GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purity:98% - 99.9%Color and Shape:SolidMolecular weight:5218.88VKGILS-NH2 Acetate
<p>VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.</p>Formula:C30H58N8O9Purity:98.83%Color and Shape:SolidMolecular weight:674.83Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Formula:C30H27BrN4O3Purity:98.12%Color and Shape:SolidMolecular weight:571.46SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Formula:C17H13N5O2Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:319.32R243
CAS:<p>R243 is CCR8 signaling and chemotaxis inhibitor.</p>Formula:C21H27NO4Purity:99.03%Color and Shape:SolidMolecular weight:357.44Carazolol
CAS:<p>Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.</p>Formula:C18H22N2O2Purity:99% - 99.53%Color and Shape:Yellowish SolidMolecular weight:298.38Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formula:C25H27N3O2SPurity:99.06% - 99.96%Color and Shape:SolidMolecular weight:433.57Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Formula:C12H17NO9Purity:97.32% - 99.97%Color and Shape:SolidMolecular weight:319.27Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Formula:C25H29ClF6N2O3Color and Shape:SolidMolecular weight:554.951-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:<p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>Formula:C9H15N3OPurity:95%Color and Shape:SolidMolecular weight:181.23Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85SAG hydrochloride (912545-86-9(free base))
CAS:<p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>Formula:C28H29Cl2N3OSPurity:99.19% - 99.77%Color and Shape:SolidMolecular weight:526.52Lidamidine Hydrochloride
CAS:Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formula:C11H17ClN4OColor and Shape:SolidMolecular weight:256.73Ablukast
CAS:<p>Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.</p>Formula:C28H34O8Purity:98.58%Color and Shape:SolidMolecular weight:498.56Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Formula:C32H51F3N8O9Purity:99.88%Color and Shape:SolidMolecular weight:748.79D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Formula:C20H23N5Purity:98.82%Color and Shape:SolidMolecular weight:333.43Pentagastrin
CAS:Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormula:C37H49N7O9SPurity:96.98% - 99.49%Color and Shape:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMolecular weight:767.89ACEPROMAZINE MALEATE
CAS:<p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>Formula:C23H26N2O5SPurity:98.87% - 99.51%Color and Shape:Off White Or Yellow Crystalline PowderMolecular weight:442.53Bombesin acetate(31362-50-2 free base)
CAS:<p>Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).</p>Formula:C73H114N24O20SPurity:98.44%Color and Shape:SolidMolecular weight:1679.92Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Formula:C26H29N5O3SPurity:99.49% - 99.843%Color and Shape:SolidMolecular weight:491.61N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Formula:C9H15N3O3Purity:98%Color and Shape:SolidMolecular weight:213.23Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Formula:C36H45NO7Purity:98% - 98.24%Color and Shape:White SolidMolecular weight:603.75Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.495-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurity:99.13%Color and Shape:SolidMolecular weight:280.36Sonidegib
CAS:<p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>Formula:C26H26F3N3O3Purity:98% - 99.97%Color and Shape:SolidMolecular weight:485.5A-381393
CAS:<p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>Formula:C20H24N4Purity:99.00%Color and Shape:SolidMolecular weight:320.43AZD-4818
CAS:<p>AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Formula:C27H32Cl2N2O7Purity:99.01%Color and Shape:SolidMolecular weight:567.46Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Formula:C21H24ClN2NaO4SPurity:99.82%Color and Shape:SolidMolecular weight:458.93Elinzanetant
CAS:<p>Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.</p>Formula:C33H35F7N4O3Purity:98% - 99.13%Color and Shape:SolidMolecular weight:668.64Ropinirole hydrochloride
CAS:<p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>Formula:C16H24N2O·HClPurity:99.87% - 99.98%Color and Shape:Off-White SolidMolecular weight:296.84β-CGRP, human acetate
<p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>Formula:C164H271N51O50S3Purity:99.35%Color and Shape:SolidMolecular weight:3853.46Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formula:C40H42ClN5O7Purity:97.94% - 98.4%Color and Shape:SolidMolecular weight:740.24Diphenhydramine
CAS:<p>Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.</p>Formula:C17H21NOPurity:98.07%Color and Shape:SolidMolecular weight:255.35BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Formula:C59H80N14O13Purity:95.3%Color and Shape:SolidMolecular weight:1193.35Cetirizine Impurity B dihydrochloride
CAS:<p>Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.</p>Formula:C19H23Cl3N2O2Purity:99.24%Color and Shape:SolidMolecular weight:417.76Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84Endothelin-2 (49-69), human
CAS:Endothelin-2 (49-69), human (Human endothelin-2) is a 21-amino acid vasoactive peptide that binds to G-protein-linked transmembrane receptors, ET-RA and ET-RB.Formula:C115H160N26O32S4Purity:98.26%Color and Shape:SolidMolecular weight:2546.92JK184
CAS:<p>JK184 is a potent Hedgehog (Hh) pathway inhibitor.</p>Formula:C19H18N4OSPurity:98.93% - 99.89%Color and Shape:SolidMolecular weight:350.44[D-Phe12,Leu14]-Bombesin acetate
<p>[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Formula:C77H118N22O20Purity:98.41% - 99.14%Color and Shape:SolidMolecular weight:1671.9Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formula:C17H25N3O2S·C4H6O5Purity:99.95%Color and Shape:Pale Yellow SolidMolecular weight:469.55Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.734i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Formula:C16H12ClN3OPurity:99.49%Color and Shape:SolidMolecular weight:297.74Vicriviroc maleate
CAS:<p>Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.</p>Formula:C32H42F3N5O6Purity:98.16% - 98.37%Color and Shape:SolidMolecular weight:649.7Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Formula:C22H23N3O3SPurity:98.77%Color and Shape:SolidMolecular weight:409.5Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33Regadenoson
CAS:<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.35PF-4136309
CAS:PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formula:C29H31F3N6O3Purity:98.85% - 99.47%Color and Shape:SolidMolecular weight:568.59Tripelennamine citrate
CAS:<p>Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.</p>Formula:C22H29N3O7Color and Shape:SolidMolecular weight:447.488SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35LGnRH-III, lamprey acetate(147859-97-0 free base)
<p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>Formula:C61H78N18O16Purity:99.66%Color and Shape:SolidMolecular weight:1319.38Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54Etrasimod
CAS:<p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purity:99.89%Color and Shape:SolidMolecular weight:239.27Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Formula:C18H19N3O·HClPurity:99.78%Color and Shape:White PowderMolecular weight:329.82Diquafosol tetrasodium
CAS:<p>Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear film</p>Formula:C18H22N4Na4O23P4Purity:98.25% - 99.97%Color and Shape:SolidMolecular weight:878.23ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37MRT-81
CAS:<p>MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.</p>Formula:C31H29N3O5SPurity:99.72%Color and Shape:SolidMolecular weight:555.64Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formula:C24H32ClNO3Purity:99.57% - 99.77%Color and Shape:SolidMolecular weight:417.97Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Formula:C36H55F3N8O12SPurity:>99.99%Color and Shape:SolidMolecular weight:880.93NPY 5RA972
CAS:<p>NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist</p>Formula:C21H25N3O2Purity:99.02% - 99.56%Color and Shape:SolidMolecular weight:351.44VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Formula:C38H73N21O10S2HClPurity:>99.99%Color and Shape:SolidMolecular weight:1353.33Mini Gastrin I, human acetate
<p>Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.</p>Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Procaterol hydrochloride hydrate
CAS:Short-acting β2-adrenergic receptor agonist used to treat asthma.Formula:C32H48Cl2N4O7Purity:99.71% - 99.97%Color and Shape:SolidMolecular weight:671.65N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8SBI-115
CAS:<p>SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5</p>Formula:C14H13ClN2O4SPurity:99.53% - 99.78%Color and Shape:SolidMolecular weight:340.78GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formula:C25H29N5OPurity:99.2%Color and Shape:SolidMolecular weight:415.53Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Formula:C46H65N13O11S2Purity:99.65%Color and Shape:SolidMolecular weight:1040.22SB297006
CAS:<p>SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.</p>Formula:C18H18N2O5Purity:99.59%Color and Shape:SolidMolecular weight:342.35AC-55541
CAS:<p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36TS-011
CAS:<p>N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.</p>Formula:C11H14ClN3O2Purity:99.48%Color and Shape:SolidMolecular weight:255.7RE-640
CAS:<p>NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.</p>Formula:C20H16Cl2N4Purity:99.60% - 99.87%Color and Shape:SolidMolecular weight:383.27Litorin acetate(55749-97-8 Free base)
<p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Chlorprothixene
CAS:<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Formula:C23H21F7N4O3Purity:98% - 99.68%Color and Shape:Off-White To Light Yellow Cyrstalline SolidMolecular weight:534.43CCG215022
CAS:<p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>Formula:C26H22FN7O3Purity:97.63% - 99.69%Color and Shape:SolidMolecular weight:499.5Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3Glasdegib
CAS:<p>Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.</p>Formula:C21H22N6OPurity:98.72%Color and Shape:SolidMolecular weight:374.44Siponimod
CAS:<p>Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.</p>Formula:C29H35F3N2O3Purity:97.08% - 99.40%Color and Shape:SolidMolecular weight:516.59GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formula:C28H36N4O2S·HClPurity:99.51%Color and Shape:SolidMolecular weight:529.14BX471
CAS:<p>BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.</p>Formula:C21H24ClFN4O3Purity:98% - 99.94%Color and Shape:SolidMolecular weight:434.89Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formula:C22H26N2O4Purity:98% - 99.9%Color and Shape:SolidMolecular weight:382.45BMS-813160
CAS:<p>BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.</p>Formula:C25H40N8O2Purity:99.66% - 99.79%Color and Shape:SolidMolecular weight:484.64Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21EST64454 hydrochloride
CAS:<p>EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.</p>Formula:C18H23ClF2N4O2Purity:99.15%Color and Shape:SolidMolecular weight:400.85Tolnapersine
CAS:<p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>Formula:C21H26N2OPurity:98%Color and Shape:SolidMolecular weight:322.44idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formula:C20H19F5N2OPurity:99.73%Color and Shape:SolidMolecular weight:398.37Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Formula:C19H23NO3·CH4O3SPurity:99.18% - 99.87%Color and Shape:Tan Or Off-White Cyrstalline SolidMolecular weight:409.5Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81PF-06291874
CAS:<p>PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.</p>Formula:C26H28F3N3O4Purity:99.12% - 99.27%Color and Shape:SolidMolecular weight:503.51Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Formula:C13H16N2O2Purity:98% - 99.89%Color and Shape:Pale Yellow Leaflets From Benzene SolidMolecular weight:232.28Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Formula:C20H26N2O7SPurity:99.86% - 99.9%Color and Shape:SolidMolecular weight:438.49Serotonin hydrochloride
CAS:<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Formula:C10H13ClN2OPurity:98.05% - 99.93%Color and Shape:White To Cream PowderMolecular weight:212.676
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