GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Balovaptan
CAS:Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.Formula:C22H24ClN5OPurity:99.88%Color and Shape:SolidMolecular weight:409.91Erenumab
CAS:<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Purity:99.43% (SEC-HPLC) - > 95%Color and Shape:LiquidMolecular weight:146.2 kDaML604086
CAS:<p>ML604086 suppresses CCL1 mediated chemotaxis and enhances intracellular Ca2 concentrations.</p>Formula:C27H32N4O4SPurity:99.91%Color and Shape:SolidMolecular weight:508.63Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White Crystalline PowderMolecular weight:341.43YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Formula:C33H37N5O5SPurity:99.67%Color and Shape:SolidMolecular weight:615.74PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Formula:C25H37Cl2N3O2Purity:99.68%Color and Shape:SolidMolecular weight:482.49Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Purity:97.76%Color and Shape:SoildSergliflozin A
CAS:<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Formula:C20H24O7Purity:99.43%Color and Shape:SolidMolecular weight:376.4Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H11ClFNO2Purity:99.98%Color and Shape:SoildMolecular weight:231.65Dexchlorpheniramine Maleate
CAS:<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Formula:C20H23ClN2O4Purity:99.58%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:390.86Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formula:C17H19ClF3NOPurity:99.6% - 99.98%Color and Shape:White To Off-White Crystalline Solid White To Off-White PowderMolecular weight:345.787Ticagrelor
CAS:<p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>Formula:C23H28F2N6O4SPurity:98.08% - 99.77%Color and Shape:SolidMolecular weight:522.57Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purity:98% - 99.82%Color and Shape:SolidMolecular weight:425.91hGPR91 antagonist 1
CAS:<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Formula:C31H23F4N3OPurity:98.89%Color and Shape:SolidMolecular weight:529.53Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Formula:C16H15FN6OSPurity:98.62% - 99.7%Color and Shape:SolidMolecular weight:358.39Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurity:99.85%Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Molecular weight:320.88Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Formula:C17H19ClN4OPurity:99.90%Color and Shape:Off-White PowderMolecular weight:330.81Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.Purity:> 95%Color and Shape:LiquidMolecular weight:146.28 kDaFluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Formula:C17H18F3NOPurity:99.07% - 99.28%Color and Shape:SolidMolecular weight:309.33Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purity:99.46%Color and Shape:White To Off-White SolidMolecular weight:525.59Latanoprostene bunod
CAS:<p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>Formula:C27H41NO8Purity:99.33% - 99.69%Color and Shape:SolidMolecular weight:507.62Tabernanthalog fumarate
CAS:<p>Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.</p>Formula:C18H22N2O5Purity:99.83%Color and Shape:SoildMolecular weight:346.38Gevotroline
CAS:<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Formula:C19H20FN3Purity:98.65%Color and Shape:SolidMolecular weight:309.38SBI-477
CAS:<p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>Formula:C24H25N3O6SPurity:99.3%Color and Shape:SolidMolecular weight:483.54Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purity:99.97%Color and Shape:SolidMolecular weight:311.89JNJ-18038683
CAS:<p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>Formula:C26H28ClN3O7Purity:97.29%Color and Shape:SolidMolecular weight:529.97Senktide acetate
<p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>Formula:C42H59N7O13SPurity:98.26%Color and Shape:SolidMolecular weight:902.02Pramipexole
CAS:<p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>Formula:C10H17N3SPurity:98% - 99.96%Color and Shape:SolidMolecular weight:211.33Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurity:99.22% - 99.92%Color and Shape:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMolecular weight:387.9Buflomedil hydrochloride
CAS:<p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>Formula:C17H26ClNO4Purity:99.7% - 99.91%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:343.85CCR2-RA-[R]
CAS:<p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>Formula:C18H19ClFNO3Purity:99.7%Color and Shape:SolidMolecular weight:351.8Labetalol
CAS:<p>Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.</p>Formula:C19H24N2O3Purity:99.87% - 99.89%Color and Shape:SolidMolecular weight:328.41Avexitide acetate
CAS:<p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>Formula:C155H246N40O53SPurity:96.64% - 98.65%Color and Shape:SolidMolecular weight:3549.91L-741626
CAS:<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Formula:C20H21ClN2OPurity:98.57%Color and Shape:SolidMolecular weight:340.85[Leu15]-Gastrin I, human
CAS:[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.Formula:C98H126N20O31Purity:98.02% - 98.84%Color and Shape:SolidMolecular weight:2080.16Imidazolidinyl urea
CAS:<p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>Formula:C11H16N8O8Purity:98.6%Color and Shape:White Fluid Powder With Slight Characteristic OdorMolecular weight:388.29Xylometazoline hydrochloride
CAS:<p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>Formula:C16H24N2·HClPurity:99.77% - 99.87%Color and Shape:White To Off-White Crystalline PowderMolecular weight:280.84Antazoline hydrochloride
CAS:<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Formula:C17H19N3·HClPurity:98% - 99.53%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:301.82Paroxetine hydrochloride
CAS:<p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>Formula:C19H21ClFNO3Purity:98% - 99.99%Color and Shape:White Crystalline PowderMolecular weight:365.826Promethazine
CAS:<p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>Formula:C17H20N2SPurity:99.76%Color and Shape:CrystalsMolecular weight:284.42Isoxsuprine hydrochloride
CAS:<p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>Formula:C18H24ClNO3Purity:99.38%Color and Shape:Crystals From Water SolidMolecular weight:337.84Metaraminol tartrate
CAS:<p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Formula:C13H19NO8Purity:99.68%Color and Shape:White PowderMolecular weight:317.29Nardeterol HCl
<p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>Formula:C20H25ClFN3O2Purity:97.72% - 98.65%Color and Shape:SoildMolecular weight:393.88Duloxetine hydrochloride
CAS:<p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>Formula:C18H20ClNOSPurity:99.93% - >99.99%Color and Shape:White Or White Crystalline PowderMolecular weight:333.88Anamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Formula:C31H42N6O3Purity:99.35% - 99.94%Color and Shape:SolidMolecular weight:546.7Glycerol phenylbutyrate
CAS:Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).Formula:C33H38O6Purity:98.54% - 99.74%Color and Shape:SolidMolecular weight:530.65Spiperone
CAS:<p>Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.</p>Formula:C23H26FN3O2Purity:99.34% - 99.91%Color and Shape:SolidMolecular weight:395.47Ifenprodil Tartrate
CAS:<p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>Formula:C21H27NO2C4H6O6Purity:99.02% - 99.55%Color and Shape:SolidMolecular weight:400.49Aripiprazole Lauroxil
CAS:<p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>Formula:C36H51Cl2N3O4Purity:99.64%Color and Shape:SolidMolecular weight:660.71Labetalol hydrochloride
CAS:<p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>Formula:C19H25ClN2O3Purity:99.54% - 99.85%Color and Shape:SolidMolecular weight:364.87CCX140
CAS:<p>CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.</p>Formula:C20H13ClF3N5O3SPurity:99.66% - 99.95%Color and Shape:SolidMolecular weight:495.86JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formula:C11H19N5Purity:98.33% - 99.62%Color and Shape:SolidMolecular weight:221.3J-113863
CAS:<p>J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).</p>Formula:C30H37Cl2IN2O2Purity:95.11%Color and Shape:SolidMolecular weight:655.44Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Formula:C20H23ClN2O5Purity:99.97%Color and Shape:Off-White SolidMolecular weight:406.86UCM-1306
CAS:<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Formula:C14H14FNO2SPurity:99.98%Color and Shape:SoildMolecular weight:279.33Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formula:C34H36Cl2N6O5S·2ClHPurity:99.17% - 99.58%Color and Shape:SoildMolecular weight:784.58Carvedilol EP IMpurity E
CAS:<p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>Formula:C9H14ClNO2Purity:99.53%Color and Shape:White To Almost White Solid CrystallineMolecular weight:203.666Enrasentan
CAS:Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure and protects myocardial function.Formula:C29H30O8Purity:97.9% - 98.39%Color and Shape:SolidMolecular weight:506.54Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Formula:C30H32ClN3O8SPurity:98.46% - 99.89%Color and Shape:SolidMolecular weight:630.11Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formula:C22H24ClN3O5Purity:99.69%Color and Shape:White To Of-White SolidMolecular weight:445.9Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Formula:C18H25ClN4OPurity:99.88% - 99.93%Color and Shape:White To Off-White Crystalline SolidMolecular weight:348.87Nepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Formula:C15H14N2O2Purity:98.94% - 99.43%Color and Shape:SolidMolecular weight:254.28MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Formula:C27H25N3O4S2Purity:97.44%Color and Shape:SolidMolecular weight:519.64Tropanserin
CAS:<p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>Formula:C17H23NO2Purity:99.74%Color and Shape:SolidMolecular weight:273.37Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Formula:C22H23ClN2O2Purity:99.71% - 99.98%Color and Shape:White PowderMolecular weight:382.88PF-04995274
CAS:<p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>Formula:C23H32N2O6Purity:99.52%Color and Shape:SolidMolecular weight:432.51Cloperastine hydrochloride
CAS:<p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>Formula:C20H25Cl2NOPurity:97.74% - 99.42%Color and Shape:SolidMolecular weight:366.33INCB-9471
CAS:<p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>Formula:C30H40F3N5O2Purity:98.80%Color and Shape:SolidMolecular weight:559.666Sumatriptan succinate
CAS:<p>Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.</p>Formula:C18H27N3O6SPurity:97.53% - 99.51%Color and Shape:White PowderMolecular weight:413.49BF-1
CAS:<p>BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.</p>Formula:C22H25NO2SPurity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:367.50Carbazochrome sodium sulfonate
CAS:<p>Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.</p>Formula:C10H11N4NaO5SPurity:99.63%Color and Shape:Orange Yellow Crystalline PowderMolecular weight:322.03Midodrine hydrochloride
CAS:<p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>Formula:C12H19ClN2O4Purity:99.79% - >99.99%Color and Shape:Crystalline SolidMolecular weight:290.74Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Formula:C4H7NO2SPurity:99.99%Color and Shape:SolidMolecular weight:133.17Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formula:C26H28Cl2F2N2Purity:99.53% - 99.89%Color and Shape:White Crystalline Powder Odorless And TastelessMolecular weight:477.42Rebamipide
CAS:<p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>Formula:C19H15ClN2O4Purity:99.48% - 99.61%Color and Shape:White PowderMolecular weight:370.79Tolnaftate
CAS:<p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>Formula:C19H17NOSPurity:98.85%Color and Shape:White PowderMolecular weight:307.41Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Formula:C23H29ClFN3O4Purity:99.77%Color and Shape:White To Slightly Biege Powder SolidMolecular weight:465.95Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Formula:C17H22ClNOPurity:99.86%Color and Shape:White SolidMolecular weight:291.82ONC206
CAS:<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Formula:C23H22F2N4OPurity:99.38% - 99.81%Color and Shape:SolidMolecular weight:408.44Dapoxetine hydrochloride
CAS:<p>Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.</p>Formula:C21H23NO·HClPurity:99.70% - 99.91%Color and Shape:White To Off-White Crystalline SolidMolecular weight:341.87Delequamine
CAS:<p>Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.</p>Formula:C18H26N2O3SPurity:99.39%Color and Shape:SolidMolecular weight:350.48Carebastine
CAS:<p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>Formula:C32H37NO4Purity:99.16%Color and Shape:Off-White SolidMolecular weight:499.64CE3F4
CAS:<p>CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).</p>Formula:C11H10Br2FNOPurity:97.15% - 98.06%Color and Shape:SolidMolecular weight:351.01Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Formula:C17H20N4SPurity:99.86% - ≥95%Color and Shape:Yellowish Crystalline PowderMolecular weight:312.43PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C31H30FN5O4Purity:97.19% - 99.56%Color and Shape:SolidMolecular weight:555.6MK-0812 Succinate
CAS:<p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>Formula:C28H40F3N3O7Purity:98.62% - 99.93%Color and Shape:SolidMolecular weight:587.63Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Formula:C12H17Cl2NOPurity:99.38%Color and Shape:SolidMolecular weight:262.18NF-56-EJ40 hydrochloride
CAS:<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Formula:C27H31Cl2N3O3Purity:99.33%Color and Shape:SoildMolecular weight:516.46Vabicaserin hydrochloride
CAS:<p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>Formula:C15H21ClN2Purity:98.32%Color and Shape:SolidMolecular weight:264.79Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurity:99.64%Color and Shape:Light Yellow To Yellow SolidMolecular weight:396.51Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Formula:C18H23Cl2NOPurity:98.04% - >99.99%Color and Shape:Antihypertensive DrugMolecular weight:340.3HJC0197
CAS:<p>HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.</p>Formula:C19H21N3OSPurity:98.05%Color and Shape:SolidMolecular weight:339.45Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Formula:C21H25ClN2O3Purity:98% - 99.94%Color and Shape:White PowderMolecular weight:388.89Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purity:99.32% - >99.99%Color and Shape:White Crystalline SolidMolecular weight:883.09RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Formula:C21H22ClF3N2O2Purity:98.95%Color and Shape:SolidMolecular weight:426.86AM095 free acid
CAS:<p>AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).</p>Formula:C27H24N2O5Purity:99.88%Color and Shape:SolidMolecular weight:456.49Bufotenidine hydrochloride(487-91-2 Free base)
CAS:<p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>Formula:C13H19ClN2OPurity:99.88%Color and Shape:SolidMolecular weight:254.76Propafenone
CAS:<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Formula:C21H27NO3Purity:99.02%Color and Shape:SolidMolecular weight:341.44Capeserod
CAS:<p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>Formula:C23H25ClN4O4Purity:98.10% - 99.94%Color and Shape:SolidMolecular weight:456.92Leronlimab
CAS:<p>Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.</p>Purity:SDS-PAGE:95.0%;SEC-HPLC:99.6%Color and Shape:LiquidMolecular weight:146.66 kDaTiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formula:C15H24N2O4S·HClPurity:99.4% - 99.77%Color and Shape:SolidMolecular weight:364.89(S)-(-)-Atenolol
CAS:<p>(S)-(-)-Atenolol has beta-adrenergic blocking effects.</p>Formula:C14H22N2O3Purity:99.31% - 99.81%Color and Shape:SolidMolecular weight:266.34RS 15385-198
CAS:<p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>Formula:C18H26N2O3SPurity:>99.99%Color and Shape:SoildMolecular weight:350.48Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purity:99.79%Color and Shape:SolidMolecular weight:353.29CI 169369
CAS:<p>CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.</p>Formula:C19H21ClN2SPurity:98.97%Color and Shape:SoildMolecular weight:344.9Alarelin Acetate
CAS:<p>Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.</p>Formula:C56H78N16O12Purity:99.81% - >99.99%Color and Shape:White PowderMolecular weight:1167.34(±) Clopidogrel hydrogen sulfate
CAS:<p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>Formula:C16H16ClNO2S·H2SO4Purity:98.67% - 99.04%Color and Shape:Colorless To Light Yellow LiquidMolecular weight:419.9ESI-05
CAS:<p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>Formula:C16H18O2SPurity:97.22%Color and Shape:SolidMolecular weight:274.38Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Formula:C21H27NO2Purity:99.58%Color and Shape:White Crystalline PowderMolecular weight:325.44Proglumide
CAS:<p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>Formula:C18H26N2O4Purity:99.4% - 99.45%Color and Shape:White Crystalline PowderMolecular weight:334.41Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Formula:C18H29ClN2O4Purity:99.92% - >99.99%Color and Shape:White Or Slightly Off-White Crystalline Powder SolidMolecular weight:372.89Apelin-13
CAS:<p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>Formula:C69H111N23O16SPurity:96.81%Color and Shape:SolidMolecular weight:1550.83(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formula:C22H24ClF4N5OSPurity:98.36%Color and Shape:SoildMolecular weight:517.97Azacyclonol
CAS:<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Formula:C18H21NOPurity:99.46%Color and Shape:Solid PowderMolecular weight:267.37Sulpiride
CAS:<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Formula:C15H23N3O4SPurity:99.94%Color and Shape:White Crystalline PowderMolecular weight:341.43MRGPRX1 agonist 1
CAS:<p>MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).</p>Formula:C23H21N3O4SPurity:99.95%Color and Shape:SolidMolecular weight:435.5Prasugrel
CAS:Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent THROMBOSIS in patients with ACUTE CORONARY SYNDROME;Formula:C20H20FNO3SPurity:99.62% - 99.82%Color and Shape:White SolidMolecular weight:373.44Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Formula:C18H25N3O6Purity:99.66%Color and Shape:SolidMolecular weight:379.41Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purity:98.41% - 99.96%Color and Shape:White Crystalline Powder; Odourless Or Almost OdourlessMolecular weight:403.53Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formula:C16H20N2·C4H4O4Purity:99.85%Color and Shape:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CMolecular weight:356.42Desvenlafaxine
CAS:<p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>Formula:C16H25NO2Purity:99.46% - 99.81%Color and Shape:White Crystalline PowderMolecular weight:263.38CYM50308
CAS:<p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>Formula:C20H21F2N3O2SPurity:99.43% - 99.77%Color and Shape:SolidMolecular weight:405.46Clopidogrel hydrogen sulfate
CAS:<p>Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.</p>Formula:C16H16ClNO2S·H2SO4Purity:99.57% - 99.79%Color and Shape:SolidMolecular weight:419.9Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurity:99% - 99.99%Color and Shape:SolidMolecular weight:312.842-(1-Piperazinyl)pyrimidine
CAS:<p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>Formula:C8H12N4Purity:98.46%Color and Shape:Liquid - Crystal - LumpMolecular weight:164.21Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurity:99.84% - 99.92%Color and Shape:White SolidMolecular weight:332.87Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Formula:C24H26N2O2Purity:98.88% - 99.68%Color and Shape:SolidMolecular weight:374.48Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formula:C24H27FN2O4Purity:99.42%Color and Shape:SolidMolecular weight:426.48Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formula:C28H32ClN3O8SPurity:99.78%Color and Shape:Off-White PowderMolecular weight:606.09Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Formula:C23H23NO5SPurity:99.25% - 99.73%Color and Shape:SolidMolecular weight:425.50BMY 25368 HCl
CAS:BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.Formula:C19H26ClN3O3Purity:98.73% - 99.81%Color and Shape:SoildMolecular weight:379.88Retatrutide
CAS:<p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>Formula:C221H342N46O68Purity:98.31%Color and Shape:SolidMolecular weight:4732.09GTS-21 dihydrochloride
CAS:<p>GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.</p>Formula:C19H20N2O2·2HClPurity:98.54% - >99.99%Color and Shape:SolidMolecular weight:381.3Vibozilimod
CAS:<p>Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .</p>Formula:C29H36ClN3O5Purity:99.97%Color and Shape:SolidMolecular weight:542.072',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Formula:C10H13N5O2Purity:99.55%Color and Shape:White SolidMolecular weight:235.24Dazmegrel HCl
Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.Formula:C16H18ClN3O2Purity:98.30%Color and Shape:SolidMolecular weight:319.79Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Formula:C21H22ClNPurity:98.75% - 99.84%Color and Shape:SolidMolecular weight:323.86Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Formula:C10H7KN6OPurity:98.91% - 99.63%Color and Shape:Crystals From Dimethylformamide Crystalline SolidMolecular weight:266.31Tolnapersine TFA
<p>Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.</p>Formula:C23H27F3N2O3Purity:99.14%Color and Shape:SoildMolecular weight:436.47Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formula:C84H107ClN18O18Purity:98.66%Color and Shape:SolidMolecular weight:1692.34Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Formula:C22H28Cl2F3N3OSPurity:99.23%Color and Shape:Off-White SolidMolecular weight:510.44Cloroperone
CAS:<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Formula:C22H23ClFNO2Purity:98.40%Color and Shape:SoildMolecular weight:387.88JMV 2959 hydrochloride (925238-89-7 free base)
CAS:<p>JMV 2959 hydrochloride (925238-89-7 free base) is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.</p>Formula:C30H33ClN6O2Purity:98.09%Color and Shape:SolidMolecular weight:545.08Mianserin hydrochloride
CAS:Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formula:C18H21ClN2Purity:99.63% - 99.82%Color and Shape:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMolecular weight:300.83Bucumolol
CAS:<p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>Formula:C17H23NO4Purity:99.66%Color and Shape:SoildMolecular weight:305.37Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Formula:C13H23ClN4O3SPurity:99.30% - 99.49%Color and Shape:SolidMolecular weight:350.86Mizolastine
CAS:<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Formula:C24H25FN6OPurity:98% - 99.75%Color and Shape:SolidMolecular weight:432.49SR59230A
CAS:<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Formula:C23H29NO6Purity:98.84%Color and Shape:SolidMolecular weight:415.48ALLO-2
CAS:ALLO-2 is a Inhibitor of Drug-Resistant Smo Mutant.It inhibits Smo agonist Hh-Ag1.5-induced luciferase expression in TM3-Gli-Luc cells with IC50 of 6 nM.Formula:C18H12F3N5OPurity:99.19%Color and Shape:SolidMolecular weight:371.32Carboprost tromethamine
CAS:<p>Carboprost tromethamine, a synthetic 15-methyl analogue of prostaglandin F2α, effectively promotes uterine contractions and significantly reduces bleeding</p>Formula:C25H47NO8Purity:>99.99%Color and Shape:SolidMolecular weight:489.64Dynarrestin
CAS:Dynarrestin inhibits cytoplasmic dynein 1/2, preventing microtubule sliding without affecting ATP hydrolysis or ciliogenesis.Formula:C22H23F2N3O2SPurity:99.64%Color and Shape:SolidMolecular weight:431.5Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Formula:C17H21NO3·HClPurity:99% - 99.52%Color and Shape:SolidMolecular weight:323.82Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.Formula:C225H347N48O68NaPurity:99.69%Color and Shape:SoildMolecular weight:4835.51Carteolol hydrochloride
CAS:Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.Formula:C16H24N2O3·HClPurity:99.84% - 99.91%Color and Shape:SolidMolecular weight:328.83Itopride hydrochloride
CAS:<p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>Formula:C20H27ClN2O4Purity:99.59%Color and Shape:White Or Pale Brownish CrystalMolecular weight:394.9Nicergoline
CAS:<p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>Formula:C24H26BrN3O3Purity:98% - 99.80%Color and Shape:SolidMolecular weight:484.39EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Formula:C23H26N4O4SPurity:99.11%Color and Shape:SolidMolecular weight:454.54Amisulpride
CAS:Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formula:C17H27N3O4SPurity:99.97% - 99.99%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:369.48Solabegron
CAS:<p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>Formula:C23H23ClN2O3Purity:97.89%Color and Shape:SolidMolecular weight:410.89Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Formula:C20H24ClNPurity:97% - 99.94%Color and Shape:Crystals White To Off-White PowderMolecular weight:313.86REV 5901A
CAS:<p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>Formula:C22H26ClNO2Purity:98.04%Color and Shape:SoildMolecular weight:371.90Sarizotan 2HCl
CAS:<p>Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.</p>Formula:C22H23Cl2FN2OPurity:98.83%Color and Shape:SoildMolecular weight:421.346-Iodopravadoline
CAS:<p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>Formula:C23H25IN2O3Purity:99.29%Color and Shape:Off-White SolidMolecular weight:504.36Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Formula:C13H16N2Purity:97.85% - 99.77%Color and Shape:SolidMolecular weight:200.28Retatrutide sodium salt
<p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>Purity:99.97%Color and Shape:SoildEvatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formula:C25H28N2O5SPurity:97.09%Color and Shape:SolidMolecular weight:468.57Terbutaline
CAS:Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterolFormula:C12H19NO3Purity:99.12%Color and Shape:SolidMolecular weight:225.3Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formula:C21H28N2O5Purity:99.61%Color and Shape:5 1 (Ntp 1992)Molecular weight:388.46Azelastine hydrochloride
CAS:<p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>Formula:C22H24ClN3O·HClPurity:98% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:418.36Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurity:99.94%Color and Shape:SolidMolecular weight:217.65Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Formula:C26H35NO7Purity:97.12% - 98.38%Color and Shape:SolidMolecular weight:473.56Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purity:99.85%Color and Shape:SolidMolecular weight:367.5Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Formula:C20H22BrFN2OPurity:99.81%Color and Shape:White Crystalline PowderMolecular weight:405.304Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurity:99.55%Color and Shape:Tan SolidMolecular weight:412.94Chlorpheniramine maleate
CAS:<p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>Formula:C20H23ClN2O4Purity:99.64% - 99.98%Color and Shape:Odorless White Crystalline Solid Or White Powder With A Bitter TasteMolecular weight:390.87Ziprasidone hydrochloride monohydrate
CAS:<p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>Formula:C21H21ClN4OS·HCl·H2OPurity:98% - 99.83%Color and Shape:Off-White PowderMolecular weight:467.12Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Formula:C31H38N2OPurity:97.49%Color and Shape:SolidMolecular weight:454.65Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Formula:C31H37N3O10SPurity:99.39% - 99.48%Color and Shape:SolidMolecular weight:643.71Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formula:C21H23N3OSPurity:99.61%Color and Shape:SolidMolecular weight:365.49Ornidazole
CAS:<p>Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.</p>Formula:C7H10ClN3O3Purity:99.47%Color and Shape:Crystalline SolidMolecular weight:219.63Desipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formula:C18H23ClN2Purity:99.58% - 99.94%Color and Shape:White To Off-White PowderMolecular weight:302.842Roluperidone
CAS:<p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>Formula:C22H23FN2O2Purity:96.46% - 97.77%Color and Shape:SolidMolecular weight:366.43Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formula:C14H22BrN3O2Purity:99.95%Color and Shape:SolidMolecular weight:344.25Bromperidol
CAS:<p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>Formula:C21H23BrFNO2Purity:99.89%Color and Shape:Tan SolidMolecular weight:420.32[D-Pro2] Spantide I TFA
<p>[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].</p>Formula:C75H108N20O13·xC2HF3O2Purity:98%Color and Shape:SolidCB2R agonist 3
<p>CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [</p>Purity:98%Color and Shape:Odour SolidHL2-m5
CAS:HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formula:C70H101N15O24S3Color and Shape:SolidMolecular weight:1632.83Mibenratide TFA
<p>Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].</p>Purity:98%Color and Shape:Odour SolidJmv 167
CAS:<p>Jmv 167 is an antagonist of the Cholecystokinin receptor.</p>Formula:C51H68N8O14SPurity:98%Color and Shape:SolidMolecular weight:1049.21(Leu31,Pro34)-Peptide YY (human) (TFA)
<p>"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a derivative of Peptide YY that acts as a</p>Formula:C195H296N54O56·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4292.75 (free base)Galanin-Like Peptide (rat)
CAS:<p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>Formula:C288H461N87O83SPurity:98%Color and Shape:SolidMolecular weight:6502.34LTD4 antagonist 2
CAS:<p>LTD4 antagonist 2 (compound 6) functions as a leukotriene D4 (LTD4) antagonist with an IC50 of 2.8 μM for the cysteinyl leukotriene 1 receptor (CysLT1R). Additionally, it acts as an agonist for the G protein-coupled bile acid receptor 1 (GPBAR1), making it applicable for research into colitis, metabolic syndrome, and other GPBAR1- and CysLT1R-related diseases.</p>Formula:C17H13NO3Color and Shape:SolidMolecular weight:279.29Pafenolol
CAS:<p>Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.</p>Formula:C18H31N3O3Purity:98.33%Color and Shape:SolidMolecular weight:337.46Tetrapeptide-1
CAS:<p>Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].</p>Formula:C20H36N4O6Purity:98%Color and Shape:SolidMolecular weight:428.52AD353
<p>AD353 is a selective sigma-1 receptor ligand. It demonstrates high efficacy in models of capsaicin-induced allodynia and PGE2-induced mechanical hyperalgesia. Additionally, AD353 exhibits favorable pharmacokinetic properties.</p>Formula:C23H30N2O2Color and Shape:SolidMolecular weight:366.5CB2 receptor agonist 9
CAS:<p>CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.</p>Formula:C16H23N3O2SColor and Shape:SolidMolecular weight:321.44SBI-810
CAS:<p>SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.</p>Formula:C27H34N4O2Color and Shape:SolidMolecular weight:446.59
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