CymitQuimica logo
Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

Show 34 more subcategories

Found 8626 products of "Metabolism"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Avasimibe

    CAS:
    <p>Avasimibe (PD-148515): Oral ACAT inhibitor, prevents arterial cholesterol buildup; IC50: 3.3 μM. Hinders CYP2C9/1A2/2C19; IC50: 2.9/13.9/26.5 μM.</p>
    Formula:C29H43NO4S
    Purity:98.39% - 99.91%
    Color and Shape:Solid
    Molecular weight:501.72
  • UK-371804

    CAS:
    <p>UK-371804: potent uPA blocker; candidate for chronic skin ulcer preclinical studies.</p>
    Formula:C14H16ClN5O4S
    Purity:95.81% - 99.77%
    Color and Shape:Solid
    Molecular weight:385.83
  • UC-1728

    CAS:
    <p>UC-1728 (t-TUCB) is an effective rabbit soluble epoxide hydrolase inhibitor (IC50: 2 nM on rabbit liver).</p>
    Formula:C21H21F3N2O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:438.4
  • OU749

    CAS:
    <p>OU749 is a γ-glutamyl transferase (GGT) inhibitor with an intrinsic Ki of 17.6 μM.</p>
    Formula:C16H15N3O3S2
    Purity:99.50%
    Color and Shape:Solid
    Molecular weight:361.44
  • Conduritol B epoxide

    CAS:
    <p>Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase).</p>
    Formula:C6H10O5
    Purity:99.85% - ≥98%
    Color and Shape:White Crystalline Solid
    Molecular weight:162.14
  • ML-​226

    CAS:
    <p>ML226 is a α/β hydrolase domain-containing protein 11 (ABHD11) inhibitor that inhibits ABHD11 in vitro and in situ.</p>
    Formula:C23H26N4O2
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:390.48
  • PF-07038124

    CAS:
    <p>PF-07038124 inhibits PDE4B2 (IC50=0.5 nM), IFNγ (IC50=1.06 nM), IL4 (IC50=4.1 nM), and IL-13 (IC50=125 nM).</p>
    Formula:C18H22BNO4
    Color and Shape:Solid
    Molecular weight:327.18
  • N6022

    CAS:
    <p>N6022(IC50 of 8 nM) is an effective, reversible, and selective S-Nitrosoglutathione reductase(GSNOR) inhibitor.</p>
    Formula:C24H22N4O3
    Purity:98.24% - 98.32%
    Color and Shape:Solid
    Molecular weight:414.46
  • LJ570

    CAS:
    <p>LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)</p>
    Formula:C27H22O3
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:394.46
  • URB602

    CAS:
    <p>URB602 is a specific monoacylglycerol lipase (MGL) inhibitor, which inhibits rat brain MGL (IC50: 28±4 μM) through a noncompetitive mechanism.</p>
    Formula:C19H21NO2
    Purity:99.64% - 99.9%
    Color and Shape:Off-White Solid
    Molecular weight:295.38
  • Fenretinide

    CAS:
    <p>Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.</p>
    Formula:C26H33NO2
    Purity:98% - 99.68%
    Color and Shape:Yellow Powder
    Molecular weight:391.55
  • CD437

    CAS:
    <p>CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.</p>
    Formula:C27H26O3
    Purity:98.92% - 99.63%
    Color and Shape:Solid
    Molecular weight:398.49
  • BPTES

    CAS:
    <p>BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.</p>
    Formula:C24H24N6O2S3
    Purity:95.83% - 99.64%
    Color and Shape:Solid
    Molecular weight:524.68
  • MPO-IN-28

    CAS:
    <p>MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.</p>
    Formula:C11H13N5O
    Purity:98.04%
    Color and Shape:Solid
    Molecular weight:231.25
  • HA130

    CAS:
    <p>HA130 is a selective ATX (autotaxin) inhibitor.</p>
    Formula:C24H19BFNO5S
    Purity:98.26% - ≥95%
    Color and Shape:Solid
    Molecular weight:463.29
  • EAAT2 activator 1

    CAS:
    <p>EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein</p>
    Formula:C16H11ClFN3S
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:331.8
  • 1-Cyclohexyl-3-dodecyl urea

    CAS:
    <p>1-Cyclohexyl-3-dodecyl urea (NCND) is a highly selective soluble epoxide hydrolase (sEH) inhibitor.</p>
    Formula:C19H38N2O
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:310.52
  • ASP-9521

    CAS:
    <p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>
    Formula:C19H26N2O3
    Purity:95.11% - 96.96%
    Color and Shape:Solid
    Molecular weight:330.42
  • Pinaverium bromide

    CAS:
    <p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>
    Formula:C26H41Br2NO4
    Purity:99.52%
    Color and Shape:White Crystalline Powder
    Molecular weight:591.42
  • Nitrofurazone

    CAS:
    <p>Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria.</p>
    Formula:C6H6N4O4
    Purity:99.87%
    Color and Shape:Pale Yellow Needles Solution) 6 0 - 6 5 Alkaline Solutions Are Dark Orange (Ntp 1992)
    Molecular weight:198.14
  • Linrodostat

    CAS:
    <p>Linrodostat (BMS-986205) is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.</p>
    Formula:C24H24ClFN2O
    Purity:99.54% - 99.71%
    Color and Shape:Solid
    Molecular weight:410.91
  • PF-06282999

    CAS:
    <p>PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potentially useful for the treatment of cardiovascular diseases.</p>
    Formula:C13H12ClN3O3S
    Purity:98.15% - 98.28%
    Color and Shape:Solid
    Molecular weight:325.77
  • NS-638

    CAS:
    <p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>
    Formula:C15H11ClF3N3
    Purity:98.44%
    Color and Shape:Solid
    Molecular weight:325.72
  • Pentamidine

    CAS:
    <p>Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor</p>
    Formula:C19H24N4O2
    Purity:98.64% - 99.67%
    Color and Shape:Crystallizes As Colorless Plates From Water Solid
    Molecular weight:340.42
  • 2-hydroxymethyl benzoic acid

    CAS:
    <p>2-hydroxymethyl benzoic acid is a principal metabolite of the phthalidyl moiety in man.</p>
    Formula:C8H8O3
    Purity:98.36%
    Color and Shape:Solid
    Molecular weight:152.15
  • Alrestatin

    CAS:
    <p>Alrestatin (AY-22284) is a specific inhibitor of aldose reductase and attenuates glucose-induced angiotensin II production in rat vascular smooth muscle in</p>
    Formula:C14H9NO4
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:255.2256
  • GOT1 inhibitor-1

    CAS:
    <p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>
    Formula:C19H19ClN4O
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:354.83
  • SR3335

    CAS:
    <p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>
    Formula:C13H9F6NO3S2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:405.34
  • AZ876

    CAS:
    <p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>
    Formula:C24H29N3O3S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:439.57
  • SR8278

    CAS:
    <p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>
    Formula:C18H19NO3S2
    Purity:99.44% - 99.73%
    Color and Shape:Solid
    Molecular weight:361.48
  • BRL-50481

    CAS:
    <p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>
    Formula:C9H12N2O4S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:244.27
  • Toloxatone

    CAS:
    <p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>
    Formula:C11H13NO3
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:207.23
  • U-104

    CAS:
    <p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>
    Formula:C13H12FN3O3S
    Purity:98.76% - 99.88%
    Color and Shape:Solid
    Molecular weight:309.32
  • Gonadorelin Acetate (33515-09-2 free base)

    CAS:
    <p>Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) is hypothalamic neuropeptide which plays a key role in the control of</p>
    Formula:C59H83N17O17
    Purity:99.42% - 99.46%
    Color and Shape:White Or Off-White Powder
    Molecular weight:1302.39
  • GSK805

    CAS:
    <p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>
    Formula:C23H18Cl2F3NO4S
    Purity:98% - ≥95%
    Color and Shape:Solid
    Molecular weight:532.36
  • 2-Bromo-4'-hydroxyacetophenone

    CAS:
    <p>2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).</p>
    Formula:C8H7BrO2
    Purity:98.64%
    Color and Shape:Clear Colorless To Light Yellow Liquid
    Molecular weight:215.04
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Formula:C11H13N
    Purity:95.64% - 97.21%
    Color and Shape:Solid
    Molecular weight:159.23
  • FG-2216

    CAS:
    <p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>
    Formula:C12H9ClN2O4
    Purity:97.1% - >99.99%
    Color and Shape:Solid
    Molecular weight:280.66
  • KPT9274

    CAS:
    KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.
    Formula:C35H29F3N4O3
    Purity:99.75% - 99.93%
    Color and Shape:Solid
    Molecular weight:610.62
  • LOX-IN-3 dihydrochloride

    CAS:
    <p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>
    Formula:C13H15Cl2FN2O2S
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:353.24
  • Cobicistat

    CAS:
    <p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>
    Formula:C40H53N7O5S2
    Purity:97.36% - 99.62%
    Color and Shape:Solid
    Molecular weight:776.02
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Formula:C15H35N2O6P
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:370.42
  • ARM1

    CAS:
    <p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>
    Formula:C16H14N2S
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:266.36
  • (±)-Amiflamine

    CAS:
    <p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>
    Formula:C12H20N2
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:192.3
  • Bempedoic acid

    CAS:
    <p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>
    Formula:C19H36O5
    Purity:99.85% - 99.94%
    Color and Shape:Solid
    Molecular weight:344.49
  • 1-Ethynylpyrene

    CAS:
    <p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>
    Formula:C18H10
    Purity:98.48%
    Color and Shape:Solid
    Molecular weight:226.27
  • Suvecaltamide

    CAS:
    <p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>
    Formula:C20H23F3N2O2
    Purity:99.29% - 99.70%
    Color and Shape:Solid
    Molecular weight:380.4
  • Diflubenzuron

    CAS:
    <p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>
    Formula:C14H9ClF2N2O2
    Purity:99.58% - 99.96%
    Color and Shape:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective Insecticide
    Molecular weight:310.68
  • GSK1016790A

    CAS:
    <p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>
    Formula:C28H32Cl2N4O6S2
    Purity:97.37% - 99.38%
    Color and Shape:Solid
    Molecular weight:655.61
  • DHBP dibromide

    CAS:
    <p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>
    Formula:C24H38Br2N2
    Purity:99.73%
    Color and Shape:Yellow To Yellow-Green Powder Or Flakes
    Molecular weight:514.38