Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(51 products)
- Calcium Channel(493 products)
- Chloride channel(49 products)
- GABA Receptor(336 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(276 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2277 products of "Membrane Transporter/Ion Channel"
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GABAA receptor agent 1
CAS:<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formula:C13H8ClN3O2Purity:99.31%Color and Shape:SolidMolecular weight:273.67Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Vinpocetine
CAS:<p>Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).</p>Formula:C22H26N2O2Purity:99.85% - 99.98%Color and Shape:White Crystalline SolidMolecular weight:350.45FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Formula:C13H11N3OPurity:98.75%Color and Shape:SolidMolecular weight:225.25Hydrochlorothiazide
CAS:<p>Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。</p>Formula:C7H8ClN3O4S2Purity:99.43% - 99.50%Color and Shape:Crystals Physical Description Crystals Or White Powder (Ntp 1992)Molecular weight:297.74Riparin III
CAS:<p>Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.</p>Formula:C16H17NO4Purity:95.13%Color and Shape:SolidMolecular weight:287.31FFN 206 dihydrochloride
CAS:<p>FFN 206 dihydrochloride: fluorescent VMAT2 marker, detects subcellular sites, non-inhibitory to DAT.</p>Formula:C12H15ClN2O2Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:254.71Piracetam
CAS:<p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>Formula:C6H10N2O2Purity:97.16%Color and Shape:Crystals From Isopropanol SolidMolecular weight:142.16Afoxolaner
CAS:<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Formula:C26H17ClF9N3O3Purity:99.1% - 99.38%Color and Shape:SolidMolecular weight:625.87Flufenamic acid
CAS:<p>Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.</p>Formula:C14H10F3NO2Purity:98.68%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:281.23Alinidine
CAS:<p>Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.</p>Formula:C12H13Cl2N3Purity:98.91% - >99.99%Color and Shape:SolidMolecular weight:270.16Flindokalner
CAS:<p>Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.</p>Formula:C16H10ClF4NO2Purity:99.96%Color and Shape:SolidMolecular weight:359.7Glibenclamide
CAS:<p>Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.</p>Formula:C23H28ClN3O5SPurity:99.05% - 99.75%Color and Shape:SolidMolecular weight:494.00Gabapentin
CAS:<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Formula:C9H17NO2Purity:99.55% - 99.91%Color and Shape:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidMolecular weight:171.24BMS-394136
CAS:<p>BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.</p>Formula:C24H21Cl2FN4OPurity:98.19% - 98.67%Color and Shape:SolidMolecular weight:471.35Phenazopyridine hydrochloride
CAS:<p>Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.</p>Formula:C11H12ClN5Purity:99.27%Color and Shape:Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionMolecular weight:249.7RUVBL1/2 ATPase-IN-1
CAS:<p>RUVBL1/2 ATPase-IN-1 inhibits RUVBL1/2 ATPase (IC50: 6.0/7.7 μM); useful in cancer research.</p>Formula:C28H28F3N5OPurity:99.92%Color and Shape:SolidMolecular weight:507.55Endovion
CAS:<p>Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.</p>Formula:C16H9BrF6N6OPurity:98.51%Color and Shape:SolidMolecular weight:495.18NS8593 hydrochloride
CAS:<p>NS8593 hydrochloride (NS8593 HCl) is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels) .</p>Formula:C17H18ClN3Purity:99.77%Color and Shape:SolidMolecular weight:299.8Ropivacaine
CAS:<p>Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.</p>Formula:C17H26N2OPurity:97.75% - >99.99%Color and Shape:SolidMolecular weight:274.40Dyclonine hydrochloride
CAS:<p>Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .</p>Formula:C18H27NO2·HClPurity:99.35%Color and Shape:White Crystalline SolidMolecular weight:325.87(Z)-Capsaicin
CAS:<p>(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer of</p>Formula:C18H27NO3Purity:97.33% - 98.91%Color and Shape:SolidMolecular weight:305.41Nicorandil
CAS:<p>Nicorandil (SG-75)(Ikorel) acts by relaxing the smooth muscle of the blood vessels, especially those of the venous system.</p>Formula:C8H9N3O4Purity:98.14% - >99.99%Color and Shape:White Or Off-White PowderMolecular weight:211.17Tuvatexib
CAS:<p>Tuvatexib is a small molecule VDAC/HK2 dual modulator.</p>Formula:C21H23NO3Purity:97.29% - 99.80%Color and Shape:SolidMolecular weight:337.41Broflanilide
CAS:<p>Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.</p>Formula:C25H14BrF11N2O2Purity:99.82%Color and Shape:SolidMolecular weight:663.29NS1652
CAS:<p>NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.</p>Formula:C15H11F3N2O3Purity:99.62%Color and Shape:SolidMolecular weight:324.25BI-749327
CAS:<p>BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).</p>Formula:C23H21F3N4O2Purity:99.68%Color and Shape:SolidMolecular weight:442.43Zamicastat
CAS:<p>Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).</p>Formula:C21H21F2N3OSPurity:99.58%Color and Shape:SolidMolecular weight:401.47Pramocaine hydrochloride
CAS:<p>Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.</p>Formula:C17H27NO3·HClPurity:99.15% - 99.61%Color and Shape:Crystals White Or Off White Crystalline PowderMolecular weight:329.86VU0134992 hydrochloride
CAS:<p>VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).</p>Formula:C20H32BrClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:447.84NBQX disodium
CAS:<p>NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.</p>Formula:C12H6N4Na2O6SPurity:97.6% - 98.22%Color and Shape:SolidMolecular weight:380.2415Clorsulon
CAS:<p>Clorsulon (L631529) is utilized for the treatment of Fasciola hepatica infections in calves and sheep.</p>Formula:C8H8Cl3N3O4S2Purity:99.66% - 99.87%Color and Shape:White To Off-White Crystalline PowderMolecular weight:380.66Miconazole
CAS:<p>Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.</p>Formula:C18H14Cl4N2OPurity:98% - >99.99%Color and Shape:SolidMolecular weight:416.13Omeprazole
CAS:<p>Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.</p>Formula:C17H19N3O3SPurity:98.43% - 98.48%Color and Shape:White SolidMolecular weight:345.42Pivagabine
CAS:<p>Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.</p>Formula:C9H17NO3Purity:99.87%Color and Shape:SolidMolecular weight:187.24Phenelzine sulfate
CAS:<p>Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.</p>Formula:C8H14N2O4SPurity:98.38% - 99.83%Color and Shape:SolidMolecular weight:234.27Ropivacaine hydrochloride
CAS:<p>Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activity</p>Formula:C17H26N2O·HClPurity:99.85% - 99.95%Color and Shape:SolidMolecular weight:310.86Oxybutynin
CAS:<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Formula:C22H31NO3Purity:97.81% - 99.57%Color and Shape:White To Off-White Crystalline PowderMolecular weight:357.49N-Acetylprocainamide
CAS:<p>N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmic</p>Formula:C15H23N3O2Purity:99.65% - 99.74%Color and Shape:SolidMolecular weight:277.36VU591 hydrochloride
CAS:<p>VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.</p>Formula:C16H13ClN6O5Purity:98.93% - 99.22%Color and Shape:SolidMolecular weight:404.76Emamectin Benzoate
CAS:<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Formula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256Acetohexamide
CAS:<p>Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.</p>Formula:C15H20N2O4SPurity:99.19% - 99.85%Color and Shape:Crystals From 90% Aq EthanolMolecular weight:324.40Hydroxyhexamide
CAS:<p>Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.</p>Formula:C15H22N2O4SPurity:98.91%Color and Shape:SolidMolecular weight:326.41Gliclazide
CAS:<p>Gliclazide (SE1702), an oral antihyperglycemic agent, belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating beta-cells of the</p>Formula:C15H21N3O3SPurity:99.58%Color and Shape:SolidMolecular weight:323.41NS5806
CAS:<p>NS5806 activates K+ currents, slows KV4.2/4.3 decay with KChIP2, and boosts KV4.3/KChIP2 peaks (EC50=5.3μM).</p>Formula:C16H8Br2F6N6OPurity:97.95%Color and Shape:SolidMolecular weight:574.07Meticrane
CAS:<p>Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.</p>Formula:C10H13NO4S2Purity:99.16%Color and Shape:SolidMolecular weight:275.34BIIB 722 Mesylate
CAS:<p>BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.</p>Formula:C19H23F3N6O5SPurity:99.57%Color and Shape:SoildMolecular weight:504.483VU591
CAS:VU591 is a selective extra-renal potassium channel inhibitor with an IC₅₀ of 0.24 μM.Formula:C16H12N6O5Purity:99.29% - 99.53%Color and Shape:SolidMolecular weight:368.3Gut restricted-7
CAS:<p>Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.</p>Formula:C25H40FNaO6SPurity:98.81% - 99.27%Color and Shape:SolidMolecular weight:510.64Omeprazole metabolite Omeprazole sulfone
CAS:<p>Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.</p>Formula:C17H19N3O4SPurity:99.87%Color and Shape:SolidMolecular weight:361.42Nikethamide
CAS:<p>Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of end</p>Formula:C10H14N2OPurity:99.42%Color and Shape:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Molecular weight:178.23Eleclazine hydrochloride
CAS:<p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>Formula:C21H17ClF3N3O3Purity:99.86%Color and Shape:SolidMolecular weight:451.83Phenformin hydrochloride
CAS:<p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>Formula:C10H16ClN5Purity:97.11% - 99.80%Color and Shape:Lactic AcidosisMolecular weight:241.72NS19504
CAS:<p>NS19504 is an activator of Ca2+-activated K+ channel with EC50 of 11.0 µM.</p>Formula:C10H9BrN2SPurity:99.87%Color and Shape:SolidMolecular weight:269.16Omeprazole sulfide
CAS:<p>Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.</p>Formula:C17H19N3O2SPurity:98.83%Color and Shape:White To Slightly Collored Solid Solid CrystallineMolecular weight:329.42ICA-27243
CAS:<p>ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.</p>Formula:C12H7ClF2N2OPurity:99.54%Color and Shape:SolidMolecular weight:268.65Baclofen
CAS:<p>Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.</p>Formula:C10H12ClNO2Purity:98% - >99.99%Color and Shape:1992)Molecular weight:213.66Azosemide
CAS:<p>Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).</p>Formula:C12H11ClN6O2S2Purity:99.84%Color and Shape:SolidMolecular weight:370.84NMDA-IN-1
CAS:<p>NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).</p>Formula:C20H23ClFN3OPurity:99.57%Color and Shape:SolidMolecular weight:375.87L-Cycloserine
CAS:<p>L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.</p>Formula:C3H6N2O2Purity:99.45% - 99.92%Color and Shape:Crystals White PowderMolecular weight:102.09Linoleoyl glycine
CAS:<p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>Formula:C20H35NO3Purity:98.96%Color and Shape:SolidMolecular weight:337.5Glipizide
CAS:<p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>Formula:C21H27N5O4SPurity:99.67% - 99.75%Color and Shape:SolidMolecular weight:445.541-EBIO
CAS:<p>1-EBIO (1-EBIO) is a calium channel agonist.</p>Formula:C9H10N2OPurity:98.75%Color and Shape:SolidMolecular weight:162.19FFN 511
CAS:<p>Fluorescent false neurotransmitter (FFN)</p>Formula:C17H20N2O2Purity:98%Color and Shape:SolidMolecular weight:284.35Clomethiazole
CAS:<p>Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.</p>Formula:C6H8ClNSPurity:99.06%Color and Shape:SolidMolecular weight:161.65TRPV4 agonist-1 free base
CAS:<p>TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).</p>Formula:C25H22F2N4O2Purity:99.79%Color and Shape:SolidMolecular weight:448.46Ethaverine hydrochloride
CAS:<p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>Formula:C24H30ClNO4Purity:99.66% - 99.90%Color and Shape:SolidMolecular weight:431.96T16Ainh-A01
CAS:T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.Formula:C19H20N4O3S2Purity:97.18% - 98.15%Color and Shape:SolidMolecular weight:416.52Vocacapsaicin hydrochloride
CAS:<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Formula:C26H42ClN3O4Purity:99.66% - 99.80%Color and Shape:SolidMolecular weight:496.08ATP synthase inhibitor 1
CAS:<p>ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.</p>Formula:C17H18ClN3O3S2Purity:99.83%Color and Shape:SolidMolecular weight:411.93GFB-8438
CAS:<p>GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).</p>Formula:C16H14ClF3N4O2Purity:99.58%Color and Shape:SolidMolecular weight:386.76Repaglinide
CAS:<p>Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.</p>Formula:C27H36N2O4Purity:99.73% - >99.99%Color and Shape:White To Off-White SolidMolecular weight:452.59Domperidone EP Impurity A
CAS:<p>Domperidone EP Impurity A is used as pharmaceutical intermediates.</p>Formula:C12H14ClN3OPurity:99.97%Color and Shape:SolidMolecular weight:251.71Sulfacarbamide
CAS:<p>Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.</p>Formula:C7H9N3O3SPurity:95.6% - 99.72%Color and Shape:SolidMolecular weight:215.23Econazole
CAS:<p>Econazole ((±)-Econazol) is an imidazole derivative that is commonly used as a topical antifungal agent.</p>Formula:C18H15Cl3N2OPurity:98.11% - 99.97%Color and Shape:SolidMolecular weight:381.68Ornidazole (Levo-)
CAS:<p>Ornidazole (Levo-) (Levornidazole) is the levo-isomer of Ornidazole.</p>Formula:C7H10ClN3O3Purity:99.8%Color and Shape:SolidMolecular weight:219.63Tertiapin-Q
CAS:<p>Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).</p>Formula:C106H175N35O24S4Purity:98.06% - 98.09%Color and Shape:SolidMolecular weight:2452CGP37157
CAS:<p>CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release from</p>Formula:C15H11Cl2NOSPurity:99.92%Color and Shape:SolidMolecular weight:324.22Manidipine dihydrochloride
CAS:<p>Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).</p>Formula:C35H40Cl2N4O6Purity:99.76% - 99.86%Color and Shape:SolidMolecular weight:683.62D-AP5
CAS:<p>D-AP5 (D-APV) is a NMDA receptor antagonist.</p>Formula:C5H12NO5PPurity:98.77% - >99.99%Color and Shape:White Fine Crystalline PowderMolecular weight:197.13Etifoxine hydrochloride
CAS:<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Formula:C17H18Cl2N2OPurity:99.36%Color and Shape:SolidMolecular weight:337.24CRAC intermediate 2
CAS:<p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>Formula:C11H7F6N3Purity:99.69%Color and Shape:SolidMolecular weight:295.18PF-04885614
CAS:<p>PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.</p>Formula:C13H14F3N3OPurity:98.02%Color and Shape:SolidMolecular weight:285.27Tolazamide
CAS:<p>Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.</p>Formula:C14H21N3O3SPurity:98% - >99.99%Color and Shape:SolidMolecular weight:311.40Devapamil
CAS:<p>Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.</p>Formula:C26H36N2O3Purity:99.63%Color and Shape:SolidMolecular weight:424.58Vigabatrin
CAS:<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Formula:C6H11NO2Purity:99.47% - 99.88%Color and Shape:SolidMolecular weight:129.16LAU159
CAS:<p>LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).</p>Formula:C17H12ClN3O2Purity:98.7% - 99.38%Color and Shape:SolidMolecular weight:325.75Oxiracetam
CAS:<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16Permethrin
CAS:<p>Permethrin (NRDC-143) is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.</p>Formula:C21H20Cl2O3Purity:99.37% - 99.54%Color and Shape:Colorless Crystals To A Viscous Liquid; Color White To Pale Yellow Permethrin Is A Pale Brown Liquid Relatively Water Insoluble Used As An InsecticideMolecular weight:391.29AR-C155858
CAS:<p>AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).</p>Formula:C21H27N5O5SPurity:98.96% - 99.42%Color and Shape:SolidMolecular weight:461.53Oxybutynin chloride
CAS:<p>Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.</p>Formula:C22H32ClNO3Purity:99.27% - >99.99%Color and Shape:White PowderMolecular weight:393.96BMS-191095
CAS:<p>BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.</p>Formula:C22H21ClN4O2Purity:>99.99%Color and Shape:SolidMolecular weight:408.88DCEBIO
CAS:<p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>Formula:C9H8Cl2N2OPurity:99.89%Color and Shape:SolidMolecular weight:231.08Chlormezanone
CAS:<p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>Formula:C11H12ClNO3SPurity:99.89% - >99.99%Color and Shape:Crystals SolidMolecular weight:273.74Isoguvacine hydrochloride
CAS:<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Formula:C6H10ClNO2Purity:99.59%Color and Shape:SolidMolecular weight:163.6Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formula:C12H21NO8SPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:339.36IA-Alkyne
CAS:<p>IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.</p>Formula:C8H12INOPurity:99.76%Color and Shape:SolidMolecular weight:265.09Eact
CAS:<p>Eact is a potent TMEM16A activator that also triggers TRPV1, causing itch, pain, and heat sensitivity.</p>Formula:C22H24N2O5SPurity:98.14%Color and Shape:SolidMolecular weight:428.5TPC2-A1-P
CAS:<p>TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).</p>Formula:C20H21BrF3NO3Purity:98.49%Color and Shape:SolidMolecular weight:460.29Chlorpropamide
CAS:<p>Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary</p>Formula:C10H13ClN2O3SPurity:98.90%Color and Shape:Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Molecular weight:276.74NaV1.7 inhibitor-1
CAS:<p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>Formula:C23H30FNO4SPurity:99.89%Color and Shape:SolidMolecular weight:435.55Nav1.8-IN-4
CAS:<p>Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.</p>Formula:C20H14F4N2O3Purity:99.83%Color and Shape:SoildMolecular weight:406.33Halothane
CAS:<p>Halothane (Anestan) 可以减弱内皮依赖性舒张作用。</p>Formula:C2HBrClF3Purity:98.50% - >99.99%Color and Shape:Colorless Volatile Liquid Density 1 875 G / Cm3 Boiling Point 122 4°F (50 2°C) NoncombustibleMolecular weight:197.38Pentetrazol
CAS:<p>Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.</p>Formula:C6H10N4Purity:99.7% - >99.99%Color and Shape:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Molecular weight:138.17E 0747 FA
<p>E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.</p>Formula:C22H30ClN3O6Purity:98.54%Color and Shape:SolidMolecular weight:467.94Flumazenil
CAS:<p>Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous</p>Formula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.29Tocainide hydrochloride
CAS:<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Formula:C11H17ClN2OPurity:97%Color and Shape:SolidMolecular weight:228.72ML418
CAS:<p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>Formula:C19H24ClN3O3Purity:99.3%Color and Shape:SolidMolecular weight:377.87Lansoprazole
CAS:<p>Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISON</p>Formula:C16H14F3N3O2SPurity:99.18% - 99.84%Color and Shape:White Crystalline PowderMolecular weight:369.364-Aminopyridine
CAS:<p>4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.</p>Formula:C5H6N2Purity:91.61%Color and Shape:SolidMolecular weight:94.11CIQ
CAS:<p>CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.</p>Formula:C26H26ClNO5Purity:99.5%Color and Shape:SolidMolecular weight:467.94Torsemide
CAS:<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Formula:C16H20N4O3SPurity:99.81%Color and Shape:Crystalline SolidMolecular weight:348.42VU6036720
<p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>Formula:C20H22ClFN4O2SPurity:98.1%Color and Shape:SoildMolecular weight:436.93DSP-2230
CAS:<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Formula:C20H20F3N5O2Purity:97.14%Color and Shape:SolidMolecular weight:419.4URAT1 inhibitor 7
CAS:<p>URAT1 inhibitor 7, a uric acid transporter protein URAT1 inhibitor.URAT1 inhibitor 7 inhibits CYP2C9 and can be used in the study of hyperuricemia and gout.</p>Formula:C19H10ClFN4O3SPurity:97.65%Color and Shape:SoildMolecular weight:428.82Suloctidil
CAS:Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.Formula:C20H35NOSPurity:99.75% - >99.99%Color and Shape:SolidMolecular weight:337.56NS13001
CAS:<p>NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).</p>Formula:C17H16ClN7Purity:99.55%Color and Shape:SolidMolecular weight:353.81Linopirdine
CAS:<p>Linopirdine (DuP 996) is a TRPV1 agonist.</p>Formula:C26H21N3OPurity:99.45% - 99.78%Color and Shape:SolidMolecular weight:391.46Methocarbamol
CAS:<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Formula:C11H15NO5Purity:99.96%Color and Shape:Crystals From Benzene SolidMolecular weight:241.24Trichlormethiazide
CAS:<p>Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.</p>Formula:C8H8Cl3N3O4S2Purity:98.8% - 99.54%Color and Shape:SolidMolecular weight:380.66Fluxametamide
CAS:<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26γ-Aminobutyric acid
CAS:<p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>Formula:C4H9NO2Purity:99.95%Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMolecular weight:103.12QX-314 chloride
CAS:<p>QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.</p>Formula:C16H27ClN2OPurity:99.73%Color and Shape:SolidMolecular weight:298.85Cycloleucine
CAS:<p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>Formula:C6H11NO2Purity:99.90%Color and Shape:SolidMolecular weight:129.16Cromolyn sodium
CAS:<p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>Formula:C23H14Na2O11Purity:99.4% - 99.95%Color and Shape:Colorless Crystals From Ethanol + Ether White Crystalline PowderMolecular weight:512.33Diphenidol hydrochloride
CAS:<p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>Formula:C21H28ClNOPurity:99.15% - 99.33%Color and Shape:Crystals Soluble In Methanol WaterMolecular weight:345.91Ciclopirox olamine
CAS:<p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>Formula:C14H24N2O3Purity:99.16% - >99.99%Color and Shape:White To Yellow Solid Solid Particulate/PowderMolecular weight:268.35Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Formula:C13H9Cl2N3OSPurity:98.87% - 99.74%Color and Shape:SolidMolecular weight:326.2Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Formula:C66H92F3N19O24Purity:99.89%Color and Shape:SolidMolecular weight:1592.55BMS-195270
CAS:<p>BMS-195270 is a bio-active chemical.</p>Formula:C15H9ClF3N3O2Purity:98.7%Color and Shape:SolidMolecular weight:355.7Flavoxate hydrochloride
CAS:<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formula:C24H26ClNO4Purity:99.78%Color and Shape:White SolidMolecular weight:427.92Tocainide
CAS:<p>Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.</p>Formula:C11H16N2OPurity:99.84%Color and Shape:SolidMolecular weight:192.26Celivarone
CAS:<p>Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.</p>Formula:C34H47NO4Purity:99.53%Color and Shape:SolidMolecular weight:533.74MRZ 2-514
CAS:<p>MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki</p>Formula:C11H6BrN3O3Purity:98.459%Color and Shape:SolidMolecular weight:308.09Prilocaine hydrochloride
CAS:<p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>Formula:C13H21ClN2OPurity:99.97%Color and Shape:Needles White Or Off White Crystalline PowderMolecular weight:256.77Z433927330
CAS:<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Formula:C20H20N4O3Purity:99.78%Color and Shape:SolidMolecular weight:364.4Bupivacaine hydrochloride
CAS:<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Formula:C18H28N2O·HClPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:324.89NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formula:C20H24ClN3OPurity:99.56%Color and Shape:SolidMolecular weight:357.88Bemegride
CAS:<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Formula:C8H13NO2Purity:99.89%Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Molecular weight:155.19IK1 inhibitor PA-6
CAS:<p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>Formula:C31H32N4O2Purity:98.9%Color and Shape:SolidMolecular weight:492.61Elexacaftor
CAS:<p>Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.</p>Formula:C26H34F3N7O4SPurity:98.87% - 99.87%Color and Shape:SolidMolecular weight:597.65NS3623
CAS:<p>NS3623 is an activator of human ether-a-go-go-related gene potassium channels.</p>Formula:C15H10BrF3N6OPurity:97.06%Color and Shape:SolidMolecular weight:427.18Lotilaner
CAS:<p>Lotilaner is a parasiticide.</p>Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76EN6
CAS:<p>EN6, a small molecule, activates autophagy by modifying ATP6V1A, inhibiting mTORC1 and enhancing lysosomal function to clear TDP-43 aggregates.</p>Formula:C19H14F2N4O2Purity:95.74% - 97.04%Color and Shape:SolidMolecular weight:368.34Mebeverine hydrochloride
CAS:<p>Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut</p>Formula:C25H35NO5Purity:99.81% - 99.81%Color and Shape:SolidMolecular weight:429.55Ethosuximide
CAS:<p>Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by</p>Formula:C7H11NO2Purity:98.87% - 99.72%Color and Shape:Crystals From Acetone And Ether SolidMolecular weight:141.17MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formula:C25H25N3O2Purity:99.77% - 99.8%Color and Shape:SolidMolecular weight:399.48DMT1 blocker 2
CAS:<p>Compound 12f, a DMT1 blocker, inhibits DMT1 with a 0.83 IC50, potentially blocking intestinal iron absorption.</p>Formula:C16H13N3OPurity:99.68%Color and Shape:SolidMolecular weight:263.29AZD 7009
CAS:<p>AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.</p>Formula:C23H34N4O5Purity:98.42% - 98.51%Color and Shape:SoildMolecular weight:446.54Moxidectin
CAS:<p>Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.</p>Formula:C37H53NO8Purity:97.38%Color and Shape:Appearance White Or Pale Yellow Amorphous PowderMolecular weight:639.82Phenibut
CAS:<p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22γ-DGG acetate(6729-55-1 free base)
CAS:<p>gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.</p>Formula:C9H16N2O7Purity:99.81%Color and Shape:SolidMolecular weight:264.23GET73
CAS:<p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>Formula:C13H16F3NO2Purity:99.54%Color and Shape:SolidMolecular weight:275.27Etimizol
CAS:<p>Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.</p>Formula:C9H14N4O2Purity:99%Color and Shape:SolidMolecular weight:210.23Oxybuprocaine hydrochloride
CAS:<p>Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.</p>Formula:C17H29ClN2O3Purity:>99.99%Color and Shape:White Crystalline PowderMolecular weight:344.88DCPIB
CAS:<p>DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM</p>Formula:C22H28Cl2O4Purity:99.79% - 99.87%Color and Shape:SolidMolecular weight:427.36Doxapram hydrochloride hydrate
CAS:<p>Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.</p>Formula:C24H33ClN2O3C24H30N2O2·ClH·H2OPurity:99.64% - >99.99%Color and Shape:SolidMolecular weight:432.99Glimepiride
CAS:<p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>Formula:C24H34N4O5SPurity:97.84% - 98.87%Color and Shape:White Cyrstalline SolidMolecular weight:490.62Disopyramide
CAS:<p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>Formula:C21H29N3OPurity:99.62%Color and Shape:SolidMolecular weight:339.473,4,5-Trimethoxycinnamic acid
CAS:<p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>Formula:C12H14O5Purity:98.91%Color and Shape:SolidMolecular weight:238.24Butamben
CAS:<p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>Formula:C11H15NO2Purity:99.43%Color and Shape:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Molecular weight:193.24Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Formula:C16H17N2NaO4SPurity:98.11%Color and Shape:White To Off-White Crystalline PowderMolecular weight:356.375,5-Dimethyloxazolidine-2,4-dione
CAS:<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Formula:C5H7NO3Purity:99.12%Color and Shape:Drypowder PelletslargecrystalsMolecular weight:129.11Leptomycin A
CAS:<p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>Formula:C32H46O6Purity:98%Color and Shape:SolidMolecular weight:526.7EVT-401
<p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>Formula:C22H20F4N2O3Color and Shape:SolidMolecular weight:436.4Cavα2δ-IN-1
CAS:<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Formula:C18H27N5OColor and Shape:SolidMolecular weight:329.448Nitrazolam
CAS:<p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>Formula:C17H13N5O2Color and Shape:SolidMolecular weight:319.32Elgodipine
CAS:<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Formula:C29H33FN2O6Purity:98.95% - 99.50%Color and Shape:SolidMolecular weight:524.58GS-9191 PM
<p>GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.</p>Formula:C11H16N6OPurity:99.79%Color and Shape:SoildMolecular weight:248.28TRPA1 Antagonist 3
CAS:<p>TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.</p>Formula:C11H8ClN3Color and Shape:SolidMolecular weight:217.66(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Formula:C6H11NO2Color and Shape:SolidMolecular weight:129.16GsMTx4
CAS:<p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>Formula:C185H273N49O45S6Purity:98%Color and Shape:SolidMolecular weight:4095.84BeKm-1
CAS:<p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>Formula:C174H261N51O52S6Purity:98%Color and Shape:SolidMolecular weight:4091.65GeX-2
CAS:<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Formula:C103H169N43O27Color and Shape:SolidMolecular weight:2441.72α,β-Methylene-ATP dilithium
CAS:<p>α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.</p>Formula:C11H16Li2N5O12P3Color and Shape:SolidMolecular weight:517.07GpTx-1 TFA
<p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.</p>Color and Shape:Odour SolidWAY-326766
CAS:<p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>Formula:C21H23N3O5Purity:98.76%Color and Shape:SolidMolecular weight:397.42AChE/Aβ-IN-1
<p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>Formula:C20H25BrN4Color and Shape:SolidMolecular weight:401.34Anisatin
<p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>Formula:C15H20O8Color and Shape:SolidMolecular weight:328.317Trans (2,3)-Dihydrotetrabenazine
CAS:<p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>Formula:C19H29NO3Purity:98%Color and Shape:SolidMolecular weight:319.44LRRK2-IN-15
<p>LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.</p>Color and Shape:Odour SolidTP-050
CAS:<p>TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.</p>Formula:C16H15ClF2N6OColor and Shape:SolidMolecular weight:380.78Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Formula:C20H18O6Color and Shape:SolidMolecular weight:354.358Jingzhaotoxin-XII TFA
<p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>Color and Shape:Odour Solid3-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Formula:C3H10NO2PColor and Shape:SolidMolecular weight:123.092Huwentoxin I
CAS:<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Formula:C161H246N48O44S6Purity:98%Color and Shape:SolidMolecular weight:3750.36LY-466195
CAS:<p>LY-466195 is a competitive antagonist of GLUK5 receptor.</p>Formula:C16H24F2N2O4Color and Shape:SolidMolecular weight:346.37Hyp9
CAS:<p>Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].</p>Formula:C18H26O5Color and Shape:SolidMolecular weight:322.40AChE/Aβ-IN-2
<p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>Formula:C20H25ClN4Color and Shape:SolidMolecular weight:356.89Chlorotoxin TFA
<p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>Formula:C160H250F3N53O49S11Color and Shape:SolidMolecular weight:4109.74JAMI1001A
CAS:<p>JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.</p>Formula:C16H17F3N4O3SColor and Shape:SolidMolecular weight:402.39SLC26A3-IN-2
CAS:<p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>Formula:C19H13ClN2O2SPurity:99.86%Color and Shape:SolidMolecular weight:368.84Homocarnosine
CAS:<p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>Formula:C10H16N4O3Color and Shape:SolidMolecular weight:240.26Idactamab
CAS:<p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>Purity:> 95%Color and Shape:LiquidMolecular weight:146.2 kDaAnticonvulsant agent 9
<p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>Formula:C22H24N4O2Color and Shape:SolidMolecular weight:376.45Crofelemer
CAS:<p>Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.</p>Color and Shape:Solid2,4,6-Tri-tert-butylphenol
CAS:<p>2,4,6-Tri-tert-butylphenol inhibits the Ca2+ ATPase activity of human red blood cell membranes and can be used in related research in the field of life sciences.</p>Formula:C18H30OPurity:99.55%Color and Shape:SolidMolecular weight:262.43Bendroflumethiazide
CAS:<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Formula:C15H14F3N3O4S2Purity:98% - >99.99%Color and Shape:Crystals From Dioxane SolidMolecular weight:421.41Levamlodipine besylate Hemipentahydrate
CAS:<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formula:C20H25ClN2O5·C6H6O3SH2OColor and Shape:SolidMolecular weight:1224.18Analgesic/antidepressant agent-1
<p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>Formula:C22H25ClN2O2Color and Shape:SolidMolecular weight:384.9
