
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Trimipramine maleate
CAS:<p>Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.</p>Formula:C24H30N2O4Purity:99.47%Color and Shape:SolidMolecular weight:410.51JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formula:C11H19N5Purity:98.33% - 99.62%Color and Shape:SolidMolecular weight:221.3Carteolol hydrochloride
CAS:Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.Formula:C16H24N2O3·HClPurity:99.84% - 99.91%Color and Shape:SolidMolecular weight:328.83(±) Clopidogrel hydrogen sulfate
CAS:<p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>Formula:C16H16ClNO2S·H2SO4Purity:98.67% - 99.04%Color and Shape:Colorless To Light Yellow LiquidMolecular weight:419.9Ziprasidone hydrochloride monohydrate
CAS:<p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>Formula:C21H21ClN4OS·HCl·H2OPurity:98% - 99.83%Color and Shape:Off-White PowderMolecular weight:467.12NS-2028
CAS:NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.Formula:C9H5BrN2O3Purity:99.44%Color and Shape:A Crystalline SolidMolecular weight:269.05Volagidemab
CAS:<p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>Purity:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)Color and Shape:LiquidLofepramine
CAS:<p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>Formula:C26H27ClN2OPurity:98.38%Color and Shape:Crystals From Methanol Or Acetone SolidMolecular weight:418.96Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Formula:C21H25ClN2O3Purity:98% - 99.94%Color and Shape:White PowderMolecular weight:388.89BIBO3304 TFA
CAS:<p>BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).</p>Formula:C31H36F3N7O5Purity:99.5%Color and Shape:SolidMolecular weight:643.66[Leu15]-Gastrin I, human
CAS:[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.Formula:C98H126N20O31Purity:98.02% - 98.84%Color and Shape:SolidMolecular weight:2080.16Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Formula:C16H15FN6OSPurity:98.62% - 99.7%Color and Shape:SolidMolecular weight:358.39Carboprost tromethamine
CAS:<p>Carboprost tromethamine, a synthetic 15-methyl analogue of prostaglandin F2α, effectively promotes uterine contractions and significantly reduces bleeding</p>Formula:C25H47NO8Purity:>99.99%Color and Shape:SolidMolecular weight:489.64Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24Terazosin hydrochloride
CAS:<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Formula:C19H26ClN5O4Purity:99.69% - 99.91%Color and Shape:SolidMolecular weight:423.89Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formula:C15H17NO2Purity:99.92%Color and Shape:White SolidMolecular weight:243.3Bufotenidine hydrochloride(487-91-2 Free base)
CAS:<p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>Formula:C13H19ClN2OPurity:99.88%Color and Shape:SolidMolecular weight:254.76Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Formula:C19H20N2C10H8O6S2Purity:99.35% - 99.96%Color and Shape:White Or Almost White CrystallineMolecular weight:420.52Flopropione
CAS:<p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>Formula:C9H10O4Purity:99.93%Color and Shape:SolidMolecular weight:182.17SR59230A
CAS:<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Formula:C23H29NO6Purity:98.84%Color and Shape:SolidMolecular weight:415.48SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formula:C9H14ClNOSPurity:99.86% - 99.99%Color and Shape:SolidMolecular weight:219.73Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Formula:C44H43ClN2O8Purity:99.49%Color and Shape:SolidMolecular weight:763.27Ifenprodil Tartrate
CAS:<p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>Formula:C21H27NO2C4H6O6Purity:99.02% - 99.55%Color and Shape:SolidMolecular weight:400.49Mefexamide hydrochloride
CAS:<p>Mefexamide hydrochloride is a central stimulant.</p>Formula:C15H25ClN2O3Purity:99.95%Color and Shape:SolidMolecular weight:316.83Ozagrel
CAS:<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formula:C13H12N2O2Purity:97.90% - 99.38%Color and Shape:White PowderMolecular weight:228.25Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurity:99.85%Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Molecular weight:320.88Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formula:C24H27FN2O4Purity:99.42%Color and Shape:SolidMolecular weight:426.48Clozapine
CAS:<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formula:C18H19ClN4Purity:99.91% - 99.93%Color and Shape:Yellow Crystals From Acetone-Petroleum Ether SolidMolecular weight:326.82Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formula:C19H27NO3Purity:98% - 99.91%Color and Shape:White To Off-White White To Off-White SolidMolecular weight:317.42Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purity:98% - 99.82%Color and Shape:SolidMolecular weight:425.91Cefaclor monohydrate
CAS:<p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>Formula:C15H16ClN3O5SPurity:97.36% - 99.9%Color and Shape:White Crystaling PowderMolecular weight:385.82Triflupromazine hydrochloride
CAS:Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.Formula:C18H20ClF3N2SPurity:99.76% - 99.82%Color and Shape:CrystalsMolecular weight:388.88Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Formula:C17H19ClN4OPurity:99.90%Color and Shape:Off-White PowderMolecular weight:330.81Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formula:C14H22BrN3O2Purity:99.95%Color and Shape:SolidMolecular weight:344.252-(1-Piperazinyl)pyrimidine
CAS:<p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>Formula:C8H12N4Purity:98.46%Color and Shape:Liquid - Crystal - LumpMolecular weight:164.21Propafenone
CAS:<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Formula:C21H27NO3Purity:99.02%Color and Shape:SolidMolecular weight:341.44Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Formula:C12H17Cl2NOPurity:99.38%Color and Shape:SolidMolecular weight:262.18Apelin-13
CAS:<p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>Formula:C69H111N23O16SPurity:96.81%Color and Shape:SolidMolecular weight:1550.83Xylometazoline hydrochloride
CAS:<p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>Formula:C16H24N2·HClPurity:99.77% - 99.87%Color and Shape:White To Off-White Crystalline PowderMolecular weight:280.84Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formula:C21H28N2O5Purity:99.61%Color and Shape:5 1 (Ntp 1992)Molecular weight:388.46Lamotrigine
CAS:<p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>Formula:C9H7Cl2N5Purity:99.76% - 99.95%Color and Shape:White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMolecular weight:256.09Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurity:99.55%Color and Shape:Tan SolidMolecular weight:412.94Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formula:C21H20ClNO5Purity:99.28%Color and Shape:SolidMolecular weight:401.84DREADD agonist 21
CAS:<p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>Formula:C17H18N4Purity:99.94%Color and Shape:SolidMolecular weight:278.35Azasetron hydrochloride
CAS:<p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>Formula:C17H20ClN3O3·HClPurity:99.50%Color and Shape:SolidMolecular weight:386.27JP1302 dihydrochloride
CAS:<p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>Formula:C24H26Cl2N4Purity:99.61%Color and Shape:SolidMolecular weight:441.4Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formula:C21H23N3OSPurity:99.61%Color and Shape:SolidMolecular weight:365.49Pamabrom
CAS:Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.Formula:C11H18BrN5O3Purity:99.84% - >99.99%Color and Shape:CoaMolecular weight:348.2Carvedilol EP IMpurity E
CAS:<p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>Formula:C9H14ClNO2Purity:99.53%Color and Shape:White To Almost White Solid CrystallineMolecular weight:203.666Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formula:C25H28N2O5SPurity:97.09%Color and Shape:SolidMolecular weight:468.57Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.Purity:> 95%Color and Shape:LiquidMolecular weight:146.28 kDaPHM-27 (human) acetate
<p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>Formula:C137H215F3N34O42SPurity:99.20%Color and Shape:SoildMolecular weight:3099.44Prostaglandin E1
CAS:<p>Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.</p>Formula:C20H34O5Purity:99.78% - >99.99%Color and Shape:SolidMolecular weight:354.48Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurity:99.64%Color and Shape:Light Yellow To Yellow SolidMolecular weight:396.51DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formula:C22H20Cl2N4OSPurity:99.95%Color and Shape:SoildMolecular weight:459.39Benserazide hydrochloride
CAS:<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Formula:C10H15N3O5·HClPurity:98.63% - 99.74%Color and Shape:White Crystalline SolidMolecular weight:293.7Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25PF-5190457
CAS:<p>PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).</p>Formula:C29H32N6OSPurity:99.34%Color and Shape:SolidMolecular weight:512.67L-741626
CAS:<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Formula:C20H21ClN2OPurity:98.57%Color and Shape:SolidMolecular weight:340.85Efloxate
CAS:<p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>Formula:C19H16O5Purity:99.66%Color and Shape:SolidMolecular weight:324.33Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formula:C34H36Cl2N6O5S·2ClHPurity:99.17% - 99.58%Color and Shape:SoildMolecular weight:784.58Gevotroline
CAS:<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Formula:C19H20FN3Purity:98.65%Color and Shape:SolidMolecular weight:309.38Senktide acetate
<p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>Formula:C42H59N7O13SPurity:98.26%Color and Shape:SolidMolecular weight:902.02Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purity:98.76% - 99.75%Color and Shape:SolidMolecular weight:471.67hGPR91 antagonist 1
CAS:<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Formula:C31H23F4N3OPurity:98.89%Color and Shape:SolidMolecular weight:529.53Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Formula:C19H27N5O4·HClPurity:99.78%Color and Shape:White To Off-White SolidMolecular weight:425.91Naluzotan hydrochloride
CAS:<p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>Formula:C23H39ClN4O3SPurity:99.96%Color and Shape:SolidMolecular weight:487.1Proglumide
CAS:<p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>Formula:C18H26N2O4Purity:99.4% - 99.45%Color and Shape:White Crystalline PowderMolecular weight:334.41TSHR antagonist S37
CAS:TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).Formula:C25H20N2O3S2Purity:98.35%Color and Shape:SolidMolecular weight:460.57Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Formula:C10H7KN6OPurity:98.91% - 99.63%Color and Shape:Crystals From Dimethylformamide Crystalline SolidMolecular weight:266.31Mifentidine
CAS:<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Formula:C13H16N4Purity:98.34% - 99.73%Color and Shape:SolidMolecular weight:228.29Oxeladin citrate
CAS:<p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>Formula:C26H41NO10Purity:97.23%Color and Shape:SolidMolecular weight:527.6Salmeterol
CAS:<p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>Formula:C25H37NO4Purity:99.2% - 99.9%Color and Shape:SolidMolecular weight:415.57Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purity:99.46%Color and Shape:White To Off-White SolidMolecular weight:525.59(Rac)-MGV354
CAS:<p>(Rac)-MGV354: a racemic sGC activator; EC50s <0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>Formula:C35H37N5O3Purity:99.26%Color and Shape:SolidMolecular weight:575.7Phentolamine mesylate
CAS:Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.Formula:C17H19N3O·CH4O3SPurity:99.87% - >99.99%Color and Shape:By The Metabolic Processes Of Bacillus Subtilis And LicheniformisMolecular weight:377.46Cloroperone
CAS:<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Formula:C22H23ClFNO2Purity:98.40%Color and Shape:SoildMolecular weight:387.88Solabegron
CAS:<p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>Formula:C23H23ClN2O3Purity:97.89%Color and Shape:SolidMolecular weight:410.89Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Formula:C18H19N3O·HCl·2H2OPurity:99.92%Color and Shape:White Crystal PowderMolecular weight:365.86Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formula:C18H30ClN3O5Purity:99.53% - 99.61%Color and Shape:White SolidMolecular weight:403.91Mizolastine
CAS:<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Formula:C24H25FN6OPurity:98% - 99.75%Color and Shape:SolidMolecular weight:432.49Adenosine A1 receptor activator T62
CAS:<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Formula:C19H31ClF3NO3Purity:99.55%Color and Shape:SolidMolecular weight:413.9(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Formula:C20H29N3O8Purity:99.72%Color and Shape:SoildMolecular weight:439.46Tropanserin
CAS:<p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>Formula:C17H23NO2Purity:99.74%Color and Shape:SolidMolecular weight:273.37Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Formula:C17H22ClNOPurity:99.86%Color and Shape:White SolidMolecular weight:291.82Duloxetine hydrochloride
CAS:<p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>Formula:C18H20ClNOSPurity:99.93% - >99.99%Color and Shape:White Or White Crystalline PowderMolecular weight:333.88(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formula:C22H24ClF4N5OSPurity:98.36%Color and Shape:SoildMolecular weight:517.97Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Formula:C24H26N2O2Purity:98.88% - 99.68%Color and Shape:SolidMolecular weight:374.48Metoclopramide hydrochloride
CAS:<p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>Formula:C14H22ClN3O2·HClPurity:99.99%Color and Shape:White To Off-White PowderMolecular weight:336.26Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFormula:C32H40ClNO4Purity:>99.99%Color and Shape:White Crystalline PowderMolecular weight:538.12Dexpramipexole dihydrochloride
CAS:<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Formula:C10H19Cl2N3SPurity:99.75% - 99.88%Color and Shape:SolidMolecular weight:284.25Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Formula:C18H25N3O6Purity:99.66%Color and Shape:SolidMolecular weight:379.41Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formula:C15H24N2O4S·HClPurity:99.4% - 99.77%Color and Shape:SolidMolecular weight:364.89Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formula:C28H32ClN3O8SPurity:99.78%Color and Shape:Off-White PowderMolecular weight:606.09PF-610355 HCl
<p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>Formula:C19H22ClN7O6Purity:97.97%Color and Shape:SolidMolecular weight:479.87Nepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Formula:C15H14N2O2Purity:98.94% - 99.43%Color and Shape:SolidMolecular weight:254.28Latanoprostene bunod
CAS:<p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>Formula:C27H41NO8Purity:99.33% - 99.69%Color and Shape:SolidMolecular weight:507.62NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formula:C20H24ClN3OPurity:99.56%Color and Shape:SolidMolecular weight:357.88Rimonabant hydrochloride
CAS:<p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>Formula:C22H22Cl4N4OPurity:98.24% - 99.5%Color and Shape:Off-White To White Crystalline PowderMolecular weight:500.25Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Formula:C20H22BrFN2OPurity:99.81%Color and Shape:White Crystalline PowderMolecular weight:405.304SBI-477
CAS:<p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>Formula:C24H25N3O6SPurity:99.3%Color and Shape:SolidMolecular weight:483.54Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Indusatumab
CAS:<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Purity:> 95% - > 95%Color and Shape:LiquidMolecular weight:145.18 kDaAnamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Formula:C31H42N6O3Purity:99.35% - 99.94%Color and Shape:SolidMolecular weight:546.7Tripelennamine hydrochloride
CAS:<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Formula:C16H21N3·HClPurity:99.54% - 99.81%Color and Shape:White SolidMolecular weight:291.82PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C31H30FN5O4Purity:97.19% - 99.56%Color and Shape:SolidMolecular weight:555.62-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Formula:C11H9BrOPurity:98.51%Color and Shape:White To Off-White PowderMolecular weight:237.09Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Formula:C23H29ClFN3O4Purity:99.77%Color and Shape:White To Slightly Biege Powder SolidMolecular weight:465.95Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Formula:C19H21N·HClPurity:98.54% - 99.98%Color and Shape:SolidMolecular weight:299.84Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Purity:97.76%Color and Shape:SoildNylidrin hydrochloride
CAS:<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Formula:C19H26ClNO2Purity:99.35%Color and Shape:SolidMolecular weight:335.87Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Formula:C56H82N16O19S2Purity:98.50% - 99.69%Color and Shape:SolidMolecular weight:1347.5Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Purity:SDS-PAGE:95% SEC-HPLC:98.90%Color and Shape:LiquidMolecular weight:146.43 kDaLafutidine
CAS:<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Formula:C22H29N3O4SPurity:98.55%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.55Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Formula:C18H26ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:367.87Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:White Crystalline PowderMolecular weight:313.86Erenumab
CAS:<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Purity:99.43% (SEC-HPLC) - > 95%Color and Shape:LiquidMolecular weight:146.2 kDaTalastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Formula:C19H21N3OPurity:98.50% - 99.44%Color and Shape:SolidMolecular weight:307.39Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Formula:C10H13NO4Purity:98.95% - 99.86%Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White FineMolecular weight:211.21Desipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formula:C18H23ClN2Purity:99.58% - 99.94%Color and Shape:White To Off-White PowderMolecular weight:302.842EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Formula:C23H26N4O4SPurity:99.11%Color and Shape:SolidMolecular weight:454.54Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formula:C17H19ClF3NOPurity:99.6% - 99.98%Color and Shape:White To Off-White Crystalline Solid White To Off-White PowderMolecular weight:345.787Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Sergliflozin A
CAS:<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Formula:C20H24O7Purity:99.43%Color and Shape:SolidMolecular weight:376.4Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:463.79Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Formula:C28H32N2O7Purity:99.03% - 99.67%Color and Shape:SolidMolecular weight:508.56ML-180
CAS:<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Formula:C20H25ClN4O2Purity:99.74%Color and Shape:SolidMolecular weight:388.89CD80-IN-3
CAS:<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Formula:C17H10FN3O3Purity:98.08%Color and Shape:SolidMolecular weight:323.28CYM 50769
CAS:<p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>Formula:C24H17ClN2O3Purity:98% - 99.08%Color and Shape:SolidMolecular weight:416.86Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Formula:C19H25F3N2O6Purity:99.92% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:434.41Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.282% - 99.76%Color and Shape:Colorless To Pink SolidMolecular weight:495.53Metaproterenol hemisulfate
CAS:<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Formula:C11H17NO3·5H2O4SPurity:98.53% - 99.74%Color and Shape:SolidMolecular weight:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Formula:C21H24ClNOPurity:99.77% - >99.99%Color and Shape:White To Slightly Yellowish Crystalline SolidMolecular weight:341.88Urapidil hydrochloride
CAS:<p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>Formula:C20H29N5O3·HClPurity:99.58%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:423.94Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formula:C21H25N3O2SPurity:99.14% - 99.63%Color and Shape:White To Off-White Crystalline PowderMolecular weight:383.51JNJ-18038683
CAS:<p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>Formula:C26H28ClN3O7Purity:97.29%Color and Shape:SolidMolecular weight:529.97PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Formula:C25H37Cl2N3O2Purity:99.68%Color and Shape:SolidMolecular weight:482.49Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Formula:C31H37N3O10SPurity:99.39% - 99.48%Color and Shape:SolidMolecular weight:643.71Naftopidil
CAS:<p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>Formula:C24H28N2O3Purity:99.60% - 99.97%Color and Shape:White Crystalline PowderMolecular weight:392.49Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Formula:C21H27NO2Purity:99.58%Color and Shape:White Crystalline PowderMolecular weight:325.44Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Formula:C18H25ClN4OPurity:99.88% - 99.93%Color and Shape:White To Off-White Crystalline SolidMolecular weight:348.87Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H11ClFNO2Purity:99.98%Color and Shape:SoildMolecular weight:231.65Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purity:99.85%Color and Shape:SolidMolecular weight:367.5Fosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Formula:C9H15ClNO5PPurity:99.84%Color and Shape:SolidMolecular weight:283.65NF-56-EJ40 hydrochloride
CAS:<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Formula:C27H31Cl2N3O3Purity:99.33%Color and Shape:SoildMolecular weight:516.46Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White Crystalline PowderMolecular weight:341.43Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Formula:C17H18F3NOPurity:99.07% - 99.28%Color and Shape:SolidMolecular weight:309.33Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Formula:C163H273N49O44Purity:96.87%Color and Shape:SolidMolecular weight:3623.21Diphenylpyraline hydrochloride
CAS:<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Formula:C19H23NO·HClPurity:98.72%Color and Shape:SolidMolecular weight:317.85Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurity:99.76%Color and Shape:White PowderMolecular weight:352.32Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Formula:C28H30N2O8Purity:99.7% - >99.99%Color and Shape:PowderMolecular weight:522.55Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Formula:C17H20N4SPurity:99.86% - ≥95%Color and Shape:Yellowish Crystalline PowderMolecular weight:312.43CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Formula:C15H18Cl2N4OPurity:99.5%Color and Shape:SolidMolecular weight:341.24Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Formula:C19H23Cl2N5OPurity:99.5% - 99.52%Color and Shape:SolidMolecular weight:408.33MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Formula:C24H26F3N3O4Purity:99.98%Color and Shape:SolidMolecular weight:477.48Antazoline hydrochloride
CAS:<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Formula:C17H19N3·HClPurity:98% - 99.53%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:301.82Brefonalol HCl
<p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>Formula:C22H29ClN2O2Purity:99.45%Color and Shape:SolidMolecular weight:388.93Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:Colourless Flake Crystalline SolidMolecular weight:448.39YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Formula:C33H37N5O5SPurity:99.67%Color and Shape:SolidMolecular weight:615.74Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Formula:C26H35NO7Purity:98.53% - 99.43%Color and Shape:CoaMolecular weight:473.57KGA-2727
CAS:<p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>Formula:C26H40N4O8Purity:98.46%Color and Shape:SolidMolecular weight:536.62(3aR,9aR)-Fluparoxan
CAS:<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H10FNO2Purity:97.82%Color and Shape:SoildMolecular weight:195.19Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Formula:C16H21N3O2Purity:99.69% - 99.91%Color and Shape:White Or Kind Of White PowderMolecular weight:287.36Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purity:99.32% - >99.99%Color and Shape:White Crystalline SolidMolecular weight:883.09AH 6809
CAS:<p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>Formula:C17H14O5Purity:97.59%Color and Shape:SolidMolecular weight:298.29Phenothiazine
CAS:<p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>Formula:C12H9NSPurity:99.95%Color and Shape:Yellow Solid PelletsMolecular weight:199.27Noradrenaline bitartrate
CAS:<p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>Formula:C12H19NO10Purity:99.53% - >99.99%Color and Shape:SolidMolecular weight:337.28ESI-05
CAS:<p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>Formula:C16H18O2SPurity:97.22%Color and Shape:SolidMolecular weight:274.38Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Formula:C4H7NO2SPurity:99.99%Color and Shape:SolidMolecular weight:133.17Centanafadine hydrochloride
CAS:Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).Formula:C15H16ClNPurity:99.65%Color and Shape:SolidMolecular weight:245.75Talipexole dihydrochloride
CAS:<p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>Formula:C10H17Cl2N3SPurity:99.89%Color and Shape:Light Yellow SolidMolecular weight:282.23LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Formula:C30H58ClN7O8SPurity:98.02% - 99.31%Color and Shape:SolidMolecular weight:712.34(R)-Elagolix
CAS:<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Formula:C32H30F5N3O5Purity:99.08%Color and Shape:SolidMolecular weight:631.59Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Formula:C31H38N2OPurity:97.49%Color and Shape:SolidMolecular weight:454.65Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Formula:C13H16N2Purity:97.85% - 99.77%Color and Shape:SolidMolecular weight:200.28RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Formula:C21H22ClF3N2O2Purity:98.95%Color and Shape:SolidMolecular weight:426.86Filorexant
CAS:<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Formula:C24H25FN4O2Purity:98.88%Color and Shape:SolidMolecular weight:420.48Levodropropizine
CAS:<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Formula:C13H20N2O2Purity:99.87% - 99.93%Color and Shape:White Or Off White Crystalline PowderMolecular weight:236.31Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurity:99.84% - 99.92%Color and Shape:White SolidMolecular weight:332.87Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purity:99.79%Color and Shape:SolidMolecular weight:353.29Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Formula:C16H26ClNO3Purity:99.94% - ≥95%Color and Shape:SolidMolecular weight:315.84Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Formula:C21H22CL2N4OSPurity:97.97% - 99.82%Color and Shape:SolidMolecular weight:449.4Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Formula:C26H27N5O2Purity:99.61%Color and Shape:Light Yellow SolidMolecular weight:441.52Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Formula:C22H34Cl2N2O2Purity:98.55%Color and Shape:SolidMolecular weight:429.42Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Formula:C24H28ClN5O3Purity:99.57% - 99.77%Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)Molecular weight:469.96Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurity:99.94%Color and Shape:SolidMolecular weight:217.65Methoxamine hydrochloride
CAS:<p>Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.</p>Formula:C11H18ClNO3Purity:99.84% - >99.99%Color and Shape:Colorless Or White Plate-Like Crystals Or White Crystalline Powder SolidMolecular weight:247.719Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurity:99.90%Color and Shape:SolidMolecular weight:320.88Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Formula:C18H29ClN2O4Purity:99.92% - >99.99%Color and Shape:White Or Slightly Off-White Crystalline Powder SolidMolecular weight:372.89Pizotifen
CAS:<p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>Formula:C19H21NSPurity:99.93%Color and Shape:SolidMolecular weight:295.44Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Formula:C59H79N15O21S6Purity:97.93% - 98.71%Color and Shape:SolidMolecular weight:1526.74MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Formula:C27H25N3O4S2Purity:97.44%Color and Shape:SolidMolecular weight:519.64Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formula:C15H20N2O2·HClPurity:99.64% - 99.92%Color and Shape:SolidMolecular weight:296.79Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formula:C84H107ClN18O18Purity:98.66%Color and Shape:SolidMolecular weight:1692.34Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purity:99.4% - 99.97%Color and Shape:SolidMolecular weight:461.81Olinciguat
CAS:<p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>Formula:C21H16F5N7O3Purity:99.33% - 99.71%Color and Shape:SolidMolecular weight:509.39Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Ogerin
CAS:<p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>Formula:C17H17N5OPurity:99.5% - 99.75%Color and Shape:SolidMolecular weight:307.35

