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Cell Cycle/Checkpoint
Subcategories of "Cell Cycle/Checkpoint"
Aurora Kinase
CDK
Cell Cycle Arrest
Chk
c-Myc
Dynamin
DYRK
Ferroptosis
HSP
Integrin
Kinesin
KSP
LIM Kinase
Microtubule Associated
PKC
PLK
Rho
ROCK
Wee1
Show 13 more subcategories
Products of "Cell Cycle/Checkpoint"
SB743921
CAS:940929-33-9
SB-743921 is an effective inhibitor of kinesin spindle protein, KSP, (Ki =0.1 nM).
Formula:
C31H34Cl2N2O3
Purity:
95.58%
Color and Shape:
solid
Molecular weight:
553.52
Estimated delivery in United States, on Monday 7 Feb 2022
Roscovitine
CAS:186692-46-6
Roscovitine is a potent inhibitor of Cdk2/cyclin E (IC50: 0.1 µM). It also inhibits Cdk7/cyclin …
Formula:
C19H26N6O
Purity:
98.00%
Color and Shape:
White To Off-White Solid
Molecular weight:
354.45
Estimated delivery in United States, on Monday 7 Feb 2022
CCG1423
CAS:285986-88-1
CCG-1423, a selective RhoA pathway inhibitor, suppresses SRF-mediated transcription.
Formula:
C18H13ClF6N2O3
Purity:
99.63%
Color and Shape:
solid
Molecular weight:
454.75
Estimated delivery in United States, on Monday 7 Feb 2022
CDK2-IN-4
CAS:2079895-42-2
CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM …
Formula:
C23H18N6O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
442.49
Estimated delivery in United States, on Monday 7 Feb 2022
(1S,3R,5R)-PIM447 dihydrochloride
(1S,3R,5R)-PIM447 (dihydrochloride) an inhibitor of PIM(IC50 of 0.095 μM for Pim1, 0.522 μM for Pim2 …
Formula:
C24H25Cl2F3N4O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
513.38
Estimated delivery in United States, on Monday 7 Feb 2022
CDK4/6-IN-2
CAS:1800506-48-2
CDK4/6-IN-2 is a potent CDK4 and CDK6 inhibitor (IC50s: 2.7 and 16 nM) extracted from …
Formula:
C27H32F2N8
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
506.59
Estimated delivery in United States, on Monday 7 Feb 2022
CDK inhibitor II
CAS:1269815-17-9
CDK-IN-2 is a potent and specific CDK9 inhibitor (IC50: <8 nM).
Formula:
C18H19ClFN3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
363.81
Estimated delivery in United States, on Monday 7 Feb 2022
XL413
CAS:1169558-38-6
XL-413 is an orally bioavailable cell division cycle 7 homolog (CDC7) kinase inhibitor with potential …
Formula:
C14H12ClN3O2
Purity:
98.0%
Color and Shape:
solid
Molecular weight:
289.06
Estimated delivery in United States, on Monday 7 Feb 2022
Digeranyl bisphosphonate
CAS:878143-03-4
Digeranyl bisphosphonate is a potent inhibitor of geranylgeranylpyrophosphate (GGPP) synthase.
Formula:
C21H34Na4O6P2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
536.4
Estimated delivery in United States, on Monday 7 Feb 2022
Atuveciclib
Atuveciclib (BAY-1143572) is a potent and highly selective, oral PTEFb/CDK9 inhibitor. It inhibits CDK9/CycT1 (IC50: …
Formula:
C18H18FN5O2S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
387.43
Estimated delivery in United States, on Monday 7 Feb 2022
CCT244747
CAS:1404095-34-6
CCT244747 is a CHK1 inhibitor (IC50: 7.7 nM) and also abrogates G2 checkpoint (IC50: 29 …
Formula:
C20H24N8O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
408.46
Estimated delivery in United States, on Monday 7 Feb 2022
EHT 5372
CAS:1425945-60-3
EHT 5372 is a strong DYRKs family kinases of inhibitor (IC50s: 0.22, 0.28 nM for …
Formula:
C18H14FN5O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
383.4
Estimated delivery in United States, on Monday 7 Feb 2022
Adavosertib
CAS:955365-80-7
MK-1775 is a small molecule inhibitor of the checkpoint kinase WEE1 (IC50: 5.2 nM). It …
Formula:
C27H32N8O2
Purity:
98.65%
Color and Shape:
solid
Molecular weight:
500.6
Estimated delivery in United States, on Monday 7 Feb 2022
RKI1447
CAS:1342278-01-6
RKI-1447 is a potent inhibitor of ROCK1 and ROCK2. It has anti-invasive and antitumor activities.
Formula:
C16H14N4O2S
Purity:
99.73%
Color and Shape:
solid
Molecular weight:
326.37
Estimated delivery in United States, on Monday 7 Feb 2022
Roniciclib
CAS:1223498-69-8
Roniciclib is an inhibitor of pan-cyclin dependent kinase (IC50s: 5-25 nM for CDK1, CDK2, CDK3, …
Formula:
C18H21F3N4O3S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
430.44
Estimated delivery in United States, on Monday 7 Feb 2022
KSI-3716
CAS:1151813-61-4
KSI-3716 is an inhibitor of c-Myc.
Formula:
C17H11BrCl2N2O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
426.09
Estimated delivery in United States, on Monday 7 Feb 2022
IIIM-290
CAS:2213468-64-3
IIIM-290 is an oral CDK inhibitor (IC50s: 90 and 94 nM for CDK2/A and CDK9/T1).
Formula:
C23H21Cl2NO5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
462.32
Estimated delivery in United States, on Monday 7 Feb 2022
AZ-Dyrk1B-33
CAS:1679330-37-0
AZ-Dyrk1B-33 is a potent and selective Dyrk1B kinase inhibitor. With an IC50 of 7 nM[1].
Formula:
C19H16N4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
300.36
Estimated delivery in United States, on Monday 7 Feb 2022
Ribociclib hydrochloride
CAS:1211443-80-9
Ribociclib hydrochloride is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively). …
Formula:
C23H31ClN8O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
471
Estimated delivery in United States, on Monday 7 Feb 2022
Indomethacin-D4
CAS:87377-08-0
Indomethacin-D4 is a deuterium labeled Indomethacin. Indomethacin is a potent and nonselective inhibitor of COX1 …
Formula:
C19H12D4ClNO4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
361.81
Estimated delivery in United States, on Monday 7 Feb 2022
THZ2
CAS:1604810-84-5
THZ2, an analog of THZ1, is a potent and selective CDK7 inhibitor(IC50:13.9 nM),with the potential …
Formula:
C31H28ClN7O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
566.05
Estimated delivery in United States, on Monday 7 Feb 2022
HMN214
CAS:173529-46-9
HMN-214(IVX214) is a potent PLK1 inhibitor with an average IC50 of 0.12 μM.
Formula:
C22H20N2O5S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
424.47
Estimated delivery in United States, on Monday 7 Feb 2022
Ginsenoside C-K
CAS:39262-14-1
Ginsenoside C-K is a bacterial metabolite of G-Rb1 exhibiting anti-inflammatory effects by reducing iNOS and …
Formula:
C36H62O8
Purity:
99.65%
Color and Shape:
solid
Molecular weight:
622.88
Estimated delivery in United States, on Monday 7 Feb 2022
GRGDSP acetate(91037-75-1 free base)
GRGDSP acetate is a synthetic linear RGD peptide and is an integrin inhibitor.
Formula:
C24H41N9O12
Purity:
99.77%
Color and Shape:
solid
Molecular weight:
647.64
Estimated delivery in United States, on Monday 7 Feb 2022
Samuraciclib hydrochloride
CAS:1805789-54-1
Samuraciclib hydrochloride is a potent, selective, ATP competitive and oral active CDK7 inhibitor with IC50 …
Formula:
C22H31ClN6O
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
430.97
Estimated delivery in United States, on Monday 7 Feb 2022
BRD6989
CAS:642008-81-9
BRD6989 is an analog of the natural product cortistatin A (dCA). Which inhibits CDK8 and …
Formula:
C16H16N4
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
264.33
Estimated delivery in United States, on Monday 7 Feb 2022
A205804
CAS:251992-66-2
A-205804 is a specific and effective inhibitor of E-selectin( IC50=20 nM ) and ICAM-1(IC50=25 nM) …
Formula:
C15H12N2OS2
Purity:
98.52%
Color and Shape:
solid
Molecular weight:
300.41
Estimated delivery in United States, on Monday 7 Feb 2022
INDY
CAS:1169755-45-6
INDY is a ATP-competitive inhibitor of Dyrk1A and Dyrk1B (IC50s: 0.24 μM and 0.23 μM). …
Formula:
C12H13NO2S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
235.3
Estimated delivery in United States, on Monday 7 Feb 2022
Ribociclib succinate
CAS:1374639-75-4
Ribociclib succinate is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively). …
Formula:
C27H36N8O5
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
552.63
Estimated delivery in United States, on Monday 7 Feb 2022
Volasertib
CAS:755038-65-4
Volasertib (BI-6727) is a potent inhibitor of PLK1 (IC50: 0.87 nM), inducing mitotic arrest and …
Formula:
C34H50N8O3
Purity:
99.72%
Color and Shape:
solid
Molecular weight:
618.81
Estimated delivery in United States, on Monday 7 Feb 2022
DYRKs-IN-1
CAS:1387090-01-8
DYRKs-IN-1 has antitumor activity. DYRKs-IN-1 is a potent DYRKs (Dual-specificity tyrosine-phosphorylation-regulated kinases) inhibitor with IC50s …
Formula:
C30H30ClN7O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
588.06
Estimated delivery in United States, on Monday 7 Feb 2022
LDC4297
CAS:1453834-21-3
LDC4297 is a potent and selective CDK7 inhibitor.
Formula:
C23H28N8O
Molecular weight:
432.52
Estimated delivery in United States, on Monday 7 Feb 2022
SY-1365
CAS:1816989-16-8
SY-1365 is a highly selective covalent CDK7 inhibitor. SY-1365 possesses therapeutic potential in both hematological …
Formula:
C31H35ClN8O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
587.12
Estimated delivery in United States, on Monday 7 Feb 2022
UAMC3203
CAS:2271358-64-4
UAMC-3203 is a potent and selective Ferroptosis inhibitor (IC50: 12 nM).
Formula:
C25H37N5O2S
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
471.66
Estimated delivery in United States, on Monday 7 Feb 2022
STF083010
CAS:307543-71-1
STF-083010 is a selective inhibitor of the IRE1 endonuclease.
Formula:
C15H11NO3S2
Purity:
98.85%
Color and Shape:
solid
Molecular weight:
317.38
Estimated delivery in United States, on Monday 7 Feb 2022
SB-218078
CAS:135897-06-2
SB-218078 is less potently inhibits Cdc2 (IC50: 250 nM) and PKC (IC50: 1000 nM). SB-218078 …
Formula:
C24H15N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
393.39
Estimated delivery in United States, on Monday 7 Feb 2022
GSK461364
CAS:929095-18-1
GSK461364(Ki=2.2 nM) inhibits purified Plk1 .The specificity of GSK461364 for Plk1 is more than 1000-fold …
Formula:
C27H28F3N5O2S
Purity:
99.50%
Color and Shape:
solid
Molecular weight:
543.6
Estimated delivery in United States, on Monday 7 Feb 2022
RGD peptide GRGDNP(2TFA)
CAS:114681-65-1
RGD peptide GRGDNP(2TFA) is a integrin-ligand interactions inhibitor.
Formula:
C23H38N10O10
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
614.61
Estimated delivery in United States, on Monday 7 Feb 2022
CAN508
CAS:140651-18-9
CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM. It …
Formula:
C9H10N6O
Molecular weight:
218.22
Estimated delivery in United States, on Monday 7 Feb 2022
EHT 1864
CAS:754240-09-0
EHT 1864 is a effective Rac family GTPase inhibitor for Rac1/Rac1b/Rac2/Rac3 (Kd: 40/50/60/250 nM).
Formula:
C25H29Cl2F3N2O4S
Purity:
99.42%
Color and Shape:
solid
Molecular weight:
581.47
Estimated delivery in United States, on Monday 7 Feb 2022
Rho-Kinase-IN-1
CAS:1035094-83-7
Rho-Kinase-IN-1 is a inhibitor of Rho kinase (ROCK) with Ki values of 30.5 and 3.9 …
Formula:
C20H24N4S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
352.5
Estimated delivery in United States, on Monday 7 Feb 2022
Y-27632 dihydrochloride
CAS:129830-38-2
Y-27632 is a selective inhibitor of ROCKs including p160ROCK (Ki: 140 nM) and ROCK2 (IC50: …
Formula:
C14H21N3O·2HCl
Purity:
99.91%
Color and Shape:
solid
Molecular weight:
320.26
Estimated delivery in United States, on Monday 7 Feb 2022
Levomefolate calcium
CAS:151533-22-1
Levomefolate calcium is an artificial form of folate. It is a coenzymated form of folic …
Formula:
C20H23CaN7O6
Color and Shape:
Off-White To Pale Yellow Solid
Molecular weight:
497.52
Estimated delivery in United States, on Monday 7 Feb 2022
Prexasertib
CAS:1234015-52-1
Prexasertib is an inhibitor of checkpoint kinase 1 (chk1) with potential antineoplastic activity.
Formula:
C18H19N7O2
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
365.4
Estimated delivery in United States, on Monday 7 Feb 2022
TC-S 7005
CAS:1082739-92-1
TC-S 7005 is an inhibitor of Polo-like kinases (IC50s: 4 nM, 24 nM and 214 …
Formula:
C21H17N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
359.38
Estimated delivery in United States, on Monday 7 Feb 2022
SCH-1473759
CAS:1094069-99-4
SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A …
Formula:
C20H26N8OS
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
426.54
Estimated delivery in United States, on Monday 7 Feb 2022
SU-9516
CAS:666837-93-0
SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.
Formula:
C13H11N3O2
Molecular weight:
241.24
Estimated delivery in United States, on Monday 7 Feb 2022
CDK4/6-IN-4
CAS:2138499-06-4
CDK4/6-IN-4 is a selective CDK4/6 inhibitor and the active metabolite of Abemaciclib.
Formula:
C27H32F2N8O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
522.59
Estimated delivery in United States, on Monday 7 Feb 2022
1-Piperidinecarboxylic acid, 4-[[5-methyl-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]-, 1-[(2E)-4-(dimethylamino)-1-oxo-2-buten-1-yl]-3-pyrrolidinyl ester
CAS:2326428-25-3
1-Piperidinecarboxylic acid, 4-[[5-methyl-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]-, 1-[(2E)-4-(dimethylamino)-1-oxo-2-buten-1-yl]-3-pyrrolidinyl ester is a novel CDK7 inhibitors.
Formula:
C26H39N7O3
Molecular weight:
497.64
Estimated delivery in United States, on Monday 7 Feb 2022
CLK-IN-T3
CAS:2109805-56-1
CLK-IN-T3 is a potent inhibitor of CDC-like kinase (CLK) (IC50s: 0.67 nM, 15 nM, and …
Formula:
C28H30N6O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
482.58
Estimated delivery in United States, on Monday 7 Feb 2022
Pyridoxine
CAS:65-23-6
Pyridoxine is the 4-methanol form of vitamin B6 and is converted to pyridoxal 5-phosphate in …
Formula:
C8H11NO3
Purity:
99.18%
Color and Shape:
Platelets Or Thick Birefringent Rods From Alcohol + Acetone Solid
Molecular weight:
169.18
Estimated delivery in United States, on Monday 7 Feb 2022
RWJ 50271
CAS:162112-37-0
RWJ 50271 is a selective lymphocyte function-associated antigen-1/intercellular adhesion molecule-1(LFA-1/ICAM-1) interaction inhibitor( IC50 of 5.0 …
Formula:
C18H17F3N4O2S
Purity:
99.22%
Color and Shape:
solid
Molecular weight:
410.41
Estimated delivery in United States, on Monday 7 Feb 2022
DYRKs-IN-2
CAS:1386980-04-6
DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM …
Formula:
C32H38ClN9O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
632.16
Estimated delivery in United States, on Monday 7 Feb 2022
Purvalanol B
CAS:212844-54-7
Purvalanol B is a CDK inhibitor that inhibits Cdk2/cyclin A, Cdk2/cyclin E, Cdk5/p35, and Cdk2/cyclin …
Formula:
C20H25ClN6O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
432.9
Estimated delivery in United States, on Monday 7 Feb 2022
LDC000067
CAS:1073485-20-7
LDC000067 is a highly specific and selective CDK9 inhibitor with an IC50 value of 44±10 …
Formula:
C18H18N4O3S
Purity:
99.07%
Color and Shape:
solid
Molecular weight:
370.43
Estimated delivery in United States, on Monday 7 Feb 2022
Simurosertib
CAS:1330782-76-7
Simurosertib is a selective and ATP-competitive cell division cycle 7 kinase inhibitor (IC50: <0.3 nM).
Formula:
C17H19N5OS
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
341.43
Estimated delivery in United States, on Monday 7 Feb 2022
Poloxin
CAS:321688-88-4
Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: …
Formula:
C18H19NO3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
297.35
Estimated delivery in United States, on Monday 7 Feb 2022
Deferoxamine Mesylate
CAS:138-14-7
Deferoxamine is an iron-chelating agent that binds free iron in a stable complex. It also …
Formula:
C26H52N6O11S
Purity:
99.65%
Color and Shape:
White To Off-White Powder
Molecular weight:
656.79
Estimated delivery in United States, on Monday 7 Feb 2022
TC-Mps1-12
CAS:1206170-62-8
TC-Mps1-12 is an effective and selective inhibitor of monopolar spindle 1 (IC50: 6.4 nM) .
Formula:
C17H20N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
324.38
Estimated delivery in United States, on Monday 7 Feb 2022
ZINC00881524
CAS:557782-81-7
ZINC00881524 is an effective and specific ROCK inhibitor.
Formula:
C21H20N2O3S
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
380.46
Estimated delivery in United States, on Monday 7 Feb 2022
NS13001
CAS:1063331-94-1
NS13001 is a potent, selective, orally active allosteric positive modulator of SK channels (small conductance …
Formula:
C17H16ClN7
Purity:
99.55%
Color and Shape:
solid
Molecular weight:
353.81
Estimated delivery in United States, on Monday 7 Feb 2022
BDP5290
CAS:1817698-21-7
BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, …
Formula:
C17H18ClN7O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
371.82
Estimated delivery in United States, on Monday 7 Feb 2022
BI 2536
CAS:755038-02-9
BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM). It has 4- and 11-fold greater …
Formula:
C28H39N7O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
521.66
Estimated delivery in United States, on Monday 7 Feb 2022
AS2863619
CAS:2241300-51-4
AS2863619 is an orally active inhibitor of cyclin-dependent kinase 8 (CDK8) and CDK19 (IC50s of …
Formula:
C16H14Cl2N8O
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
405.24
Estimated delivery in United States, on Monday 7 Feb 2022
(±)-BAY-1251152
CAS:1610358-53-6
(±)-BAY-1251152 is a racemic mixture of BAY-1251152. BAY-1251152 is highly selective inhibitor of PTEF/CDK9.
Formula:
C19H18F2N4O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
404.43
Estimated delivery in United States, on Monday 7 Feb 2022
FIT-039
CAS:1113044-49-7
FIT-039 is a selective and ATP-competitive, orally active inhibitor of CDK9( IC50 : 5.8 μM;CDK9/cyclin …
Formula:
C17H18FN3S
Molecular weight:
315.41
Estimated delivery in United States, on Monday 7 Feb 2022
Trilaciclib hydrochloride
CAS:1977495-97-8
Trilaciclib hydrochloride is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 …
Formula:
C24H32Cl2N8O
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
519.47
Estimated delivery in United States, on Monday 7 Feb 2022
CDK9-IN-9
CAS:2246956-84-1
CDK9-IN-9 is a potent and selective CDK9 inhibitor (IC50: 1.8 nM) with anti-cancer activity. It …
Formula:
C22H23F2N5O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
459.51
Estimated delivery in United States, on Monday 7 Feb 2022
PROTAC CDK2/9 Degrader-1
CAS:2408641-24-5
PROTAC CDK2/9 Degrader-1 is a potent CDK2 and CDK9 dual degrader(DC50 of 62 nM and …
Formula:
C40H41N13O7
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
815.84
Estimated delivery in United States, on Monday 7 Feb 2022
Tripolin A
CAS:1148118-92-6
Tripolin A is a specific non-ATP competitive inhibitor of Aurora A kinase(Aurora A and Aurora …
Formula:
C15H11NO3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
253.25
Estimated delivery in United States, on Monday 7 Feb 2022
CDK8-IN-4
CAS:1613638-82-6
CDK8-IN-4 is an inhibitor of CDK8 (IC50: 0.2 nM).
Formula:
C20H18N4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
330.38
Estimated delivery in United States, on Monday 7 Feb 2022
Palbociclib hydrochloride
CAS:827022-32-2
Palbociclib (PD-0332991) is a selective inhibitor of CDK4/6 (IC50s: 11/16 nM). It exhibits no inhibition …
Formula:
C24H29N7O2·HCl
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
483.99
Estimated delivery in United States, on Monday 7 Feb 2022
Rac1 Inhibitor W56 acetate(1095179-01-3 free base)
Peptide comprising residues 45-60 of the guanine nucleotide exchange factor (GEF) recognition/activation site of Rac1; …
Formula:
C76H121N19O25S
Molecular weight:
1732.95
Estimated delivery in United States, on Monday 7 Feb 2022
Liproxstatin-1
CAS:950455-15-9
Liproxstatin-1 is a potent ferroptosis inhibitor.
Formula:
C19H21ClN4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
340.85
Estimated delivery in United States, on Monday 7 Feb 2022
Bimosiamose disodium
CAS:187269-60-9
Bimosiamose disodium has anti-inflammatory effects[1]. Bimosiamose disodium (TBC-1269Z) is a nonoligosaccharide pan-selectin inhibitor with IC50s …
Formula:
C46H52Na2O16
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
906.88
Estimated delivery in United States, on Monday 7 Feb 2022
Ferrostatin-1
CAS:347174-05-4
Ferrostatin-1 is a potent ferroptosis inhibitor (EC50: 60 nM).
Formula:
C15H22N2O2
Purity:
99.68%
Color and Shape:
solid
Molecular weight:
262.35
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P180
CAS:211555-08-7
WHI-P180 is a potent EGFR and Cdk2 inhibitors with IC50 of 4.0 and 1.0 uM, …
Formula:
C16H15N3O3
Purity:
97.74%
Color and Shape:
solid
Molecular weight:
297.31
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06873600
CAS:2185857-97-8
PF-06873600 is a selective and orally bioavailable cyclin-dependent kinase (CDK) inhibitor(CDK2, CDK4 and CDK6 with …
Formula:
C20H27F2N5O4S
Purity:
98.77%
Color and Shape:
Solid
Molecular weight:
471.52
Estimated delivery in United States, on Monday 7 Feb 2022
UAMC-3203 hydrochloride
CAS:2271358-65-5
UAMC-3203 hydrochloride is a potent and selective Ferroptosis inhibitor with an IC50 of 12 nM.
Formula:
C25H38ClN5O2S
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
508.12
Estimated delivery in United States, on Monday 7 Feb 2022
Tricin
CAS:520-32-1
Tricin can inhibit human cytomegalovirus (HCMV) replication by inhibiting CDK9. Tricin inhibits the proliferation and …
Formula:
C17H14O7
Molecular weight:
330.29
Estimated delivery in United States, on Monday 7 Feb 2022
ILK-IN-3
CAS:6975-75-3
ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.
Formula:
C10H12N6O
Purity:
99.88%
Color and Shape:
solid
Molecular weight:
232.24
Estimated delivery in United States, on Monday 7 Feb 2022
THZ1
CAS:1604810-83-4
THZ1 is a novel selective and potent covalent CDK7 inhibitor.
Formula:
C31H28ClN7O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
566.05
Estimated delivery in United States, on Monday 7 Feb 2022
CHK1-IN-3
CAS:2097252-39-4
CHK1-IN-2 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM).
Formula:
C20H23N9O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
405.46
Estimated delivery in United States, on Monday 7 Feb 2022
TH 257
CAS:2244678-29-1
TH 257 is a Potent and selective allosteric LIMK 1/2 inhibitor(LIMK1 and LIMK2, IC50 of …
Formula:
C24H26N2O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
422.5
Estimated delivery in United States, on Monday 7 Feb 2022
Eg5 Inhibitor V, trans-24
CAS:869304-55-2
Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be …
Formula:
C26H21N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
423.46
Estimated delivery in United States, on Monday 7 Feb 2022
Gracillin
CAS:19083-00-2
Gracillin can induce cell cycle arrest, oxidative stress, and apoptosis in HL60 cells, and has …
Formula:
C45H72O17
Purity:
99.86%
Color and Shape:
solid
Molecular weight:
885.05
Estimated delivery in United States, on Monday 7 Feb 2022
Abemaciclib Metabolites M2
CAS:1231930-57-6
Abemaciclib Metabolites M2 is a metabolite of abemaciclib, acts as a potent CDK4 and CDK6 …
Formula:
C25H28F2N8
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
478.54
Estimated delivery in United States, on Monday 7 Feb 2022
Cdc7-IN-1
CAS:1402055-25-7
Cdc7-IN-1 is a highly selective and ATP competitive inhibitor of Cdc7 kinase (IC50: 0.6 nM …
Formula:
C21H16ClN3O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
409.82
Estimated delivery in United States, on Monday 7 Feb 2022
iRGD peptide
CAS:1392278-76-0
iRGD peptide is a 9-amino acid cyclic peptide (sequence: CRGDKGPDC) and a molecular mimicry agent …
Formula:
C35H57N13O14S2
Purity:
98.77%
Color and Shape:
Solid
Molecular weight:
948.04
Estimated delivery in United States, on Monday 7 Feb 2022
CHK-IN-1
CAS:1278405-51-8
CHK-IN-1 is a CHK1 and CHK2 inhibitor, has anti-proliferative activities.
Formula:
C18H19ClFN5OS
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
407.89
Estimated delivery in United States, on Monday 7 Feb 2022
CDKI-73
CAS:1421693-22-2
CDKI-73 is a potent CDK9 inhibitor (Ki: 4 nM). It shows selective toxicity to CLL …
Formula:
C15H15FN6O2S2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
394.45
Estimated delivery in United States, on Monday 7 Feb 2022
-glycosidase-IN-1
CAS:176485-27-1
-glycosidase-IN-1 is a piperidine derivative, and is an inhibitor of -glycosidase. It has hypoglycemic activity.
Formula:
C13H23NO5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
273.33
Estimated delivery in United States, on Monday 7 Feb 2022
Ilorasertib hydrochloride
CAS:1847485-91-9
Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora …
Formula:
C25H22ClFN6O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
525
Estimated delivery in United States, on Monday 7 Feb 2022
OSU-T315
CAS:1333146-24-9
OSU-T315 is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 …
Formula:
C30H30F3N5O
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
533.6
Estimated delivery in United States, on Monday 7 Feb 2022
LY2835219
CAS:1231930-82-7
LY2835219 is a specific and effective inhibitor of CDK4(IC50=2 nM) and CDK6(IC50=10 nM).
Formula:
C27H32F2N8·CH4O3S
Purity:
99.10%
Color and Shape:
solid
Molecular weight:
602.7
Estimated delivery in United States, on Monday 7 Feb 2022
AS2863619 free base
CAS:2241300-50-3
AS2863619 free base enables the conversion of antigen-specific effector/memory T cells into Foxp3+ regulatory T …
Formula:
C16H12N8O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
332.32
Estimated delivery in United States, on Monday 7 Feb 2022
EN4 MYC inhibitor
CAS:1197824-15-9
EN4 MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It …
Formula:
C25H24N2O4
Purity:
98.19%
Molecular weight:
416.47
Estimated delivery in United States, on Monday 7 Feb 2022
E7820
CAS:289483-69-8
E7820 is an angiogenesis inhibitor by suppressing integrin a2 (a cell adhesion molecule expressed on …
Formula:
C17H12N4O2S
Purity:
98.48%
Color and Shape:
solid
Molecular weight:
336.37
Estimated delivery in United States, on Monday 7 Feb 2022
CLK1-IN-1
CAS:2123491-32-5
CLK1-IN-1 is a potent and selective inhibitor of the Cdc2-like kinase 1 (CLK1; IC50: 2 …
Formula:
C24H16FN5O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
409.42
Estimated delivery in United States, on Monday 7 Feb 2022
CWHM-12
CAS:1564286-55-0
CWHM-12 is a potent inhibitor of V integrins (IC50s of 0.2/0.8/1.5/1.8 nM for v8/v3/v6/v1).
Formula:
C26H32BrN5O6
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
590.47
Estimated delivery in United States, on Monday 7 Feb 2022
