochloride
CAS:Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formula:C24H28N2O3·2HClPurity:99.76%Color and Shape:White SolidMolecular weight:465.41GR-73632
CAS:<p>Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).</p>Formula:C40H59N7O6SPurity:99.68%Color and Shape:SolidMolecular weight:766Vazegepant hydrochloride
CAS:Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.Formula:C36H47ClN8O3Purity:98.93%Color and Shape:SolidMolecular weight:675.33-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Formula:C21H25Cl2NOPurity:99.03%Color and Shape:SolidMolecular weight:378.33Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:299.80GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formula:C25H29N5OPurity:99.2%Color and Shape:SolidMolecular weight:415.53TGR5 Receptor Agonist
CAS:TGR5 is a potent TGR5(GPCR19) agonist.Formula:C18H14Cl2N2O2Purity:99.77% - ≥95%Color and Shape:SolidMolecular weight:361.22Droxidopa
CAS:Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formula:C9H11NO5Purity:97.27% - 99.88%Color and Shape:SolidMolecular weight:213.19Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purity:95.00%Color and Shape:SolidMolecular weight:261.7Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21SHU 9119 acetate
SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.Formula:C56H75N15O11Purity:99.8%Color and Shape:SolidMolecular weight:1134.29Ranitidine
CAS:<p>Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).</p>Formula:C13H22N4O3SPurity:99.52%Color and Shape:Solid SolidMolecular weight:314.40TG4-155
CAS:<p>TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.</p>Formula:C23H26N2O4Purity:97.2%Color and Shape:SolidMolecular weight:394.46[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C77H118N22O20Purity:98.41% - 99.14%Color and Shape:SolidMolecular weight:1671.9Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Formula:C17H20BrNOColor and Shape:SolidMolecular weight:334.25JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formula:C27H27Cl2N5O3SPurity:99.54% - 99.84%Color and Shape:SolidMolecular weight:572.51Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurity:97.71% - 99.78%Color and Shape:SolidMolecular weight:4186.57Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Formula:C37H56F7N6O16PPurity:98% - 99.03%Color and Shape:SolidMolecular weight:1004.83Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formula:C17H27ClN2O4SPurity:≥95%Color and Shape:White Or Yellowish PowderMolecular weight:390.93MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Formula:C27H21F3N2O3Purity:99.54% - 99.59%Color and Shape:SolidMolecular weight:478.46Darbufelone mesylate
CAS:Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formula:C19H28N2O5S2Purity:96.81% - 99.92%Color and Shape:SolidMolecular weight:428.57Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Formula:C26H29N5O3SPurity:99.49% - 99.843%Color and Shape:SolidMolecular weight:491.61Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36Galanin (1-16), mouse, porcine, rat
CAS:Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.Formula:C78H116N20O21Purity:98.65%Color and Shape:White PowderMolecular weight:1669.88Atrasentan
CAS:Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.Formula:C29H38N2O6Purity:97.65% - 99.08%Color and Shape:SolidMolecular weight:510.62Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purity:97.41%Color and Shape:SolidMolecular weight:244.38ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Formula:C29H29ClN4O2Purity:99.88%Color and Shape:SolidMolecular weight:501.02EST64454 Maleic acid salt
CAS:EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.Formula:C22H26F2N4O6Purity:97.54%Color and Shape:SolidMolecular weight:480.46Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Formula:C20H20FNO3S·HClPurity:99.39% - 99.79%Color and Shape:SolidMolecular weight:409.9Fenoprofen Calcium
CAS:Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.Formula:C30H26CaO6Purity:99.24% - 99.66%Color and Shape:SolidMolecular weight:522.6Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Formula:C10H17N3S·2HCl·H2OPurity:99.68%Color and Shape:White To Off-White Crystalline PowderMolecular weight:302.26Vanoxerine dihydrochloride
CAS:Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Formula:C28H34Cl2F2N2OPurity:98.16% - 98.35%Color and Shape:White SolidMolecular weight:523.49Phosphorylcholine chloride
CAS:Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integralFormula:C5H15ClNO4PPurity:99.481% - 99.85%Color and Shape:SolidMolecular weight:219.6Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purity:98.25%Color and Shape:SolidMolecular weight:233.18Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Formula:C15H19Cl2N3O3SPurity:98.48%Color and Shape:SolidMolecular weight:392.3BisfluoroModafinil
CAS:CRL-40940 is a selective dopaminergic reuptake inhibitorFormula:C15H13F2NO2SPurity:99.19%Color and Shape:SolidMolecular weight:309.33Endothelin-2 (49-69), human
CAS:Endothelin-2 (49-69), human (Human endothelin-2) is a 21-amino acid vasoactive peptide that binds to G-protein-linked transmembrane receptors, ET-RA and ET-RB.Formula:C115H160N26O32S4Purity:98.26%Color and Shape:SolidMolecular weight:2546.92(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Formula:C14H20ClNO3Purity:97.76%Color and Shape:SolidMolecular weight:285.77A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Formula:C32H41N5O10Purity:97.69%Color and Shape:SolidMolecular weight:655.7GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formula:C27H20N4O2Purity:98.23%Color and Shape:SolidMolecular weight:432.47SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Montelukast sodium
CAS:<p>Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.</p>Formula:C35H35ClNNaO3SPurity:99.14% - 99.89%Color and Shape:White To Off-White Crystalline PowderMolecular weight:608.17Exenatide
CAS:Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.Formula:C186H286N50O62SPurity:99.42%Color and Shape:SolidMolecular weight:4247Indacaterol
CAS:<p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>Formula:C24H28N2O3Purity:99.96%Color and Shape:SolidMolecular weight:392.49(R)-Propranolol hydrochloride
CAS:(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.Formula:C16H22ClNO2Purity:98.63% - 99.01%Color and Shape:SolidMolecular weight:295.8Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formula:C17H18ClN3OPurity:99.95%Color and Shape:SolidMolecular weight:315.8Montelukast
CAS:Montelukast (Singular), oral asthma med, linked to rare liver injury.Formula:C35H36ClNO3SPurity:98.56% - >99.99%Color and Shape:SolidMolecular weight:586.18Dobutamine
CAS:Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38BI-6015
CAS:<p>BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.</p>Formula:C15H13N3O4SPurity:99.81%Color and Shape:SolidMolecular weight:331.35Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formula:C47H76N14O12Purity:97.09%Color and Shape:SolidMolecular weight:1029.19Montelukast dicyclohexylamine
CAS:Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.Formula:C47H59ClN2O3SColor and Shape:SolidMolecular weight:767.5LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Formula:C30H34N4OPurity:98.65%Color and Shape:SolidMolecular weight:466.62Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Formula:C59H83N13O14S2Purity:99.7%Color and Shape:SolidMolecular weight:1262.5RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71Dexmedetomidine
CAS:Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formula:C13H16N2Purity:99% - >99.99%Color and Shape:SolidMolecular weight:200.28Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formula:C12H14N2·HClPurity:99.97%Color and Shape:SolidMolecular weight:222.71AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.739-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.37%Color and Shape:SolidMolecular weight:163.18LY 78335
CAS:LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.Formula:C8H10Cl3NPurity:99.30% - 99.81%Color and Shape:SolidMolecular weight:226.531-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Formula:C13H13NO5Purity:99.55%Color and Shape:SolidMolecular weight:263.255-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formula:C11H16ClNOPurity:98.5%Color and Shape:SolidMolecular weight:213.7Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Haloperidol decanoate
CAS:Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.Formula:C31H41ClFNO3Purity:99.57% - 99.72%Color and Shape:SolidMolecular weight:530.11WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formula:C25H34N4O2·C4H4O4Purity:98.44% - 99.46%Color and Shape:SolidMolecular weight:538.64H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.79Istradefylline
CAS:Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurity:99.83%Color and Shape:SolidMolecular weight:286.35Rizatriptan benzoate
CAS:<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Formula:C22H25N5O2Purity:99% - 99.79%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.47Sarpogrelate
CAS:Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.Formula:C24H31NO6Color and Shape:SolidMolecular weight:429.51ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Formula:C22H25N3O3Purity:98.4% - 99.42%Color and Shape:SolidMolecular weight:379.45MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurity:99.35%Color and Shape:SolidMolecular weight:292.36Fipamezole HCl
CAS:Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.Formula:C14H16ClFN2Color and Shape:SolidMolecular weight:266.74Tirzepatide Acetate(2023788-19-2 free base)
Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.Formula:C227H352N48O70Purity:97.3% - 98.05%Color and Shape:SolidMolecular weight:4873.5S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formula:C31H34N2O4Purity:99.77%Color and Shape:SolidMolecular weight:498.61Donitriptan Mesylate
CAS:Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formula:C24H29N5O5SColor and Shape:SolidMolecular weight:499.58C14TKL-1 acetate
C14TKL-1 acetate is a NK1 receptor agonist.Formula:C65H102N20O15S2Purity:98.56%Color and Shape:SolidMolecular weight:1467.75Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formula:C95H160N34O29Purity:98.25%Color and Shape:SolidMolecular weight:2242.5Droxidopa hydrochloride
CAS:Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.Formula:C9H12ClNO5Color and Shape:SolidMolecular weight:249.65Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormula:C21H32O2Purity:99.59% - 99.92%Color and Shape:SolidMolecular weight:316.48EST64454 free base
CAS:EST64454: σ1R antagonist for pain, high solubility, permeable, BCS class I, metabolically stable.Formula:C18H22F2N4O2Color and Shape:SolidMolecular weight:364.39Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05Bupranolol HCl
CAS:Bupranolol: non-selective beta blocker, no ISA, strong membrane stabilizer, fast gut absorption, high first-pass metabolism, 2-4hr half-life.Formula:C14H23Cl2NO2Color and Shape:SolidMolecular weight:308.243Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formula:C17H25N3O2SPurity:99.85%Color and Shape:Light Yellow Or White PowerMolecular weight:335.46BMS 182874 hydrochloride
CAS:BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formula:C17H20ClN3O3SPurity:97.01%Color and Shape:SolidMolecular weight:381.88Facinicline (free base)
CAS:Facinicline (free base) is a partial agonist of the nicotinic alpha-7 (α7) receptor. It is used for the oral treatment of Alzheimer's.Formula:C15H18N4OColor and Shape:SolidMolecular weight:270.33Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49FK962
CAS:<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Formula:C14H17FN2O2Purity:99.89%Color and Shape:SolidMolecular weight:264.3Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Formula:C24H40NaO4Purity:99.66% - 99.96%Color and Shape:SolidMolecular weight:415.56N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Formula:C9H15N3O3Purity:98%Color and Shape:SolidMolecular weight:213.23Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purity:99.24%Color and Shape:SolidMolecular weight:485.96BD 1008 dihydrobromide
CAS:<p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>Formula:C15H24Br2Cl2N2Purity:97.81%Color and Shape:SolidMolecular weight:463.08R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purity:99.52%Color and Shape:SolidMolecular weight:865.93Siramesine
CAS:Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potentFormula:C30H31FN2OPurity:98%Color and Shape:SolidMolecular weight:454.58Ibrolipim
CAS:<p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>Formula:C19H20BrN2O4PPurity:98.04%Color and Shape:SolidMolecular weight:451.25Vercirnon sodium
CAS:Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formula:C22H21ClN2NaO4SColor and Shape:SolidMolecular weight:467.92AM211
CAS:AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)Formula:C27H27F3N2O4Purity:≥95%Color and Shape:SolidMolecular weight:500.51nifenalol.HCl
CAS:Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72Phentolamine hydrochloride
CAS:Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].Formula:C17H20ClN3OColor and Shape:SolidMolecular weight:317.82HCGRP-(8-37) acetate
<p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>Formula:C141H234N44O40Purity:99.29%Color and Shape:SolidMolecular weight:3185.64Praliciguat
CAS:Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formula:C21H14F8N6O2Purity:98.82%Color and Shape:SolidMolecular weight:534.36[Sar9] Substance P acetate(77128-75-7 free base)
[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.Formula:C66H104N18O15SPurity:96.67%Color and Shape:SolidMolecular weight:1421.71carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59Pranlukast hemihydrate
CAS:<p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>Formula:C27H23N5O40·5H2OPurity:99.28%Color and Shape:SolidMolecular weight:490.52SB-649868
CAS:SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).Formula:C26H24FN3O3SPurity:99.53%Color and Shape:SolidMolecular weight:477.55GW627368
CAS:GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.Formula:C30H28N2O6SPurity:99.75% - 99.92%Color and Shape:SolidMolecular weight:544.62RS 100329
CAS:RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formula:C20H25F3N4O3Color and Shape:SolidMolecular weight:426.43Methiothepin mesylate
CAS:Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formula:C21H28N2O3S3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:452.65Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Formula:C28H37N3O3Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:463.61Flibanserin
CAS:<p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>Formula:C20H21F3N4OPurity:99.37% - 99.93%Color and Shape:White PowderMolecular weight:390.4Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43RBC8
CAS:RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.Formula:C25H20N4O3Purity:98.44% - 99.81%Color and Shape:SolidMolecular weight:424.45ENMD-1068 HBr
CAS:ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.Formula:C15H30BrN3O2Color and Shape:SolidMolecular weight:364.32KB-5492 anhydrous
CAS:KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.Formula:C27H34N2O10Color and Shape:SolidMolecular weight:546.57A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45ICI 118,551 hydrochloride
CAS:ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3Formula:C17H28ClNO2Purity:99.296% - 99.76%Color and Shape:SolidMolecular weight:313.86DPCPX
CAS:DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormula:C16H24N4O2Purity:99.23% - 99.93%Color and Shape:White SolidMolecular weight:304.39AM1241
CAS:<p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>Formula:C22H22IN3O3Purity:98.937% - 99.1%Color and Shape:SolidMolecular weight:503.33JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormula:C20H34Cl2N2OPurity:99.51%Color and Shape:SolidMolecular weight:389.41-Oleoyl lysophosphatidic acid sodium
CAS:1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formula:C21H40O7P·NaPurity:98.75% - 99.24%Color and Shape:SolidMolecular weight:458.51BAY 41-2272
CAS:<p>BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.</p>Formula:C20H17FN6Purity:99.54%Color and Shape:SolidMolecular weight:360.39Nifenalol
CAS:Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.Formula:C11H16N2O3Purity:98%Color and Shape:SolidMolecular weight:224.26Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formula:C21H30N4O4Purity:99.52%Color and Shape:SolidMolecular weight:402.49Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Formula:C25H26Cl3N7OPurity:99.79% - ≥95%Color and Shape:SolidMolecular weight:546.88PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formula:C21H29Cl2N3O4SPurity:98.5%Color and Shape:SolidMolecular weight:490.44Terutroban
CAS:<p>Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.</p>Formula:C20H22ClNO4SPurity:99.53%Color and Shape:SolidMolecular weight:407.91JNJ-31020028
CAS:<p>JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).</p>Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68Syk Inhibitor II dihydrochloride dihydrate
CAS:Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formula:C14H21Cl2F3N6O3Color and Shape:SolidMolecular weight:449.26ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37TC-G 1005
CAS:TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).Formula:C25H25N3O2Purity:98.60% - 99.78%Color and Shape:SolidMolecular weight:399.48ML401
CAS:ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .Formula:C20H20BrClN2OPurity:99.13%Color and Shape:SolidMolecular weight:419.74Cinaciguat hydrochloride
CAS:Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.Formula:C36H40ClNO5Color and Shape:SolidMolecular weight:602.17NPS-2143 hydrochloride
CAS:NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.Formula:C24H25ClN2O2·HClPurity:99.38% - 99.67%Color and Shape:SolidMolecular weight:445.38Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Formula:C28H42F2N2O12S2Purity:99.98%Color and Shape:SolidMolecular weight:700.77Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Formula:C21H25ClN2O3Purity:99.75%Color and Shape:SolidMolecular weight:388.89Substance P (7-11)
CAS:<p>Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .</p>Formula:C31H44N6O5SPurity:98.39%Color and Shape:SolidMolecular weight:612.78SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurity:99.61%Color and Shape:SolidMolecular weight:266.3Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurity:98.86% - 99.93%Color and Shape:SolidMolecular weight:358.69RO1138452
CAS:RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).Formula:C19H23N3OPurity:97.01% - 99.34%Color and Shape:SolidMolecular weight:309.41Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Formula:C21H28N2O2·2ClHPurity:99.73%Color and Shape:SolidMolecular weight:413.39Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61BAY 41-8543
CAS:<p>BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).</p>Formula:C21H21FN8OPurity:99.86%Color and Shape:SolidMolecular weight:420.44Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Formula:C58H69F3N12O16S2Purity:99.7%Color and Shape:SolidMolecular weight:1311.36Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formula:C25H27N3O2S·xHClPurity:99.05%Color and Shape:SolidMolecular weight:433.6Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Formula:C17H11N3O6SPurity:97.74%Color and Shape:SolidMolecular weight:385.35Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formula:C24H30N2O2SPurity:99.9% - 99.92%Color and Shape:SolidMolecular weight:410.57Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852Riociguat
CAS:Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormula:C20H19FN8O2Purity:99.28% - 99.95%Color and Shape:SolidMolecular weight:422.42Procaterol hydrochloride hydrate
CAS:Short-acting β2-adrenergic receptor agonist used to treat asthma.Formula:C32H48Cl2N4O7Purity:99.71% - 99.97%Color and Shape:SolidMolecular weight:671.65Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12
![[D-Phe12,Leu14]-Bombesin acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1916L1.webp&w=3840&q=75)
![1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT8913.webp&w=3840&q=75)
![[Sar9] Substance P acetate(77128-75-7 free base)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1862L.webp&w=3840&q=75)
