GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Purity (%)

100

products per page.

+ Info
Thiethylperazine
CAS:
- 1420-55-9
Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.
Formula:C₂₂H₂₉N₃S₂
Purity:98.72%
Color and Shape:Solid
Molecular weight:399.62
Ref: TM-T61915
+ Info
Hydroxyzine D8
CAS:
- 1189480-47-4
Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
Formula:C₂₁H₂₇ClN₂O₂
Purity:98%
Color and Shape:Solid
Molecular weight:382.95
Ref: TM-T11592
+ Info
Dapagliflozin impurity
CAS:
- 960404-86-8
Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.
Formula:C₂₁H₂₅ClO₇
Color and Shape:Solid
Molecular weight:424.87
Ref: TM-T10957
+ Info
L-798106
CAS:
- 244101-02-8
L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.
Formula:C₂₇H₂₂BrNO₄S
Purity:98.97%
Color and Shape:Solid
Molecular weight:536.44
Ref: TM-T15689
+ Info
Altanserin
CAS:
- 76330-71-7
Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.
Formula:C₂₂H₂₂FN₃O₂S
Color and Shape:Solid
Molecular weight:411.49
Ref: TM-T29913
+ Info
Nadolol-d9
CAS:
- 94513-92-5
Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.
Formula:C₁₇H₂₇NO₄
Purity:98%
Color and Shape:Solid
Molecular weight:318.46
Ref: TM-T12167
+ Info
SB-408124 Hydrochloride
CAS:
- 1431697-90-3
SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).
Formula:C₁₉H₁₉ClF₂N₄O
Purity:98%
Color and Shape:Solid
Molecular weight:392.83
Ref: TM-T12844
+ Info
3-Hydroxy agomelatine
CAS:
- 166526-99-4
3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.
Formula:C₁₅H₁₇NO₃
Color and Shape:Solid
Molecular weight:259.3
Ref: TM-T10114
+ Info
BW 723C86
CAS:
- 160521-72-2
BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.
Formula:C₁₆H₁₉ClN₂OS
Purity:99.35%
Color and Shape:Solid
Molecular weight:322.85
Ref: TM-T21625
+ Info
Omidenepag
CAS:
- 1187451-41-7
Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.
Formula:C₂₃H₂₂N₆O₄S
Purity:99.67% - 99.77%
Color and Shape:Solid
Molecular weight:478.52
Ref: TM-T16389
+ Info
Pramipexole dihydrochloride
CAS:
- 104632-25-9
Pramipexole dihydrochloride could be used to treat Parkinson disease.
Formula:C₁₀H₁₈ClN₃S
Purity:98%
Color and Shape:White Crystalline Powder
Molecular weight:247.79
Ref: TM-T1476L
+ Info
L 888607
CAS:
- 860033-06-3
L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).
Formula:C₁₉H₁₅ClFNO₂S
Color and Shape:Solid
Molecular weight:375.84
Ref: TM-T15828
+ Info
TFLLR-NH2(TFA)
CAS:
- 1313730-19-6
TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)
Formula:C₃₃H₅₄F₃N₉O₈
Purity:98%
Color and Shape:Solid
Molecular weight:761.83
Ref: TM-TP1334
+ Info
BMS-986020 sodium
CAS:
- 1380650-53-2
BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.
Formula:C₂₉H₂₅N₂NaO₅
Color and Shape:Solid
Molecular weight:504.51
Ref: TM-T63439
+ Info
GSK682753A
CAS:
- 1334294-76-6
GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).
Formula:C₂₃H₂₁Cl₃N₂O₃
Color and Shape:Solid
Molecular weight:479.78
Ref: TM-T11498
+ Info
Pimozide-d4
CAS:
- 1803193-57-8
Pimozide D4 is a deuterium labeled Pimozide.
Formula:C₂₈H₂₉F₂N₃O
Purity:98%
Color and Shape:Solid
Molecular weight:465.57
Ref: TM-T12476
+ Info
Calcium-Sensing Receptor Antagonists I
CAS:
- 478963-79-0
Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.
Formula:C₂₃H₂₄N₂O₂
Color and Shape:Solid
Molecular weight:360.45
Ref: TM-T10665
+ Info
GLP-1 receptor agonist 7
CAS:
- 2736447-04-2
GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.
Formula:C₃₁H₃₀ClFN₄O₅
Color and Shape:Solid
Molecular weight:593.05
Ref: TM-T64195
+ Info
Levomepromazine
CAS:
- 60-99-1
Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.
Formula:C₁₉H₂₄N₂OS
Purity:99.15%
Color and Shape:Solid
Molecular weight:328.47
Ref: TM-T15743
+ Info
Neurotensin(8-13)
CAS:
- 60482-95-3
Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
Formula:C₃₈H₆₄N₁₂O₈
Purity:99.95%
Color and Shape:Solid
Molecular weight:816.99
Ref: TM-T7617
+ Info
Telcagepant
CAS:
- 781649-09-0
Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.
Formula:C₂₆H₂₇F₅N₆O₃
Purity:98.98% - 98.98%
Color and Shape:Solid
Molecular weight:566.52
Ref: TM-T16093
+ Info
Piribedil D8
CAS:
- 1398044-45-5
Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.
Formula:C₁₆H₁₈N₄O₂
Purity:98%
Color and Shape:Solid
Molecular weight:306.39
Ref: TM-T12486
+ Info
4-Hydroxyatomoxetine D3
CAS:
- 1217686-14-0
4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.
Formula:C₁₇H₂₁NO₂
Purity:98%
Color and Shape:Solid
Molecular weight:274.37
Ref: TM-T10144
+ Info
Apraclonidine hydrochloride
CAS:
- 73218-79-8
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.
Formula:C₉H₁₁Cl₃N₄
Purity:99.74%
Color and Shape:Solid
Molecular weight:281.57
Ref: TM-T21371
+ Info
WAY-100635
CAS:
- 162760-96-5
WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .
Formula:C₂₅H₃₄N₄O₂
Purity:98.972%
Color and Shape:Solid
Molecular weight:422.56
Ref: TM-T21561
+ Info
(S)-ZINC-3573
CAS:
- 2095596-11-3
(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.
Formula:C₁₈H₂₁N₅
Color and Shape:Solid
Molecular weight:307.401
Ref: TM-T41187
+ Info
Timapiprant sodium
CAS:
- 950688-14-9
Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.
Formula:C₂₁H₁₇FN₂NaO₂
Purity:98%
Color and Shape:Solid
Molecular weight:371.367
Ref: TM-T17099
+ Info
5-HT2B antagonist-1
CAS:
- 393129-91-4
Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.
Formula:C₁₁H₁₄BrN₅
Purity:99.965%
Color and Shape:Solid
Molecular weight:296.17
Ref: TM-T9842
+ Info
Aripiprazole (D8)
CAS:
- 1089115-06-9
Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
Formula:C₂₃H₂₇Cl₂N₃O₂
Purity:98%
Color and Shape:Solid
Molecular weight:456.44
Ref: TM-T10368
+ Info
Nefazodone
CAS:
- 83366-66-9
Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.
Formula:C₂₅H₃₂ClN₅O₂
Purity:99.85%
Color and Shape:White To Off-White Crystalline Powder
Molecular weight:470.01
Ref: TM-T21451
+ Info
SB-269970 hydrochloride
CAS:
- 261901-57-9
SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity
Formula:C₁₈H₂₈N₂O₃S·HCl
Purity:98.45%
Color and Shape:Solid
Molecular weight:388.95
Ref: TM-T6655
+ Info
Levosalbutamol Hydrochloride
CAS:
- 50293-90-8
Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.
Formula:C₁₃H₂₂ClNO₃
Purity:98%
Color and Shape:Solid
Molecular weight:275.77
Ref: TM-T1139L
+ Info
Clomipramine D3 hydrochloride
CAS:
- 1398065-86-5
Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).
Formula:C₁₉H₂₄Cl₂N₂
Color and Shape:Solid
Molecular weight:354.33
Ref: TM-T10842L
+ Info
Fipexide hydrochloride
CAS:
- 34161-23-4
Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.
Formula:C₂₀H₂₂Cl₂N₂O₄
Color and Shape:Solid
Molecular weight:425.31
Ref: TM-T22332
+ Info
Setiptiline maleate
CAS:
- 85650-57-3
Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.
Formula:C₂₃H₂₃NO₄
Purity:99.94%
Color and Shape:Solid
Molecular weight:377.43
Ref: TM-T12900L
+ Info
Propranolol-d7 hydrochloride
CAS:
- 1613439-56-7
Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.
Formula:C₁₆H₂₂ClNO₂
Purity:98%
Color and Shape:Solid
Molecular weight:302.85
Ref: TM-T12550
+ Info
Cudarolimab
CAS:
- 2244739-29-3
Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.
Purity:97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)
Color and Shape:Liquid
Ref: TM-T77153
+ Info
Lanreotide
CAS:
- 108736-35-2
Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.
Formula:C₅₄H₆₉N₁₁O₁₀S₂
Color and Shape:Solid
Molecular weight:1096.32
Ref: TM-T20534
+ Info
Agomelatine-d6
CAS:
- 1079389-42-6
Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.
Formula:C₁₅H₁₇NO₂
Purity:98%
Color and Shape:Solid
Molecular weight:249.34
Ref: TM-T10266
+ Info
Brombuterol hydrochloride
CAS:
- 21912-49-2
Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.
Formula:C₁₂H₁₉Br₂ClN₂O
Color and Shape:Solid
Molecular weight:402.56
Ref: TM-T37848
+ Info
Substance P TFA
CAS:
- 148470-19-3
Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.
Formula:C₆₅H₉₉F₃N₁₈O₁₅S
Purity:98%
Color and Shape:Solid
Molecular weight:1461.67
Ref: TM-TP2155
+ Info
Diphenylpyraline
CAS:
- 147-20-6
Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.
Formula:C₁₉H₂₃NO
Color and Shape:Solid
Molecular weight:281.39
Ref: TM-T0059L
+ Info
Etofylline clofibrate
CAS:
- 54504-70-0
Etofylline clofibrate has a hypolipidemic and antithrombotic effect and it also has an agonistic interaction with intimal PGI2.
Formula:C₁₉H₂₁ClN₄O₅
Color and Shape:Solid
Molecular weight:420.85
Ref: TM-T15256
+ Info
Vilazodone-d8
CAS:
- 1794789-93-7
Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.
Formula:C₂₆H₂₇N₅O₂
Purity:98%
Color and Shape:Solid
Molecular weight:449.57
Ref: TM-T13300
+ Info
5-HT3 antagonist 5
CAS:
- 901599-43-7
5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.
Formula:C₁₆H₁₃N₃O₂
Purity:99.84%
Color and Shape:Solid
Molecular weight:279.29
Ref: TM-T9846
+ Info
SAR247799
CAS:
- 1315311-14-8
SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.
Formula:C₂₁H₁₆ClN₃O₅
Color and Shape:Solid
Molecular weight:425.82
Ref: TM-T38716
+ Info
Tegaserod
CAS:
- 145158-71-0
Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).
Formula:C₁₆H₂₃N₅O
Purity:99.20% - 99.89%
Color and Shape:Solid
Molecular weight:301.39
Ref: TM-T60680
+ Info
(+)-Penbutolol
CAS:
- 38363-41-6
(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.
Formula:C₁₈H₂₉NO₂
Color and Shape:Solid
Molecular weight:291.43
Ref: TM-T13465
+ Info
Rebamipide-d4
CAS:
- 1219409-06-9
Rebamipide D4 is deuterium labeled Rebamipide.
Formula:C₁₉H₁₅ClN₂O₄
Purity:98%
Color and Shape:Solid
Molecular weight:374.81
Ref: TM-T19547
+ Info
Acrivastine D7
CAS:
- 172165-56-9
Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
Formula:C₂₂H₂₄N₂O₂
Purity:98%
Color and Shape:Solid
Molecular weight:355.48
Ref: TM-T10241
+ Info
4-Hydroxypropranolol-d7 hydrochloride
CAS:
- 1219804-03-1
Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.
Formula:C₁₆H₂₂ClNO₃
Purity:98%
Color and Shape:Solid
Molecular weight:318.85
Ref: TM-T10149
+ Info
Haloperidol (D4')
CAS:
- 136765-35-0
Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.
Formula:C₂₁H₂₃ClFNO₂
Purity:98%
Color and Shape:Solid
Molecular weight:379.89
Ref: TM-T11536
+ Info
Ivabradine-d6 hydrochloride
CAS:
- 2070009-63-9
Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.
Formula:C₂₇H₃₇ClN₂O₅
Purity:98%
Color and Shape:Solid
Molecular weight:511.08
Ref: TM-T11694
+ Info
Clozapine-d8
CAS:
- 1185053-50-2
Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.
Formula:C₁₈H₁₉ClN₄
Color and Shape:Solid
Molecular weight:334.87
Ref: TM-TMIH-0166
+ Info
Ipragliflozin (L-Proline)
CAS:
- 951382-34-6
Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.
Formula:C₂₆H₃₀FNO₇S
Color and Shape:Solid
Molecular weight:519.58
Ref: TM-T11667
+ Info
Ramelteon-d5
CAS:
- 1134159-63-9
Ramelteon-d5 is a deuterated compound of Ramelteon.
Formula:C₁₆H₁₆D₅NO₂
Color and Shape:Solid
Molecular weight:264.37
Ref: TM-TMIH-0486
+ Info
Bombesin
CAS:
- 31362-50-2
Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.
Formula:C₇₁H₁₁₀N₂₄O₁₈S
Color and Shape:While Lyophilized Powder
Molecular weight:1619.85
Ref: TM-TP1281
+ Info
Cariprazine D6
CAS:
- 1308278-67-2
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
Formula:C₂₁H₂₆D₆Cl₂N₄O
Purity:98%
Color and Shape:Solid
Molecular weight:433.45
Ref: TM-T10681
+ Info
Lysosphingomyelin (d18:1)
CAS:
- 1670-26-4
Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.
Formula:C₂₃H₄₉N₂O₅P
Color and Shape:Solid
Molecular weight:464.628
Ref: TM-T38000
+ Info
β2AR/M-receptor agonist-2
CAS:
- 1017857-38-3
β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).
Formula:C₃₆H₄₉ClN₄O₇S
Color and Shape:Solid
Molecular weight:717.31
Ref: TM-T72226
+ Info
Cefaclor
CAS:
- 53994-73-3
Cefaclor (Panoral) is a cephalosporin antibiotic.
Formula:C₁₅H₁₄ClN₃O₄S
Purity:99.03% - 99.98%
Color and Shape:Solid
Molecular weight:367.81
Ref: TM-T6436
+ Info
Diacetolol D7
CAS:
- 1346604-19-0
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
Formula:C₁₆H₂₄N₂O₄
Purity:98%
Color and Shape:Solid
Molecular weight:315.42
Ref: TM-T11036
+ Info
R121919
CAS:
- 195055-03-9
R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.
Formula:C₂₂H₃₂N₆
Purity:99.75%
Color and Shape:Solid
Molecular weight:380.53
Ref: TM-T16713
+ Info
Dehydroaripiprazole
CAS:
- 129722-25-4
Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.
Formula:C₂₃H₂₅Cl₂N₃O₂
Purity:98.7%
Color and Shape:Solid
Molecular weight:446.37
Ref: TM-T10989
+ Info
ST-836 hydrochloride
CAS:
- 1415564-68-9
ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .
Formula:C₂₃H₃₅ClN₄OS
Purity:98%
Color and Shape:Solid
Molecular weight:451.07
Ref: TM-T13025L
+ Info
Thioridazine
CAS:
- 50-52-2
Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.
Formula:C₂₁H₂₆N₂S₂
Color and Shape:Solid
Molecular weight:370.57
Ref: TM-T61476
+ Info
Antazoline phosphate
CAS:
- 154-68-7
Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.
Formula:C₁₇H₂₂N₃O₄P
Purity:98%
Color and Shape:Coa
Molecular weight:363.35
Ref: TM-T21020
+ Info
Lecirelin
CAS:
- 61012-19-9
Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.
Formula:C₅₉H₈₄N₁₆O₁₂
Color and Shape:Solid
Molecular weight:1209.4
Ref: TM-TP1434
+ Info
MRGPRX4 modulator-2
CAS:
- 2492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].
Formula:C₁₅H₉ClF₄O₃
Purity:99.24%
Color and Shape:Solid
Molecular weight:348.68
Ref: TM-T61183
+ Info
ML 00253764
CAS:
- 681847-92-7
melanocortin MC4 receptor antagonist
Formula:C₁₈H₁₈BrFN₂O
Color and Shape:Solid
Molecular weight:377.25
Ref: TM-T22989
+ Info
Clorprenaline
CAS:
- 3811-25-4
Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.
Formula:C₁₁H₁₆ClNO
Purity:98.9%
Color and Shape:Solid
Molecular weight:213.7
Ref: TM-T60261
+ Info
1-Phenylbiguanide HCl
CAS:
- 55-57-2
Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.
Formula:C₈H₁₂ClN₅
Purity:99.31%
Color and Shape:Solid
Molecular weight:213.67
Ref: TM-PDK0269
+ Info
Ceralifimod
CAS:
- 891859-12-4
Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).
Formula:C₂₇H₃₃NO₄
Color and Shape:Solid
Molecular weight:435.56
Ref: TM-T14930
+ Info
JNJ-10397049
CAS:
- 708275-58-5
OX2 receptor antagonist
Formula:C₁₉H₂₀Br₂N₂O₃
Color and Shape:Solid
Molecular weight:484.18
Ref: TM-T22880
+ Info
Endothelin-3 (Rat,Human) (TFA)
Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).
Formula:C₁₂₃H₁₆₉F₃N₂₆O₃₅S₄·xC₂HF₃O₂
Purity:98%
Color and Shape:Solid
Molecular weight:2757.07 (free base)
Ref: TM-TP1173
+ Info
Glucagon (1-29), bovine, human, porcine
CAS:
- 16941-32-5
Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.
Formula:C₁₅₃H₂₂₅N₄₃O₄₉S
Purity:99.56% - 99.56%
Color and Shape:Solid
Molecular weight:3482.75
Ref: TM-T15389
+ Info
TP-16
CAS:
- 2332972-26-4
TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.
Formula:C₂₄H₂₂FNO₄S
Purity:98.53% - 99.15%
Color and Shape:Solid
Molecular weight:439.5
Ref: TM-T62525
+ Info
Zaloglanstat
CAS:
- 1513852-12-4
Zaloglanstat (ISC-27864) is a selective, orally active mPGES-1 inhibitor with an IC50 of 5 nM, analgesic in osteoarthritis and inflammatory arthritis.
Formula:C₂₁H₂₀ClF₃N₄O₂
Purity:99.97%
Color and Shape:Solid
Molecular weight:452.86
Ref: TM-T39000
+ Info
Tiotidine
CAS:
- 69014-14-8
Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).
Formula:C₁₀H₁₆N₈S₂
Purity:98%
Color and Shape:Solid
Molecular weight:312.42
Ref: TM-T13163
+ Info
Gizzerosine
CAS:
- 89238-78-8
Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.
Formula:C₁₁H₂₀N₄O₂
Color and Shape:Solid
Molecular weight:240.3
Ref: TM-T31931
+ Info
3-Hydroxy agomelatine D3
CAS:
- 1079774-23-4
3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).
Formula:C₁₅H₁₇NO₃
Purity:98%
Color and Shape:Solid
Molecular weight:262.32
Ref: TM-T10113
+ Info
(Rac)-Mirabegron-d5
CAS:
- 1215807-38-7
(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.
Formula:C₂₁H₂₄N₄O₂S
Purity:98%
Color and Shape:Solid
Molecular weight:401.54
Ref: TM-T12671
+ Info
Fluvoxamine
CAS:
- 54739-18-3
Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.
Formula:C₁₅H₂₁F₃N₂O₂
Color and Shape:Solid
Molecular weight:318.33
Ref: TM-T1077L
+ Info
Fexofenadine-d6
CAS:
- 548783-71-7
Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
Formula:C₃₂H₃₉NO₄
Purity:98%
Color and Shape:Solid
Molecular weight:507.69
Ref: TM-T11276
+ Info
Flibanserin-d4
CAS:
- 2122830-90-2
Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.
Formula:C₂₀H₂₁F₃N₄O
Purity:98%
Color and Shape:Solid
Molecular weight:394.43
Ref: TM-T11295
+ Info
Doxepin D3 Hydrochloride
CAS:
- 347840-07-7
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and
Formula:C₁₉H₂₂ClNO
Purity:98%
Color and Shape:Solid
Molecular weight:318.86
Ref: TM-T11088
+ Info
NBI-27914
CAS:
- 184241-44-9
NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.
Formula:C₁₈H₂₀Cl₄N₄
Purity:99.47% - 99.64%
Color and Shape:Solid
Molecular weight:434.19
Ref: TM-T62444
+ Info
Paliperidone Palmitate
CAS:
- 199739-10-1
Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.
Formula:C₃₉H₅₇FN₄O₄
Purity:98%
Color and Shape:Solid
Molecular weight:664.89
Ref: TM-T19950
+ Info
Tulobuterol-d9 HCl
CAS:
- 1325559-14-5
Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.
Formula:C₁₂H₁₀D₉Cl₂NO
Molecular weight:273.25
Ref: TM-TMIH-0589
+ Info
(R)-Praziquantel-d11
CAS:
- 1399880-38-6
(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.
Formula:C₁₉H₂₄N₂O₂
Purity:98%
Color and Shape:Solid
Molecular weight:323.47
Ref: TM-T12638
+ Info
SB-674042
CAS:
- 483313-22-0
SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.
Formula:C₂₄H₂₁FN₄O₂S
Purity:99.9%
Color and Shape:Solid
Molecular weight:448.51
Ref: TM-T16854
+ Info
Emedastine Difumarate
CAS:
- 87233-62-3
Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.
Formula:C₂₅H₃₄N₄O₉
Color and Shape:Solid
Molecular weight:534.56
Ref: TM-T21388
+ Info
PSB-0739
CAS:
- 1052087-90-7
PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.
Formula:C₂₆H₁₇N₃Na₂O₈S₂
Purity:98%
Color and Shape:Solid
Molecular weight:609.54
Ref: TM-T23195
+ Info
Mozavaptan hydrochloride
CAS:
- 138470-70-9
Mozavaptan is a vasopressin receptor antagonist.
Formula:C₂₇H₃₀ClN₃O₂
Color and Shape:Solid
Molecular weight:464
Ref: TM-T21465
+ Info
SUN B8155
CAS:
- 345893-91-6
SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.
Formula:C₁₄H₁₅N₃O₃
Purity:99.38% - 99.38%
Color and Shape:Solid
Molecular weight:273.29
Ref: TM-T23406
+ Info
Bromperidol hydrochloride
CAS:
- 59453-24-6
Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.
Formula:C₂₁H₂₄BrClFNO₂
Color and Shape:Solid
Molecular weight:456.78
Ref: TM-T62840
+ Info
GLP-1 receptor agonist 2
CAS:
- 2230197-64-3
GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:C₃₀H₃₁ClFN₅O₄
Color and Shape:Solid
Molecular weight:580.05
Ref: TM-T11407
+ Info
Aramisulpride
CAS:
- 71675-90-6
Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.
Formula:C₁₇H₂₇N₃O₄S
Color and Shape:Solid
Molecular weight:369.48
Ref: TM-T40825
+ Info
Tetrahexyldecyl ascorbate
CAS:
- 183476-82-6
Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.
Formula:C₇₀H₁₂₈O₁₀
Purity:98%
Color and Shape:Solid
Molecular weight:1129.76
Ref: TM-T20174
+ Info
MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.
Formula:C₁₅H₂₀F₃N₃O₄
Color and Shape:Solid
Molecular weight:363.332
Ref: TM-T204444
+ Info
Alosetron D3 Hydrochloride
CAS:
- 1189919-71-8
Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
Formula:C₁₇H₁₉ClN₄O
Purity:98%
Color and Shape:Solid
Molecular weight:333.83
Ref: TM-T19190
+ Info
RU-SKI 43 Hydrochloride
CAS:
- 1782573-67-4
RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.
Formula:C₂₂H₃₁ClN₂O₂S
Purity:98%
Color and Shape:Solid
Molecular weight:423.01
Ref: TM-T12797L
+ Info
Dexloxiglumide
CAS:
- 119817-90-2
Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.
Formula:C₂₁H₃₀Cl₂N₂O₅
Color and Shape:Solid
Molecular weight:461.38
Ref: TM-T15105
+ Info
Revdofilimab
CAS:
- 2230138-89-1
Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.
Purity:98.80% - 98.80%
Color and Shape:Liquid
Ref: TM-T77181
+ Info
SKF-82958 hydrobromide
CAS:
- 74115-01-8
SKF-82958 hydrobromide is a D1/D5 receptor full agonist.
Formula:C₁₉H₂₁BrClNO₂
Purity:98%
Color and Shape:Solid
Molecular weight:410.73
Ref: TM-T16892
+ Info
Benoxathian hydrochloride
CAS:
- 92642-97-2
Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.
Formula:C₁₉H₂₄ClNO₄S
Color and Shape:Solid
Molecular weight:397.91
Ref: TM-T61889
+ Info
Quetiapine-d4 hemifumarate
CAS:
- 1217310-65-0
Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.
Formula:C₂₅H₂₉N₃O₆S
Purity:98%
Color and Shape:White Solid
Molecular weight:503.61
Ref: TM-T12618L
+ Info
LY223982
CAS:
- 117423-74-2
LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.
Formula:C₃₀H₃₀O₇
Purity:99.86%
Color and Shape:Solid
Molecular weight:502.56
Ref: TM-T15803
+ Info
YNT-185 dihydrochloride
CAS:
- 1804978-82-2
Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.
Formula:C₃₃H₃₉Cl₂N₅O₅S
Color and Shape:Solid
Molecular weight:688.67
Ref: TM-T37112
+ Info
Cetirizine D4
CAS:
- 1219803-84-5
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
Formula:C₂₁H₂₅ClN₂O₃
Purity:98%
Color and Shape:Solid
Molecular weight:392.91
Ref: TM-T10769
+ Info
GB-88
CAS:
- 1416435-96-5
GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.
Formula:C₃₂H₄₂N₄O₄
Color and Shape:Solid
Molecular weight:546.7
Ref: TM-T11370
+ Info
Bradykinin (1-5)
CAS:
- 23815-89-6
Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.
Formula:C₂₇H₄₀N₈O₆
Color and Shape:Solid
Molecular weight:572.66
Ref: TM-TP1725
+ Info
Virodhamine
CAS:
- 287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.
Formula:C₂₂H₃₇NO₂
Purity:98%
Color and Shape:Soild
Molecular weight:347.53
Ref: TM-T64371
+ Info
Methyldopate
CAS:
- 6014-30-8
Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.
Formula:C₁₂H₁₇NO₄
Color and Shape:Solid
Molecular weight:239.27
Ref: TM-T36206
+ Info
Ziprasidone amino acid
CAS:
- 1159977-64-6
Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.
Formula:C₂₁H₂₃ClN₄O₂S
Color and Shape:Solid
Molecular weight:430.95
Ref: TM-T73961
+ Info
Doxazosin D8
CAS:
- 1126848-44-9
Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.
Formula:C₂₃H₂₅N₅O₅
Purity:98%
Color and Shape:Solid
Molecular weight:459.52
Ref: TM-T19297
+ Info
TS-011
CAS:
- 339071-18-0
N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.
Formula:C₁₁H₁₄ClN₃O₂
Purity:99.48%
Color and Shape:Solid
Molecular weight:255.7
Ref: TM-T13215
+ Info
Takeda103A
CAS:
- 865609-72-9
Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
Formula:C₂₄H₂₃F₂N₇O
Purity:97.17%
Color and Shape:Solid
Molecular weight:463.48
Ref: TM-T24850
+ Info
Albiglutide TFA (782500-75-8 free base)
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
Formula:C₁₅₀H₂₂₅F₃N₄₀O₄₇
Purity:>99.99%
Color and Shape:Solid
Molecular weight:3397.63
Ref: TM-TP1796
+ Info
Dexmedetomidine hydrochloride
CAS:
- 145108-58-3
Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:C₁₃H₁₆N₂·HCl
Purity:99.94% - 99.94%
Color and Shape:White Or Almost White Crystalline Powder
Molecular weight:236.74
Ref: TM-T6466
+ Info
Eformoterol Hemifumarate
CAS:
- 43229-80-7
Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma
Formula:C₁₉H₂₄N₂O₄C₄H₄O₄
Purity:99.86% - >99.99%
Color and Shape:White Powder
Molecular weight:402.4
Ref: TM-T6505
+ Info
Protease-Activated Receptor-2, amide
CAS:
- 190383-13-2
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
Formula:C₂₈H₅₄N₈O₇
Purity:>99.99%
Color and Shape:Solid
Molecular weight:614.78
Ref: TM-T7513
+ Info
Cinaciguat
CAS:
- 329773-35-5
Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:C₃₆H₃₉NO₅
Purity:98% - 99.18%
Color and Shape:Solid
Molecular weight:565.7
Ref: TM-T1984
+ Info
JD-5037
CAS:
- 1392116-14-1
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
Formula:C₂₇H₂₇Cl₂N₅O₃S
Purity:99.54% - 99.84%
Color and Shape:Solid
Molecular weight:572.51
Ref: TM-T4453
+ Info
TC-G 1005
CAS:
- 1415407-60-1
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).
Formula:C₂₅H₂₅N₃O₂
Purity:98.60% - 99.78%
Color and Shape:Solid
Molecular weight:399.48
Ref: TM-T8818
+ Info
C14TKL-1 acetate
C14TKL-1 acetate is a NK1 receptor agonist.
Formula:C₆₅H₁₀₂N₂₀O₁₅S₂
Purity:98.56%
Color and Shape:Solid
Molecular weight:1467.75
Ref: TM-TP2227L
+ Info
5-HT1A modulator 2 hydrochloride
CAS:
- 3880-76-0
5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.
Formula:C₁₁H₁₆ClNO
Purity:98.5%
Color and Shape:Solid
Molecular weight:213.7
Ref: TM-T37197
+ Info
Prasugrel Hydrochloride
CAS:
- 389574-19-0
Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
Formula:C₂₀H₂₀FNO₃S·HCl
Purity:99.39% - 99.79%
Color and Shape:Solid
Molecular weight:409.9
Ref: TM-T6952
+ Info
Fosaprepitant dimeglumine
CAS:
- 265121-04-8
Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.
Formula:C₃₇H₅₆F₇N₆O₁₆P
Purity:98% - 99.03%
Color and Shape:Solid
Molecular weight:1004.83
Ref: TM-T1790
+ Info
3-CPMT
CAS:
- 14008-79-8
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
Formula:C₂₁H₂₅Cl₂NO
Purity:99.03%
Color and Shape:Solid
Molecular weight:378.33
Ref: TM-T22508
+ Info
PSB-SB-487
CAS:
- 1399049-81-0
PSB-SB-487 is antagonist of GPR55.
Formula:C₂₆H₃₂O₄
Purity:98.53%
Color and Shape:Solid
Molecular weight:408.53
Ref: TM-T8975
+ Info
PNU-282987
CAS:
- 123464-89-1
PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).
Formula:C₁₄H₁₈Cl₂N₂O
Purity:99% - >99.99%
Color and Shape:Solid
Molecular weight:301.21
Ref: TM-T2422
+ Info
SSR240612
CAS:
- 464930-42-5
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,
Formula:C₄₂H₅₃ClN₄O₇S
Purity:98.59% - 99.16%
Color and Shape:Solid
Molecular weight:793.41
Ref: TM-T5048
+ Info
GSK189254A
CAS:
- 720690-73-3
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
Formula:C₂₁H₂₅N₃O₂
Purity:98.71% - 99.858%
Color and Shape:Solid
Molecular weight:351.44
Ref: TM-TQ0066
+ Info
[Sar9,Met(O2)11]-Substance P
CAS:
- 110880-55-2
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
Formula:C₆₄H₁₀₀N₁₈O₁₅S
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1393.66
Ref: TM-T7828
+ Info
JNJ-37822681
CAS:
- 935776-74-2
JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.
Formula:C₁₇H₁₇F₅N₄
Purity:99.84%
Color and Shape:Solid
Molecular weight:372.34
Ref: TM-T27677
+ Info
Exendin-4 acetate
CAS:
- 914454-01-6
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
Formula:C₁₈₆H₂₈₆N₅₀O₆₂S
Purity:98.48% - 99.78%
Color and Shape:Solid
Molecular weight:4247
Ref: TM-T8748
+ Info
Clomipramine
CAS:
- 303-49-1
Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.
Formula:C₁₉H₂₃ClN₂
Purity:99.31% - 99.71%
Color and Shape:Solid
Molecular weight:314.85
Ref: TM-T21013
+ Info
Clebopride malate
CAS:
- 57645-91-7
Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.
Formula:C₂₄H₃₀ClN₃O₇
Purity:99.52%
Color and Shape:Solid
Molecular weight:507.96
Ref: TM-T7569
+ Info
Aprocitentan
CAS:
- 1103522-45-7
Aprocitentan (ACT-132577) is ETA and ETB antagonist .
Formula:C₁₆H₁₄Br₂N₆O₄S
Purity:99.17%
Color and Shape:Solid
Molecular weight:546.19
Ref: TM-T7817
+ Info
Ertugliflozin
CAS:
- 1210344-57-2
PF-04971729 (Ertugliflozin (PF-04971729)) is a potent and selective inhibitor of the sodium-dependent glucose cotransporter 2 (SGLT2).
Formula:C₂₂H₂₅ClO₇
Purity:99.89% - 99.96%
Color and Shape:Solid
Molecular weight:436.88
Ref: TM-T4999
+ Info
R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).
Formula:C₅₉H₈₂F₃N₁₃O₁₄
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1254.36
Ref: TM-TP1933
+ Info
Fluoroclebopride
CAS:
- 154540-49-5
Fluoroclebopride is a dopamine (DA) D2 receptor ligand.
Formula:C₂₀H₂₃ClFN₃O₂
Purity:99.68% - 99.91%
Color and Shape:Solid
Molecular weight:391.87
Ref: TM-T3187
+ Info
Zafirlukast
CAS:
- 107753-78-6
Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and anti-inflammatory effects. Cost-effective and quality-assured.
Formula:C₃₁H₃₃N₃O₆S
Purity:99% - 99.83%
Color and Shape:Solid
Molecular weight:575.68
Ref: TM-T6736
+ Info
BQ-123
CAS:
- 136553-81-6
BQ-123 is a selective endothelin A receptor (ETA) antagonist with IC50 of 7.3 nM. Phase 2.
Formula:C₃₁H₄₂N₆O₇
Purity:99.22% - ≥95%
Color and Shape:Solid
Molecular weight:610.7
Ref: TM-T6792
+ Info
OS-3-106
CAS:
- 1580000-17-4
OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.
Formula:C₂₅H₃₀N₄O₂S
Purity:99.4% - 99.57%
Color and Shape:Solid
Molecular weight:450.6
Ref: TM-T8959
+ Info
8-Hydroxy-DPAT hydrobromide
CAS:
- 76135-31-4
8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.
Formula:C₁₆H₂₆BrNO
Purity:98.90% - 99.09%
Color and Shape:Solid
Molecular weight:328.29
Ref: TM-T22534
+ Info
SDZ WAG 994
CAS:
- 130714-47-5
SDZ WAG 994 is an A1 adenosine receptor agonist.
Formula:C₁₇H₂₅N₅O₄
Purity:99.82%
Color and Shape:Solid
Molecular weight:363.41
Ref: TM-T23347
+ Info
LY255283
CAS:
- 117690-79-6
LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.
Formula:C₁₉H₂₈N₄O₃
Purity:99.18%
Color and Shape:Solid
Molecular weight:360.45
Ref: TM-T22946
+ Info
Dynamin inhibitory peptide Acetate
Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin.
Formula:C₄₉H₈₄N₁₈O₁₆
Purity:97.28%
Color and Shape:Solid
Molecular weight:1181.3
Ref: TM-T21798L
+ Info
Fexofenadine hydrochloride
CAS:
- 153439-40-8
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,
Formula:C₃₂H₃₉NO₄·HCl
Purity:99.39% - ≥95%
Color and Shape:Solid
Molecular weight:538.13
Ref: TM-T1470
+ Info
Physalaemin acetate
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
Formula:C₆₀H₈₈N₁₄O₁₈S
Purity:99.13%
Color and Shape:Solid
Molecular weight:1325.49
Ref: TM-T19518L
+ Info
Tofogliflozin (hydrate)
CAS:
- 1201913-82-7
Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).
Formula:C₂₂H₂₈O₇
Purity:97.03% - 98.78%
Color and Shape:Solid
Molecular weight:404.45
Ref: TM-T5016
+ Info
Triptorelin acetate(57773-63-4 free base)
CAS:
- 140194-24-7
Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.
Formula:C₆₆H₈₆N₁₈O₁₅
Purity:99.90%
Color and Shape:White Powder
Molecular weight:1371.53
Ref: TM-T21410
+ Info
Myristicin
CAS:
- 607-91-0
Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formula:C₁₁H₁₂O₃
Purity:99.828%
Color and Shape:Liquid
Molecular weight:192.21
Ref: TM-T9113
+ Info
GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:C₅₁H₆₅N₉O₁₀
Purity:97.86%
Color and Shape:Solid
Molecular weight:964.12
Ref: TM-T22811L
+ Info
Hypidone hydrochloride
CAS:
- 1339058-04-6
Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor
Formula:C₁₈H₂₃ClN₂O₂
Purity:99.82% - 99.93%
Color and Shape:Solid
Molecular weight:334.84
Ref: TM-T3648
+ Info
Acrivastine
CAS:
- 87848-99-5
Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
Formula:C₂₂H₂₄N₂O₂
Purity:99.73% - >99.99%
Color and Shape:Solid
Molecular weight:348.44
Ref: TM-T4551
+ Info
Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
Formula:C₃₇H₄₈F₆N₈O₁₁
Purity:98.54%
Color and Shape:Solid
Molecular weight:894.81
Ref: TM-T7740
+ Info
BML-190
CAS:
- 2854-32-2
BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。
Formula:C₂₃H₂₃ClN₂O₄
Purity:97.70%
Color and Shape:Solid
Molecular weight:426.89
Ref: TM-T6417
+ Info
(±)-Ibipinabant
CAS:
- 362519-49-1
(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.
Formula:C₂₃H₂₀Cl₂N₄O₂S
Purity:99.28% - 99.83%
Color and Shape:Solid
Molecular weight:487.4
Ref: TM-T4654
+ Info
Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
Purity:98%
Color and Shape:Liquid
Molecular weight:N/A
Ref: TM-TP1148L
+ Info
Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
Purity:99.24%
Color and Shape:Liquid
Molecular weight:N/A
Ref: TM-TP1976L
+ Info
BRL 54443
CAS:
- 57477-39-1
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
Formula:C₁₄H₁₈N₂O
Purity:98.07%
Color and Shape:Solid
Molecular weight:230.31
Ref: TM-T2459
+ Info
BIBO3304
CAS:
- 191868-13-0
BIBO3304: Selective NPY Y1 blocker, IC50 of 0.38nM (human), 0.72nM (rat); curbs hunger from NPY/fasting when injected centrally.
Formula:C₂₉H₃₅N₇O₃
Color and Shape:Solid
Molecular weight:529.63
Ref: TM-T26800
+ Info
Ufenamate
CAS:
- 67330-25-0
Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseases
Formula:C₁₈H₁₈F₃NO₂
Purity:99.89%
Color and Shape:Solid
Molecular weight:337.34
Ref: TM-T4966
+ Info
Pergolide mesylate
CAS:
- 66104-23-2
Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.
Formula:C₂₀H₃₀N₂O₃S₂
Purity:99.70%
Color and Shape:White To Off-White Solid
Molecular weight:410.59
Ref: TM-T2226
+ Info
Cutamesine dihydrochloride
CAS:
- 165377-44-6
Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.
Formula:C₂₃H₃₂N₂O₂·2HCl
Purity:99.96%
Color and Shape:Solid
Molecular weight:441.43
Ref: TM-T3597
+ Info
Maropitant
CAS:
- 147116-67-4
Maropitant is a selective neurokinin (NK1) receptor antagonist.
Formula:C₃₂H₄₀N₂O
Purity:97.35% - 99.75%
Color and Shape:Solid
Molecular weight:468.67
Ref: TM-T7209
+ Info
α-MSH
CAS:
- 581-05-5
α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
Formula:C₇₇H₁₀₉N₂₁O₁₉S
Purity:99.10% - 99.67%
Color and Shape:White Powder
Molecular weight:1664.89
Ref: TM-T7813
+ Info
CID 16020046
CAS:
- 834903-43-4
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
Formula:C₂₅H₁₉N₃O₄
Purity:99.03%
Color and Shape:Solid
Molecular weight:425.44
Ref: TM-T4478
+ Info
NIBR189
CAS:
- 1599432-08-2
NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)
Formula:C₂₁H₂₁BrN₂O₃
Purity:97%
Color and Shape:Colourless
Molecular weight:429.31
Ref: TM-T7156
+ Info
PNU 22394 hydrochloride
CAS:
- 15923-42-9
PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
Formula:C₁₃H₁₇ClN₂
Purity:97.83%
Color and Shape:Solid
Molecular weight:236.74
Ref: TM-T23168
+ Info
Alcaftadine
CAS:
- 147084-10-4
Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
Formula:C₁₉H₂₁N₃O
Purity:98% - 98.65%
Color and Shape:Solid
Molecular weight:307.39
Ref: TM-T2533
+ Info
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and
Formula:C₇₆H₁₀₃N₂₁O₁₈S
Purity:99.75%
Color and Shape:Solid
Molecular weight:1630.82
Ref: TM-TP1893L1
+ Info
PAR-2-IN-1
CAS:
- 1690176-75-0
PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
Formula:C₁₂H₁₄ClN₃O₂
Purity:99.75%
Color and Shape:Solid
Molecular weight:267.71
Ref: TM-T8917
+ Info
Bosentan (hydrate)
CAS:
- 157212-55-0
Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.
Formula:C₂₇H₂₉N₅O₆S·H₂O
Purity:99.31% - 99.86%
Color and Shape:White Powder
Molecular weight:569.63
Ref: TM-T6265
+ Info
Bexagliflozin
CAS:
- 1118567-05-7
Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.
Formula:C₂₄H₂₉ClO₇
Purity:98.99% - 99.89%
Color and Shape:Solid
Molecular weight:464.94
Ref: TM-T7217
+ Info
GW 405833
CAS:
- 180002-83-9
GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective
Formula:C₂₃H₂₄Cl₂N₂O₃
Purity:99.82% - 99.93%
Color and Shape:Solid
Molecular weight:447.35
Ref: TM-T7705
+ Info
Epinastine
CAS:
- 80012-43-7
Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.
Formula:C₁₆H₁₅N₃
Purity:99.94%
Color and Shape:Solid
Molecular weight:249.31
Ref: TM-T60366
+ Info
6-fluoro-DL-Tryptophan
CAS:
- 7730-20-3
6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.
Formula:C₁₁H₁₁FN₂O₂
Purity:99.25%
Color and Shape:Off-White Powder
Molecular weight:222.22
Ref: TM-T7694
+ Info
HS 014 acetate(207678-81-7 free base)
HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.
Formula:C₇₃H₉₈N₂₀O₁₉S₂
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1623.83
Ref: TM-TP2015L
+ Info
Sertindole
CAS:
- 106516-24-9
Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).
Formula:C₂₄H₂₆ClFN₄O
Purity:99.87% - 99.92%
Color and Shape:Off-White To Pale Yellow Solid
Molecular weight:440.94
Ref: TM-T5858
+ Info
GLPG2938
CAS:
- 2130996-00-6
GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and
Formula:C₂₀H₁₉F₆N₇O₂
Purity:98.25%
Color and Shape:Solid
Molecular weight:503.4
Ref: TM-T9199
+ Info
Dioxopromethazine hydrochloride
CAS:
- 15374-15-9
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
Formula:C₁₇H₂₀N₂O₂S·HCl
Purity:99.58%
Color and Shape:Solid
Molecular weight:352.88
Ref: TM-T3723
+ Info
Nomifensine
CAS:
- 24526-64-5
Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.
Formula:C₁₆H₁₈N₂
Purity:99.83% - ≥95%
Color and Shape:Solid
Molecular weight:238.33
Ref: TM-T7308
+ Info
A-582941 dihydrochloride
CAS:
- 848591-90-2
A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial
Formula:C₁₇H₂₂Cl₂N₄
Purity:99.55%
Color and Shape:Solid
Molecular weight:353.29
Ref: TM-T22016
+ Info
Elagolix sodium
CAS:
- 832720-36-2
Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
Formula:C₃₂H₂₉F₅N₃NaO₅
Purity:99.71%
Color and Shape:Solid
Molecular weight:653.57
Ref: TM-T5031
+ Info
Bimatoprost
CAS:
- 155206-00-1
Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular
Formula:C₂₅H₃₇NO₄
Purity:98% - >99.99%
Color and Shape:Crystalline Solid
Molecular weight:415.57
Ref: TM-T2538
+ Info
Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct
Formula:C₄₀H₆₇N₇O₁₀
Purity:99.95%
Color and Shape:Solid
Molecular weight:805.9
Ref: TM-TP1085L
+ Info
Chlorphenoxamine
CAS:
- 77-38-3
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Formula:C₁₈H₂₂ClNO
Purity:99.44% - 99.85%
Color and Shape:Solid
Molecular weight:303.83
Ref: TM-T7564
+ Info
UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.
Formula:C₅₂H₆₈N₁₀O₁₄S₂
Purity:99.78%
Color and Shape:Solid
Molecular weight:1121.29
Ref: TM-TP2104L
+ Info
Vorapaxar
CAS:
- 618385-01-6
Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
Formula:C₂₉H₃₃FN₂O₄
Purity:98.77% - 99.93%
Color and Shape:Solid
Molecular weight:492.58
Ref: TM-T7013
+ Info
Octreotide Acetate
CAS:
- 79517-01-4
Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.
Formula:C₅₁H₇₀N₁₀O₁₂S₂
Purity:99.03% - 99.87%
Color and Shape:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised Solid
Molecular weight:1079.3
Ref: TM-T4119
+ Info
Betahistine
CAS:
- 5638-76-6
Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.
Formula:C₈H₁₂N₂
Purity:99.87% - 99.87%
Color and Shape:Yellowish Liquid Liquid Liquid
Molecular weight:136.19
Ref: TM-T4195
+ Info
Sotagliflozin
CAS:
- 1018899-04-1
Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potential
Formula:C₂₁H₂₅ClO₅S
Purity:99% - 99.86%
Color and Shape:Solid
Molecular weight:424.94
Ref: TM-T3547
+ Info
M617 acetate
M617 acetate is a selective agonist of galanin receptor 1 (GAL1).
Formula:C₁₁₂H₁₆₁N₂₉O₂₈
Purity:96.02%
Color and Shape:Solid
Molecular weight:2361.65
Ref: TM-TP1993L
+ Info
HS024
CAS:
- 212370-59-7
HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.
Formula:C₅₈H₇₉N₁₉O₁₀S₂
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1266.5
Ref: TM-TP1898
+ Info
SB-222200
CAS:
- 174635-69-9
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
Formula:C₂₆H₂₄N₂O
Purity:97.13%
Color and Shape:Solid
Molecular weight:380.48
Ref: TM-T16849
+ Info
Guanabenz Acetate
CAS:
- 23256-50-0
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.
Formula:C₈H₈Cl₂N₄·C₂H₄O₂
Purity:99% - 99.66%
Color and Shape:White Solid From Acetonitrile White Solid
Molecular weight:291.13
Ref: TM-T6522