GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Motilin (26-47), human, porcine
CAS:Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formula:C120H188N34O35SPurity:98%Color and Shape:SolidMolecular weight:2699.07AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Formula:C27H23ClN2O5Purity:98.06% - 99.79%Color and Shape:SolidMolecular weight:490.93Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formula:C66H87N17O14Purity:99.84%Color and Shape:SolidMolecular weight:1342.5Asapiprant
CAS:Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.Formula:C24H27N3O7SPurity:99.64%Color and Shape:SolidMolecular weight:501.55SB297006
CAS:<p>SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.</p>Formula:C18H18N2O5Purity:99.59%Color and Shape:SolidMolecular weight:342.35SLF1081851 TFA
CAS:SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.Formula:C23H34F3N3O3Color and Shape:SolidMolecular weight:457.538Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Formula:C21H24Cl2FNO2Color and Shape:SolidMolecular weight:412.33Vercirnon
CAS:<p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>Formula:C22H21ClN2O4SPurity:99.23%Color and Shape:SolidMolecular weight:444.93RS102895
CAS:<p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>Formula:C21H21F3N2O2Purity:97.64% - 99.80%Color and Shape:SolidMolecular weight:390.4BMS-813160
CAS:BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formula:C25H40N8O2Purity:99.66% - 99.79%Color and Shape:SolidMolecular weight:484.64L-765314
CAS:L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.Formula:C27H34N6O5Purity:99.73%Color and Shape:SolidMolecular weight:522.65-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formula:C4H6N2O3Purity:99.99%Color and Shape:SolidMolecular weight:130.1PAR-2 Activating Peptide acetate
<p>PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).</p>Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.88Pimavanserin tartrate
CAS:<p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>Formula:C50H68F2N6O4·C4H6O6Purity:99.24% - 99.98%Color and Shape:SolidMolecular weight:1005.2H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:98.25% - 99.47%Color and Shape:SolidMolecular weight:404.33Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurity:99.91%Color and Shape:SolidMolecular weight:456.49Ozanimod
CAS:Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formula:C23H24N4O3Purity:98.68% - 99.58%Color and Shape:SolidMolecular weight:404.46Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66ABT-724
CAS:ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formula:C17H19N5Purity:99.73%Color and Shape:SolidMolecular weight:293.37AC-55541
CAS:<p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.95% - 99.13%Color and Shape:SolidMolecular weight:269.73ZK 756326
CAS:ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formula:C21H28N2O3Purity:99.43%Color and Shape:SolidMolecular weight:356.46Dimaprit dihydrochloride
CAS:<p>Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.</p>Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19JNJ-10229570
CAS:<p>JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland</p>Formula:C22H19N3O2SPurity:98.41%Color and Shape:SolidMolecular weight:389.47Pimozide
CAS:<p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>Formula:C28H29F2N3OPurity:99.63% - >99.99%Color and Shape:SolidMolecular weight:461.55NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formula:C28H29Cl2N3OPurity:98.79%Color and Shape:SolidMolecular weight:494.46Bevantolol hydrochloride
CAS:Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formula:C20H28ClNO4Purity:99.49%Color and Shape:SolidMolecular weight:381.9Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Formula:C14H20F6N4O7Purity:98.18%Color and Shape:SolidMolecular weight:470.32Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Formula:C21H20O9Purity:98.90% - 99.21%Color and Shape:Yellow Brown Fine PowderMolecular weight:416.38JNJ-31020028
CAS:<p>JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).</p>Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68Tetrahydrozoline hydrochloride
CAS:Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.Formula:C13H16N2·HClPurity:99.90%Color and Shape:Off-White SolidMolecular weight:236.74Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formula:C21H30N4O4Purity:99.52%Color and Shape:SolidMolecular weight:402.49CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purity:99.08% - 99.76%Color and Shape:SolidMolecular weight:751.67A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Formula:C28H37N3O3Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:463.61MK 212 hydrochloride
CAS:MK 212 hydrochloride is a 5-HT2C receptor agonistFormula:C8H11ClN4·HClPurity:99.88%Color and Shape:SolidMolecular weight:235.12Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:98.87%Color and Shape:SolidMolecular weight:478.47S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Formula:C20H24ClN3O2Purity:98% - 99.84%Color and Shape:SolidMolecular weight:373.87MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Formula:C27H21F3N2O3Purity:99.54% - 99.59%Color and Shape:SolidMolecular weight:478.46Indacaterol
CAS:<p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>Formula:C24H28N2O3Purity:99.96%Color and Shape:SolidMolecular weight:392.49Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formula:C16H26N2O2Purity:99.52%Color and Shape:SolidMolecular weight:278.39Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formula:C21H19Cl2N3O6S3Purity:99.09%Color and Shape:SolidMolecular weight:576.49Pentagastrin
CAS:Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormula:C37H49N7O9SPurity:96.98% - 99.49%Color and Shape:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMolecular weight:767.89Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Formula:C38H73N21O10S2HClPurity:>99.99%Color and Shape:SolidMolecular weight:1353.33Mini Gastrin I, human acetate
<p>Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.</p>Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColor and Shape:SolidMolecular weight:445.96SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Formula:C16H17NO2·HClPurity:99.1% - 99.51%Color and Shape:SolidMolecular weight:291.77MK-571 sodium
CAS:MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formula:C26H27ClN2O3S2·NaPurity:97.86% - 99.58%Color and Shape:SolidMolecular weight:537.07Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formula:C23H24FN3O2Purity:99.2%Color and Shape:SolidMolecular weight:393.45Taprenepag
CAS:Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).Formula:C24H22N4O5SPurity:98.89% - 99.15%Color and Shape:SolidMolecular weight:478.52Tetracosactide acetate
CAS:Cosyntropin (acetate) stimulates the release of corticosteroids such as cortisol from the adrenal gland.Formula:C138H214N40O33SPurity:99.76%Color and Shape:SolidMolecular weight:2993.54Exo1
CAS:Exo1 is an inhibitor of the exocytic pathwayFormula:C15H12FNO3Purity:98.75%Color and Shape:SolidMolecular weight:273.26Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Formula:C11H12N2O2Purity:99.68%Color and Shape:SolidMolecular weight:204.23Isoxsuprine Free Base
CAS:Isoxsuprine Free Base relaxes uterine/vascular muscles, dilates arteries, treats peripheral vascular disease, and premature labor.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Moxisylyte
CAS:Moxisylyte (thymoxamine) treats erectile dysfunction, Reynaud's syndrome, and reverses eye mydriasis; it's an α1-adrenergic blocker.Formula:C16H25NO3Color and Shape:SolidMolecular weight:279.37Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81Solabegron HCl
CAS:Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.Formula:C23H24Cl2N2O3Color and Shape:SolidMolecular weight:447.35Phosphorylcholine chloride
CAS:Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integralFormula:C5H15ClNO4PPurity:99.481% - 99.85%Color and Shape:SolidMolecular weight:219.6Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purity:99.89%Color and Shape:SolidMolecular weight:239.27Opromazine hydrochloride
CAS:Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.Formula:C17H20Cl2N2OSPurity:98.03%Color and Shape:SolidMolecular weight:371.32Vortioxetine
CAS:<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formula:C21H27N3Purity:98%Color and Shape:SolidMolecular weight:321.46GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formula:C25H29N5OPurity:99.2%Color and Shape:SolidMolecular weight:415.53Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purity:99.52%Color and Shape:SolidMolecular weight:865.93Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurity:99.04%Color and Shape:SolidMolecular weight:436.95Bupranolol HCl
CAS:Bupranolol: non-selective beta blocker, no ISA, strong membrane stabilizer, fast gut absorption, high first-pass metabolism, 2-4hr half-life.Formula:C14H23Cl2NO2Color and Shape:SolidMolecular weight:308.243Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26BD 1008 Free Base
CAS:BD 1008 Free Base: Sigma-1 receptor antagonist, Kᵢ = 2 ± 1 nM, 4x more selective for sigma-1 than sigma-2.Formula:C15H22Cl2N2Color and Shape:SolidMolecular weight:301.25Lanreotide acetate
CAS:Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndromeFormula:C56H73N11O12S2Purity:>99.99%Color and Shape:SolidMolecular weight:1156.39Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFormula:C23H27ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:431.93SANT-1
CAS:SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formula:C23H27N5Purity:99.98% - >99.99%Color and Shape:SolidMolecular weight:373.49C-021
CAS:C 021 dihydrochloride is a potent CCR4 antagonist.Formula:C27H41N5O2Purity:99.74% - 99.90%Color and Shape:SolidMolecular weight:467.65[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formula:C69H108N22O16SPurity:99.71%Color and Shape:SolidMolecular weight:1533.8Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formula:C12H14N2·HClPurity:99.97%Color and Shape:SolidMolecular weight:222.71Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Formula:C63H104N22O17SPurity:98.33%Color and Shape:SolidMolecular weight:1473.72S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Formula:C23H24FN3O3Purity:99.07% - 99.9%Color and Shape:SolidMolecular weight:409.45Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Formula:C23H21F7N4O3Purity:98% - 99.68%Color and Shape:Off-White To Light Yellow Cyrstalline SolidMolecular weight:534.43Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formula:C4H3F7OPurity:98%Color and Shape:Less Oil Colorless OilMolecular weight:200.05ML-SI3
CAS:CCG-143140 is a GLP-1 receptor inverse agonists.Formula:C23H31N3O3SPurity:99.75%Color and Shape:SolidMolecular weight:429.58PF-4136309
CAS:PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formula:C29H31F3N6O3Purity:98.85% - 99.47%Color and Shape:SolidMolecular weight:568.59PGS-IN-1
CAS:<p>PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).</p>Formula:C19H26O3Purity:99.39%Color and Shape:SolidMolecular weight:302.41Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Formula:C17H25N7O4Purity:99.74%Color and Shape:SolidMolecular weight:391.42β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurity:99.64%Color and Shape:SolidMolecular weight:2720.97AC 187 Acetate
<p>AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.</p>Formula:C129H209N37O42Purity:99.71%Color and Shape:SolidMolecular weight:2950.26HhAntag
CAS:HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activityFormula:C24H23ClN4O3Purity:95.73%Color and Shape:SolidMolecular weight:450.92ML401
CAS:ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .Formula:C20H20BrClN2OPurity:99.13%Color and Shape:SolidMolecular weight:419.74ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84FK962
CAS:<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Formula:C14H17FN2O2Purity:99.89%Color and Shape:SolidMolecular weight:264.3SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Formula:C28H28ClN3OSPurity:97.37% - 98.88%Color and Shape:SolidMolecular weight:490.06
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