GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purity:98.76% - 99.75%Color and Shape:SolidMolecular weight:471.67Mefexamide hydrochloride
CAS:<p>Mefexamide hydrochloride is a central stimulant.</p>Formula:C15H25ClN2O3Purity:99.95%Color and Shape:SolidMolecular weight:316.83Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formula:C18H30ClN3O5Purity:99.53% - 99.61%Color and Shape:White SolidMolecular weight:403.91Moxonidine
CAS:<p>Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.</p>Formula:C9H12ClN5OPurity:99.81% - 99.94%Color and Shape:CrystalMolecular weight:241.68YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Formula:C33H37N5O5SPurity:99.67%Color and Shape:SolidMolecular weight:615.74Apelin-13
CAS:<p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>Formula:C69H111N23O16SPurity:96.81%Color and Shape:SolidMolecular weight:1550.83Avexitide acetate
CAS:<p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>Formula:C155H246N40O53SPurity:96.64% - 98.65%Color and Shape:SolidMolecular weight:3549.91Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Formula:C21H22ClNPurity:98.75% - 99.84%Color and Shape:SolidMolecular weight:323.86Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24Efloxate
CAS:<p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>Formula:C19H16O5Purity:99.66%Color and Shape:SolidMolecular weight:324.33Dexpramipexole dihydrochloride
CAS:<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Formula:C10H19Cl2N3SPurity:99.75% - 99.88%Color and Shape:SolidMolecular weight:284.25Sarizotan 2HCl
CAS:<p>Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.</p>Formula:C22H23Cl2FN2OPurity:98.83%Color and Shape:SoildMolecular weight:421.34Cinnarizine
CAS:<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Formula:C26H28N2Purity:99.94%Color and Shape:SolidMolecular weight:368.51Phentolamine mesylate
CAS:Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.Formula:C17H19N3O·CH4O3SPurity:99.87% - >99.99%Color and Shape:By The Metabolic Processes Of Bacillus Subtilis And LicheniformisMolecular weight:377.46Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurity:99.55%Color and Shape:Tan SolidMolecular weight:412.94AM-8123
CAS:AM-8123: oral APJ agonist, potent, inhibits cAMP, activates Gα, key for cardiovascular research.Formula:C27H33N7O5SPurity:99.59% - 99.76%Color and Shape:SolidMolecular weight:567.66Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Formula:C10H16N6SPurity:99.82%Color and Shape:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Molecular weight:252.34GTS-21 dihydrochloride
CAS:<p>GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.</p>Formula:C19H20N2O2·2HClPurity:98.54% - >99.99%Color and Shape:SolidMolecular weight:381.3UCM-1306
CAS:<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Formula:C14H14FNO2SPurity:99.98%Color and Shape:SoildMolecular weight:279.33Azacyclonol
CAS:<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Formula:C18H21NOPurity:99.46%Color and Shape:Solid PowderMolecular weight:267.37Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.Formula:C20H24Cl2N4O2Purity:99.01% - 99.40%Color and Shape:SoildMolecular weight:423.34Bufotenidine hydrochloride(487-91-2 Free base)
CAS:<p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>Formula:C13H19ClN2OPurity:99.88%Color and Shape:SolidMolecular weight:254.76Orphenadrine hydrochloride
CAS:Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formula:C18H23NO·HClPurity:99.88%Color and Shape:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Molecular weight:305.85Volagidemab
CAS:<p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>Purity:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)Color and Shape:LiquidSEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formula:C9H14ClNOSPurity:99.86% - 99.99%Color and Shape:SolidMolecular weight:219.73Adenosine A1 receptor activator T62
CAS:<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Formula:C4H7NO2SPurity:99.99%Color and Shape:SolidMolecular weight:133.17Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Formula:C31H38N2OPurity:97.49%Color and Shape:SolidMolecular weight:454.65MRGPRX1 agonist 1
CAS:<p>MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).</p>Formula:C23H21N3O4SPurity:99.95%Color and Shape:SolidMolecular weight:435.5Paroxetine hydrochloride
CAS:<p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>Formula:C19H21ClFNO3Purity:98% - 99.99%Color and Shape:White Crystalline PowderMolecular weight:365.826Astemizole
CAS:<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Formula:C28H31FN4OPurity:98.24% - 99.67%Color and Shape:White Crystals SolidMolecular weight:458.57Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Formula:C18H23Cl2NOPurity:98.04% - >99.99%Color and Shape:Antihypertensive DrugMolecular weight:340.3PIT
CAS:<p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>Formula:C20H16N2O5SPurity:98.63%Color and Shape:SolidMolecular weight:396.42Somatostatin acetate
<p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>Purity:99.11%Color and Shape:Odour SolidPrasugrel
CAS:Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent THROMBOSIS in patients with ACUTE CORONARY SYNDROME;Formula:C20H20FNO3SPurity:99.62% - 99.82%Color and Shape:White SolidMolecular weight:373.44GANT 58
CAS:<p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>Formula:C24H16N4SPurity:99.53%Color and Shape:SolidMolecular weight:392.48Labetalol hydrochloride
CAS:<p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>Formula:C19H25ClN2O3Purity:99.54% - 99.85%Color and Shape:SolidMolecular weight:364.87Roluperidone
CAS:<p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>Formula:C22H23FN2O2Purity:96.46% - 97.77%Color and Shape:SolidMolecular weight:366.43(S)-(-)-Atenolol
CAS:<p>(S)-(-)-Atenolol has beta-adrenergic blocking effects.</p>Formula:C14H22N2O3Purity:99.31% - 99.81%Color and Shape:SolidMolecular weight:266.34Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Formula:C26H27N5O2Purity:99.61%Color and Shape:Light Yellow SolidMolecular weight:441.52Famotidine
CAS:Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.Formula:C8H15N7O2S3Purity:98.93% - 99.91%Color and Shape:White To Off-White Crystalline PowderMolecular weight:337.45Strontium ranelate
CAS:<p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>Formula:C12H6N2O8S·2SrPurity:98.97%Color and Shape:Crystalline SolidMolecular weight:513.49Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25Oxeladin citrate
CAS:<p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>Formula:C26H41NO10Purity:97.23%Color and Shape:SolidMolecular weight:527.6Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purity:99.85%Color and Shape:SolidMolecular weight:367.5AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formula:C23H22N8OPurity:98.09% - >99.99%Color and Shape:SolidMolecular weight:426.47Heptaminol hydrochloride
CAS:<p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>Formula:C8H20ClNOPurity:98.61%Color and Shape:White Crystalline PowderMolecular weight:181.71Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formula:C15H20N2O2·HClPurity:99.64% - 99.92%Color and Shape:SolidMolecular weight:296.79Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formula:C21H28N2O5Purity:99.61%Color and Shape:5 1 (Ntp 1992)Molecular weight:388.46Gevotroline
CAS:<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Formula:C19H20FN3Purity:98.65%Color and Shape:SolidMolecular weight:309.38Solabegron
CAS:<p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>Formula:C23H23ClN2O3Purity:97.89%Color and Shape:SolidMolecular weight:410.89Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formula:C22H24ClN3O5Purity:99.69%Color and Shape:White To Of-White SolidMolecular weight:445.9Ifenprodil Tartrate
CAS:<p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>Formula:C21H27NO2C4H6O6Purity:99.02% - 99.55%Color and Shape:SolidMolecular weight:400.49Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Formula:C22H28Cl2F3N3OSPurity:99.23%Color and Shape:Off-White SolidMolecular weight:510.446-Iodopravadoline
CAS:<p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>Formula:C23H25IN2O3Purity:99.29%Color and Shape:Off-White SolidMolecular weight:504.36DSP-4 hydrochloride
CAS:<p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>Formula:C11H16BrCl2NPurity:99.9%Color and Shape:SolidMolecular weight:313.06Sulpiride
CAS:<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Formula:C15H23N3O4SPurity:99.94%Color and Shape:White Crystalline PowderMolecular weight:341.43Monatepil 2maleate
Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.Formula:C32H34FN3O5SPurity:98%Color and Shape:SolidMolecular weight:591.69PHM-27 (human) acetate
<p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>Formula:C137H215F3N34O42SPurity:99.20%Color and Shape:SoildMolecular weight:3099.44Luzindole
CAS:<p>Luzindole (N-0774) is a selective melatonin receptor antagonist.</p>Formula:C19H20N2OPurity:98.53%Color and Shape:Off-White Amorphous SolidMolecular weight:292.37Pramipexole
CAS:<p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>Formula:C10H17N3SPurity:98% - 99.96%Color and Shape:SolidMolecular weight:211.33Betaxolol hydrochloride
CAS:<p>Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.</p>Formula:C18H30ClNO3Purity:99.48% - 99.56%Color and Shape:SolidMolecular weight:343.89Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Formula:C30H32ClN3O8SPurity:98.46% - 99.89%Color and Shape:SolidMolecular weight:630.11Terbutaline
CAS:Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterolFormula:C12H19NO3Purity:99.12%Color and Shape:SolidMolecular weight:225.3Lesopitron HCl
CAS:<p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>Formula:C15H22Cl2N6Purity:97.05% - 99.89%Color and Shape:SoildMolecular weight:357.28Clopidogrel hydrogen sulfate
CAS:<p>Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.</p>Formula:C16H16ClNO2S·H2SO4Purity:99.57% - 99.79%Color and Shape:SolidMolecular weight:419.9Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formula:C24H27FN2O4Purity:99.42%Color and Shape:SolidMolecular weight:426.48Isoprenaline hydrochloride
CAS:Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.Formula:C11H18ClNO3Purity:98% - 99.65%Color and Shape:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Molecular weight:247.719Ciliobrevin D
CAS:<p>Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.</p>Formula:C17H8Cl3N3O2Purity:98.09%Color and Shape:SolidMolecular weight:392.62Tabernanthalog fumarate
CAS:<p>Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.</p>Formula:C18H22N2O5Purity:99.83%Color and Shape:SoildMolecular weight:346.38CE3F4
CAS:<p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>Formula:C11H10Br2FNOPurity:97.15% - 98.06%Color and Shape:SolidMolecular weight:351.01CYM50308
CAS:<p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>Formula:C20H21F2N3O2SPurity:99.43% - 99.77%Color and Shape:SolidMolecular weight:405.46Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurity:99% - 99.99%Color and Shape:SolidMolecular weight:312.84Seganserin
CAS:<p>Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.</p>Formula:C29H27F2N3OPurity:99.22%Color and Shape:SolidMolecular weight:471.54Ebalzotan
CAS:<p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>Formula:C19H30N2O2Purity:98.09% - 99.41%Color and Shape:SolidMolecular weight:318.45Ornidazole
CAS:<p>Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.</p>Formula:C7H10ClN3O3Purity:99.47%Color and Shape:Crystalline SolidMolecular weight:219.63Fenclozine Maleate
CAS:<p>Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain.</p>Formula:C45H47ClN2O12Purity:98.47%Color and Shape:SoildMolecular weight:843.314Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Formula:C18H25N3O6Purity:99.66%Color and Shape:SolidMolecular weight:379.41Orforglipron
CAS:<p>Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1</p>Formula:C48H48F2N10O5Purity:99.47% - 99.8%Color and Shape:SolidMolecular weight:882.96Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Formula:C12H17Cl2NOPurity:99.38%Color and Shape:SolidMolecular weight:262.18INCB-9471
CAS:<p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>Formula:C30H40F3N5O2Purity:98.80%Color and Shape:SolidMolecular weight:559.666Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purity:99.97%Color and Shape:SolidMolecular weight:311.89Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurity:99.84% - 99.92%Color and Shape:White SolidMolecular weight:332.87Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formula:C19H27NO3Purity:98% - 99.91%Color and Shape:White To Off-White White To Off-White SolidMolecular weight:317.42Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Formula:C16H15FN6OSPurity:98.62% - 99.7%Color and Shape:SolidMolecular weight:358.39ML-180
CAS:<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Formula:C20H25ClN4O2Purity:99.74%Color and Shape:SolidMolecular weight:388.89Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Formula:C17H19ClN4OPurity:99.90%Color and Shape:Off-White PowderMolecular weight:330.81Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formula:C14H22BrN3O2Purity:99.95%Color and Shape:SolidMolecular weight:344.25BIBO3304 TFA
CAS:<p>BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).</p>Formula:C31H36F3N7O5Purity:99.5%Color and Shape:SolidMolecular weight:643.66RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Formula:C21H22ClF3N2O2Purity:98.95%Color and Shape:SolidMolecular weight:426.86TSHR antagonist S37
CAS:TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).Formula:C25H20N2O3S2Purity:98.35%Color and Shape:SolidMolecular weight:460.57Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Formula:C24H26N2O2Purity:98.88% - 99.68%Color and Shape:SolidMolecular weight:374.48Tripelennamine hydrochloride
CAS:<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Formula:C16H21N3·HClPurity:99.54% - 99.81%Color and Shape:White SolidMolecular weight:291.82Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Purity:SDS-PAGE:95% SEC-HPLC:98.90%Color and Shape:LiquidMolecular weight:146.43 kDaNepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Formula:C15H14N2O2Purity:98.94% - 99.43%Color and Shape:SolidMolecular weight:254.28Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formula:C17H19ClF3NOPurity:99.6% - 99.98%Color and Shape:White To Off-White Crystalline Solid White To Off-White PowderMolecular weight:345.787Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.Purity:> 95%Color and Shape:LiquidMolecular weight:146.28 kDaProstaglandin E1
CAS:<p>Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.</p>Formula:C20H34O5Purity:99.78% - >99.99%Color and Shape:SolidMolecular weight:354.48Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Formula:C19H27N5O4·HClPurity:99.78%Color and Shape:White To Off-White SolidMolecular weight:425.91
