CymitQuimica logo
Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

Show 34 more subcategories

Found 8595 products of "Metabolism"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Izonsteride

    CAS:
    <p>Izonsteride (LY320236) is a selective and potent 5alpha reductase inhibitor with dual action on the type I and type II isoforms of the enzyme.Izonsteride is</p>
    Formula:C24H26N2OS2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:422.61
  • HTS07545

    CAS:
    <p>HTS07545, an SQOR inhibitor (IC50: 30nM), slows H2S breakdown, researched for heart failure.</p>
    Formula:C22H18N2O3
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:358.39
  • Mopidamol

    CAS:
    <p>Mopidamol (RA 233) is a phosphodiesterase inhibitor, a dipyridamole derivative, with anticancer activity that prevents retinal vascular defects in experimental</p>
    Formula:C19H31N7O4
    Purity:99.05% - 99.78%
    Color and Shape:Solid
    Molecular weight:421.49
  • Xanthine oxidoreductase-IN-4

    CAS:
    <p>Xanthine oxidoreductase-IN-4: oral XOR inhibitor, IC50 of 29.3 nM, potential for hyperuricemia research.</p>
    Formula:C16H15N5O2
    Purity:98.25%
    Color and Shape:Soild
    Molecular weight:309.32
  • Cevoglitazar

    CAS:
    <p>Cevoglitazar (LBM-642) is a PPARɑ agonist and PPARγ agonist. Cevoglitazar potently reduces food intake and body weight in obese mice and cynomolgus monkeys.</p>
    Formula:C27H21F3N2O6S
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:558.53
  • Tanimilast

    CAS:
    <p>Tanimilast (CHF-6001) is a potent PDE4 inhibitor with IC50 of 0.026 nM, used topically for obstructive lung disease.</p>
    Formula:C30H30Cl2F2N2O8S
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:687.54
  • Zifaxaban

    CAS:
    <p>Zifaxaban (TY-602) is an oral selective factor Xa inhibitor with an IC50 of 11.1 nM, highly specific over other serine proteases, used in thrombosis studies.</p>
    Formula:C20H16ClN3O4S
    Purity:97.46% - 99.82%
    Color and Shape:Solid
    Molecular weight:429.88
  • Fluorobexarotene

    CAS:
    <p>Fluorobexarotene, a potent RXR agonist, has 75% higher affinity than Bexarotene with Ki of 12 nM and EC50 of 43 nM for RXRα.</p>
    Formula:C24H27FO2
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:366.47
  • BMS 753

    CAS:
    <p>BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).</p>
    Formula:C21H21NO4
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:351.4
  • MAO-B-IN-8

    CAS:
    <p>MAO-B-IN-8 is a highly potent and reversible inhibitor of monoamine oxidase-B (MAO-B), which also exhibits inhibitory effects on the microglial production of</p>
    Formula:C18H16O6
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:328.32
  • Malic enzyme inhibitor ME1

    CAS:
    <p>Malic enzyme inhibitor ME1 (ME1) is a specific inhibitor of Malic enzyme (IC50 = 0.15 μM). Malic enzyme inhibitor ME1 reduces cell viability/metabolic activity.</p>
    Formula:C20H21N3O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:351.4
  • Vatanidipine

    CAS:
    <p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>
    Formula:C41H42N4O6
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:686.8
  • PD173212

    CAS:
    <p>PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).</p>
    Formula:C38H53N3O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:599.85
  • KT182

    CAS:
    <p>KT182 is a selective and  potent inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells.</p>
    Formula:C27H26N4O2
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:438.52
  • uk-50001

    CAS:
    <p>UK-50001 is a PDE4 inhibitor for treating inflammation, allergies, respiratory issues, and wounds.</p>
    Formula:C26H24F3N3O4
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:499.48
  • UCM05

    CAS:
    <p>UCM05 is a potent FASN and FtsZ inhibitor active against HER2+ breast cancer and B. subtilis (MIC 100 μM), but not E. coli.</p>
    Formula:C24H16O10
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:464.38
  • CYP1B1-IN-5

    CAS:
    <p>CYP1B1-IN-5: selective CYP1B1 inhibitor, IC50 = 4.7 nM, useful for metabolism disease research.</p>
    Formula:C14H8INO2
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:349.12
  • 4-Hydroxymephenytoin

    CAS:
    <p>4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.</p>
    Formula:C12H14N2O3
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:234.25
  • AChE/BChE/MAO-B-IN-1

    CAS:
    <p>AChE/BChE/MAO-B-IN-1 is a reversible, non-time-dependent inhibitor of AChE, BChE and MAO-B that crosses the blood-brain barrier and exhibits inhibitory effects</p>
    Formula:C20H24N2O2
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:324.42
  • PTP1B-IN-3

    CAS:
    <p>PTP1B-IN-3 是一种具有有选择性和高效性的 PTP1B 抑制剂,具有抗癌活性,抑制 PTP1B 和 TCPTP 。PTP1B-IN-3 可用于研究糖尿病。</p>
    Formula:C12H7BrF2NO3P
    Purity:99.31% - 99.97%
    Color and Shape:Solid
    Molecular weight:362.06
  • BAY-4931

    CAS:
    <p>BAY-4931 is a powerful, covalent, and selective inverse-agonist of PPARγ, exhibiting an IC50 value of 0.17 nM.</p>
    Formula:C22H16ClN3O4
    Purity:99.47%
    Color and Shape:Soild
    Molecular weight:421.83
  • SERCA2a activator 1

    CAS:
    <p>SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.</p>
    Formula:C32H29N3O4S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:551.66
  • AZD-0284

    CAS:
    <p>AZD-0284 is an inverse agonist of the nuclear receptor RORγ. In development for the treatment of plaque psoriasis vulgaris and respiratory tract disorders[1].</p>
    Formula:C21H18F6N2O5S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:524.43
  • PDE4B-IN-2

    CAS:
    <p>PDE4B-IN-2 (A 33), an oral PDE4B inhibitor, IC50: 15 nM; less potent on PDE4D (IC50: 1.7 µM), has anti-inflammatory properties.</p>
    Formula:C19H18ClN3O2S
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:387.88
  • PKUMDL-WQ-2101

    CAS:
    <p>PKUMDL-WQ-2101 is a selective allosteric inhibitor of phosphoglycerate dehydrogenase with anti-tumor activity.</p>
    Formula:C14H11N3O6
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:317.25
  • Lecimibide

    CAS:
    <p>Lecimibide (DuP 128) is a potent and selective inhibitor of acyl coenzyme A: cholesterol acyltransferase (ACAT), which can be used to study diseases due to high</p>
    Formula:C34H40F2N4OS
    Purity:99.44% - 99.87%
    Color and Shape:Solid
    Molecular weight:590.77
  • 5-LOX-IN-1

    CAS:
    <p>5-LOX-IN-1 is a 5-Lipoxygenase (5-LOX) inhibitor (IC50: 2.3 μM).5-LOX-IN-1 can be used for cancer research.</p>
    Formula:C20H18N2O2S
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:350.43
  • Crobenetine

    CAS:
    <p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>
    Formula:C25H33NO2
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:379.54
  • Ch55

    CAS:
    <p>Ch55, a potent HL60 cell differentiator (EC50=200nM), binds well to RAR-α/β, useful for cancer research.</p>
    Formula:C24H28O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:364.48
  • Isolithocholic Acid

    CAS:
    <p>Isolithocholic Acid, a bile acid isomer, forms through microbial metabolism of Lithocholic acid or its 3α-sulfate.</p>
    Formula:C24H40O3
    Purity:99.56% - 99.84%
    Color and Shape:Solid
    Molecular weight:376.57
  • Dasantafil

    CAS:
    <p>Dasantafil (SCH446132) is a small molecule phosphodiesterase-5A (PDE5A) inhibitor used to treat genitourinary disorders and study erectile dysfunction.</p>
    Formula:C22H28BrN5O5
    Purity:99.4% - 99.50%
    Color and Shape:Solid
    Molecular weight:522.39
  • hCAII-IN-9

    CAS:
    <p>hCAII-IN-9 inhibits hCA II/IX/XII with IC50s of 1.18, 0.17, 2.99 μM; not BBB permeable.</p>
    Formula:C15H16ClN3O5S2
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:417.89
  • MK-0873

    CAS:
    <p>MK-0873 is a novel and potent selective phosphodiesterase 4 (PDE4) inhibitor.</p>
    Formula:C25H18N4O3
    Purity:98.40%
    Color and Shape:Solid
    Molecular weight:422.44
  • EWP 815

    CAS:
    <p>EWP 815, a disulfiram analog, inhibits Ins(1,4)P2, Ins(1,4,5)P3 phosphatases, and dopamine β-hydroxylase.</p>
    Formula:C12H22N4S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.59
  • PHGDH-IN-3

    CAS:
    <p>PHGDH-IN-3, an oral PHGDH blocker with 2.8 μM IC50, may help in cancer research.</p>
    Formula:C24H18FN3O4S2
    Purity:97.24% - 98.55%
    Color and Shape:Solid
    Molecular weight:495.55
  • OSMI-4

    CAS:
    <p>OSMI-4 is a low nanomolar O-GlcNAc transferase (OGT) inhibitor that can be used to study OGT inhibition in different human cell lines.Cost-effective and quality-assured.</p>
    Formula:C27H26ClN3O7S2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:604.09
  • TDO-IN-1

    CAS:
    <p>TDO-IN-1 is a tryptophan 2,3-dioxygenase (TDO) inhibitor with antitumor activity that acts by reversing local immune tolerance in tumor tissues.</p>
    Formula:C16H13F3N4O2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:350.3
  • Atibeprone

    CAS:
    <p>Atibeprone is a MAO-B inhibitor with antidepressant activity for the study of Parkinson's disease.</p>
    Formula:C17H18N2O3S
    Purity:99.18% - 99.86%
    Color and Shape:Solid
    Molecular weight:330.4
  • Nanterinone

    CAS:
    <p>Nanterinone: oral phosphodiesterase inhibitor, improves acute heart failure hemodynamics.</p>
    Formula:C15H15N3O
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:253.3
  • CYP1B1-IN-4

    CAS:
    <p>CYP1B1-IN-4: 2,4-diarylthiazole, selective CYP1B1 inhibitor (IC50=0.2 nM), low cytotoxicity, stable in liver microsomes.</p>
    Formula:C18H14N2O2S
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:322.38
  • Troriluzole

    CAS:
    <p>Troriluzole is a glutamate modulator with anticancer activity and is used in the study of spinocerebellar ataxia.</p>
    Formula:C15H16F3N5O4S
    Purity:97.14%
    Color and Shape:Solid
    Molecular weight:419.38
  • Farglitazar

    CAS:
    <p>Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer used in the study of diabetes.</p>
    Formula:C34H30N2O5
    Purity:99.4% - 99.52%
    Color and Shape:Solid
    Molecular weight:546.61
  • CM037

    CAS:
    <p>CM037 (A-37) is a selective ALDH1A1 (acetaldehyde dehydrogenase 1A1) inhibitor (IC50; 4.6 µM) with antitumor activity and may be used in studies to eliminate</p>
    Formula:C21H25N3O3S2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:431.57
  • C75

    CAS:
    <p>C75 is an inhibitor synthetic fatty-acid synthase (FASN) and inhibits prostate cancer cells PC3 (IC50: 35 μM).</p>
    Formula:C14H22O4
    Purity:98.84% - >99.99%
    Color and Shape:Solid
    Molecular weight:254.32
  • IPN60090

    CAS:
    <p>IPN60090: potent oral GLS1 inhibitor, IC50 of 31 nM, potential for anticancer and immunomodulation.</p>
    Formula:C24H27F3N8O3
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:532.52
  • Qc1

    CAS:
    <p>Qc1 is an inhibitor of threonine dehydrogenase (TDH) inhibitor and can be used in studies about metabolic diseases.</p>
    Formula:C23H16F3N3O2S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:455.45
  • S-2474

    CAS:
    <p>S-2474, an inhibitor of COX-2 and 5-lipoxygenase, has anti-inflammatory and neuroprotective activities, and inhibits cell death.</p>
    Formula:C20H31NO3S
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:365.53
  • AGN 196996

    CAS:
    <p>AGN 196996: strong RARα inhibitor (Ki: 2 nM), weak for RARβ/γ (Ki: 1087/8523 nM).</p>
    Formula:C24H20BrNO5
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:482.32
  • EMD-503982

    CAS:
    <p>EMD-503982 is a potential Factor Xa and Factor VIIa inhibitor with anticancer activity for the study of thromboembolic and neurologic diseases.</p>
    Formula:C22H23ClN4O5
    Purity:97.09% - 99.81%
    Color and Shape:Solid
    Molecular weight:458.90
  • Fumarate hydratase-IN-1

    CAS:
    <p>Fumarate hydratase-IN-1 is a cell-permeable fumarate hydratase inhibitor with antiproliferative activity and can be used to study cellular activity.</p>
    Formula:C27H30N2O4
    Purity:98.96% - 99.49%
    Color and Shape:Solid
    Molecular weight:446.54
  • Utreloxastat

    CAS:
    <p>Utreloxastat (PTC857) is a novel 15-lipoxygenase inhibitor that can be used to study amyotrophic lateral sclerosis<br>.</p>
    Formula:C18H28O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:276.41
  • Carbonic anhydrase inhibitor 6

    CAS:
    <p>Carbonic anhydrase inhibitor 6 is an hCA inhibitor that inhibits hCA IX, hCA II, hCA XII, and hCA I. It is used in the study of lupus erythematosus.</p>
    Formula:C26H25N3O5S
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:491.56
  • Cholesterol 24-hydroxylase-IN-1

    CAS:
    <p>Cholesterol 24-hydroxylase-IN-1 is a cholesterol 24-hydroxylase (CH24H or CYP46A1) inhibitor used in the study of neurological disorders such as epilepsy.</p>
    Formula:C17H23N5O
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:313.40
  • Giripladib

    CAS:
    <p>Giripladib (PLA695/PLX-695) blocks radiation-boosted phosphorylation of ERK and Akt in endothelial cells.</p>
    Formula:C41H36ClF3N2O4S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:745.25
  • AMG-1694

    CAS:
    <p>AMG-1694 disrupts GK-GKRP complex, enhancing GK activity with 7 nM IC50; normalizes glucose in diabetic rodents without affecting normoglycemic animals.</p>
    Formula:C23H30F3N3O4S2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:533.63
  • Chloramphenicol succinate

    CAS:
    <p>Chloramphenicol succinate is a bacteriostatic antibiotic. CPSA is a competitive substrate and inhibitor of succinate dehydrogenase (SDH),can be oxidized by.</p>
    Formula:C15H16Cl2N2O8
    Purity:95.32%
    Color and Shape:Physical Description White Powder (Ntp 1992)
    Molecular weight:423.2
  • Pradefovir

    CAS:
    <p>Pradefovir (Remofovir) is a prodrug for chronic HBV, converting to PMEA in the liver with a Km of 60 μM and clearance of 359 ml/min.</p>
    Formula:C17H19ClN5O4P
    Purity:97.50%
    Color and Shape:Solid
    Molecular weight:423.79
  • G6PD activator AG1

    CAS:
    <p>G6PD activator AG1 is a G6PD agonist that promotes G6PD oligomerization to a catalytically competent form.</p>
    Formula:C24H30N4S2
    Purity:98.38% - 99.51%
    Color and Shape:Solid
    Molecular weight:438.65
  • Autotaxin-IN-3

    CAS:
    <p>Autotaxin-IN-3 is an inhibitor of Autotaxin (IC50 = 2.4 nM) which is responsible for the increase in lysophosphatidic acid in ascites and plasma.</p>
    Formula:C22H21N9O2
    Purity:99.54% - 99.79%
    Color and Shape:Solid
    Molecular weight:443.46
  • Luciferase-IN-1

    CAS:
    <p>Luciferase-IN-1 is a luciferase inhibitor that can be used to study bacterial and fungal infections.</p>
    Formula:C15H14N2S
    Purity:97.84%
    Color and Shape:Solid
    Molecular weight:254.35
  • hCAI/II-IN-6

    CAS:
    <p>hCAI/II-IN-6 is a selective and orally active inhibitor of human carbonic anhydrase (CA).</p>
    Formula:C19H24N4O3S
    Purity:97.07%
    Color and Shape:Solid
    Molecular weight:388.48
  • Salnacedin

    CAS:
    <p>Salnacedin (G-201) treats immune, skin, and musculoskeletal issues, suitable for acne, dermatitis, and psoriasis research.</p>
    Formula:C12H13NO5S
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:283.3
  • CX-157

    CAS:
    <p>CX-157 (KP 157) is a novel monoamine oxidase-A (MAO-A) inhibitor for the study of depression-like neurological disorders and cancer.</p>
    Formula:C14H8F4O4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:348.27
  • ALDH1A3-IN-2

    CAS:
    <p>ALDH1A3-IN-2 is a potent ALDH1A3 inhibitor with an IC50 of 0.30 μM.ALDH1A3-IN-2 has potential for cancer disease research.</p>
    Formula:C13H17NO
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:203.28
  • IQB-782

    CAS:
    <p>IQB-782 is a mucolytic agent with mucolytic expectorant activity for the study of obstructive lung disease.</p>
    Formula:C4H9N3O2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:163.2
  • PC945

    CAS:
    <p>PC945 (Opelconazole) is an antifungal compound that inhibits CYP51A/CYP51B and can be used to study fungal infections of the lungs.</p>
    Formula:C38H37F3N6O3
    Purity:98.89% - 99.37%
    Color and Shape:Solid
    Molecular weight:682.73
  • Lifarizine

    CAS:
    <p>Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.</p>
    Formula:C29H32N4
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:436.59
  • RPR107393 free base

    CAS:
    <p>NVP-BAG956 (BAG956) is a PI3K/PDK inhibitor that inhibits PI3Kδ, and can be used to study melanoma.</p>
    Formula:C22H22N2O
    Purity:99.13% - 99.57%
    Color and Shape:Solid
    Molecular weight:330.42
  • Cronidipine

    CAS:
    <p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>
    Formula:C30H32ClN3O8
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:598.04
  • IGP-1

    CAS:
    <p>iGP-1 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>
    Formula:C17H15N3O3
    Purity:99.12% - 99.15%
    Color and Shape:Solid
    Molecular weight:309.32
  • Ibiglustat (L-Malic acid)

    CAS:
    <p>Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.</p>
    Formula:C24H30FN3O7S
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:523.57
  • Indeglitazar

    CAS:
    <p>Indeglitazar (PPM 204) is orally available pan-agonist of PPAR (PPAR subtypes alpha (α), delta (δ), and gamma (γ)).</p>
    Formula:C19H19NO6S
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:389.42
  • IHVR-17028

    CAS:
    <p>IHVR-17028 is a potent broad-spectrum ERα-glucosidase I (α-glucosidase? I) inhibitor with IC50 of 0.24 μM and antiviral activity.</p>
    Formula:C23H44N2O5
    Purity:97.90%
    Color and Shape:Solid
    Molecular weight:428.61
  • MM 11253

    CAS:
    <p>MM 11253 is a RARγ antagonist with IC50 of 44nM.</p>
    Formula:C28H30O2S2
    Purity:99.41%
    Color and Shape:Solid
    Molecular weight:462.67
  • Dirlotapide

    CAS:
    <p>Dirlotapide (CP742033), an intestinal MTP inhibitor, cuts weight in diabetic dogs by lowering food intake and raising peptide YY.</p>
    Formula:C40H33F3N4O3
    Purity:98.47% - 99.62%
    Color and Shape:Solid
    Molecular weight:674.71
  • NecroX-5

    CAS:
    <p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>
    Formula:C27H39N3O9S3
    Purity:99.944%
    Color and Shape:Solid
    Molecular weight:645.81
  • K-111

    CAS:
    <p>K-111 is a PPAR alpha agonist. K-111 improves insulin resistance, reducing bodyweight, and ameliorating atherogenic dyslipidemia.</p>
    Formula:C18H25Cl3O2
    Purity:99.64% - 99.88%
    Color and Shape:Solid
    Molecular weight:379.75
  • Diproteverine HCl

    CAS:
    <p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>
    Formula:C26H36ClNO4
    Purity:98.55% - 99.84%
    Color and Shape:Solid
    Molecular weight:462.02
  • JJKK 048

    CAS:
    <p>JJKK 048 is a potent and selective MAGL inhibitor.</p>
    Formula:C23H22N4O5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:434.44
  • BPDA2

    CAS:
    <p>BPDA2 selectively inhibits SHP2 (IC50=92nM) over SHP1/1B (33.39/40.71μM), curbs RTKs, and hampers SHP2-driven breast cancer cell traits.</p>
    Formula:C24H30O5
    Purity:99.80%
    Color and Shape:Solid
    Molecular weight:398.49
  • NAAD sodium salt

    CAS:
    <p>NAAD sodium salt (NAAD Na salt) is a substrate of nicotinamide adenine dinucleotide synthase and can be used in studies about the specificity and kinetics of</p>
    Formula:C21H25N6NaO15P2
    Purity:98.6% - 99.87%
    Color and Shape:Solid
    Molecular weight:686.4
  • 11-cis-Vaccenyl acetate

    CAS:
    <p>11-cis-Vaccenyl acetate ((Z)-Octadec-11-enyl acetate) activates olfactory neurons located in the T1 sensilla on the antenna and mediates aggregation behavior in</p>
    Formula:C20H38O2
    Purity:96.53% - 99.95%
    Color and Shape:Liquid
    Molecular weight:310.51
  • A-69412

    CAS:
    <p>A-69412 is a reversible 5-lipoxygenase inhibitor, potentially treating ulcerative colitis and asthma.</p>
    Formula:C7H10N2O3
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:170.17
  • LY 517717

    CAS:
    <p>LY 517717 is an orally active inhibitor of coagulation factor Xa with antithrombotic activity for the study of venous thromboembolism (VTE).</p>
    Formula:C27H33N5O2
    Purity:99.77% - 99.88%
    Color and Shape:Solid
    Molecular weight:459.58
  • JNJ-42226314

    CAS:
    <p>JNJ-42226314 is a MAGL inhibitor with anti-injury effects and has shown efficacy in neuropathic pain and inflammatory pain models.</p>
    Formula:C26H24FN5O2S
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:489.56
  • Imanixil

    CAS:
    <p>Imanixil boosts LDLR, cuts cholesterol and VLDL production, reducing atherosclerosis.</p>
    Formula:C17H17F3N6O2
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:394.35
  • DS16570511

    CAS:
    <p>DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.</p>
    Formula:C30H25Cl2N3O4
    Purity:98.34% - 98.45%
    Color and Shape:Solid
    Molecular weight:562.44
  • AC-261066

    CAS:
    <p>AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.</p>
    Formula:C17H20FNO4S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:353.41
  • SR2211

    CAS:
    <p>SR2211 is a specific modulator and an inverse agonist of RORγ(IC50 = 320 nM, Ki = 105 nM).</p>
    Formula:C26H24F7N3O
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:527.48
  • Xanthine oxidoreductase-IN-3

    CAS:
    <p>Xanthine oxidoreductase-IN-3, an oral XOR inhibitor with IC50 of 26.3 nM, is useful for acute hyperuricemia research.</p>
    Formula:C14H10ClN5O
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:299.72
  • sEH inhibitor-7

    CAS:
    <p>sEH inhibitor-7 is a soluble epoxide hydrolase (sEH) inhibitor that inhibits sEH in human and mouse with IC 50 s of 6.2 μM and 0.15 μM, respectively.</p>
    Formula:C15H21NO2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:247.33
  • Xanthine oxidoreductase-IN-5

    CAS:
    <p>Xanthine oxidoreductase-IN-5: oral XOR inhibitor; IC50 55 nM; for acute hyperuricemia research.</p>
    Formula:C17H17N5O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:323.35
  • PKM2 activator 2

    CAS:
    <p>PKM2 activator 2 is a pyruvate kinase M2 (PKM2) activator with an AC 50 value of 66 nM.PKM2 activator 2 has anti-tumor proliferative properties and attenuates</p>
    Formula:C20H18F2N2O4S2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:452.49
  • CYP1B1-IN-1

    CAS:
    <p>CYP1B1-IN-1 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with potential anticancer and antitumor activity for breast cancer research.</p>
    Formula:C19H11ClO2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:306.74
  • IDH2R140Q-IN-2

    CAS:
    <p>IDH2R140Q-IN-2 is an IDH2R140Q inhibitor indicated for the study of acute myeloid leukaemia (AML).</p>
    Formula:C21H18F6N6O
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:484.4
  • NCGC 607

    CAS:
    <p>NCGC 607 is a a noninhibitory chaperone of glucocerebrosidase (GCase).</p>
    Formula:C24H22IN3O4
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:543.35
  • JNJ-40355003

    CAS:
    <p>JNJ-40355003 is a FAAH inhibitor that increases plasma levels of fatty acid amides in rats, dogs, and crabs.</p>
    Formula:C23H23ClN4O2
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:422.91
  • Esuprone

    CAS:
    <p>Esuprone (LU-43839) is a novel reversible and highly selective MAO-A inhibitor with anticonvulsant activity for the treatment of depression.</p>
    Formula:C13H14O5S
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:282.31
  • Clopimozide

    CAS:
    <p>Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.</p>
    Formula:C28H28ClF2N3O
    Purity:98.19% - >99.99%
    Color and Shape:Solid
    Molecular weight:495.99
  • Filaminast

    CAS:
    <p>Filaminast (UNII-CDD69JC61J) is an analog of a phosphodiesterase 4 inhibitor (PDE4 inhibitor) and roliplam, which is used as an anti-asthma drug.</p>
    Formula:C15H20N2O4
    Purity:98.53% - 98.93%
    Color and Shape:Solid
    Molecular weight:292.33
  • Ladostigil

    CAS:
    <p>Ladostigil is an oral cholinesterase &amp; MAO-B inhibitor used for depression and Alzheimer's studies.</p>
    Formula:C16H20N2O2
    Purity:97.48%
    Color and Shape:Solid
    Molecular weight:272.34
  • Dalvastatin

    CAS:
    <p>Dalvastatin (RG-12561) is an orally available inhibitor of HMG-CoA reductase and cholesterol-lowering synthesis.Dalvastatin competitively inhibits rat hepatic</p>
    Formula:C24H31FO3
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:386.5
  • GAC0003A4

    CAS:
    <p>GAC0003A4 is an LXR inverse agonist with antitumor activity for the study of advanced pancreatic cancer and other recalcitrant malignancies.</p>
    Formula:C20H24N2O3
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:340.42
  • ML 209

    CAS:
    <p>ML-209 is an antagonist of retinoic acid receptor-related orphan receptor γt (RORγt; IC50= 1.1 μM in a reporter assay).1It inhibits RORγt-induced transcription</p>
    Formula:C25H31NO6
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:441.52
  • LDL-IN-3

    CAS:
    <p>LDL-IN-3 shows anti-atherosclerotic and antioxidant activities.</p>
    Formula:C24H36O3Si
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:400.63
  • CYP4A11/CYP4F2-IN-1

    CAS:
    <p>CYP4A11/CYP4F2-IN-1 is a cytochrome P450 (CYP) 4A11 and CYP4F2 inhibitor for the study of kidney disease and cardiovascular disease.</p>
    Formula:C15H15N3OS
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:285.36
  • Aleplasinin

    CAS:
    <p>Aleplasinin (PAZ 417) is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolytic</p>
    Formula:C28H27NO3
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:425.52
  • IMPDH2-IN-2

    CAS:
    <p>IMPDH2-IN-2 is an IMPDH inhibitor with antimicrobial activity and potential anti-tuberculosis activity for the study of inflammation and immune dysfunction.</p>
    Formula:C21H15Cl2N3O3
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:428.27
  • Acetyl-L-carnitine

    CAS:
    <p>Acetyl-L-carnitine, an amino-acid supplement, crosses the blood-brain barrier to aid in neuroinflammation and Alzheimer's.</p>
    Formula:C9H17NO4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:203.24
  • Didesethyl chloroquine

    CAS:
    <p>Didesethyl chloroquine, a chloroquine metabolite, is an effective myocardial inhibitor and antimalarial.</p>
    Formula:C14H18ClN3
    Purity:98.11%
    Color and Shape:Solid
    Molecular weight:263.77
  • ARRY-403

    CAS:
    <p>ARRY-403 is a novel glucokinase activator that reduces fasting and postprandial blood glucose in patients with type 2 diabetes.</p>
    Formula:C20H18N6O3S2
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:454.52
  • Sultiame

    CAS:
    <p>Sultiame is an inhibitor of carbonic anhydrase. Sultiame can be used in antiepileptic research.</p>
    Formula:C10H14N2O4S2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:290.36
  • PDE IV-IN-1

    CAS:
    <p>PDE IV-IN-1 is a potent phosphodiesterase 4 (PDE4) inhibitor with anti-inflammatory activity for the treatment of asthma, chronic obstructive pulmonary disease</p>
    Formula:C20H23ClN4O2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:386.88
  • Clozic

    CAS:
    <p>Clozic (ICI 55897) exhibits reversible anti-proliferative effects and can be used in studies about serving as a potential anti-arthritic agent.</p>
    Formula:C17H17ClO3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:304.77
  • Imigliptin

    CAS:
    <p>Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.</p>
    Formula:C21H24N6O
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:376.46
  • Lauroyl lysine

    CAS:
    <p>Lauroyl lysine (N6-Lauroyl-L-lysine) functions as skin and hair conditioning agents and as surfactants-cleansing agents in personal care products.</p>
    Formula:C18H36N2O3
    Purity:99.18%
    Color and Shape:White To Off-White Solid With Characteristic Faint Odor
    Molecular weight:328.49
  • HSD-016

    CAS:
    <p>HSD-016: Oral 11β-HSD1 inhibitor, active in humans, mice, rats (IC50: 11, 1, 8 nM), potential for type 2 diabetes research.</p>
    Formula:C21H21F7N2O3S
    Purity:99.40% - >99.99%
    Color and Shape:Solid
    Molecular weight:514.46
  • DSM421

    CAS:
    <p>DSM421 (DSM-421) is a dihydrodehydrogenase inhibitor (DHODH) that is in preclinical development as a potential treatment option for malaria and has shown</p>
    Formula:C14H11F5N6
    Purity:98.23% - 99.82%
    Color and Shape:Solid
    Molecular weight:358.27
  • Bupicomide

    CAS:
    <p>Bupicomide is a dopamine β-hydroxylase inhibitor with antihypertensive and vasodilatory activity and may be used in the study of hypertension.</p>
    Formula:C10H14N2O
    Purity:99.84% - >99.99%
    Color and Shape:Solid
    Molecular weight:178.23
  • Tigulixostat

    CAS:
    <p>Tigulixostat (LC350189) is a novel xanthine oxidase inhibitor (XOI) that reduces uric acid production and may be used to study gout-related diseases.</p>
    Formula:C16H14N4O2
    Purity:98.22% - 99.71%
    Color and Shape:Solid
    Molecular weight:294.31
  • AM 374

    CAS:
    <p>AM 374 (HDSF), a fatty acid amide hydrolase (FAAH) inhibitor, demonstrates the capacity to inhibit amidase activity, boasting an IC50 value of 13 nM.</p>
    Formula:C16H33FO2S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:308.5
  • SAK3

    CAS:
    <p>SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.</p>
    Formula:C20H23N3O4
    Purity:98.37% - 99.43%
    Color and Shape:Solid
    Molecular weight:369.41
  • Olorofim

    CAS:
    <p>Olorofim(F-901318)is a new selective antifungal compound that inhibits Aspergillus fumigatus DHODH (IC50: 44 nM). Cost-effective and quality-assured.</p>
    Formula:C28H27FN6O2
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:498.55
  • BRD7389

    CAS:
    <p>BRD7389 is an inhibitor of RSK family kinase with IC50s of 1.5 μM, 2.4 μM, and 1.2 μM for RSK1, RSK2, and RSK3, respectively.</p>
    Formula:C24H18N2O2
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:366.41
  • AA 2379

    CAS:
    <p>N6-Allyladenosine (N Allyladenosine) is a nucleoside analog with antimicrobial activity and anticancer activity.</p>
    Formula:C15H23N5O4
    Purity:97.78% - 98.87%
    Color and Shape:Solid
    Molecular weight:337.37
  • Lidorestat

    CAS:
    <p>Lidorestat (IDD-676) is an aldose reductase inhibitor (IC50: 5 nM) with effective, selective and oral activity.</p>
    Formula:C18H11F3N2O2S
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:376.35
  • L-Threonine derivative-1

    CAS:
    <p>L-Threonine derivative-1 is acetylsalicylic acid-L-threonine ester with potential analgesic activity.</p>
    Formula:C13H15NO6
    Purity:97.03% - 98.91%
    Color and Shape:Solid
    Molecular weight:281.26
  • AICAR monophosphate

    CAS:
    <p>AICAR monophosphate (Aica ribonucleotide) is a purine precursor with antineoplastic activity and can be used in studies about type 2 diabetes.</p>
    Formula:C9H15N4O8P
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:338.21
  • Verofylline

    CAS:
    <p>Verofylline (Verofyllinum) is an orally available, long-acting, multiacting, methylxanthine-substituted bronchodilator with inhibitory effects on PDE4 for the</p>
    Formula:C12H18N4O2
    Purity:98.33% - 98.83%
    Color and Shape:Solid
    Molecular weight:250.3
  • Benitrobenrazide

    CAS:
    <p>Benitrobenrazide (Hexokinase 2 inhibitor 1) is a novel orally available hexokinase 2 (HK2) inhibitor with anticancer and antitumor activity for cancer research.</p>
    Formula:C14H11N3O6
    Purity:96.87%
    Color and Shape:Solid
    Molecular weight:317.25
  • Isomazole

    CAS:
    <p>Isomazole is a novel orally available phosphodiesterase (PDE) inhibitor with calcium-sensitizing properties that inhibits PDE3 and PDE4.</p>
    Formula:C14H13N3O2S
    Purity:98.66%
    Color and Shape:Solid
    Molecular weight:287.34
  • Dovramilast

    CAS:
    <p>Dovramilast (CC-11050) is a PDE4 inhibitor that reduces the production of pro-inflammatory mediators in lupus erythematosus.</p>
    Formula:C24H28N2O6S
    Purity:98.75% - 99.62%
    Color and Shape:Solid
    Molecular weight:472.55
  • Nampt activator-2

    CAS:
    <p>Nampt activator-2: Potent NAMPT activator (EC50: 0.023 μM), binds CYP2C9 (0.060 μM), 2D6 (0.41 μM), 2C19 (0.59 μM); useful in metabolic disease research.</p>
    Formula:C17H15ClN4O3S
    Purity:98.30% - 98.33%
    Color and Shape:Solid
    Molecular weight:390.84
  • MLS000544460

    CAS:
    <p>MLS000544460 is a highly selective and reversible Eya2 phosphatase inhibitor (Kd: 2.0 μM, IC50: 4 μM).MLS000544460 exhibits inhibitory effects on Eya2</p>
    Formula:C17H12FN3O2S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:341.36
  • GSK205

    CAS:
    <p>GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.</p>
    Formula:C24H25BrN4S
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:481.45
  • JNJ-DGAT2-A

    CAS:
    <p>JNJ-DGAT2-A, a specific inhibitor of DGAT2(IC50 = 0.14 μM), can be used in studies about the synthesis of triglycerides.</p>
    Formula:C24H16BrFN4O2S
    Purity:98.3%
    Color and Shape:Solid
    Molecular weight:523.38
  • Allopurinol riboside

    CAS:
    <p>Allopurinol riboside, an allopurinol metabolite, inhibits purine nucleoside phosphorylase in parasites with a Ki of 277 μM.</p>
    Formula:C10H12N4O5
    Purity:99.46% - 99.73%
    Color and Shape:Solid
    Molecular weight:268.23
  • BAY-0069

    CAS:
    <p>BAY-0069 is a potent and selective PPARγ transactivator that inhibits human PPARγ and murine PPARγ with IC50s of 6.3 nM and 24 nM, respectively.BAY-0069 can be</p>
    Formula:C22H16BrN3O4
    Purity:99.41%
    Color and Shape:Soild
    Molecular weight:466.28
  • 5-ALA benzyl ester hydrochloride

    CAS:
    <p>5-ALA benzyl ester hydrochloride: a photodetection agent that promotes PPIX in colon cancer cells.</p>
    Formula:C12H16ClNO3
    Purity:98.39% - 99.38%
    Color and Shape:Solid
    Molecular weight:257.71
  • PBRM

    CAS:
    <p>PBRM (17β-HSD1-IN-2) is a selective covalent inhibitor of 17β-HSD1, used in breast cancer and endometriosis research.</p>
    Formula:C28H34BrNO2
    Purity:99.56% - 99.59%
    Color and Shape:Solid
    Molecular weight:496.48
  • NG-497

    CAS:
    <p>NG-497, a selective inhibitor of human ATGL, blocks lipolysis in adipocytes and aids cancer research.</p>
    Formula:C18H21NO4
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:315.36
  • AZ3976

    CAS:
    <p>AZ3976 is an inhibitor of PAI-1 with an IC50 of 16 μM in a plasma clot lysis assay. AZ3976 displays profibrinolytic activities.</p>
    Formula:C15H19N5O3
    Purity:98.14%
    Color and Shape:Solid
    Molecular weight:317.34
  • Carbazeran

    CAS:
    <p>Carbazeran (UK-31,557) is an inhibitor of PDE2 and PDE3 and can be used for studies about metabolic diseases.</p>
    Formula:C18H24N4O4
    Purity:99.3%
    Color and Shape:Solid
    Molecular weight:360.41
  • Lonapalene

    CAS:
    <p>Lonapalene is a topically effective inhibitor of 5-lipoxygenase.</p>
    Formula:C16H15ClO6
    Purity:98.67% - 99.33%
    Color and Shape:Solid
    Molecular weight:338.74
  • Libenzapril

    CAS:
    <p>Libenzapril (CGS 16617) is a potent angiotensin-converting enzyme inhibitor used to study myocardial injury.</p>
    Formula:C18H25N3O5
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:363.41
  • BMS-823778

    CAS:
    <p>BMS-823778 is a potent inhibitor of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1) for the study of type 2 diabetes.</p>
    Formula:C18H18ClN3O
    Purity:99.39% - 99.75%
    Color and Shape:Solid
    Molecular weight:327.81
  • S19-1035


    <p>S19-1035: potent AKR1C3 inhibitor with 3.04 nM IC50, useful for tumor research.</p>
    Formula:C19H17ClN2O3
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:356.80
  • VU0155069

    CAS:
    <p>VU0155069, a selective PLD1 inhibitor (IC50: 46 nM), halts cancer cell migration in transwell assays.</p>
    Formula:C26H27ClN4O2
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:462.97
  • Opc 8490

    CAS:
    <p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>
    Formula:C30H35N3O10
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:597.61
  • BW-1370U87

    CAS:
    <p>BW-1370U87 is an MAO-A inhibitor increasing brain amines, showing promise in depression models.</p>
    Formula:C14H12O3S
    Purity:99.82% - 99.89%
    Color and Shape:Solid
    Molecular weight:260.31
  • MFI8

    CAS:
    <p>MFI8 is a compound that regulates mitochondrial fission and can be used to study aging.</p>
    Formula:C16H18ClNO
    Purity:99.08% - 99.78%
    Color and Shape:Solid
    Molecular weight:275.77
  • YM 511

    CAS:
    <p>YM 511 is a specific non-steroidal aromatase inhibitor with IC50s of 0.4 and 0.12 nM, minimally affecting other steroids.</p>
    Formula:C16H12BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:354.2
  • Lifibrol

    CAS:
    <p>Lifibrol (U-83860) is an inhibitor of cholesterol synthesis.Lifibrol has anticholesterol and hypolipidemic properties and promotes the conversion of LDL Apo B-</p>
    Formula:C21H26O4
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:342.43
  • NNC 05-2090 hydrochloride

    CAS:
    <p>NNC 05-2090 HCl: BGT-1 inhibitor, IC50 = 10.6 μM, potential for epilepsy, neurological research.</p>
    Formula:C27H31ClN2O2
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:451
  • 1,2-Dimyristoyl-sn-glycero-3-PA sodium

    CAS:
    <p>DMPA, a derivative of phosphatidic acid (PA), constitutes a significant component of cellular membranes.</p>
    Formula:C31H59Na2O8P
    Color and Shape:Solid
    Molecular weight:636.758
  • (S,R)-WT IDH1 Inhibitor 2

    CAS:
    <p>(S,R)-WT IDH1 Inhibitor 2: selectively targets mutant IDH1; IC50 - R132G: 2.9 nM, R132C: 3.8 nM, R132H: 4.6 nM, WT: 46 nM; potential for AML treatment.</p>
    Formula:C28H28FN5O3
    Color and Shape:Solid
    Molecular weight:501.55
  • Diflumidone sodium

    CAS:
    <p>Diflumidone sodium is a non-steroidal agent with anti-inflammatory activity.</p>
    Formula:C14H10F2NNaO3S
    Color and Shape:Solid
    Molecular weight:333.29
  • H-0104 Dihydrochloride

    CAS:
    <p>H-0104 Dihydrochloride is an inhibitor of ROCK that acts by applying potent intraocular pressure (IOP)-lowering effects into the eyes of monkeys.</p>
    Formula:C15H20BrCl2N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.21
  • Glyoxalase I inhibitor 3

    CAS:
    <p>Compound 22g: potent GLO1 inhibitor; IC50=0.011 μM; potential for depression, anxiety research.</p>
    Formula:C22H21N3O3
    Color and Shape:Solid
    Molecular weight:375.42
  • Glycosidase-IN-2

    CAS:
    <p>Glycosidase-IN-2 is a glycosidase inhibitor with hypoglycemic activity.</p>
    Formula:C13H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.33
  • Iomazenil

    CAS:
    <p>Iomazenil is an antagonist and partial inverse agonist of benzodiazepine and potential therapy for alcohol abuse.</p>
    Formula:C15H14IN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.19
  • sPLA2 inhibitor 1

    CAS:
    <p>KH064 is a sPLA2-IIA inhibitor of oral activity.</p>
    Formula:C31H37NO4
    Color and Shape:Solid
    Molecular weight:487.63
  • sEH/AChE-IN-4

    CAS:
    <p>sEH/AChE-IN-4-15 is a dual sEH and AChE inhibitor crossing the BBB, with IC50s: 3.1 nM (hsEH), 1660 nM (hAChE), 179 nM (hBChE), 14.5 nM (msEH), 102 nM (mAChE).</p>
    Formula:C35H39ClF3N5O3
    Color and Shape:Solid
    Molecular weight:670.16
  • NUCC-0223619

    CAS:
    <p>NUCC-0223619 is an IDO1 inhibitor that induces the degradation of IDO protein and can be involved in the synthesis of PROTAC.</p>
    Formula:C24H24ClFN2O2
    Color and Shape:Solid
    Molecular weight:426.91
  • Lignoceroyl Ethanolamide

    CAS:
    <p>Lignoceroyl ethanolamide, a fatty N-acyl ethanolamine within the endocannabinoid family, is derived from lignoceric acid, which is found in relatively high concentrations in rat cerebrospinal fluid. However, the specific function and significance of this metabolite remain unclear.</p>
    Formula:C26H53NO2
    Color and Shape:Solid
    Molecular weight:411.715
  • Pactimibe sulfate

    CAS:
    <p>Pactimibe sulfate is a dual ACAT1/2 inhibitor with anti-atherogenic potential, reducing plasma cholesterol.</p>
    Formula:C50H82N4O10S
    Color and Shape:Solid
    Molecular weight:931.28
  • 2-Stearoyl-sn-glycero-3-PC

    CAS:
    <p>2-Stearoyl-sn-glycero-3-phosphatidylcholine (2-Stearoyl-sn-glycero-3-PC) is a lysophospholipid characterized by the presence of stearic acid at the sn-2 position. This compound has been identified in the myocardium of rabbits.</p>
    Formula:C26H54NO7P
    Color and Shape:Solid
    Molecular weight:523.68
  • ERX-41

    CAS:
    <p>ERX-41 is an orally active, stereospecific small molecule that targets lysosomal acid lipase A (LIPA).</p>
    Formula:C38H48N4O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:704.81
  • BAY-7081


    <p>BAY-7081 is a cyanopyridone-based compound that functions as a potent, selective, and orally active PDE9A inhibitor, demonstrating an inhibition concentration (</p>
    Formula:C19H27ClN4O
    Color and Shape:Solid
    Molecular weight:362.9
  • HIF-2α-IN-6

    CAS:
    <p>HIF-2α-IN-6 (117) is a HIF-2α inhibitor [1].</p>
    Formula:C15H13F4NO3S
    Color and Shape:Solid
    Molecular weight:363.33
  • ICMT-IN-15

    CAS:
    <p>ICMT-IN-15 (compound 51) serves as an ICMT inhibitor with an IC50 value of 0.032 μM [1].</p>
    Formula:C21H25ClFNO
    Color and Shape:Solid
    Molecular weight:361.88
  • VT-1598 tosylate

    CAS:
    <p>VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.</p>
    Formula:C38H28F4N6O5S
    Color and Shape:Solid
    Molecular weight:756.72
  • GPX4-IN-2

    CAS:
    <p>GPX4-IN-2 is a potent inhibitor of GPX4, exhibiting antiproliferative activity. It holds potential for cancer research applications.</p>
    Formula:C30H40N2O
    Color and Shape:Solid
    Molecular weight:444.65
  • Celgosivir

    CAS:
    <p>Celgosivir (6 O-butanoyl castanospermine) is an inhibitor of α-glucosidase I. In vitro assay, it inhibits bovine viral diarrhoea virus (BVDV) ( IC50: 1.27 μM ).</p>
    Formula:C12H21NO5
    Purity:98.03%
    Color and Shape:Solid
    Molecular weight:259.3
  • BMS-962212

    CAS:
    <p>BMS-962212: reversible, selective FXIa blocker, well-tolerated, quick PD effect, rapid clearance, alters clotting time/activity.</p>
    Formula:C32H28ClFN8O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.07
  • PF-915275

    CAS:
    <p>PF-915275 inhibits 11βHSD1 in humans (Ki=2.3 nM, EC50=15 nM) and affects cortisone-cortisol conversion in hepatocytes.</p>
    Formula:C18H14N4O2S
    Purity:99.58% - 99.61%
    Color and Shape:Solid
    Molecular weight:350.39
  • 4BAB

    CAS:
    <p>4BAB (compound 29) is an irreversible inhibitor of glyoxalase I (GLO1) and exhibits anticancer activity.</p>
    Formula:C18H28BrN3O10S
    Color and Shape:Solid
    Molecular weight:558.4
  • Ac-VDVAD-CHO

    CAS:
    <p>Ac-VDVAD-CHO is an inhibitor of caspase-2 and caspase-3 (IC50: 46 nM for caspase-2 and 15 nM for caspase-3) [1].</p>
    Formula:C23H37N5O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:543.57
  • Aladotril

    CAS:
    <p>Aladotril is an inhibitor of neutral endopeptidase. Its prodrug is aladotrilat.</p>
    Formula:C21H23NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.48
  • JW 618

    CAS:
    <p>JW 618 is a selective inhibitor of ABHD6, demonstrating inhibition concentrations (IC50 values) of 38 nM for mouse ABHD6 and 13 nM for rat ABHD6, indicating its potent activity across species [1].</p>
    Formula:C17H14F6N2O2
    Color and Shape:Solid
    Molecular weight:392.3
  • Thioquinapiperifil

    CAS:
    <p>Thioquinapiperifil is a type of phosphodiesterase-5 (PDE-5) inhibitor found in dietary supplements.</p>
    Formula:C24H28N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.58
  • ALP/Carbonic anhydrase-IN-1

    CAS:
    <p>Compound 1e, also known as ALP/Carbonic anhydrase-IN-1, is a dual inhibitor targeting both carbonic anhydrase (CA) isozymes II, IX, and XII, as well as alkaline</p>
    Formula:C15H16N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:224.3
  • Dasatinib analog-1

    CAS:
    <p>Dasatinib analog-1 (compound 5826) demonstrates inhibition of CYP3A4 activity, presenting a K_i value of 5.4 μM, and effectively prevents the formation of glutathione adducts [1].</p>
    Formula:C22H25ClFN7O2S
    Color and Shape:Solid
    Molecular weight:506
  • 9-OAHSA

    CAS:
    <p>Branched fatty acid esters of hydroxy fatty acids (FAHFAs) are a class of endogenous lipids whose levels are modulated by fasting and high-fat diets and are linked to insulin sensitivity. These compounds typically consist of a C-16 or C-18 fatty acid, such as palmitoleic, palmitic, oleic, or stearic acid, esterified to a hydroxylated C-16 or C-18 lipid. One specific form of FAHFA, known as 9-OAHSA, involves the esterification of oleic acid to 9-hydroxy stearic acid. Within the FAHFA family, OAHSAs notably represent the predominant form found in the serum of glucose-tolerant AG4OX mice, which uniquely overexpress the Glut4 glucose transporter in adipose tissue.</p>
    Formula:C36H68O4
    Color and Shape:Solid
    Molecular weight:564.936
  • RORγt modulator 4

    CAS:
    <p>RORγt modulator 4 is a RORγt modulator that regulates IL-17A production activity in cells derived from mouse spleen.</p>
    Formula:C26H27N3O4S
    Color and Shape:Solid
    Molecular weight:477.58
  • ICMT-IN-25

    CAS:
    <p>ICMT-IN-25 (compound 37) serves as a potent inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting an IC50 value of 0.025 μM [1].</p>
    Formula:C21H26ClNO
    Color and Shape:Solid
    Molecular weight:343.89
  • cis-Clopidogrel-MP derivative

    CAS:
    <p>cis-Clopidogrel-MP derivative, also Clopidogrel-MP-AM, is a 3'-methoxyacetophenone Clopidogrel metabolite and oral P2Y12 receptor platelet inhibitor.</p>
    Formula:C25H26ClNO6S
    Color and Shape:Solid
    Molecular weight:503.99
  • ICMT-IN-26

    CAS:
    <p>ICMT-IN-26 (compound 38) acts as an ICMT inhibitor with an IC50 value of 0.36 μM [1].</p>
    Formula:C21H26ClNO
    Color and Shape:Solid
    Molecular weight:343.89
  • Quercetin 7-glucuronide

    CAS:
    <p>Quercetin 7-glucuronide (Quercetin 7-O-β-glucuronide), a Quercetin metabolite found in Madagascarian Uncarina species, has the capability to inhibit LDL</p>
    Formula:C21H18O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:478.36
  • LFHP-1c

    CAS:
    <p>LFHP-1c, a neuroprotective PGAM5 inhibitor, demonstrates efficacy in preserving blood-brain barrier integrity following ischemic stroke.</p>
    Formula:C55H64N6O4
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:873.13
  • CYP17-IN-1

    CAS:
    <p>CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.</p>
    Formula:C18H17FN2S
    Purity:99.14% - 99.83%
    Color and Shape:Solid
    Molecular weight:312.4
  • α-Glucosidase-IN-29

    CAS:
    <p>α-Glucosidase-IN-29 (compound 19) is an inhibitor of α-glucosidases, exhibiting an IC50 value of 1.21 μM and a Ki of 1.80 μM.</p>
    Formula:C33H30Br2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:698.4
  • C18 ((±)-2'-hydroxy) Ceramide (d18:1/18:0)

    CAS:
    <p>C18 ((±)-2'-hydroxy) Ceramide (d18:1/18:0) is a lipid molecule that can be used in life science related research. The CAS number of C18 ((±)-2'-hydroxy) Ceramide (d18:1/18:0) is 34249-41-7.</p>
    Formula:C36H71NO4
    Color and Shape:Solid
    Molecular weight:581.967
  • 7,12-Diketolithocholic Acid

    CAS:
    <p>7,12-Diketolithocholic acid, a bile acid, exhibits elevated plasma levels in patients experiencing cholestasis.</p>
    Formula:C24H36O5
    Color and Shape:Solid
    Molecular weight:404.54
  • Quetiapine sulfoxide hydrochloride


    <p>Quetiapine sulfoxide hydrochloride is a main metabolite of Quetiapinem. Quetiapine is a 5-HT receptors agonist and a dopamine receptor antagonist.</p>
    Formula:C21H26ClN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.97
  • ICMT-IN-14

    CAS:
    <p>ICMT-IN-14 (compound 50) serves as an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 of 0.025 μM [1].</p>
    Formula:C21H25ClFNO
    Color and Shape:Solid
    Molecular weight:361.88
  • MLS000545091

    CAS:
    <p>MLS000545091 is a potent and selective human epithelial 15-lipoxygenase-2 mixed-type inhibitor.</p>
    Formula:C14H15ClN2O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:262.73
  • PF-04957325

    CAS:
    <p>PF-04957325 is an inhibitor of PDE8.PF-04957325 has an IC50 of 0.7 nM for PDE8A.PF-04957325 can be used for the study of autoimmune encephalomyelitis.</p>
    Formula:C14H15F3N8OS
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:400.38
  • Lp-PLA2-IN-13

    CAS:
    <p>Lp-PLA2-IN-13 (compound 15), a potent Lp-PLA2 inhibitor, holds potential for research in neurodegenerative-related diseases [1].</p>
    Formula:C22H17F5N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.39
  • VULM 1457

    CAS:
    <p>VULM 1457 is a potent ACAT inhibitor.</p>
    Formula:C25H27N3O3S
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:449.57