Cell Cycle/Checkpoint
Cell cycle/checkpoint inhibitors are compounds that disrupt the normal progression of the cell cycle, particularly at key regulatory checkpoints. These inhibitors are crucial for studying cell division, understanding cancer cell proliferation, and developing anti-cancer therapies. By targeting specific phases of the cell cycle, these inhibitors can induce cell cycle arrest, leading to apoptosis or senescence in rapidly dividing cells. At CymitQuimica, we offer a diverse range of high-quality cell cycle/checkpoint inhibitors to support your research in cancer biology, cell biology, and drug development.
Subcategories of "Cell Cycle/Checkpoint"
- Aurora Kinase(114 products)
- CDK(545 products)
- Cell Cycle Arrest(5 products)
- Chk(48 products)
- DYRK(47 products)
- Dynamin(27 products)
- Ferroptosis(226 products)
- HSP(179 products)
- Integrin(249 products)
- Kinesin(87 products)
- LIM Kinase(20 products)
- Microtubule Associated(274 products)
- PKC(124 products)
- PLK(25 products)
- ROCK(62 products)
- Rho(6 products)
- Wee1(14 products)
- c-Myc(76 products)
Show 10 more subcategories
Found 3859 products of "Cell Cycle/Checkpoint"
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TH1760
CAS:TH1760 inhibits NUDT15 (IC50=25nM); boosts 6-thioguanine efficacy in leukemia by raising 6-thio-(d)GTP.Formula:C20H18N4O5SPurity:97.31%Color and Shape:SoildMolecular weight:426.45Sulfameter
CAS:Sulfameter (Sulfametoxydiazine) is a long-acting sulfonamide antibacterial agent used to treat urinary tract infections and leprosy.Formula:C11H12N4O3SPurity:99.46% - 99.90%Color and Shape:Crystalline SolidMolecular weight:280.3Tegafur
CAS:Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity.Formula:C8H9FN2O3Purity:99.16% - 99.89%Color and Shape:White Crystalline PowderMolecular weight:200.17Upamostat
CAS:Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.Formula:C32H47N5O6SPurity:99.41%Color and Shape:SolidMolecular weight:629.81Ref: TM-T13257
1mg64.00€2mg94.00€5mg145.00€10mg226.00€25mg379.00€50mg538.00€100mg730.00€1mL*10mM (DMSO)163.00€ATN-161 acetate
CAS:ATN-161 acetate, a pentapeptide compound derived from the synergistic region of fibronectin, is an integrin-alpha5 antagonist with antitumor activity.Formula:C25H39N9O10SPurity:98.27%Color and Shape:SoildMolecular weight:657.7Ref: TM-T10398L
1mg190.00€5mg471.00€10mg663.00€25mg1,036.00€50mg1,429.00€100mg1,830.00€200mg2,498.00€Abituzumab
CAS:Abituzumab (DI17E6) is a humanized monoclonal antibody targeting integrin alphaV, exhibiting anti-cancer activity and can be used in prostate cancer research.Purity:>95%Color and Shape:LiquidMolecular weight:144.58 kDaBT173
CAS:BT173 is a novel inhibitor of homeodomain interacting protein kinase 2 (HIPK2 ), attenuating renal fibrosis through suppression of the TGF-ß1/Smad3 pathway.Formula:C18H12BrN3O2Purity:98.247%Color and Shape:SolidMolecular weight:382.21MKC8866
CAS:MKC8866, a selective IRE1 RNase inhibitor with an IC50 of 0.29 μM, curbs breast and prostate cancer cell growth.Formula:C18H19NO7Purity:99.28% - 99.854%Color and Shape:SolidMolecular weight:361.35Ref: TM-T15594
1mg84.00€2mg109.00€5mg177.00€10mg250.00€25mg423.00€50mg557.00€100mg760.00€200mg1,018.00€1mL*10mM (DMSO)192.00€N-Dodecyl-β-D-maltoside
CAS:N-Dodecyl-β-D-maltoside (Lauryl Maltoside) has also been employed in applications such as in the purification and stabilization of RNA polymerase and theFormula:C24H46O11Purity:99.18% - >99.99%Color and Shape:White PowderMolecular weight:510.62Tinengotinib
CAS:Tinengotinib is a multikinase inhibitor that targets a series of kinases , including Aurora kinases A/B, JAK1/2, FGFR1/2/3, VEGFRs, and many other kinases.Formula:C20H19ClN6OPurity:99.05%Color and Shape:SolidMolecular weight:394.86Osalmid
CAS:Osalmid (Oxaphenamide) is a choleretic drug, inhibits ribonucleotide reductase activity by targeting ribonucleotide reductase small subunit M2 (RRM2).Formula:C13H11NO3Purity:99.08% - 99.6%Color and Shape:White CrystalMolecular weight:229.23Foscarnet sodium
CAS:Foscarnet sodium (Phosphonoformate) is an antiviral agent used in the treatment of cytomegalovirus retinitis.Formula:CNa3O5PPurity:98.52%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:191.95Doxifluridine
CAS:Doxifluridine (AMC 0101) is a fluoropyrimidine derivative and oral prodrug of the antineoplastic agent 5-fluorouracil (5-FU) with antitumor activity.Formula:C9H11FN2O5Purity:99.47% - 99.86%Color and Shape:White SolidMolecular weight:246.19Foralumab
CAS:Foralumab (NI-0401) is a human anti-CD3 monoclonal antibody for the study of COVID-19 infection.Purity:96.7% (SDS-PAGE); 96.4% (SEC-HPLC) - 96.7% (SDS-PAGE); 96.4% (SEC-HPLC)Color and Shape:LiquidMolecular weight:146.59 kDaGemifloxacin mesylate
CAS:Gemifloxacin mesylate (Gemifloxacin mesylate) inhibits activities of DNA gyrase and topoisomerase IV, thereby inhibiting DNA replication and eventuallyFormula:C19H24FN5O7SPurity:97.24% - ≥95%Color and Shape:Beige SolidMolecular weight:485.49Teplizumab
CAS:Teplizumab (MGA-031) is a humanized monoclonal antibody against CD3 that slows the loss of beta cell function.Teplizumab is used to treat type 1 diabetes.Purity:SDS-PAGE:95.8%;SEC-HPLC:99.7%Color and Shape:LiquidMolecular weight:145.79 kDaCarmofur
CAS:Carmofur (HCFU) is a highly potent acid ceramidase inhibitor, used in the treatment of breast and colorectal cancer.Formula:C11H16FN3O3Purity:98.53% - 99.98%Color and Shape:SolidMolecular weight:257.26Orbofiban TFA
CAS:Orbofiban TFA is an orally active GPIIb/IIIa platelet receptor antagonist with inhibitory effects on platelet aggregation for the study of unstable coronaryFormula:C19H24F3N5O6Purity:97.21% - 98.72%Color and Shape:SolidMolecular weight:475.42Centrinone
CAS:Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).Formula:C26H25F2N7O6S2Purity:98.76%Color and Shape:SolidMolecular weight:633.65DNA2 inhibitor C5
CAS:DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.Formula:C10H6N2O5Purity:99.05%Color and Shape:SolidMolecular weight:234.16Ref: TM-T15146
1mg57.00€2mg80.00€5mg113.00€10mg178.00€25mg409.00€50mg605.00€100mg860.00€500mg1,728.00€1mL*10mM (DMSO)112.00€RWJ 50271
CAS:RWJ 50271 inhibits LFA-1/ICAM-1 interaction with IC50 5.0 μM in HL60 cells.Formula:C18H17F3N4O2SPurity:99.09%Color and Shape:SolidMolecular weight:410.41Ref: TM-T12783
1mg120.00€5mg295.00€10mg447.00€25mg707.00€50mg964.00€100mg1,243.00€200mg1,693.00€1mL*10mM (DMSO)326.00€Ledoxantrone trihydrochloride
CAS:Ledoxantrone trihydrochloride is a Top II inhibitor with anticancer activity and is used in the study of digestive disorders and urologic disorders.Formula:C21H30Cl3N5OSPurity:98.13%Color and Shape:SoildMolecular weight:506.92Arg-Gly-Asp-Ser acetate
Arg-Gly-Asp-Ser acetate targets integrin, binding pro-caspase-8, -9, -3, but not -1; inhibits receptor function.Formula:C17H31N7O10Purity:98.14%Color and Shape:SolidMolecular weight:493.47GRL0617
CAS:GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM).Formula:C20H20N2OPurity:99.31%Color and Shape:SolidMolecular weight:304.39Ref: TM-T11464
1mg34.00€5mg74.00€10mg105.00€25mg178.00€50mg313.00€100mg500.00€500mg1,063.00€1mL*10mM (DMSO)82.00€P 218
CAS:P 218 is a novel DHFR inhibitor with antimalarial activity and antifolate effects and can be used to study Buruli ulcer.Formula:C18H25ClN4O4Purity:98.83%Color and Shape:SoildMolecular weight:396.87Procarbazine hydrochloride
CAS:Procarbazine hydrochloride (NSC-77213 HCl) is the hydrochloride salt of a methylhydrazine derivative with antineoplastic and mutagenic activities.Formula:C12H19N3O·HClPurity:96.99% - ≥98%Color and Shape:(Ntp 1992)Molecular weight:257.76Rifabutin
CAS:Rifabutin (LM-427), a semisynthetic ansamycin, blocks bacterial RNA synthesis by inhibiting RNA polymerase.Formula:C46H62N4O11Purity:98.87% - 99.7%Color and Shape:Red-Violet Crystalline PowderMolecular weight:847.00C527
CAS:C527 is a is a pan DUB enzyme inhibitor. Which has a high potency for the USP1/UAF1 complex (IC50=0.88 μM).Formula:C17H8FNO3Purity:97.22%Color and Shape:SolidMolecular weight:293.25Monalizumab
CAS:Monalizumab, a humanized antibody, enhances NK cell function by inhibiting NKG2A; used in HNSCC studies.Purity:95% - >95.0% (SDS-PAGE); 100% (SEC-HPLC)Color and Shape:LiquidMolecular weight:147 kDaAbrilumab
CAS:Abrilumab (MEDI-7183) is a fully human monoclonal antibody against α4β7 that inhibits the α4β7 integrin.Purity:98.5% (SDS-PAGE); 99% (SEC-HPLC) - 98.5% (SDS-PAGE); 99% (SEC-HPLC)Color and Shape:LiquidMolecular weight:143.80 kDaEnrofloxacin
CAS:Enrofloxacin (BAY-Vp2674) is a veterinary antibacterial agent, used in poultry.
Formula:C19H22FN3O3Purity:99.43% - >99.99%Color and Shape:Pale Yellow CrystalsMolecular weight:359.39Rifaximin
CAS:Rifaximin: an oral semi-synthetic antibiotic from rifamycin SV; targets bacterial RNA polymerase to halt growth.Formula:C43H51N3O11Purity:99.18% - 99.40%Color and Shape:Red-Orange Crystalline PowderMolecular weight:785.88hSMG-1 inhibitor 11j
CAS:hSMG-1 inhibitor 11j: pyrimidine, IC50=0.11 nM, >455x selective vs. mTOR/PI3Kα/γ/CDK1/CDK2; cancer research use.
Formula:C27H28ClN7O3SPurity:99.22% - 99.65%Color and Shape:SolidMolecular weight:566.07Levofloxacin hydrate
CAS:Levofloxacin hydrate (Cravit hydrate) is a third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity.Formula:C18H20FN3O4H2OPurity:98.26%Color and Shape:Pale Yellow SolidMolecular weight:370.38Procaine
CAS:Procaine (Vitamin H3) is a slow-acting ester local anesthetic with a short effect, used for infiltration, nerve, and spinal blocks.
Formula:C13H20N2O2Purity:99.57% - 99.73%Color and Shape:Anhydrous Plates Tables From Ligroin Or Ether SolidMolecular weight:236.31ATN-161 trifluoroacetate salt
CAS:ATN-161 TFA salt, a new integrin α5β1 inhibitor, curbs angiogenesis, liver metastases growth, enhances survival in mice.Formula:C25H36F3N9O10SPurity:98% - 99.98%Color and Shape:SolidMolecular weight:711.67Hu7691 free base
CAS:Hu7691 free base is an Akt inhibitor that inhibits Akt1, Akt2 and Akt3 and induces differentiation of neuroblastoma cells.Formula:C22H21F3N4OPurity:98.89%Color and Shape:SolidMolecular weight:414.423BMVC-8C3O
CAS:BMVC-8C3O is a DNA G-quadruplex (G4) ligand.Cost-effective and quality-assured.Formula:C42H53I3N4O3Purity:99.72%Color and Shape:SolidMolecular weight:1042.61Ref: TM-T13584
1mg101.00€5mg192.00€10mg285.00€25mg462.00€50mg623.00€100mg858.00€200mg1,153.00€1mL*10mM (DMSO)371.00€TK216
CAS:TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.Formula:C19H15Cl2NO3Purity:97.22%Color and Shape:SolidMolecular weight:376.23Trimethoprim
CAS:Trimethoprim (NSC-106568) inhibits dihydrofolate reductase, CYP2C8, and OCT2 - an antibacterial agent.Formula:C14H18N4O3Purity:99.80% - 99.81%Color and Shape:White To Yellowish PowderMolecular weight:290.32NMDI14
CAS:NMDI14 is an inhibitor of nonsense mediated RNA decay (NMD).Formula:C21H25N3O4SPurity:97.79% - 99.37%Color and Shape:SolidMolecular weight:415.51Ref: TM-T12235
1mg35.00€5mg74.00€10mg119.00€25mg236.00€50mg356.00€100mg537.00€200mg762.00€1mL*10mM (DMSO)84.00€BAY-524
CAS:BAY-524 is an inhibitor of Bub1(IC50 = 450 nM.human Bub1 in the presence of 2 mM ATP).Formula:C24H24F2N6O3Purity:98.68% - 99.57%Color and Shape:SolidMolecular weight:482.48Ref: TM-T14505
1mg96.00€5mg177.00€10mg298.00€25mg482.00€50mg658.00€100mg892.00€1mL*10mM (DMSO)178.00€Pazufloxacin Mesylate
CAS:Pazufloxacin Mesylate (T-3762) is a fluoroquinolone antibiotic.Formula:C16H15FN2O4·CH4O3SPurity:99.88% - 99.93%Color and Shape:Crystalline SolidMolecular weight:414.4Nedaplatin
CAS:Nedaplatin, a cisplatin derivative, induces tumor DNA damage (IC50: 94 μM) through platinum-DNA cross-links, causing apoptosis.Formula:C2H8N2O3PtPurity:99.88% - >99.99%Color and Shape:Straw Yellow PowderMolecular weight:303.17GSK-3 inhibitor 4
CAS:Orally active GSK-3 inhibitor 4 targets GSK-3α/β, CDK2/5 (IC50: 0.45-0.68 μM) and may aid in Alzheimer's research by lowering Tau protein.Formula:C22H15F2N5OPurity:99.82%Color and Shape:SoildMolecular weight:403.38Ref: TM-T77341
1mg315.00€5mg873.00€10mg1,080.00€25mg1,431.00€50mg1,783.00€100mg2,250.00€500mg3,537.00€Tenofovir diphosphate TEA
CAS:Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.Formula:C9H16N5O10P3·C6H15NPurity:93.45% - 98.51%Color and Shape:SolidMolecular weight:548.36RG7800
CAS:RG7800 (RO6885247) has the potential for spinal muscular atrophy treatment. RG7800 is an SMN2 splicing modifier.Formula:C24H28N6OPurity:99.44%Color and Shape:SolidMolecular weight:416.52Y-33075 dihydrochloride
CAS:Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM).Formula:C16H18Cl2N4OPurity:98.88% - 99.89%Color and Shape:SolidMolecular weight:353.25Ref: TM-T13384L
1mg34.00€5mg66.00€10mg102.00€25mg192.00€50mg341.00€100mg510.00€200mg732.00€1mL*10mM (DMSO)78.00€GSK-626616
CAS:GSK-626616: strong, oral DYRK3 inhibitor (IC50: 0.7 nM), affects DYRK family, may treat anemia.Formula:C18H10Cl2N4OSPurity:98.27%Color and Shape:SolidMolecular weight:401.27BAY-2402234
CAS:BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.Formula:C21H18ClF5N4O4Purity:98.9%Color and Shape:SolidMolecular weight:520.84Ref: TM-T14501
1mg170.00€2mg234.00€5mg349.00€10mg537.00€25mg858.00€50mg1,161.00€100mg1,558.00€1mL*10mM (DMSO)401.00€Diaveridine
CAS:Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.Formula:C13H16N4O2Purity:99.10%Color and Shape:White SolidMolecular weight:260.29Enoxacin hydrate
CAS:Enoxacin hydrate (AT-2266 hydrate) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent.Formula:C15H17FN4O3H2OPurity:99.50%Color and Shape:SolidMolecular weight:347.34AZ1495
CAS:AZ1495: oral IRAK4 inhibitor (IC50: 5 nM), IRAK1 (23 nM), treats MYD88L265P DLBCL.Formula:C21H31N5O2Purity:98.81%Color and Shape:SolidMolecular weight:385.5Ref: TM-T14367
1mg93.00€5mg156.00€10mg245.00€25mg349.00€50mg494.00€100mg750.00€200mg1,009.00€1mL*10mM (DMSO)170.00€Ribociclib succinate
CAS:Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).Formula:C27H36N8O5Purity:99.9%Color and Shape:SolidMolecular weight:552.63Ref: TM-T15732
2mg34.00€5mg49.00€10mg70.00€25mg92.00€50mg109.00€100mg165.00€200mg258.00€500mg459.00€1mL*10mM (DMSO)60.00€JH-RE-06
CAS:JH-RE-06 disrupts mutagenic translesion synthesis (TLS) by preventing the recruitment of mutagenic POLζ.Formula:C20H16Cl3N3O4Purity:99.29%Color and Shape:SolidMolecular weight:468.72Ref: TM-T15611
1mg44.00€5mg93.00€10mg152.00€25mg334.00€50mg587.00€100mg1,044.00€1mL*10mM (DMSO)95.00€DHODH-IN-11
CAS:DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.Formula:C15H11N3O2Purity:98.14%Color and Shape:SolidMolecular weight:265.27AZ-Dyrk1B-33
CAS:AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.Formula:C19H16N4Purity:99.91%Color and Shape:SolidMolecular weight:300.36Ref: TM-T14364
1mg44.00€5mg92.00€10mg147.00€25mg289.00€50mg419.00€100mg583.00€200mg787.00€1mL*10mM (DMSO)100.00€Pyrimethamine
CAS:Pyrimethamine (Pirimecidan) is a competitive inhibitor of dihydrofolate reductase (DHFR), used as an antimalarial drug.Formula:C12H13ClN4Purity:99.67%Color and Shape:CrystalsMolecular weight:248.71Mps1-IN-3
CAS:Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).Formula:C26H31N7O4SPurity:99.25%Color and Shape:SolidMolecular weight:537.63Ref: TM-T16130
2mg34.00€5mg54.00€10mg87.00€25mg149.00€50mg255.00€100mg384.00€200mg538.00€1mL*10mM (DMSO)64.00€HBX 19818
CAS:HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).Formula:C25H28ClN3OPurity:97.71%Color and Shape:SolidMolecular weight:421.96Ref: TM-T15464
1mg35.00€5mg80.00€10mg111.00€25mg177.00€50mg253.00€100mg353.00€200mg502.00€1mL*10mM (DMSO)89.00€TAME hydrochloride
CAS:TAME hydrochloride (Tos-Arg-OMe HCl) is a kind od amino acid derivatives.Formula:C14H23ClN4O4SPurity:99.11% - 99.21%Color and Shape:White Fine Crystalline PowderMolecular weight:378.87Netarsudil Dihydrochloride
CAS:Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) is an inhibitor of Rho-related protein kinase (ROCK) and norepinephrine transporter (NET) and is effective in reducing intraocular pressure (IOP).Cost-effective and quality-assured.Formula:C28H29Cl2N3O3Purity:99.94% - 99.98%Color and Shape:SolidMolecular weight:526.45GSK-1520489A
CAS:GSK-1520489A is an active PKMYT1 inhibitor.Formula:C21H23N5O3SPurity:99.85%Color and Shape:SolidMolecular weight:425.5XPW1
CAS:XPW1 is a CDK9 inhibitor with antitumor activity, inhibits DNA repair procedures, and can be used for the research of clear cell renal cell carcinoma.Formula:C36H39ClFN7O2Purity:98.08%Color and Shape:SoildMolecular weight:656.19Cyclin K degrader 1
Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.Formula:C23H17Cl2N5O2Purity:99.76%Color and Shape:SolidMolecular weight:466.32Cibisatamab
CAS:Cibisatamab, a T-cell bispecific antibody, targets CEA on cancer cells and CD3 on T-cells, inducing T-cell-mediated tumor cell killing.Purity:SDS-PAGE:99.1%;SEC-HPLC:96.5%Color and Shape:LiquidMolecular weight:191.1 kDaCirtuvivint
CAS:Cirtuvivint (SM08502) is a potent and orally active CDC-like kinase (CLK) inhibitor that can be used to study arthritis.Formula:C24H25N7OPurity:99.95% - 99.96%Color and Shape:SolidMolecular weight:427.5Butylparaben
CAS:Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.Formula:C11H14O3Purity:98.15%Color and Shape:Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)Molecular weight:194.23LY 345899
CAS:LY 345899 is a Folate analog and is a methylenetetrahydrofolate dehydrogenase and MTHFD2 inhibitor (IC50: 96 nM and 663 nM, respectively and a Ki: 18 nM for
Formula:C20H21N7O7Purity:99.7%Color and Shape:SolidMolecular weight:471.42HLM006474
CAS:HLM006474 is a pan inhibitor of E2F. This inhibits E2F4 DNA-binding (IC50: 29.8 μM in A375 cells).Formula:C25H25N3O2Purity:99.04% - 99.20%Color and Shape:SolidMolecular weight:399.48TAO Kinase inhibitor 2
CAS:TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
Formula:C25H24N2O3Purity:98.58%Color and Shape:SoildMolecular weight:400.47MYCi975
CAS:MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.Formula:C25H16Cl2F6N2O2Purity:99.3% - 99.82%Color and Shape:SolidMolecular weight:561.3Otelixizumab
CAS:Otelixizumab (ChAglyCD3) is a chimeric monoclonal antibody targeting CD3, used in research on Type 1 diabetes and autoimmune diseases.Purity:>95%Color and Shape:LiquidLerociclib dihydrochloride
CAS:Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/Formula:C26H36Cl2N8OPurity:97.4%Color and Shape:SolidMolecular weight:547.52TAK-901
CAS:TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among othersFormula:C28H32N4O3SPurity:99.02% - 99.59%Color and Shape:SolidMolecular weight:504.64Ref: TM-T2709
1mg35.00€5mg70.00€10mg104.00€25mg202.00€50mg329.00€100mg525.00€200mg748.00€1mL*10mM (DMSO)79.00€Trilaciclib hydrochloride
CAS:Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).Formula:C24H32Cl2N8OPurity:99.69% - 99.89%Color and Shape:SolidMolecular weight:519.47Hycanthone
CAS:Hycanthone (Etrenol(mesylate)) is a potent drug of antischistosomal.Formula:C20H24N2O2SPurity:98.78%Color and Shape:Yellow-Orange Powder (Ntp 1992)Molecular weight:356.48NU6140
CAS:NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).Formula:C23H30N6O2Purity:98.33%Color and Shape:SolidMolecular weight:422.52Ref: TM-T16359
2mg39.00€5mg60.00€10mg92.00€25mg177.00€50mg285.00€100mg414.00€200mg580.00€1mL*10mM (DMSO)67.00€Rifapentine
CAS:Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections.Formula:C47H64N4O12Purity:95.74% - ≥98%Color and Shape:SolidMolecular weight:877.03Vitamin D2
CAS:Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.Formula:C28H44OPurity:98.73% - 99.89%Color and Shape:Prisms From Acetone 1998)Molecular weight:396.65R-10015
CAS:R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.Formula:C20H19ClN6O2Purity:98.68%Color and Shape:SolidMolecular weight:410.86Ref: TM-T12609
1mg50.00€5mg112.00€10mg170.00€25mg280.00€50mg371.00€100mg525.00€200mg712.00€1mL*10mM (DMSO)124.00€SIBA
CAS:SIBA, a synthetic SAH analog, inhibits SAM-dependent transmethylation and blocks HSV-1 replication.Formula:C14H21N5O3SPurity:99.48%Color and Shape:SolidMolecular weight:339.41Ref: TM-T12908
1mg52.00€5mg94.00€10mg117.00€25mg220.00€50mg329.00€100mg469.00€200mg652.00€1mL*10mM (DMSO)104.00€Abciximab
CAS:Abciximab: chimeric antibody, anti-platelet, blocks glycoprotein IIb/IIIa, vitronectin, Mac-1.Purity:SDS-PAGE:95.2%;SEC-HPLC:95.9%Color and Shape:LiquidMolecular weight:95.18 kDaPaprotrain
CAS:Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.Formula:C16H11N3Purity:99.91%Color and Shape:SolidMolecular weight:245.28Ref: TM-T12359
5mg46.00€10mg58.00€25mg92.00€50mg160.00€100mg236.00€200mg353.00€500mg580.00€1mL*10mM (DMSO)49.00€SU056
CAS:SU056 is a YB-1 inhibitor that induces cell-cycle arrest, apoptosis, and inhibits ovarian cancer cell migration.
Formula:C20H16FNO5Purity:99.89%Color and Shape:SoildMolecular weight:369.34DI-87
CAS:DI-87 (TRE-515) is a novel and orally available dCK (deoxycytidine kinase) inhibitor. DI-87 binds to dCK reduces the production of dNTP inhibits tumor growth.Formula:C23H30N6O3S2Purity:99.76%Color and Shape:SolidMolecular weight:502.65MALAT1-IN-1
CAS:MALAT1-IN-1 is an effective dose-dependent Malat1 inhibitor, not altering Neat1 expression.Formula:C19H21N3O2Purity:99.58%Color and Shape:SolidMolecular weight:323.39Ref: TM-T16007
5mg39.00€10mg63.00€25mg120.00€50mg224.00€100mg432.00€200mg623.00€1mL*10mM (DMSO)44.00€Metarrestin
CAS:Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis.
Formula:C31H30N4OPurity:99.45%Color and Shape:SolidMolecular weight:474.6Ref: TM-T12006
1mg40.00€2mg52.00€5mg88.00€10mg144.00€25mg298.00€50mg512.00€100mg740.00€500mg1,539.00€Nadifloxacin
CAS:Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.Formula:C19H21FN2O4Purity:99.03% - 99.7%Color and Shape:Off-White Crystalline SolidMolecular weight:360.38Pefloxacin Mesylate Dihydrate
CAS:Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).Formula:C17H20FN3O3·CH4O3S·2H2OPurity:99.79%Color and Shape:SolidMolecular weight:465.49Ceftriaxone sodium hydrate
CAS:Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.Formula:C18H16N8Na2O7S3·5H2OPurity:99.77% - 99.78%Color and Shape:White Or Almost White Crystalline Powder OdorlessMolecular weight:661.6Ribavirin
CAS:Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formula:C8H12N4O5Purity:99.09% - 99.83%Color and Shape:Less Solid Colourless SolidMolecular weight:244.20PTBP1-RNA-binding inhibitor P6 TFA
PTBP1-RNA-binding inhibitor P6 TFA is a stapled peptide inhibitor of PTBP1, used to inhibit RNA alternative splicing events regulated by PTBP1.Color and Shape:Odour SolidCa2+ channel agonist 1
CAS:Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.Formula:C19H26N6OPurity:97.71%Color and Shape:SolidMolecular weight:354.45Ref: TM-T10659
1mg97.00€5mg188.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)217.00€CDK2-IN-4
CAS:CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM for CDK2/cyclin A.Formula:C23H18N6O2SPurity:97.24% - 99.10%Color and Shape:SolidMolecular weight:442.49Ref: TM-T14916
1mg82.00€5mg192.00€10mg304.00€25mg522.00€50mg713.00€100mg1,018.00€1mL*10mM (DMSO)212.00€Cinoxacin
CAS:Cinoxacin (Compound 64716), an older synthetic antimicrobial, was related to the quinolone class of antibiotics.Formula:C12H10N2O5Purity:99.62% - 99.98%Color and Shape:SolidMolecular weight:262.22Famciclovir
CAS:Famciclovir (BRL 42810) inhibits Herpes virus DNA polymerase by mimicking nucleosides.Formula:C14H19N5O4Purity:99.85% - 99.99%Color and Shape:Off-White PowderMolecular weight:321.33MKC9989
CAS:MKC9989 is an inhibitor of Hydroxy aryl aldehydes (HAA). MKC9989 also inhibits IRE1α with an IC50 of 0.23 to 44 μM.Formula:C17H20O7Purity:99.3%Color and Shape:SolidMolecular weight:336.34Ref: TM-T12071
1mg51.00€5mg156.00€10mg226.00€25mg376.00€50mg543.00€100mg730.00€1mL*10mM (DMSO)140.00€BRD6989
CAS:BRD6989, a cortistatin A analog, inhibits CDK8/19, enhances IL-10, and binds CDK8 with a 200 nM IC50.Formula:C16H16N4Purity:99.43%Color and Shape:SolidMolecular weight:264.33Ref: TM-T14778
1mg34.00€5mg66.00€10mg92.00€25mg177.00€50mg268.00€100mg398.00€200mg575.00€1mL*10mM (DMSO)73.00€Procaine hydrochloride
CAS:Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.Formula:C13H20N2O2·HClPurity:99.1% - 99.22%Color and Shape:White Crystalline PowderMolecular weight:272.77
