GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(58 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5982 products of "GPCR/G-Protein"
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Bimatoprost
CAS:Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular
Formula:C25H37NO4Purity:98% - >99.99%Color and Shape:Crystalline SolidMolecular weight:415.57Azaphen dihydrochloride monohydrate
CAS:Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formula:C16H23Cl2N5O2Purity:99.85%Color and Shape:SolidMolecular weight:388.295-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurity:99.13%Color and Shape:SolidMolecular weight:280.36Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formula:C11H21NColor and Shape:SolidMolecular weight:167.29Pancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.Purity:97.53%Color and Shape:SolidMolecular weight:N/ARef: TM-TP1044L
1mg215.00€5mg510.00€10mg692.00€25mg1,009.00€50mg1,378.00€100mg1,863.00€200mg2,520.00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purity:99.95%Color and Shape:SolidMolecular weight:805.9Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
2mg39.00€5mg58.00€10mg93.00€25mg167.00€50mg250.00€100mg408.00€200mg585.00€1mL*10mM (DMSO)81.00€Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formula:C21H29ClN2O5Purity:99.52%Color and Shape:SolidMolecular weight:424.92MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8Ref: TM-T9330
1mg35.00€2mg50.00€5mg74.00€10mg105.00€25mg178.00€50mg313.00€100mg485.00€1mL*10mM (DMSO)82.00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formula:C114H174N34O31Purity:99.05%Color and Shape:SolidMolecular weight:2516.81Ref: TM-TP2279L
1mg77.00€2mg97.00€5mg156.00€10mg225.00€25mg375.00€50mg535.00€100mg730.00€200mg938.00€Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purity:99.93%Color and Shape:SolidMolecular weight:1035.15CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.Formula:C143H235N41O45SPurity:97.12%Color and Shape:SolidMolecular weight:3280.76Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formula:C13H13ClN2OPurity:99.61% - >99.99%Color and Shape:Yellow To Slightly Green Crystalline PowderMolecular weight:248.71Preladenant
CAS:Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormula:C25H29N9O3Purity:98.02% - 99.68%Color and Shape:SolidMolecular weight:503.56Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formula:C76H117N19O22SPurity:95.43%Color and Shape:SolidMolecular weight:1680.94Ziprasidone mesylate
CAS:Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.Formula:C22H25ClN4O4S2Color and Shape:SolidMolecular weight:509.04Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formula:C18H22ClNOPurity:99.44% - 99.85%Color and Shape:SolidMolecular weight:303.83Ref: TM-T7564
2mg35.00€5mg51.00€10mg81.00€25mg106.00€50mg147.00€100mg207.00€200mg306.00€1mL*10mM (DMSO)63.00€Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4Formula:C59H69F3N12O12Purity:99.22%Color and Shape:SolidMolecular weight:1195.25Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66ONO-AE3-208
CAS:ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.
Formula:C24H21FN2O3Purity:98.04% - 99.55%Color and Shape:SolidMolecular weight:404.43Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purity:99.33%Color and Shape:SolidMolecular weight:430.97Ref: TM-T9833
1mg90.00€5mg215.00€10mg340.00€25mg618.00€50mg879.00€100mg1,224.00€500mg2,457.00€1mL*10mM (DMSO)236.00€Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43Scyliorhinin II acetate
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.Formula:C79H123N21O28S3Purity:99.06%Color and Shape:SolidMolecular weight:1911.14GBR 12935
CAS:GBR-12935: selective dopamine inhibitor, used in Parkinson's research.Formula:C28H34N2OColor and Shape:SolidMolecular weight:414.58Dapiprazole Hydrochloride
CAS:Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.Formula:C19H28ClN5Purity:99.75% - 99.93%Color and Shape:SolidMolecular weight:361.92UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formula:C52H68N10O14S2Purity:99.78%Color and Shape:SolidMolecular weight:1121.29Vorapaxar
CAS:Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).Formula:C29H33FN2O4Purity:98.77% - 99.93%Color and Shape:SolidMolecular weight:492.58Ref: TM-T7013
1mg74.00€5mg145.00€10mg202.00€25mg344.00€50mg472.00€100mg677.00€200mg937.00€1mL*10mM (DMSO)160.00€Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formula:C51H70N10O12S2Purity:99.03% - 99.87%Color and Shape:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMolecular weight:1079.3AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formula:C23H31ClN2O2Purity:99.71%Color and Shape:SolidMolecular weight:402.96M 1145 acetate
M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; >90x affinity vs GAL1, 76x vs GalR3. Enhances galanin signal.Formula:C130H209N37O34Purity:99.1%Color and Shape:SolidMolecular weight:2834.28Ref: TM-TP1991L
1mg248.00€5mg532.00€10mg712.00€25mg1,054.00€50mg1,425.00€100mg1,928.00€200mg2,593.00€Regadenoson hydrate
CAS:Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.Formula:C15H20N8O6Purity:98%Color and Shape:SolidMolecular weight:408.37Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Ref: TM-T5520L
1mg52.00€5mg90.00€10mg150.00€25mg291.00€50mg437.00€100mg642.00€500mg1,359.00€1mL*10mM (DMSO)251.00€Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purity:>99.99%Color and Shape:SolidMolecular weight:1024.18FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Formula:C23H25Cl2N3OSPurity:99.62%Color and Shape:SolidMolecular weight:462.44Ref: TM-T21667
1mg52.00€5mg111.00€10mg169.00€25mg323.00€50mg512.00€100mg740.00€500mg1,539.00€1mL*10mM (DMSO)123.00€Betahistine
CAS:Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formula:C8H12N2Purity:99.87% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19Loxapine hydrochloride
CAS:Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Formula:C18H19Cl2N3OColor and Shape:SolidMolecular weight:364.27AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formula:C17H21N5O2SPurity:99.81%Color and Shape:SolidMolecular weight:359.45Ref: TM-T5179
1mg37.00€2mg50.00€5mg77.00€10mg114.00€25mg225.00€50mg335.00€100mg484.00€1mL*10mM (DMSO)85.00€ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.Formula:C77H123N25O19S2Purity:97.2%Color and Shape:SolidMolecular weight:1767.09BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formula:C22H33Cl2N3O3Purity:97.32% - 99.08%Color and Shape:SolidMolecular weight:458.425'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formula:C12H16N6O4Purity:98.95% - ≥95%Color and Shape:PowderMolecular weight:308.29LRGILS-NH2 acetate
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.Formula:C29H56N10O7Purity:96.65%Color and Shape:SolidMolecular weight:656.82Mebhydrolin
CAS:Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Color and Shape:SolidMolecular weight:472.97Sotagliflozin
CAS:Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potentialFormula:C21H25ClO5SPurity:99% - 99.86%Color and Shape:SolidMolecular weight:424.94Ref: TM-T3547
1mg46.00€2mg57.00€5mg87.00€10mg131.00€25mg248.00€50mg378.00€100mg560.00€500mg1,198.00€1mL*10mM (DMSO)88.00€Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formula:C16H19BrN2Color and Shape:SolidMolecular weight:319.24M617 acetate
M617 acetate is a selective agonist of galanin receptor 1 (GAL1).Formula:C112H161N29O28Purity:96.02%Color and Shape:SolidMolecular weight:2361.65Ursodeoxycholic acid sodium
CAS:Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.
Formula:C24H40NaO4Purity:99.66% - 99.96%Color and Shape:SolidMolecular weight:415.56HS024
CAS:HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.Formula:C58H79N19O10S2Purity:>99.99%Color and Shape:SolidMolecular weight:1266.5Ozanimod
CAS:Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formula:C23H24N4O3Purity:98.68% - 99.58%Color and Shape:SolidMolecular weight:404.46Ref: TM-T6923
1mg48.00€5mg96.00€10mg144.00€25mg283.00€50mg454.00€100mg655.00€200mg929.00€500mg1,378.00€1mL*10mM (DMSO)96.00€SB-222200
CAS:SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).Formula:C26H24N2OPurity:97.13%Color and Shape:SolidMolecular weight:380.48Urapidil
CAS:Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formula:C20H29N5O3Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:387.48GSK 789472 hydrochloride
CAS:GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Formula:C15H22ClN3OPurity:99.89%Color and Shape:SolidMolecular weight:295.81Guanabenz Acetate
CAS:Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.Formula:C8H8Cl2N4·C2H4O2Purity:99% - 99.66%Color and Shape:White Solid From Acetonitrile White SolidMolecular weight:291.13NIBR-0213
CAS:NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.Formula:C27H29ClN2O3Purity:98.36% - 99.34%Color and Shape:SolidMolecular weight:464.98d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formula:C52H75N13O13S2Purity:99.86%Color and Shape:SolidMolecular weight:1154.37PF-04418948
CAS:PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.Formula:C23H20FNO5Purity:98.67% - 99.45%Color and Shape:SolidMolecular weight:409.41Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Color and Shape:SolidMolecular weight:372.72FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formula:C41H61F3N10O10Purity:99.32%Color and Shape:SolidMolecular weight:910.99Alprenolol hydrochloride
CAS:Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formula:C15H24ClNO2Purity:99.79%Color and Shape:SolidMolecular weight:285.81Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formula:C17H27Cl2NOPurity:99.72% - 99.91%Color and Shape:SolidMolecular weight:332.31Ref: TM-T7176
5mg50.00€10mg74.00€25mg124.00€50mg197.00€100mg311.00€200mg467.00€500mg747.00€1mL*10mM (DMSO)52.00€Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purity:99.8% - 99.91%Color and Shape:Off-White SolidMolecular weight:355.43Evatanepag sodium
CAS:Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formula:C25H27N2NaO5SColor and Shape:SolidMolecular weight:490.55TNCA
CAS:TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.Formula:C12H12N2O2Purity:97.33% - 97.73%Color and Shape:SolidMolecular weight:216.24Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formula:C14H17ClN4SColor and Shape:SolidMolecular weight:308.83Vorapaxar sulfate
CAS:Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.Formula:C29H35FN2O8SPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:590.66Ref: TM-T3098
1mg38.00€2mg49.00€5mg79.00€10mg119.00€25mg210.00€50mg354.00€100mg528.00€500mg1,159.00€1mL*10mM (DMSO)99.00€Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Formula:C65H102N16O25Purity:95.55%Color and Shape:SolidMolecular weight:1507.6Ref: TM-TP1578L
1mg67.00€2mg95.00€5mg130.00€10mg185.00€25mg339.00€50mg507.00€100mg713.00€500mg1,504.00€AdipoRon hydrochloride
CAS:AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).Formula:C27H29ClN2O3Color and Shape:SolidMolecular weight:464.99Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91Ref: TM-T4635
1mg52.00€2mgTo inquire5mg111.00€10mg170.00€25mg301.00€50mg424.00€100mg605.00€200mg848.00€1mL*10mM (DMSO)124.00€L-DOPA methyl ester (hydrochloride)
CAS:L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formula:C10H14ClNO4Purity:98.69% - 99.81%Color and Shape:White SolidMolecular weight:247.6759-FLUORENOL
CAS:9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formula:C13H10OPurity:99.98%Color and Shape:Off-White Crystalline PowderMolecular weight:182.22Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46GLP-1(7-37) acetate(106612-94-6 free base)
CAS:Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formula:C99H163N27O34Purity:99.25%Color and Shape:SolidMolecular weight:2275.51Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Formula:C16H18BrNO2Purity:98.99%Color and Shape:SolidMolecular weight:336.22Pergolide
CAS:Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormula:C19H26N2SPurity:99.95%Color and Shape:SolidMolecular weight:314.49Ref: TM-T21340
2mg38.00€5mg57.00€10mg80.00€25mg116.00€50mg167.00€100mg250.00€200mg370.00€1mL*10mM (DMSO)64.00€Prasugrel Hydrochloride
CAS:Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
Formula:C20H20FNO3S·HClPurity:99.39% - 99.79%Color and Shape:SolidMolecular weight:409.9CYM 50358 hydrochloride (1314212-39-9 free base)
CAS:CYM50358 HCl is an S1P4 antagonist.Formula:C20H19Cl3N2O2Purity:99.57%Color and Shape:SolidMolecular weight:425.73Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formula:C32H39NO2Purity:99.65% - 99.99%Color and Shape:White To Off-White PowderMolecular weight:469.66LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purity:98.36%Color and Shape:SolidMolecular weight:473.93Ref: TM-T7303
2mg37.00€5mg70.00€10mg104.00€25mg216.00€50mg354.00€100mg550.00€200mg785.00€1mL*10mM (DMSO)73.00€Motilin (26-47), human, porcine
CAS:Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formula:C120H188N34O35SPurity:98%Color and Shape:SolidMolecular weight:2699.07Ref: TM-TP1425
1mg111.00€5mg334.00€10mg504.00€25mg745.00€50mg999.00€100mg1,341.00€200mg1,773.00€500µg86.00€Sitaxsentan sodium
CAS:Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.Formula:C18H14ClN2O6S2·NaPurity:98.39% - 99.01%Color and Shape:SolidMolecular weight:476.89Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formula:C28H36N4O2S·HClPurity:99.51%Color and Shape:SolidMolecular weight:529.14Ref: TM-T1735
5mg39.00€10mg59.00€25mg75.00€50mg90.00€100mg137.00€200mg213.00€500mg447.00€1mL*10mM (DMSO)54.00€Cinaciguat hydrochloride
CAS:Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.Formula:C36H40ClNO5Color and Shape:SolidMolecular weight:602.17H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:98.25% - 99.47%Color and Shape:SolidMolecular weight:404.33Ref: TM-T22834
1mg58.00€5mg113.00€10mg177.00€25mg334.00€50mg497.00€100mg708.00€1mL*10mM (DMSO)124.00€AM966
CAS:AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.
Formula:C27H23ClN2O5Purity:98.06% - 99.79%Color and Shape:SolidMolecular weight:490.93Ipragliflozin
CAS:Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
Formula:C21H21FO5SPurity:99.38% - 99.70%Color and Shape:SolidMolecular weight:404.45Bromodiphenhydramine
CAS:Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.Formula:C17H20BrNOColor and Shape:SolidMolecular weight:334.25Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21Asapiprant
CAS:Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.Formula:C24H27N3O7SPurity:99.64%Color and Shape:SolidMolecular weight:501.55Ref: TM-T5386
1mg40.00€5mg97.00€10mg156.00€25mg284.00€50mg449.00€100mg730.00€200mg938.00€1mL*10mM (DMSO)105.00€SB297006
CAS:SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.Formula:C18H18N2O5Purity:99.59%Color and Shape:SolidMolecular weight:342.35Ropinirole hydrochloride
CAS:Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formula:C16H24N2O·HClPurity:99.87% - 99.98%Color and Shape:Off-White SolidMolecular weight:296.84Ralmitaront
CAS:Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).
Formula:C17H22N4O2Purity:99.71% - 99.79%Color and Shape:SolidMolecular weight:314.38MHP
CAS:MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.Formula:C16H23NO4Purity:98.58%Color and Shape:SolidMolecular weight:293.36Ref: TM-T4658
1mg34.00€2mg46.00€5mg66.00€10mg101.00€25mg207.00€50mg334.00€100mg537.00€200mg762.00€1mL*10mM (DMSO)73.00€SANT-1
CAS:SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formula:C23H27N5Purity:99.93% - >99.99%Color and Shape:SolidMolecular weight:373.49Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Formula:C14H20F6N4O7Purity:98.18%Color and Shape:SolidMolecular weight:470.32Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Color and Shape:SolidMolecular weight:491.49Ciliobrevin A
CAS:Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formula:C17H9Cl2N3O2Purity:98.54% - 99.57%Color and Shape:SolidMolecular weight:358.18Ref: TM-T3156
2mg42.00€5mg59.00€10mg85.00€25mg168.00€50mg235.00€100mg331.00€200mg492.00€1mL*10mM (DMSO)69.00€Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38PRX-08066
CAS:PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Formula:C19H17ClFN5SPurity:97.79% - 98.07%Color and Shape:SolidMolecular weight:401.89Ref: TM-T16669
1mg60.00€5mg119.00€10mg170.00€25mg350.00€50mg522.00€100mg748.00€200mg1,026.00€1mL*10mM (DMSO)111.00€Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74CID 1375606
CAS:CID 1375606: Surrogate agonist for GPR27, conserved in vertebrates, mainly in CNS.Formula:C20H14Cl2N2O2Purity:99.41%Color and Shape:SolidMolecular weight:385.24SAG
CAS:SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.
Formula:C28H28ClN3OSPurity:97.37% - 98.88%Color and Shape:SolidMolecular weight:490.06Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Purity:98.27%Color and Shape:LiquidMolecular weight:N/ASubstance P (7-11)
CAS:Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .Formula:C31H44N6O5SPurity:98.39%Color and Shape:SolidMolecular weight:612.78Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.Purity:95.44% - 99.73%Color and Shape:SolidMolecular weight:N/AOndansetron hydrochloride
CAS:Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormula:C18H19N3O·HClPurity:99.78%Color and Shape:White PowderMolecular weight:329.82NAV-2729
CAS:NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formula:C25H17ClN4O3Purity:98.83% - 98.91%Color and Shape:SolidMolecular weight:456.88Ref: TM-T5142
2mg43.00€5mg63.00€10mg90.00€25mg193.00€50mg286.00€100mg429.00€500mg888.00€1mL*10mM (DMSO)71.00€Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purity:98.13% - 99.66%Color and Shape:SolidMolecular weight:449.54Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Pentagastrin
CAS:Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormula:C37H49N7O9SPurity:96.98% - 99.49%Color and Shape:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMolecular weight:767.89Praliciguat
CAS:Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formula:C21H14F8N6O2Purity:98.82%Color and Shape:SolidMolecular weight:534.36Ref: TM-T16569
1mg142.00€2mg207.00€5mg349.00€10mg537.00€25mg858.00€50mg1,161.00€100mg1,558.00€1mL*10mM (DMSO)409.00€Riociguat
CAS:Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormula:C20H19FN8O2Purity:99.28% - 99.95%Color and Shape:SolidMolecular weight:422.42HhAntag
CAS:HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activityFormula:C24H23ClN4O3Purity:95.73%Color and Shape:SolidMolecular weight:450.92GW842166X
CAS:GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formula:C18H17Cl2F3N4O2Purity:99.47%Color and Shape:SolidMolecular weight:449.25BD 1008 Free Base
CAS:BD 1008 Free Base: Sigma-1 receptor antagonist, Kᵢ = 2 ± 1 nM, 4x more selective for sigma-1 than sigma-2.Formula:C15H22Cl2N2Color and Shape:SolidMolecular weight:301.25Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Formula:C21H28ClN3O3SColor and Shape:SolidMolecular weight:437.98[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2Formula:C40H68N8O10Purity:99.31%Color and Shape:SolidMolecular weight:821.02Ref: TM-T38807L
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)To inquireCCG215022
CAS:CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formula:C26H22FN7O3Purity:97.63% - 99.69%Color and Shape:SolidMolecular weight:499.5Ref: TM-T3498
1mg56.00€5mg114.00€10mg178.00€25mg394.00€50mg655.00€100mg1,035.00€1mL*10mM (DMSO)127.00€Arformoterol Tartrate
CAS:Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49Ref: TM-T22245
5mg60.00€10mg87.00€25mg150.00€50mg221.00€100mg329.00€200mg487.00€1mL*10mM (DMSO)85.00€BMS 182874 hydrochloride
CAS:BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formula:C17H20ClN3O3SPurity:97.01%Color and Shape:SolidMolecular weight:381.88Ref: TM-T21790
1mg77.00€2mg92.00€5mg140.00€10mg205.00€25mg343.00€50mg477.00€100mg665.00€200mg897.00€1mL*10mM (DMSO)146.00€Tolnapersine
CAS:Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Formula:C21H26N2OPurity:98%Color and Shape:SolidMolecular weight:322.44Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formula:C14H22ClN3O2SColor and Shape:SolidMolecular weight:331.86AC 187 Acetate
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.Formula:C129H209N37O42Purity:99.71%Color and Shape:SolidMolecular weight:2950.26Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29AC-55541
CAS:AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.58%Color and Shape:SolidMolecular weight:330.44Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Ivabradine hydrochloride
CAS:Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formula:C27H37ClN2O5Purity:99% - 99.73%Color and Shape:SolidMolecular weight:505.05Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formula:C36H55F3N8O12SPurity:>99.99%Color and Shape:SolidMolecular weight:880.93DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formula:C35H56N10O15Purity:>99.99%Color and Shape:SolidMolecular weight:856.88[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formula:C69H108N22O16SPurity:99.71%Color and Shape:SolidMolecular weight:1533.8VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35Ref: TM-T29112
1mg49.00€5mg96.00€10mg124.00€25mg222.00€50mg309.00€100mg439.00€200mg592.00€1mL*10mM (DMSO)88.00€SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Ref: TM-T3183
1mg79.00€5mg152.00€10mg245.00€25mg398.00€50mg532.00€100mg735.00€200mg973.00€1mL*10mM (DMSO)166.00€GRA Ex-25
CAS:GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03Ref: TM-T7617L
1mg35.00€5mg73.00€10mg107.00€25mg207.00€50mg313.00€100mg447.00€200mg620.00€1mL*10mM (DMSO)132.00€D3-βArr
CAS:D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by directFormula:C20H23N5Purity:98.82%Color and Shape:SolidMolecular weight:333.43Cimetidine hydrochloride
CAS:Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.Formula:C10H17ClN6SColor and Shape:SolidMolecular weight:288.8Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formula:C25H18ClN5O2S2Purity:98.85% - 99.57%Color and Shape:SolidMolecular weight:520.03Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurity:94.61%Color and Shape:SolidMolecular weight:2996.45Carmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Formula:C24H26N2O2Color and Shape:SolidMolecular weight:374.48SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€1mL*10mM (DMSO)150.00€CYM2503
CAS:CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.
Formula:C45H55N5O7Purity:97.04%Color and Shape:SolidMolecular weight:777.95Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formula:C61H93N19O15SPurity:99.68% - 99.90%Color and Shape:SolidMolecular weight:1364.57Ref: TM-T22344
1mg66.00€2mg92.00€5mg177.00€10mg281.00€25mg475.00€50mg677.00€100mg888.00€1mL*10mM (DMSO)355.00€Parethoxycaine hydrochloride
CAS:Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81Ref: TM-T9397
1mg93.00€5mg182.00€10mg266.00€25mg425.00€50mg605.00€100mg803.00€200mg1,063.00€1mL*10mM (DMSO)177.00€Methyldopa hydrate
CAS:Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formula:C10H13NO4H2OPurity:99.67%Color and Shape:White SolidMolecular weight:238.24Melanotan I
CAS:Melanotan I is a non-specific melanocortin receptor (MCR) agonist, an α-melanocyte-stimulating hormone (α-MSH) analog, which is injected subcutaneously toFormula:C78H111N21O19Purity:>99.99%Color and Shape:SolidMolecular weight:1646.85ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formula:C13H16ClN3O3Purity:98.15%Color and Shape:SolidMolecular weight:297.74Ref: TM-T9193
1mg52.00€5mg116.00€10mg182.00€25mg320.00€50mg449.00€100mg615.00€200mg830.00€1mL*10mM (DMSO)128.00€BD-1047 dihydrobromide
CAS:BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormula:C13H22Br2Cl2N2Purity:98.13% - 99.39%Color and Shape:SolidMolecular weight:437.04Ref: TM-T1740
1mg37.00€2mg48.00€5mg73.00€10mg95.00€25mg168.00€50mg290.00€100mg490.00€1mL*10mM (DMSO)74.00€Adenosine receptor antagonist 4
CAS:Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formula:C10H13N3Purity:99.63% - 99.65%Color and Shape:Off-White PowderMolecular weight:175.23Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Formula:C20H33NO7Purity:99.26%Color and Shape:White Crystalline PowdeMolecular weight:399.48carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.
Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59Phosphorylcholine chloride
CAS:Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integralFormula:C5H15ClNO4PPurity:99.481% - 99.85%Color and Shape:SolidMolecular weight:219.6Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurity:99.91%Color and Shape:SolidMolecular weight:456.49Ambrisentan
CAS:Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.Formula:C22H22N2O4Purity:99.65% - 99.86%Color and Shape:SolidMolecular weight:378.42Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formula:C23H29F2N3OPurity:99.68%Color and Shape:SolidMolecular weight:401.49Ref: TM-T23733
1mg87.00€5mg178.00€10mg295.00€25mg497.00€50mg708.00€100mg964.00€500mg1,918.00€1mL*10mM (DMSO)321.00€Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate
Formula:C21H32Cl2N4OPurity:99.68% - 99.87%Color and Shape:SolidMolecular weight:427.41Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formula:C21H27N3Purity:98%Color and Shape:SolidMolecular weight:321.46Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1g505.00€10mg50.00€25mg69.00€50mg95.00€100mg124.00€200mg215.00€500mg350.00€1mL*10mM (DMSO)48.00€Thozalinone
CAS:Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.Formula:C11H12N2O2Purity:99.68%Color and Shape:SolidMolecular weight:204.231-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Formula:C40H42ClN5O7Purity:97.94% - 98.4%Color and Shape:SolidMolecular weight:740.24Fipamezole HCl
CAS:Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.Formula:C14H16ClFN2Color and Shape:SolidMolecular weight:266.74ML382
CAS:ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
Formula:C18H20N2O4SPurity:99.79%Color and Shape:SolidMolecular weight:360.43Prazosin
CAS:Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Formula:C19H21N5O4Purity:99.86%Color and Shape:White To Tan Powder SolidMolecular weight:383.4DORA-22
CAS:DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormula:C23H22F2N4O2Purity:97.67%Color and Shape:SolidMolecular weight:424.44Ref: TM-T5500
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)331.00€ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formula:C20H19F5N2OPurity:99.73%Color and Shape:SolidMolecular weight:398.37Ref: TM-T7103
1mg88.00€2mg118.00€5mg188.00€10mg254.00€25mg429.00€50mg630.00€100mg898.00€1mL*10mM (DMSO)187.00€ACTH (1-17) acetate
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).Formula:C97H149N29O25SPurity:98.53%Color and Shape:SolidMolecular weight:2153.47MEN 10207 acetate
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.Formula:C59H72N14O12Purity:99.18%Color and Shape:SolidMolecular weight:1169.29GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formula:C149H226N40O45Purity:99.85%Color and Shape:White PowderMolecular weight:3297.63Lidamidine Hydrochloride
CAS:Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formula:C11H17ClN4OColor and Shape:SolidMolecular weight:256.73Piperoxan hydrochloride
CAS:Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77Ref: TM-T4526
2mg39.00€5mg62.00€10mg92.00€25mg128.00€50mg166.00€100mg200.00€200mg299.00€1mL*10mM (DMSO)55.00€Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formula:C18H18ClN3OPurity:99.88%Color and Shape:Pale Yellowish Crystals From Petroleum Ether SolidMolecular weight:327.812-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09TG4-155
CAS:TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.
Formula:C23H26N2O4Purity:97.2%Color and Shape:SolidMolecular weight:394.46Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.Formula:C38H60F6N8O10SPurity:99%Color and Shape:SolidMolecular weight:934.99Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formula:C28H28F2N6O3Purity:99.1% - 99.99%Color and Shape:SolidMolecular weight:534.56Rolapitant hydrochloride hydrate
CAS:Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.Formula:C25H29ClF6N2O3Color and Shape:SolidMolecular weight:554.95Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formula:C15H21N5O4SColor and Shape:SolidMolecular weight:367.42M40 acetate(143896-17-7 free base)
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)Formula:C96H149N23O26Purity:99.88%Color and Shape:SolidMolecular weight:2041.38NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Laropiprant sodium
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.Color and Shape:SolidAlosetron (Hydrochloride(1:X))
CAS:Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.Formula:C17H18ClN4OColor and Shape:SolidMolecular weight:329.11691Flibanserin hydrochloride
CAS:Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formula:C20H22ClF3N4OColor and Shape:SolidMolecular weight:426.87Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).
Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Norepinephrine bitartrate salt
CAS:Norepinephrine bitartrate salt is an adrenergic neurotransmitter.Formula:C12H17NO9Purity:97.32% - 99.97%Color and Shape:SolidMolecular weight:319.27Brimonidine
CAS:Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.Formula:C11H10BrN5Purity:99.626%Color and Shape:Yellow SolidMolecular weight:292.13Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formula:C17H25ClN2O2Purity:97.91%Color and Shape:SolidMolecular weight:324.85Ref: TM-T4087
1mg39.00€5mg74.00€10mg97.00€25mg167.00€50mg239.00€100mg340.00€200mg460.00€1mL*10mM (DMSO)74.00€Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purity:98.76% - 99.79%Color and Shape:SolidMolecular weight:295.38
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