
GPCR/G-Protein
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Found 5963 products of "GPCR/G-Protein"
Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formula:C20H22N2SPurity:99.98%Color and Shape:SolidMolecular weight:322.47AdipoRon hydrochloride
CAS:AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).Formula:C27H29ClN2O3Color and Shape:SolidMolecular weight:464.992-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.Formula:C38H64F3N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:891.98Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurity:97.62%Color and Shape:SolidMolecular weight:370.28Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Formula:C20H24N2OSColor and Shape:SolidMolecular weight:340.48Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83CYM2503
CAS:CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.
Formula:C45H55N5O7Purity:97.04%Color and Shape:SolidMolecular weight:777.95SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€1mL*10mM (DMSO)150.00€ABT-724
CAS:ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formula:C17H19N5Purity:99.73%Color and Shape:SolidMolecular weight:293.37CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28GLP-1(7-37) acetate(106612-94-6 free base)
CAS:Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54Riociguat
CAS:Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormula:C20H19FN8O2Purity:99.28% - 99.95%Color and Shape:SolidMolecular weight:422.42Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Ref: TM-TQ0227
1mg50.00€5mg105.00€10mg170.00€25mg230.00€50mg289.00€100mg401.00€1mL*10mM (DMSO)107.00€JNJ-10229570
CAS:JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous glandFormula:C22H19N3O2SPurity:98.41%Color and Shape:SolidMolecular weight:389.47Ref: TM-T5464
1mg104.00€5mg178.00€10mg281.00€25mg447.00€50mg620.00€100mg802.00€1mL*10mM (DMSO)203.00€AR-M 1896 Acetate
AR-M 1896 Acetate is the selective agonist of GalR2.Formula:C56H85N13O16Purity:99.76%Color and Shape:SolidMolecular weight:1196.35Ref: TM-T21646L
1mg537.00€2mg727.00€5mg1,064.00€10mg1,454.00€25mg2,147.00€50mg2,822.00€1mL*10mM (DMSO)2,213.00€S1RA hydrochloride
CAS:S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >Formula:C20H24ClN3O2Purity:98% - 99.84%Color and Shape:SolidMolecular weight:373.87Ref: TM-T4229
1mg35.00€5mg75.00€10mg105.00€25mg205.00€50mg334.00€100mg492.00€500mg973.00€1mL*10mM (DMSO)84.00€Ipragliflozin
CAS:Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
Formula:C21H21FO5SPurity:99.38% - 99.70%Color and Shape:SolidMolecular weight:404.45EST64454 free base
CAS:EST64454: σ1R antagonist for pain, high solubility, permeable, BCS class I, metabolically stable.Formula:C18H22F2N4O2Color and Shape:SolidMolecular weight:364.39H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:98.25% - 99.47%Color and Shape:SolidMolecular weight:404.33Ref: TM-T22834
1mg58.00€5mg113.00€10mg177.00€25mg334.00€50mg497.00€100mg708.00€1mL*10mM (DMSO)124.00€GBR 12935 dihydrochloride
CAS:GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formula:C28H36Cl2N2OPurity:99.09% - ≥95%Color and Shape:SolidMolecular weight:487.5Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1g477.00€10mg48.00€25mg65.00€50mg90.00€100mg117.00€200mg203.00€500mg333.00€1mL*10mM (DMSO)46.00€9-FLUORENOL
CAS:9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formula:C13H10OPurity:99.98%Color and Shape:Off-White Crystalline PowderMolecular weight:182.22Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formula:C17H25N3O2S·C4H6O5Purity:99.95%Color and Shape:Pale Yellow SolidMolecular weight:469.55Laropiprant sodium
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.Color and Shape:SolidNamodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73Bupranolol HCl
CAS:Bupranolol: non-selective beta blocker, no ISA, strong membrane stabilizer, fast gut absorption, high first-pass metabolism, 2-4hr half-life.Formula:C14H23Cl2NO2Color and Shape:SolidMolecular weight:308.243R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purity:99.52%Color and Shape:SolidMolecular weight:865.93Dapiprazole Hydrochloride
CAS:Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.Formula:C19H28ClN5Purity:99.75% - 99.93%Color and Shape:SolidMolecular weight:361.92SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Ref: TM-T23336
1mg46.00€5mg88.00€10mg132.00€25mg266.00€50mg409.00€100mg573.00€200mg807.00€1mL*10mM (DMSO)92.00€Parethoxycaine hydrochloride
CAS:Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81Ref: TM-T9397
1mg93.00€5mg182.00€10mg266.00€25mg425.00€50mg605.00€100mg803.00€200mg1,063.00€1mL*10mM (DMSO)177.00€Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formula:C79H125N23O22Purity:98.52%Color and Shape:SolidMolecular weight:1748.98SB-423562 HCl
CAS:SB-423562 is a calcium-sensing receptor antagonist.Formula:C26H33ClN2O4Purity:98%Color and Shape:SolidMolecular weight:473HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purity:99.51%Color and Shape:SolidMolecular weight:614.57BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg84.00€5mg161.00€10mg235.00€25mg420.00€50mg605.00€100mg842.00€200mg1,134.00€1mL*10mM (DMSO)172.00€GRA Ex-25
CAS:GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61Carazolol
CAS:Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formula:C18H22N2O2Purity:99% - 99.53%Color and Shape:Yellowish SolidMolecular weight:298.38TNCA
CAS:TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.Formula:C12H12N2O2Purity:97.33% - 97.73%Color and Shape:SolidMolecular weight:216.24BMS-813160
CAS:BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formula:C25H40N8O2Purity:99.66% - 99.79%Color and Shape:SolidMolecular weight:484.64Ref: TM-T4584
1mg63.00€5mg137.00€10mg187.00€25mg341.00€50mg567.00€100mg810.00€500mg1,644.00€1mL*10mM (DMSO)145.00€Cinacalcet hydrochloride
CAS:Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-Formula:C22H23ClF3NPurity:99.96% - >99.99%Color and Shape:Off-White To Tan SolidMolecular weight:393.87Ref: TM-T2406
10mg50.00€25mg70.00€50mg88.00€100mg144.00€200mg185.00€500mg309.00€1mL*10mM (DMSO)52.00€MK-0557
CAS:MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).Formula:C22H19FN4O3Purity:99.88%Color and Shape:SolidMolecular weight:406.41Ref: TM-TQ0286
1mg34.00€5mg67.00€10mg92.00€25mg166.00€50mg264.00€100mg371.00€200mg517.00€1mL*10mM (DMSO)75.00€Desipramine
CAS:Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.Formula:C18H22N2Color and Shape:SolidMolecular weight:266.38SAX-187 hydrochloride
CAS:WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.Formula:C15H14Cl2N4O2S2Color and Shape:SolidMolecular weight:417.33Ambrisentan
CAS:Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.Formula:C22H22N2O4Purity:99.65% - 99.86%Color and Shape:SolidMolecular weight:378.42[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFormula:C23H27ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:431.93CGS 21680 Hydrochloride
CAS:CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formula:C23H29N7O6·HClPurity:96.74% - 99.53%Color and Shape:SolidMolecular weight:535.98Ref: TM-T6441
1mg38.00€2mg50.00€5mg81.00€10mg109.00€25mg215.00€50mg389.00€100mg575.00€1mL*10mM (DMSO)95.00€AC 187 Acetate
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.Formula:C129H209N37O42Purity:99.71%Color and Shape:SolidMolecular weight:2950.26Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85ML401
CAS:ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .Formula:C20H20BrClN2OPurity:99.13%Color and Shape:SolidMolecular weight:419.74Ref: TM-T8234
1mg92.00€5mg187.00€10mg305.00€25mg487.00€50mg655.00€100mg847.00€200mg1,159.00€1mL*10mM (DMSO)207.00€JNJ-31020028
CAS:JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68BMS 182874 hydrochloride
CAS:BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formula:C17H20ClN3O3SPurity:97.01%Color and Shape:SolidMolecular weight:381.88Ref: TM-T21790
1mg77.00€2mg92.00€5mg140.00€10mg205.00€25mg343.00€50mg477.00€100mg665.00€200mg897.00€1mL*10mM (DMSO)146.00€Senktide
CAS:Senktide is an agonist of tachykinin NK3 receptor.Formula:C40H55N7O11SPurity:99.84% - >99.99%Color and Shape:White PowderMolecular weight:841.97Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formula:C14H17ClN4SColor and Shape:SolidMolecular weight:308.83Levalbuterol tartrate
CAS:Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Formula:C17H27NO9Purity:99.28% - 99.98%Color and Shape:SolidMolecular weight:389.39Ref: TM-T7164
2mg34.00€5mg50.00€10mg88.00€25mg100.00€50mg124.00€100mg177.00€200mg259.00€1mL*10mM (DMSO)60.00€BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formula:C22H33Cl2N3O3Purity:97.32% - 99.08%Color and Shape:SolidMolecular weight:458.42Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formula:C21H29Cl2N3O4SPurity:98.5%Color and Shape:SolidMolecular weight:490.44FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formula:C41H61F3N10O10Purity:99.32%Color and Shape:SolidMolecular weight:910.99Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formula:C21H30N4O4Purity:99.52%Color and Shape:SolidMolecular weight:402.49Ref: TM-T21385
1mg73.00€5mg155.00€10mg240.00€25mg479.00€50mg692.00€100mg973.00€1mL*10mM (DMSO)177.00€Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurity:99.04%Color and Shape:SolidMolecular weight:436.95Zuclopenthixol dihydrochloride
CAS:Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Formula:C22H27Cl3N2OSPurity:98%Color and Shape:SolidMolecular weight:473.89HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formula:C35H51N9O14Purity:>99.99%Color and Shape:SolidMolecular weight:821.84RBC8
CAS:RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.Formula:C25H20N4O3Purity:98.44% - 99.81%Color and Shape:SolidMolecular weight:424.45Ref: TM-T6634
1mg48.00€5mg92.00€10mg156.00€25mg298.00€50mg472.00€100mg687.00€200mg938.00€1mL*10mM (DMSO)97.00€Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852RS 100329
CAS:RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formula:C20H25F3N4O3Color and Shape:SolidMolecular weight:426.43Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43Ref: TM-T7183
2mg34.00€5mg52.00€10mg73.00€25mg128.00€50mg197.00€100mg295.00€200mg442.00€1mL*10mM (DMSO)52.00€RE-640
CAS:NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.Formula:C20H16Cl2N4Purity:99.60% - 99.87%Color and Shape:SolidMolecular weight:383.27SRI-37330 hydrochloride
CAS:SRI-37330 hydrochloride is an orally active thioredoxin-interacting protein (TXNIP) inhibitor. hydrochloride can be used to study type 2 diabetes.Formula:C16H20ClF3N4O2SColor and Shape:SolidMolecular weight:424.87Hemokinin 1 (human) acetate(491851-53-7 free base)
Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.Formula:C56H88N14O16SPurity:97.82%Color and Shape:SolidMolecular weight:1245.45Peptide YY (PYY) (3-36), human
CAS:Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formula:C176H272N52O54Purity:97.76%Color and Shape:SolidMolecular weight:3980.42Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Doxazosin
CAS:Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formula:C23H25N5O5Purity:99.47% - 99.87%Color and Shape:SolidMolecular weight:451.48AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formula:C21H25ClN2Purity:99.61%Color and Shape:SolidMolecular weight:340.89Ref: TM-T26690
1mg34.00€5mg75.00€10mg114.00€25mg205.00€50mg334.00€100mg557.00€200mg790.00€1mL*10mM (DMSO)92.00€Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formula:C15H19Cl2N3O3SPurity:98.48%Color and Shape:SolidMolecular weight:392.3Ref: TM-T28972
1mg66.00€5mg130.00€10mg177.00€25mg299.00€50mg447.00€100mg623.00€200mg882.00€1mL*10mM (DMSO)137.00€Org 27569
CAS:Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormula:C24H28ClN3OPurity:>99.99% - ≥95%Color and Shape:SolidMolecular weight:409.95Tolnapersine
CAS:Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Formula:C21H26N2OPurity:98%Color and Shape:SolidMolecular weight:322.44MRT-10
CAS:MRT-10 is a Smoothened (Smo) receptor antagonist.
Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52Acitazanolast
CAS:Acitazanolast (WP-871) is an anti-allergic drug candidate.
Formula:C9H7N5O3Purity:98.25%Color and Shape:SolidMolecular weight:233.18RS-127445 hydrochloride
CAS:RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formula:C17H17ClFN3Purity:99.48%Color and Shape:SolidMolecular weight:317.79Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formula:C23H23ClN2O5SPurity:97.6% - 97.78%Color and Shape:SolidMolecular weight:474.96Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purity:98.76% - 99.79%Color and Shape:SolidMolecular weight:295.38Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formula:C21H27N3Purity:98%Color and Shape:SolidMolecular weight:321.46Evatanepag sodium
CAS:Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formula:C25H27N2NaO5SColor and Shape:SolidMolecular weight:490.55Scyliorhinin II acetate
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.Formula:C79H123N21O28S3Purity:99.06%Color and Shape:SolidMolecular weight:1911.14Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purity:99.89%Color and Shape:SolidMolecular weight:239.27Ref: TM-T9132
1mg84.00€5mg168.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)152.00€Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formula:C17H25ClN2O2Purity:97.91%Color and Shape:SolidMolecular weight:324.85Ref: TM-T4087
1mg37.00€5mg71.00€10mg92.00€25mg164.00€50mg225.00€100mg323.00€200mg437.00€1mL*10mM (DMSO)71.00€Urapidil
CAS:Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formula:C20H29N5O3Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:387.48AP1189 acetate
CAS:AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
Formula:C16H18N6O4Purity:99.95%Color and Shape:SolidMolecular weight:358.35BD1063 dhydrochloride
CAS:BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).Formula:C13H20Cl4N2Purity:99.52% - ≥95%Color and Shape:SolidMolecular weight:346.12Ref: TM-T7488
2mg46.00€5mg69.00€10mg95.00€25mg177.00€50mg321.00€100mg472.00€200mg665.00€500mg1,018.00€CAY10526
CAS:CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formula:C12H7BrO3SPurity:98.75%Color and Shape:SolidMolecular weight:311.15Cetirizine Impurity B dihydrochloride
CAS:Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.Formula:C19H23Cl3N2O2Purity:97.33%Color and Shape:SolidMolecular weight:417.76Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purity:98.13% - 99.66%Color and Shape:SolidMolecular weight:449.54TRAP-6 amide acetate
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
Formula:C36H61N11O10Purity:98.55%Color and Shape:SolidMolecular weight:807.94A-381393
CAS:A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Formula:C20H24N4Purity:99.00%Color and Shape:SolidMolecular weight:320.43Ref: TM-T5397
1mg38.00€5mg75.00€10mg111.00€25mg198.00€50mg288.00€100mg414.00€200mg583.00€1mL*10mM (DMSO)84.00€Piperoxan hydrochloride
CAS:Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77Ref: TM-T4526
2mg39.00€5mg62.00€10mg92.00€25mg128.00€50mg166.00€100mg200.00€200mg299.00€1mL*10mM (DMSO)55.00€Bucindolol hydrochloride
CAS:Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Formula:C22H26ClN3O2Color and Shape:SolidMolecular weight:399.91Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formula:C22H26N2O4Purity:98% - 99.9%Color and Shape:SolidMolecular weight:382.45Ref: TM-T6S0654
1mg62.00€2mg89.00€5mg132.00€10mg226.00€25mg384.00€50mg557.00€100mg785.00€200mg1,054.00€1mL*10mM (DMSO)146.00€[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.Formula:C190H286N54O56Purity:99.39%Color and Shape:SolidMolecular weight:4223SKF 38393 hydrochloride
CAS:SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formula:C16H17NO2·HClPurity:99.1% - 99.51%Color and Shape:SolidMolecular weight:291.77Azepexole
CAS:Azepexole is a selective α2-adrenoceptor agonist that exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor.Formula:C9H15N3OColor and Shape:SolidMolecular weight:181.23ICI 89406
CAS:ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.Formula:C19H22N4O3Purity:99.92%Color and Shape:SolidMolecular weight:354.4Secretin (33-59), rat
CAS:Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purity:99.2%Color and Shape:SolidMolecular weight:393.45BPTU
CAS:BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).Formula:C23H22F3N3O3Purity:99.37% - 99.89%Color and Shape:SolidMolecular weight:445.43Ref: TM-T4132
1mg35.00€2mg50.00€5mg69.00€10mg110.00€25mg225.00€50mg389.00€100mg577.00€1mL*10mM (DMSO)69.00€Treprostinil
CAS:Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).Formula:C23H34O5Purity:99.29%Color and Shape:SolidMolecular weight:390.51Ref: TM-T5150
1mg34.00€5mg71.00€10mg108.00€25mg221.00€50mg355.00€100mg533.00€200mg755.00€1mL*10mM (DMSO)60.00€Nelociguat
CAS:Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:C19H17FN8O2Purity:99.19%Color and Shape:SolidMolecular weight:408.39Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formula:C20H20NO4Purity:97.18% - 99.06%Color and Shape:SolidMolecular weight:338.38cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formula:C16H14O2Purity:98.15%Color and Shape:SolidMolecular weight:238.2812Ref: TM-T8586
1mg62.00€5mg123.00€10mg180.00€25mg298.00€50mg419.00€100mg567.00€200mg752.00€1mL*10mM (DMSO)111.00€Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38ML-18
CAS:ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.Formula:C32H35N5O5Purity:98.62% - >99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-T4540
1mg34.00€5mg60.00€10mg96.00€25mg170.00€50mg264.00€100mg425.00€200mg587.00€1mL*10mM (DMSO)75.00€Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
Formula:C52H77N13O13Purity:99.93%Color and Shape:SolidMolecular weight:1092.27LY 78335
CAS:LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.Formula:C8H10Cl3NPurity:99.30% - 99.81%Color and Shape:SolidMolecular weight:226.53Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29CCG-50014
CAS:CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.Formula:C16H13FN2O2SPurity:98.53%Color and Shape:SolidMolecular weight:316.35K 41498 aceate
K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for CRF1; blocks aSvg-30 effect on cAMP in cells.Purity:96.4%Color and Shape:LiquidMolecular weight:N/AAC-55541
CAS:AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formula:C11H9Cl2N3O3SPurity:99.80% - >99.99%Color and Shape:SolidMolecular weight:334.18Ref: TM-T4300
1mg34.00€5mg66.00€10mg105.00€25mg217.00€50mg334.00€100mg502.00€500mg1,063.00€1mL*10mM (DMSO)73.00€ZK 756326
CAS:ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formula:C21H28N2O3Purity:99.43%Color and Shape:SolidMolecular weight:356.46ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formula:C13H16ClN3O3Purity:98.15%Color and Shape:SolidMolecular weight:297.74Ref: TM-T9193
1mg50.00€5mg110.00€10mg172.00€25mg304.00€50mg424.00€100mg583.00€200mg785.00€1mL*10mM (DMSO)122.00€Human growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) onPurity:99.26%Color and Shape:LiquidMolecular weight:N/AChlorphenesin
CAS:Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.Formula:C9H11ClO3Purity:99.59%Color and Shape:SolidMolecular weight:202.63Netupitant
CAS:Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).Formula:C30H32F6N4OPurity:99.43%Color and Shape:SolidMolecular weight:578.59Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42Melperone
CAS:Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.Formula:C16H22FNOPurity:98.84%Color and Shape:SolidMolecular weight:263.35Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Purity:98.27%Color and Shape:LiquidMolecular weight:N/ARomifidine hydrochloride
CAS:Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.Formula:C9H10BrClFN3Color and Shape:SolidMolecular weight:294.55Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Formula:C26H28ClN5O6Color and Shape:SolidMolecular weight:541.98Mesdopetam
CAS:Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Formula:C12H18FNO3SColor and Shape:SolidMolecular weight:275.34TFLLR-NH2 2TFA(197794-83-5(free base))
TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).Formula:C35H55F6N9O10Purity:99.56%Color and Shape:SolidMolecular weight:875.87Alizapride
CAS:Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].Formula:C16H21N5O2Color and Shape:SolidMolecular weight:315.37ENMD-1068 HBr
CAS:ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.Formula:C15H30BrN3O2Color and Shape:SolidMolecular weight:364.32Dobutamine
CAS:Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formula:C149H234N40O47SPurity:98% - 99.65%Color and Shape:SolidMolecular weight:3369.76Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg38.00€2mg50.00€5mg84.00€10mg118.00€25mg220.00€50mg403.00€100mg582.00€500mg1,198.00€1mL*10mM (DMSO)120.00€Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03Ref: TM-T7617L
1mg35.00€5mg73.00€10mg107.00€25mg207.00€50mg313.00€100mg447.00€200mg620.00€1mL*10mM (DMSO)132.00€PF-4136309
CAS:PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formula:C29H31F3N6O3Purity:98.85% - 99.47%Color and Shape:SolidMolecular weight:568.59Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formula:C10H17N3SPurity:99.78%Color and Shape:SolidMolecular weight:211.33Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurity:99.04% - 99.88%Color and Shape:SolidMolecular weight:315.47Ozanimod hydrochloride
CAS:Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formula:C23H25ClN4O3Purity:99.81%Color and Shape:SolidMolecular weight:440.92Ref: TM-T62552
1mg47.00€5mg92.00€10mg137.00€25mg268.00€50mg432.00€100mg620.00€200mg875.00€1mL*10mM (DMSO)101.00€Alfuzosin
CAS:Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formula:C19H27N5O4Purity:99.64%Color and Shape:White Crystaline PowderMolecular weight:389.45Trabodenoson
CAS:Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Ref: TM-T34914
1mg40.00€5mg89.00€10mg116.00€25mg187.00€50mg285.00€100mg411.00€200mg577.00€1mL*10mM (DMSO)88.00€Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formula:(C6H14N2O2)x·xHBrColor and Shape:SolidMolecular weight:227.102Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purity:99.94%Color and Shape:SolidMolecular weight:383.49Ref: TM-TQ0315
2mg34.00€5mg50.00€10mg80.00€25mg130.00€50mg178.00€100mg284.00€200mg408.00€1mL*10mM (DMSO)55.00€CP-105696
CAS:CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.Formula:C28H28O4Purity:99.78%Color and Shape:SolidMolecular weight:428.52LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94Atogepant
CAS:Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formula:C29H23F6N5O3Purity:99.66%Color and Shape:SolidMolecular weight:603.52Ref: TM-T26682
1mg147.00€5mg250.00€10mg313.00€25mg620.00€50mg1,108.00€100mg1,611.00€200mg2,178.00€1mL*10mM (DMSO)334.00€Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formula:C20H21FN2OPurity:99.78% - 99.89%Color and Shape:SolidMolecular weight:324.39Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purity:99.41% - >99.99%Color and Shape:SolidMolecular weight:517.66Atipamezole
CAS:Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formula:C14H16N2Purity:99.88%Color and Shape:Off-White To Light Yellow Crystal PowderMolecular weight:212.29L-368,899 hydrochloride
CAS:L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formula:C26H43ClN4O5S2Purity:99.59%Color and Shape:SolidMolecular weight:591.23Ref: TM-T11794
2mg105.00€5mg147.00€10mg230.00€25mg439.00€50mg685.00€100mg964.00€1mL*10mM (DMSO)200.00€Protein deglycase DJ-1 against-1
CAS:Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formula:C24H23N3O4Purity:97.23%Color and Shape:SolidMolecular weight:417.46WIN 51,708
CAS:WIN 51,708 is an antagonist of neurokinin-1 receptor.Formula:C29H33N3OPurity:99%Color and Shape:SolidMolecular weight:439.59GAT211
CAS:GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.Formula:C22H18N2O2Purity:99.7%Color and Shape:SolidMolecular weight:342.39Ref: TM-T27405
1mg34.00€5mg66.00€10mg90.00€25mg148.00€50mg210.00€100mg310.00€500mg750.00€1mL*10mM (DMSO)73.00€Nebentan potassium
CAS:Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.Formula:C24H20KN5O5SPurity:99.05%Color and Shape:SolidMolecular weight:529.61Ref: TM-T36008
1mg52.00€2mg77.00€5mg111.00€10mg177.00€25mg313.00€50mg502.00€100mg680.00€200mg888.00€1mL*10mM (DMSO)133.00€CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formula:C25H41NO2Purity:98.78%Color and Shape:SolidMolecular weight:387.6Medetomidine
CAS:Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formula:C13H16N2Purity:99.88%Color and Shape:SolidMolecular weight:200.28Ref: TM-T21492
2mg38.00€5mg57.00€10mg77.00€25mg128.00€50mg193.00€100mg290.00€200mg447.00€1mL*10mM (DMSO)62.00€S1RA
CAS:S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formula:C20H23N3O2Purity:99.45%Color and Shape:SolidMolecular weight:337.42S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formula:C19H34O3Purity:97.05% - 98.55%Color and Shape:SolidMolecular weight:310.47UCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formula:C19H20N2O2Purity:98.88%Color and Shape:SolidMolecular weight:308.37ACT-462206
CAS:ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formula:C20H24N2O4SPurity:99.45%Color and Shape:SolidMolecular weight:388.48Ref: TM-T26559
1mg44.00€5mg93.00€10mg137.00€25mg279.00€50mg445.00€100mg707.00€500mg1,415.00€1mL*10mM (DMSO)93.00€SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purity:98.78% - 99.86%Color and Shape:SolidMolecular weight:428.41Ref: TM-T37816
1mg35.00€5mg75.00€10mg114.00€25mg260.00€50mg485.00€100mgTo inquire1mL*10mM (DMSO)84.00€Fenoterol hydrobromide
CAS:Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formula:C17H22BrNO4Purity:99.88%Color and Shape:SolidMolecular weight:384.27(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purity:99.75%Color and Shape:SolidMolecular weight:265.35Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurity:98.05% - 98.07%Color and Shape:SolidMolecular weight:261.36Maropitant citrate
CAS:Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.Formula:C38H50N2O9Purity:98.91%Color and Shape:SolidMolecular weight:678.81A2ti-1
CAS:A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.Formula:C20H22N4O2SPurity:99.86%Color and Shape:SolidMolecular weight:382.48Ref: TM-T36432
1mg94.00€5mg200.00€10mg313.00€25mg620.00€50mg982.00€100mg1,341.00€500mg2,682.00€1mL*10mM (DMSO)286.00€Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formula:C16H22ClN3O2Purity:98.97% - 99.09%Color and Shape:SolidMolecular weight:323.82Ref: TM-T38507
1mg93.00€2mg124.00€5mg200.00€10mg359.00€25mg692.00€50mg945.00€100mg1,279.00€200mg1,701.00€Opipramol
CAS:Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.Formula:C23H29N3OPurity:99.84% - 99.98%Color and Shape:SolidMolecular weight:363.5SID 7969543
CAS:SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formula:C24H24N2O7Purity:98.94%Color and Shape:SolidMolecular weight:452.465-LOX inhibitor
CAS:5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) is an itraconazole impurity, a LOX-5 inhibitor.Formula:C22H27N5O2Purity:98.01%Color and Shape:SolidMolecular weight:393.48Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formula:C15H19N5Purity:99.74%Color and Shape:SolidMolecular weight:269.35Fenoprofen
CAS:Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formula:C15H14O3Purity:98.4%Color and Shape:SolidMolecular weight:242.27Bucindolol
CAS:Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.Formula:C22H25N3O2Purity:99.9%Color and Shape:SolidMolecular weight:363.45Clopidogrel thiolactone
CAS:Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.Formula:C16H16ClNO3SPurity:98.79%Color and Shape:SolidMolecular weight:337.82Ref: TM-T5501
1mg96.00€5mg205.00€10mg326.00€25mg557.00€50mg803.00€100mg1,063.00€200mg1,459.00€1mL*10mM (DMSO)227.00€Benzylthiouracil
CAS:Benzylthiouracil (6-Benzyl-2-thiouracil) induces ANCA-associated glomerulonephritis in Graves' disease patients and is used to study hyperthyroidism.Formula:C11H10N2OSPurity:99.65%Color and Shape:SolidMolecular weight:218.28WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purity:99.96%Color and Shape:White SolidMolecular weight:538.645Ref: TM-T3453
2mg46.00€5mg66.00€10mg95.00€25mg159.00€50mg226.00€100mg334.00€500mg807.00€1mL*10mM (DMSO)79.00€(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purity:99.37%Color and Shape:SolidMolecular weight:265.35AF-710B
CAS:AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.Formula:C20H27N3OSPurity:98.62% - 99.89%Color and Shape:SolidMolecular weight:357.51Canagliflozin hemihydrate
CAS:Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.Formula:C48H52F2O11S2Purity:99.42% - 99.96%Color and Shape:SolidMolecular weight:907.05Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46Jatrorrhizine chloride
CAS:Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formula:C20H20ClNO4Purity:99.79%Color and Shape:SolidMolecular weight:373.8GRK6-IN-2
CAS:GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.
Formula:C21H21FN6Purity:98.94%Color and Shape:SolidMolecular weight:376.43BMS-986278
CAS:BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,
Formula:C22H31N5O5Purity:99.86%Color and Shape:SolidMolecular weight:445.51Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purity:99.68%Color and Shape:SolidMolecular weight:545.51Levocetirizine Dihydrochloride
CAS:Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.
Formula:C21H27Cl3N2O3Purity:99.89%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:461.81KB-5492 free base
CAS:KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formula:C23H30N2O6Purity:97.10% - 97.94%Color and Shape:SolidMolecular weight:430.49Ref: TM-T62396
2mg39.00€5mg58.00€10mg82.00€25mg119.00€50mg168.00€100mg249.00€500mg613.00€1mL*10mM (DMSO)64.00€Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purity:97.11%Color and Shape:SolidMolecular weight:333.47INCB 3284
CAS:INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formula:C26H31F3N4O4Purity:97.81% - 99.42%Color and Shape:SolidMolecular weight:520.54CGP 20712 A
CAS:CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formula:C24H29F3N4O8SPurity:99.37%Color and Shape:SolidMolecular weight:590.57Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3

