GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Ertugliflozin
CAS:PF-04971729 (Ertugliflozin (PF-04971729)) is a potent and selective inhibitor of the sodium-dependent glucose cotransporter 2 (SGLT2).Formula:C22H25ClO7Purity:99.89% - 99.96%Color and Shape:SolidMolecular weight:436.88Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.Purity:98%Color and Shape:LiquidMolecular weight:N/ACinaciguat
CAS:Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:C36H39NO5Purity:98% - 99.18%Color and Shape:SolidMolecular weight:565.7Doxazosin
CAS:Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formula:C23H25N5O5Purity:99.47% - 99.87%Color and Shape:SolidMolecular weight:451.48Dexmedetomidine hydrochloride
CAS:Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C13H16N2·HClPurity:99.94% - 99.94%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:236.74Ref: TM-T6466
5mg42.00€10mg55.00€25mg88.00€50mg159.00€100mg226.00€200mg340.00€500mg563.00€1mL*10mM (DMSO)50.00€Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formula:C11H21NColor and Shape:SolidMolecular weight:167.29Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].Purity:99.24%Color and Shape:LiquidMolecular weight:N/AConivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFormula:C32H26N4O2·HClPurity:98.33% - 99.86%Color and Shape:SolidMolecular weight:535.04Tribenoside
CAS:Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formula:C29H34O6Purity:≥98%Color and Shape:LiquidMolecular weight:478.58Haloperidol decanoate
CAS:Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.Formula:C31H41ClFNO3Purity:99.57% - 99.72%Color and Shape:SolidMolecular weight:530.11Ref: TM-T25487
5mg48.00€10mg66.00€25mg117.00€50mg170.00€100mg255.00€200mg373.00€1mL*10mM (DMSO)50.00€TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formula:C27H26N4O2SPurity:99.35% - 99.52%Color and Shape:SolidMolecular weight:470.59Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formula:C21H29ClN2O5Purity:99.52%Color and Shape:SolidMolecular weight:424.92OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.58%Color and Shape:SolidMolecular weight:330.44EST64454 hydrochloride
CAS:EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.Formula:C18H23ClF2N4O2Purity:99.15%Color and Shape:SolidMolecular weight:400.85Ref: TM-T8834
2mg42.00€5mg62.00€10mg92.00€25mg187.00€50mg304.00€100mg482.00€200mg662.00€1mL*10mM (DMSO)77.00€Ro 46-2005
CAS:Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).Formula:C23H27N3O6SPurity:98.02% - 98.8%Color and Shape:SolidMolecular weight:473.54SBI-115
CAS:SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5Formula:C14H13ClN2O4SPurity:99.53% - 99.78%Color and Shape:SolidMolecular weight:340.78Terazosin hydrochloride dihydrate
CAS:Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.922-ATHBI
CAS:2-ATHBI is a S1P lyase inhibitor.Formula:C9H14N2O5Purity:99.10%Color and Shape:SolidMolecular weight:230.22BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formula:C34H51N5NaO7Color and Shape:SolidMolecular weight:664.8Taprenepag
CAS:Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).Formula:C24H22N4O5SPurity:98.89% - 99.15%Color and Shape:SolidMolecular weight:478.52Ref: TM-T3174
1mg34.00€5mg62.00€10mg92.00€25mg178.00€50mg295.00€100mg425.00€200mg595.00€1mL*10mM (DMSO)66.00€Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:391.34Ref: TM-T16999
1mg77.00€5mg166.00€10mg260.00€25mg475.00€50mg668.00€100mg888.00€1mL*10mM (DMSO)178.00€Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Ref: TM-T5389
1mg39.00€5mg84.00€10mg117.00€25mg220.00€50mg285.00€100mg371.00€200mg530.00€1mL*10mM (DMSO)92.00€HAEGTFTSDVSSYLE
HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.
Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formula:C14H22ClN3O2SColor and Shape:SolidMolecular weight:331.86N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Ref: TM-T5158
2mg34.00€5mg48.00€10mg79.00€25mg152.00€50mg235.00€100mg344.00€200mg490.00€1mL*10mM (DMSO)58.00€Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43Chlorphenesin
CAS:Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.Formula:C9H11ClO3Purity:99.59%Color and Shape:SolidMolecular weight:202.63Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg42.00€5mg62.00€10mg88.00€25mg141.00€50mg215.00€100mg318.00€200mg442.00€1mL*10mM (DMSO)59.00€9-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.37%Color and Shape:SolidMolecular weight:163.18HPI 1
CAS:HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formula:C27H29NO6Purity:97.6%Color and Shape:SolidMolecular weight:463.52Ref: TM-T22089
1mg47.00€2mg60.00€5mg92.00€10mg135.00€25mg217.00€50mg324.00€100mg472.00€500mg1,026.00€1mL*10mM (DMSO)107.00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.Formula:C143H235N41O45SPurity:97.12%Color and Shape:SolidMolecular weight:3280.76LY 78335
CAS:LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.Formula:C8H10Cl3NPurity:99.30% - 99.81%Color and Shape:SolidMolecular weight:226.53Peptide YY (PYY) (3-36), human
CAS:Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formula:C176H272N52O54Purity:97.76%Color and Shape:SolidMolecular weight:3980.42SORT-PGRN interaction inhibitor 1
CAS:SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).Formula:C15H18N2O2Purity:98.72%Color and Shape:SolidMolecular weight:258.32Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formula:C22H32ClN3O2Color and Shape:SolidMolecular weight:405.96Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Ivabradine hydrochloride
CAS:Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formula:C27H37ClN2O5Purity:99% - 99.73%Color and Shape:SolidMolecular weight:505.05AZ3451
CAS:AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).Formula:C30H27BrN4O3Purity:98.12%Color and Shape:SolidMolecular weight:571.46Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS:Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-Formula:C24H35ClO9Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:502.98Hydroxyzine dihydrochloride
CAS:Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formula:C21H27ClN2O2·2HClPurity:99.46% - 99.79%Color and Shape:Oil PowderMolecular weight:447.83Nomifensine maleate
CAS:Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
Formula:C20H22N2O4Purity:98.46%Color and Shape:SolidMolecular weight:354.4CRT0273750
CAS:CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formula:C25H22ClF3N4O2Purity:99.91%Color and Shape:SolidMolecular weight:502.92PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Formula:C26H32O4Purity:98.53%Color and Shape:SolidMolecular weight:408.53Ref: TM-T8975
1mg35.00€5mg80.00€10mg119.00€25mg231.00€50mg344.00€100mg480.00€200mg660.00€1mL*10mM (DMSO)87.00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Ref: TM-T5031
2mg35.00€5mg52.00€10mg80.00€25mg144.00€50mg227.00€100mg359.00€200mg532.00€1mL*10mM (DMSO)74.00€Fosaprepitant dimeglumine
CAS:Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.
Formula:C37H56F7N6O16PPurity:98% - 99.03%Color and Shape:SolidMolecular weight:1004.83Dobutamine
CAS:Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Formula:C59H82F3N13O14Purity:>99.99%Color and Shape:SolidMolecular weight:1254.36Idazoxan hydrochloride
CAS:Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.Formula:C11H12N2O2·HClPurity:99.42% - 99.84%Color and Shape:SolidMolecular weight:240.69Ref: TM-T0115
2mg35.00€5mg52.00€10mg78.00€25mg133.00€50mg187.00€100mg281.00€200mg416.00€1mL*10mM (DMSO)50.00€RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formula:C25H27N3O3Purity:98.64% - 99.62%Color and Shape:SolidMolecular weight:417.5NPY 5RA972
CAS:NPY 5RA972 is a neuropeptide Y Y5 receptor antagonistFormula:C21H25N3O2Purity:99.02% - 99.56%Color and Shape:SolidMolecular weight:351.44Cimetidine hydrochloride
CAS:Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.Formula:C10H17ClN6SColor and Shape:SolidMolecular weight:288.8YIL781 hydrochloride
CAS:YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).Formula:C24H29ClFN3O2Color and Shape:SolidMolecular weight:445.96CGS 21680 Hydrochloride
CAS:CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formula:C23H29N7O6·HClPurity:96.74% - 99.53%Color and Shape:SolidMolecular weight:535.98Ref: TM-T6441
1mg38.00€2mg50.00€5mg81.00€10mg109.00€25mg215.00€50mg389.00€100mg575.00€1mL*10mM (DMSO)95.00€Montelukast dicyclohexylamine
CAS:Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.Formula:C47H59ClN2O3SColor and Shape:SolidMolecular weight:767.5MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formula:C22H28FNO3Purity:98.96%Color and Shape:SolidMolecular weight:373.46Ref: TM-T22359
1mg99.00€5mg187.00€10mg280.00€25mg434.00€50mg585.00€100mg775.00€200mg1,054.00€1mL*10mM (DMSO)222.00€Midodrine
CAS:Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formula:C12H18N2O4Purity:99.89%Color and Shape:SolidMolecular weight:254.28BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21%Color and Shape:SolidMolecular weight:372.89BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurity:98.07%Color and Shape:SolidMolecular weight:230.31DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formula:C35H56N10O15Purity:>99.99%Color and Shape:SolidMolecular weight:856.88Tetradecyl Phosphonate
CAS:Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formula:C14H31O3PPurity:99.95%Color and Shape:White To Off-White PowderMolecular weight:278.37Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.572-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.Formula:C38H64F3N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:891.98Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.Formula:C169H256N42O57Purity:98.28%Color and Shape:SolidMolecular weight:3788.14Bosentan
CAS:Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.Formula:C27H29N5O6SPurity:99.74% - 99.84%Color and Shape:Pale Yellow To Off-White SolidMolecular weight:551.614Ref: TM-T6264
10mg38.00€25mg56.00€50mg81.00€100mg127.00€200mg207.00€500mg294.00€1mL*10mM (DMSO)88.00€4i
CAS:4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formula:C16H12ClN3OPurity:99.49%Color and Shape:SolidMolecular weight:297.74Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4Formula:C59H69F3N12O12Purity:99.22%Color and Shape:SolidMolecular weight:1195.25Bimatoprost
CAS:Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocularFormula:C25H37NO4Purity:98% - >99.99%Color and Shape:Crystalline SolidMolecular weight:415.57Ref: TM-T2538
2mg34.00€5mg48.00€10mg75.00€25mg127.00€50mg219.00€100mg371.00€200mg547.00€1mL*10mM (DMSO)50.00€Blarcamesine
CAS:Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
Formula:C19H23NOPurity:99.87%Color and Shape:SolidMolecular weight:281.39MK-0557
CAS:MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).Formula:C22H19FN4O3Purity:99.88%Color and Shape:SolidMolecular weight:406.41Ref: TM-TQ0286
1mg34.00€5mg67.00€10mg92.00€25mg166.00€50mg264.00€100mg371.00€200mg517.00€1mL*10mM (DMSO)75.00€SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Ref: TM-T6979
1mg40.00€2mg51.00€5mg85.00€10mg125.00€25mg225.00€50mg364.00€100mg582.00€1mL*10mM (DMSO)86.00€OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formula:C79H125N23O22Purity:98.52%Color and Shape:SolidMolecular weight:1748.98Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03Ref: TM-T7617L
1mg35.00€5mg73.00€10mg107.00€25mg207.00€50mg313.00€100mg447.00€200mg620.00€1mL*10mM (DMSO)132.00€Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.Formula:C42H69N13O12Purity:98.37%Color and Shape:SolidMolecular weight:948.08C14TKL-1 acetate
C14TKL-1 acetate is a NK1 receptor agonist.Formula:C65H102N20O15S2Purity:98.56%Color and Shape:SolidMolecular weight:1467.75SB-649868
CAS:SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).Formula:C26H24FN3O3SPurity:99.53%Color and Shape:SolidMolecular weight:477.55Ref: TM-T5498
2mg37.00€5mg74.00€10mg116.00€25mg239.00€50mg386.00€100mg620.00€200mg832.00€1mL*10mM (DMSO)90.00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purity:99.95%Color and Shape:SolidMolecular weight:805.9Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurity:98.65% - 99.94%Color and Shape:SolidMolecular weight:342.82CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurity:98% - 99.83%Color and Shape:SolidMolecular weight:324.24Ref: TM-T4369
1mg39.00€2mg50.00€5mg78.00€10mg97.00€25mg195.00€50mg369.00€100mg550.00€1mL*10mM (DMSO)78.00€Butyrophenone
CAS:Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.Formula:C10H12OPurity:99.84%Color and Shape:Colourless To Yellow LiquidMolecular weight:148.2Ibutamoren Mesylate
CAS:Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.Formula:C28H40N4O8S2Purity:97.98% - ≥98%Color and Shape:SolidMolecular weight:624.77AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:98.87%Color and Shape:SolidMolecular weight:478.47Ref: TM-T2000
1mg35.00€2mg47.00€5mg66.00€10mg97.00€25mg180.00€50mg283.00€100mg439.00€1mL*10mM (DMSO)70.00€Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Ref: TM-TQ0227
1mg50.00€5mg105.00€10mg170.00€25mg230.00€50mg289.00€100mg401.00€1mL*10mM (DMSO)107.00€Bromodiphenhydramine
CAS:Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.Formula:C17H20BrNOColor and Shape:SolidMolecular weight:334.25Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formula:C17H20N2O2SPurity:98%Color and Shape:SolidMolecular weight:316.42ML-18
CAS:ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.Formula:C32H35N5O5Purity:98.62% - >99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-T4540
1mg34.00€5mg60.00€10mg96.00€25mg170.00€50mg264.00€100mg425.00€200mg587.00€1mL*10mM (DMSO)75.00€Lidamidine Hydrochloride
CAS:Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formula:C11H17ClN4OColor and Shape:SolidMolecular weight:256.73Vercirnon sodium
CAS:Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formula:C22H21ClN2NaO4SColor and Shape:SolidMolecular weight:467.92Bunazosin
CAS:Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45Ipragliflozin
CAS:Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
Formula:C21H21FO5SPurity:99.38% - 99.70%Color and Shape:SolidMolecular weight:404.45Laropiprant sodium
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.Color and Shape:SolidT-1095
CAS:T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).Formula:C26H28O11Purity:99.78%Color and Shape:SolidMolecular weight:516.49Ref: TM-T9590
1mg50.00€2mg71.00€5mg90.00€10mg130.00€25mg207.00€50mg370.00€100mg530.00€1mL*10mM (DMSO)127.00€Desipramine
CAS:Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.Formula:C18H22N2Color and Shape:SolidMolecular weight:266.38Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurity:99.99%Color and Shape:Crystalline SolidMolecular weight:327.90Ref: TM-T4274
10mg44.00€25mg64.00€50mg93.00€100mg110.00€200mg161.00€500mg264.00€1mL*10mM (DMSO)48.00€Guanabenz hydrochloride
CAS:Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formula:C8H9Cl3N4Purity:99.45%Color and Shape:SolidMolecular weight:267.54Secretin (33-59), rat
CAS:Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35TCS-OX2-29
CAS:TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.Formula:C23H31N3O3Purity:99.81%Color and Shape:SolidMolecular weight:397.51Ref: TM-T4965
1mg35.00€5mg70.00€10mg96.00€25mg156.00€50mg215.00€100mg303.00€200mg449.00€1mL*10mM (DMSO)77.00€Dazoxiben
CAS:Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase
Formula:C12H13ClN2O3Purity:99.99%Color and Shape:SolidMolecular weight:268.7RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.
Formula:C17H16FN3Purity:99.32%Color and Shape:SolidMolecular weight:281.33Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formula:C20H25ClN2OSPurity:99.17%Color and Shape:SolidMolecular weight:376.94Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurity:99.91%Color and Shape:SolidMolecular weight:456.49Ozanimod
CAS:Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formula:C23H24N4O3Purity:98.68% - 99.58%Color and Shape:SolidMolecular weight:404.46Ref: TM-T6923
1mg46.00€5mg90.00€10mg137.00€25mg268.00€50mg430.00€100mg622.00€200mg879.00€500mg1,305.00€1mL*10mM (DMSO)90.00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Ref: TM-T5520L
1mg52.00€5mg90.00€10mg150.00€25mg291.00€50mg437.00€100mg642.00€500mg1,359.00€1mL*10mM (DMSO)251.00€Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
2mg35.00€5mg51.00€10mg88.00€25mg120.00€50mg170.00€100mg250.00€200mg373.00€1mL*10mM (DMSO)57.00€Pimavanserin
CAS:Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55Ondansetron hydrochloride
CAS:Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormula:C18H19N3O·HClPurity:99.78%Color and Shape:White PowderMolecular weight:329.82Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.Formula:C63H104N22O17SPurity:98.33%Color and Shape:SolidMolecular weight:1473.72MHP
CAS:MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.Formula:C16H23NO4Purity:98.58%Color and Shape:SolidMolecular weight:293.36Ref: TM-T4658
1mg34.00€2mg46.00€5mg66.00€10mg101.00€25mg207.00€50mg334.00€100mg537.00€200mg762.00€1mL*10mM (DMSO)73.00€JNJ-31020028
CAS:JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68Senktide
CAS:Senktide is an agonist of tachykinin NK3 receptor.Formula:C40H55N7O11SPurity:99.84% - >99.99%Color and Shape:White PowderMolecular weight:841.97Terutroban
CAS:Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.Formula:C20H22ClNO4SPurity:99.53%Color and Shape:SolidMolecular weight:407.91Otenabant hydrochloride
CAS:Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formula:C25H26Cl3N7OPurity:99.79% - ≥95%Color and Shape:SolidMolecular weight:546.88CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purity:99.08% - 99.76%Color and Shape:SolidMolecular weight:751.67Ref: TM-T5996
1mg82.00€2mg110.00€5mg180.00€10mg258.00€25mg423.00€50mg588.00€100mg793.00€500mg1,594.00€1mL*10mM (DMSO)215.00€Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg50.00€10mg73.00€25mg138.00€50mg241.00€100mg358.00€200mg523.00€500mg822.00€1mL*10mM (DMSO)52.00€Pranlukast hemihydrate
CAS:Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.Formula:C27H23N5O40·5H2OPurity:99.28%Color and Shape:SolidMolecular weight:490.52carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59AP1189 acetate
CAS:AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
Formula:C16H18N6O4Purity:99.95%Color and Shape:SolidMolecular weight:358.35Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formula:C20H20NO4Purity:97.18% - 99.06%Color and Shape:SolidMolecular weight:338.38Talastine HCl
CAS:Talastine is an antihistamine drug.Formula:C19H22ClN3OPurity:98%Color and Shape:SolidMolecular weight:343.86Thozalinone
CAS:Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.Formula:C11H12N2O2Purity:99.68%Color and Shape:SolidMolecular weight:204.23Parethoxycaine hydrochloride
CAS:Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].Formula:C15H24ClNO3Purity:99.46%Color and Shape:SolidMolecular weight:301.81Ref: TM-T9397
1mg93.00€5mg182.00€10mg266.00€25mg425.00€50mg605.00€100mg803.00€200mg1,063.00€1mL*10mM (DMSO)177.00€Solabegron HCl
CAS:Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.Formula:C23H24Cl2N2O3Color and Shape:SolidMolecular weight:447.35Neuropeptide W-23(human)
CAS:Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2.Formula:C119H183N35O28SPurity:98.5%Color and Shape:SolidMolecular weight:2584.01Ref: TM-TP1073
1mg114.00€2mg177.00€5mg334.00€10mg485.00€25mg770.00€50mg1,035.00€100mg1,395.00€500mg2,673.00€Gastrin I (1-14), human
CAS:Gastrin I (1-14), human: a short peptide from the hormone gastrin, which regulates gastric acid secretion.Formula:C79H100N16O27Purity:98.19%Color and Shape:SolidMolecular weight:1705.73EST64454 Maleic acid salt
CAS:EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.Formula:C22H26F2N4O6Purity:97.54%Color and Shape:SolidMolecular weight:480.46Ref: TM-T9306
1mg88.00€5mg172.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)207.00€Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Formula:C26H29N5O3SPurity:99.49% - 99.843%Color and Shape:SolidMolecular weight:491.61DOPEXAMINE
CAS:Dopexamine is a dopaminergic agonistFormula:C22H32N2O2Purity:99.42%Color and Shape:SolidMolecular weight:356.5Ref: TM-T8653
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)306.00€Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purity:99.12%Color and Shape:SolidMolecular weight:307.139Ref: TM-T21970
5mg62.00€10mg90.00€25mg133.00€50mg192.00€100mg286.00€500mg687.00€1mL*10mM (DMSO)67.00€[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2Formula:C40H68N8O10Purity:99.31%Color and Shape:SolidMolecular weight:821.02Ref: TM-T38807L
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€1mL*10mM (DMSO)To inquireCarmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Formula:C24H26N2O2Color and Shape:SolidMolecular weight:374.48Vicriviroc
CAS:Vicriviroc, also known as MK4176 is a CCR5 antagonist.Formula:C28H38F3N5O2Color and Shape:SolidMolecular weight:533.63Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1g477.00€10mg48.00€25mg65.00€50mg90.00€100mg117.00€200mg203.00€500mg333.00€1mL*10mM (DMSO)46.00€CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43Ref: TM-T7183
2mg34.00€5mg52.00€10mg73.00€25mg128.00€50mg197.00€100mg295.00€200mg442.00€1mL*10mM (DMSO)52.00€Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formula:C24H29ClFNO5Color and Shape:SolidMolecular weight:465.95Exo1
CAS:Exo1 is an inhibitor of the exocytic pathwayFormula:C15H12FNO3Purity:98.75%Color and Shape:SolidMolecular weight:273.26Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9GUANABENZ
CAS:GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.Formula:C8H8Cl2N4Purity:98.31%Color and Shape:White Solid From Acetonitrile SolidMolecular weight:231.08MK-571 sodium
CAS:MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formula:C26H27ClN2O3S2·NaPurity:97.86% - 99.58%Color and Shape:SolidMolecular weight:537.07Ref: TM-T3148
2mgTo inquire5mg50.00€10mg75.00€25mg157.00€50mg270.00€100mg404.00€1mL*10mM (DMSO)63.00€E7046
CAS:E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.Formula:C22H18F5N3O4Purity:99.86%Color and Shape:SolidMolecular weight:483.4Dobutamine hydrochloride
CAS:Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227Selexipag
CAS:Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.Formula:C26H32N4O4SPurity:99.98% - >99.99%Color and Shape:SolidMolecular weight:496.62Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Color and Shape:SolidMolecular weight:310.35Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Color and Shape:SolidMolecular weight:372.72Arformoterol Tartrate
CAS:Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49Ref: TM-T22245
5mg60.00€10mg87.00€25mg150.00€50mg221.00€100mg329.00€200mg487.00€1mL*10mM (DMSO)85.00€BMS 182874 hydrochloride
CAS:BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formula:C17H20ClN3O3SPurity:97.01%Color and Shape:SolidMolecular weight:381.88Ref: TM-T21790
1mg77.00€2mg92.00€5mg140.00€10mg205.00€25mg343.00€50mg477.00€100mg665.00€200mg897.00€1mL*10mM (DMSO)146.00€5-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurity:99.13%Color and Shape:SolidMolecular weight:280.36Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Color and Shape:SolidMolecular weight:497.63Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85Regadenoson
CAS:Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.35Ref: TM-T2671
2mg47.00€5mg65.00€10mg92.00€25mg173.00€50mg273.00€100mg416.00€500mg935.00€1mL*10mM (DMSO)72.00€S1RA hydrochloride
CAS:S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >Formula:C20H24ClN3O2Purity:98% - 99.84%Color and Shape:SolidMolecular weight:373.87Ref: TM-T4229
1mg35.00€5mg75.00€10mg105.00€25mg205.00€50mg334.00€100mg492.00€500mg973.00€1mL*10mM (DMSO)84.00€AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formula:C21H24ClF2NOPurity:99.89%Color and Shape:SolidMolecular weight:379.87Ref: TM-T39429
2mg34.00€5mg49.00€10mg75.00€25mg130.00€50mg192.00€100mg295.00€200mg442.00€1mL*10mM (DMSO)50.00€Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formula:C15H20Cl2N2O3Purity:99.17%Color and Shape:SolidMolecular weight:347.24ACEPROMAZINE MALEATE
CAS:ACEPROMAZINE MALEATE is a dopamine receptor antagonistFormula:C23H26N2O5SPurity:98.87% - 99.51%Color and Shape:Off White Or Yellow Crystalline PowderMolecular weight:442.53L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
Formula:C18H22Cl4N4Purity:97.52%Color and Shape:SolidMolecular weight:436.21Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formula:C36H55F3N8O12SPurity:>99.99%Color and Shape:SolidMolecular weight:880.93ZK 756326
CAS:ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formula:C21H28N2O3Purity:99.43%Color and Shape:SolidMolecular weight:356.46Clemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formula:C19H20ClN3Purity:98% - 99.65%Color and Shape:SolidMolecular weight:325.84Ref: TM-T1822
1mg44.00€5mg87.00€10mg106.00€25mg160.00€50mg270.00€100mg487.00€500mg1,026.00€1mL*10mM (DMSO)87.00€Taladegib
CAS:Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formula:C26H24F4N6OPurity:98.75% - >99.99%Color and Shape:SolidMolecular weight:512.5CCG215022
CAS:CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formula:C26H22FN7O3Purity:97.63% - 99.69%Color and Shape:SolidMolecular weight:499.5Ref: TM-T3498
1mg56.00€5mg114.00€10mg178.00€25mg394.00€50mg655.00€100mg1,035.00€1mL*10mM (DMSO)127.00€Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3PGS-IN-1
CAS:PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formula:C19H26O3Purity:99.39%Color and Shape:SolidMolecular weight:302.41Ref: TM-T10098
1mg52.00€5mg97.00€10mg170.00€25mg369.00€50mg540.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)110.00€HhAntag
CAS:HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activityFormula:C24H23ClN4O3Purity:95.73%Color and Shape:SolidMolecular weight:450.92MRT-10
CAS:MRT-10 is a Smoothened (Smo) receptor antagonist.
Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52RE-640
CAS:NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.Formula:C20H16Cl2N4Purity:99.60% - 99.87%Color and Shape:SolidMolecular weight:383.27Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formula:C46H65N13O11S2Purity:99.65%Color and Shape:SolidMolecular weight:1040.22Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purity:99.57% - 99.77%Color and Shape:SolidMolecular weight:417.97Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45M40 acetate(143896-17-7 free base)
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)Formula:C96H149N23O26Purity:99.88%Color and Shape:SolidMolecular weight:2041.38Gastrin I (human) acetate
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (Formula:C99H128N20O33SPurity:98.84%Color and Shape:SolidMolecular weight:2158.25ML-184
CAS:ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Formula:C25H34N4O3SPurity:99.45%Color and Shape:SolidMolecular weight:470.63GBR 12935 dihydrochloride
CAS:GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formula:C28H36Cl2N2OPurity:99.09% - ≥95%Color and Shape:SolidMolecular weight:487.5GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formula:C149H226N40O45Purity:99.85%Color and Shape:White PowderMolecular weight:3297.63ACTH (1-17) acetate
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).Formula:C97H149N29O25SPurity:98.53%Color and Shape:SolidMolecular weight:2153.47PF-04418948
CAS:PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.Formula:C23H20FNO5Purity:98.67% - 99.45%Color and Shape:SolidMolecular weight:409.41Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formula:C25H27N3O2SPurity:99.06% - 99.96%Color and Shape:SolidMolecular weight:433.57Ref: TM-T2306
5mg50.00€10mg63.00€25mg75.00€50mg88.00€100mg94.00€200mg140.00€500mg259.00€1mL*10mM (DMSO)To inquireTolazoline
CAS:Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formula:C10H12N2Purity:99.52%Color and Shape:SolidMolecular weight:160.22Levalbuterol tartrate
CAS:Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Formula:C17H27NO9Purity:99.28% - 99.98%Color and Shape:SolidMolecular weight:389.39Ref: TM-T7164
2mg34.00€5mg50.00€10mg88.00€25mg100.00€50mg124.00€100mg177.00€200mg259.00€1mL*10mM (DMSO)60.00€Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formula:C149H234N40O47SPurity:98% - 99.65%Color and Shape:SolidMolecular weight:3369.76Tiprenolol
CAS:Tiprenolol is a beta adrenergic receptor antagonist.[1]Formula:C13H21NO2SPurity:99.43%Color and Shape:SolidMolecular weight:255.38Ref: TM-T50081
1mg52.00€5mg98.00€10mg146.00€25mg235.00€50mg319.00€100mg447.00€200mg587.00€1mL*10mM (DMSO)89.00€Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormula:C43H77N17O12S2Purity:99.79%Color and Shape:SolidMolecular weight:1088.32AVN-101
CAS:AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formula:C21H25ClN2Purity:99.61%Color and Shape:SolidMolecular weight:340.89Ref: TM-T26690
1mg34.00€5mg75.00€10mg114.00€25mg205.00€50mg334.00€100mg557.00€200mg790.00€1mL*10mM (DMSO)92.00€NAN-190 hydrobromide
CAS:NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:C23H28BrN3O3Purity:95.20%Color and Shape:SolidMolecular weight:474.39Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purity:>99.99%Color and Shape:SolidMolecular weight:1120.26Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurity:99.78% - >99.99%Color and Shape:SolidMolecular weight:463.871-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.
Formula:C9H15N3OPurity:95%Color and Shape:SolidMolecular weight:181.23VKGILS-NH2 Acetate
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.Formula:C30H58N8O9Purity:98.83%Color and Shape:SolidMolecular weight:674.83Ref: TM-T21699L
1mg34.00€2mg52.00€5mg65.00€10mg97.00€25mg163.00€50mg235.00€100mg349.00€200mg497.00€1mL*10mM (DMSO)97.00€Pridopidine
CAS:Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formula:C15H23NO2SPurity:95.2% - 99.89%Color and Shape:SolidMolecular weight:281.41lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurity:95.83% - 99.95%Color and Shape:SolidMolecular weight:565.7Vilazodone Hydrochloride
CAS:Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormula:C26H27N5O2·HClPurity:99.56% - >99.99%Color and Shape:SolidMolecular weight:477.99PF-06291874
CAS:PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.Formula:C26H28F3N3O4Purity:99.12% - 99.27%Color and Shape:SolidMolecular weight:503.51
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