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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Latozinemab


    Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.28 kDa
  • Dynarrestin

    CAS:
    Dynarrestin inhibits cytoplasmic dynein 1/2, preventing microtubule sliding without affecting ATP hydrolysis or ciliogenesis.
    Formula:C22H23F2N3O2S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:431.5
  • Mizolastine

    CAS:
    Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.
    Formula:C24H25FN6O
    Purity:98% - 99.75%
    Color and Shape:Solid
    Molecular weight:432.49
  • [Leu15]-Gastrin I, human

    CAS:
    [Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.
    Formula:C98H126N20O31
    Purity:98.02% - 98.84%
    Color and Shape:Solid
    Molecular weight:2080.16
  • Clomipramine hydrochloride

    CAS:
    Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.
    Formula:C19H23ClN2·HCl
    Purity:99.04% - 99.47%
    Color and Shape:White To Slightly Yellow Crystalline Powder
    Molecular weight:351.31
  • AZ084

    CAS:
    AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.
    Formula:C26H34N4O2
    Purity:97.12%
    Color and Shape:Solid
    Molecular weight:434.57
  • Volagidemab

    CAS:
    <p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>
    Purity:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)
    Color and Shape:Liquid
  • Xylometazoline hydrochloride

    CAS:
    <p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>
    Formula:C16H24N2·HCl
    Purity:99.77% - 99.87%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:280.84
  • Azasetron hydrochloride

    CAS:
    <p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>
    Formula:C17H20ClN3O3·HCl
    Purity:99.50%
    Color and Shape:Solid
    Molecular weight:386.27
  • Mefexamide hydrochloride

    CAS:
    Mefexamide hydrochloride is a central stimulant.
    Formula:C15H25ClN2O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:316.83
  • Carboprost tromethamine

    CAS:
    <p>Carboprost tromethamine, a synthetic 15-methyl analogue of prostaglandin F2α, effectively promotes uterine contractions and significantly reduces bleeding</p>
    Formula:C25H47NO8
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:489.64
  • Ogerin

    CAS:
    <p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>
    Formula:C17H17N5O
    Purity:99.5% - 99.75%
    Color and Shape:Solid
    Molecular weight:307.35
  • Vabicaserin hydrochloride

    CAS:
    Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).
    Formula:C15H21ClN2
    Purity:98.32%
    Color and Shape:Solid
    Molecular weight:264.79
  • Cinnarizine

    CAS:
    <p>Cinnarizine is a piperazine, blocks H1-receptor &amp; Ca-channels, has vasodilating &amp; antiemetic effects, may cause Parkinson-like symptoms.</p>
    Formula:C26H28N2
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:368.51
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Formula:C19H26ClN5O4
    Purity:99.69% - 99.91%
    Color and Shape:Solid
    Molecular weight:423.89
  • Agomelatine

    CAS:
    Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
    Formula:C15H17NO2
    Purity:99.92%
    Color and Shape:White Solid
    Molecular weight:243.3
  • Bufotenidine hydrochloride(487-91-2 Free base)

    CAS:
    <p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>
    Formula:C13H19ClN2O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:254.76
  • Carteolol hydrochloride

    CAS:
    Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.
    Formula:C16H24N2O3·HCl
    Purity:99.84% - 99.91%
    Color and Shape:Solid
    Molecular weight:328.83
  • Centanafadine hydrochloride

    CAS:
    Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).
    Formula:C15H16ClN
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:245.75
  • Metoclopramide hydrochloride

    CAS:
    Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
    Formula:C14H22ClN3O2·HCl
    Purity:99.99%
    Color and Shape:White To Off-White Powder
    Molecular weight:336.26
  • GR 103691

    CAS:
    <p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>
    Formula:C30H35N3O3
    Purity:98.94% - 99.29%
    Color and Shape:Solid
    Molecular weight:485.62
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Formula:C25H28N2O5S
    Purity:97.09%
    Color and Shape:Solid
    Molecular weight:468.57
  • Benserazide hydrochloride

    CAS:
    <p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>
    Formula:C10H15N3O5·HCl
    Purity:98.63% - 99.74%
    Color and Shape:White Crystalline Solid
    Molecular weight:293.7
  • Traxanox

    CAS:
    Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.
    Formula:C13H6ClN5O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:299.67
  • Domperidone

    CAS:
    <p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>
    Formula:C22H24ClN5O2
    Purity:98% - 99.82%
    Color and Shape:Solid
    Molecular weight:425.91
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Formula:C11H19N5
    Purity:98.33% - 99.62%
    Color and Shape:Solid
    Molecular weight:221.3
  • PF-4348235 2HCl


    <p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>
    Formula:C36H51Cl3N4O7S
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:790.24
  • Dexchlorpheniramine Maleate

    CAS:
    <p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>
    Formula:C20H23ClN2O4
    Purity:99.58%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:390.86
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Formula:C21H26ClN3OS
    Purity:99.3% - 99.99%
    Color and Shape:Solid
    Molecular weight:403.97
  • Astemizole

    CAS:
    <p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>
    Formula:C28H31FN4O
    Purity:98.24% - 99.67%
    Color and Shape:White Crystals Solid
    Molecular weight:458.57
  • Cefaclor monohydrate

    CAS:
    <p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>
    Formula:C15H16ClN3O5S
    Purity:97.36% - 99.9%
    Color and Shape:White Crystaling Powder
    Molecular weight:385.82
  • Triflupromazine hydrochloride

    CAS:
    Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
    Formula:C18H20ClF3N2S
    Purity:99.76% - 99.82%
    Color and Shape:Crystals
    Molecular weight:388.88
  • Alosetron hydrochloride

    CAS:
    Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.
    Formula:C17H19ClN4O
    Purity:99.90%
    Color and Shape:Off-White Powder
    Molecular weight:330.81
  • Bromopride

    CAS:
    Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.
    Formula:C14H22BrN3O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:344.25
  • 2-(1-Piperazinyl)pyrimidine

    CAS:
    2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
    Formula:C8H12N4
    Purity:98.46%
    Color and Shape:Liquid - Crystal - Lump
    Molecular weight:164.21
  • Propafenone

    CAS:
    <p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>
    Formula:C21H27NO3
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:341.44
  • Cericlamine

    CAS:
    Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.
    Formula:C12H17Cl2NO
    Purity:99.06%
    Color and Shape:Solid
    Molecular weight:262.18
  • Lofepramine

    CAS:
    <p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>
    Formula:C26H27ClN2O
    Purity:98.38%
    Color and Shape:Crystals From Methanol Or Acetone Solid
    Molecular weight:418.96
  • Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Formula:C46H54N6O8S2
    Purity:99.32% - >99.99%
    Color and Shape:White Crystalline Solid
    Molecular weight:883.09
  • Lamotrigine

    CAS:
    Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
    Formula:C9H7Cl2N5
    Purity:99.76% - 99.95%
    Color and Shape:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Molecular weight:256.09
  • Talipexole dihydrochloride

    CAS:
    Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and
    Formula:C10H17Cl2N3S
    Purity:99.89%
    Color and Shape:Light Yellow Solid
    Molecular weight:282.23
  • Evocalcet

    CAS:
    Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
    Formula:C24H26N2O2
    Purity:98.88% - 99.68%
    Color and Shape:Solid
    Molecular weight:374.48
  • Hydroxyzine Pamoate

    CAS:
    Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.
    Formula:C44H43ClN2O8
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:763.27
  • Nepafenac

    CAS:
    Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.
    Formula:C15H14N2O2
    Purity:98.94% - 99.43%
    Color and Shape:Solid
    Molecular weight:254.28
  • Pamabrom

    CAS:
    Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.
    Formula:C11H18BrN5O3
    Purity:99.84% - >99.99%
    Color and Shape:Coa
    Molecular weight:348.2
  • Ornidazole

    CAS:
    Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.
    Formula:C7H10ClN3O3
    Purity:99.47%
    Color and Shape:Crystalline Solid
    Molecular weight:219.63
  • Prostaglandin E1

    CAS:
    Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.
    Formula:C20H34O5
    Purity:99.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:354.48
  • Luzindole

    CAS:
    Luzindole (N-0774) is a selective melatonin receptor antagonist.
    Formula:C19H20N2O
    Purity:98.53%
    Color and Shape:Off-White Amorphous Solid
    Molecular weight:292.37
  • Iloperidone

    CAS:
    Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
    Formula:C24H27FN2O4
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:426.48
  • Ciproquazone

    CAS:
    Ciproquazone has analgesic activity and is used to treat spondylitis.
    Formula:C19H18N2O2
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:306.36
  • EMPA

    CAS:
    <p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>
    Formula:C23H26N4O4S
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:454.54
  • Pheniramine maleate

    CAS:
    Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.
    Formula:C16H20N2·C4H4O4
    Purity:99.85%
    Color and Shape:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
    Molecular weight:356.42
  • Aniracetam

    CAS:
    <p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>
    Formula:C12H13NO3
    Purity:99.88% - 99.89%
    Color and Shape:White Crystalline Or Crystalline Powde
    Molecular weight:219.24
  • NS-2028

    CAS:
    NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.
    Formula:C9H5BrN2O3
    Purity:99.44%
    Color and Shape:A Crystalline Solid
    Molecular weight:269.05
  • DPTN dihydrochloride

    CAS:
    DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
    Formula:C22H20Cl2N4OS
    Purity:99.95%
    Color and Shape:Soild
    Molecular weight:459.39
  • Ticagrelor

    CAS:
    <p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>
    Formula:C23H28F2N6O4S
    Purity:98.08% - 99.77%
    Color and Shape:Solid
    Molecular weight:522.57
  • PF-04995274

    CAS:
    PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.
    Formula:C23H32N2O6
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:432.51
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Formula:C10H16N6S
    Purity:99.82%
    Color and Shape:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Molecular weight:252.34
  • Naftidrofuryl oxalate

    CAS:
    <p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>
    Formula:C26H35NO7
    Purity:97.12% - 98.38%
    Color and Shape:Solid
    Molecular weight:473.56
  • Naftifine hydrochloride

    CAS:
    Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.
    Formula:C21H22ClN
    Purity:98.75% - 99.84%
    Color and Shape:Solid
    Molecular weight:323.86
  • Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Formula:C34H36Cl2N6O5S·2ClH
    Purity:99.17% - 99.58%
    Color and Shape:Soild
    Molecular weight:784.58
  • Gevotroline

    CAS:
    <p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>
    Formula:C19H20FN3
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:309.38
  • Senktide acetate


    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Formula:C42H59N7O13S
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:902.02
  • Terfenadine

    CAS:
    Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
    Formula:C32H41NO2
    Purity:98.76% - 99.75%
    Color and Shape:Solid
    Molecular weight:471.67
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Formula:C31H23F4N3O
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:529.53
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Formula:C19H27N5O4·HCl
    Purity:99.78%
    Color and Shape:White To Off-White Solid
    Molecular weight:425.91
  • Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Formula:C23H39ClN4O3S
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:487.1
  • Proglumide

    CAS:
    Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.
    Formula:C18H26N2O4
    Purity:99.4% - 99.45%
    Color and Shape:White Crystalline Powder
    Molecular weight:334.41
  • TSHR antagonist S37

    CAS:
    TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
    Formula:C25H20N2O3S2
    Purity:98.35%
    Color and Shape:Solid
    Molecular weight:460.57
  • Pemirolast potassium

    CAS:
    <p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>
    Formula:C10H7KN6O
    Purity:98.91% - 99.63%
    Color and Shape:Crystals From Dimethylformamide Crystalline Solid
    Molecular weight:266.31
  • Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Formula:C13H16N4
    Purity:98.34% - 99.73%
    Color and Shape:Solid
    Molecular weight:228.29
  • Oxeladin citrate

    CAS:
    <p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>
    Formula:C26H41NO10
    Purity:97.23%
    Color and Shape:Solid
    Molecular weight:527.6
  • Salmeterol

    CAS:
    Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
    Formula:C25H37NO4
    Purity:99.2% - 99.9%
    Color and Shape:Solid
    Molecular weight:415.57
  • Carbetapentane citrate

    CAS:
    Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.
    Formula:C20H31NO3·C6H8O7
    Purity:99.46%
    Color and Shape:White To Off-White Solid
    Molecular weight:525.59
  • (Rac)-MGV354

    CAS:
    <p>(Rac)-MGV354: a racemic sGC activator; EC50s &lt;0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>
    Formula:C35H37N5O3
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:575.7
  • Phentolamine mesylate

    CAS:
    Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.
    Formula:C17H19N3O·CH4O3S
    Purity:99.87% - >99.99%
    Color and Shape:By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
    Molecular weight:377.46
  • Brefonalol HCl


    Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
    Formula:C22H29ClN2O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:388.93
  • Apelin-13

    CAS:
    Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor
    Formula:C69H111N23O16S
    Purity:96.81%
    Color and Shape:Solid
    Molecular weight:1550.83
  • Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Formula:C18H19N3O·HCl·2H2O
    Purity:99.92%
    Color and Shape:White Crystal Powder
    Molecular weight:365.86
  • Bambuterol hydrochloride

    CAS:
    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
    Formula:C18H30ClN3O5
    Purity:99.53% - 99.61%
    Color and Shape:White Solid
    Molecular weight:403.91
  • Adenosine A1 receptor activator T62

    CAS:
    Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also
    Formula:C15H14ClNOS
    Purity:97.83%
    Color and Shape:Solid
    Molecular weight:291.8
  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.
    Formula:C20H29N3O8
    Purity:99.72%
    Color and Shape:Soild
    Molecular weight:439.46
  • Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Formula:C19H31ClF3NO3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:413.9
  • Tropanserin

    CAS:
    <p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>
    Formula:C17H23NO2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:273.37
  • Tetrahydrozoline

    CAS:
    <p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>
    Formula:C13H16N2
    Purity:97.85% - 99.77%
    Color and Shape:Solid
    Molecular weight:200.28
  • (-)-GSK598809 hydrochloride

    CAS:
    <p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>
    Formula:C22H24ClF4N5OS
    Purity:98.36%
    Color and Shape:Soild
    Molecular weight:517.97
  • Frovatriptan succinate hydrate

    CAS:
    <p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>
    Formula:C18H25N3O6
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:379.41
  • JP1302 dihydrochloride

    CAS:
    JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
    Formula:C24H26Cl2N4
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:441.4
  • (±) Clopidogrel hydrogen sulfate

    CAS:
    (±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots
    Formula:C16H16ClNO2S·H2SO4
    Purity:98.67% - 99.04%
    Color and Shape:Colorless To Light Yellow Liquid
    Molecular weight:419.9
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Formula:C21H23N3OS
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:365.49
  • Fexofenadine hydrochloride

    CAS:
    Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with
    Formula:C32H40ClNO4
    Purity:>99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:538.12
  • Dexpramipexole dihydrochloride

    CAS:
    Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine
    Formula:C10H19Cl2N3S
    Purity:99.75% - 99.88%
    Color and Shape:Solid
    Molecular weight:284.25
  • Heptaminol hydrochloride

    CAS:
    <p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>
    Formula:C8H20ClNO
    Purity:98.61%
    Color and Shape:White Crystalline Powder
    Molecular weight:181.71
  • Carvedilol EP IMpurity E

    CAS:
    <p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>
    Formula:C9H14ClNO2
    Purity:99.53%
    Color and Shape:White To Almost White Solid Crystalline
    Molecular weight:203.666
  • Prochlorperazine Maleate

    CAS:
    Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.
    Formula:C28H32ClN3O8S
    Purity:99.78%
    Color and Shape:Off-White Powder
    Molecular weight:606.09
  • PF-610355 HCl


    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Formula:C19H22ClN7O6
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:479.87
  • Promethazine hydrochloride

    CAS:
    Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
    Formula:C17H20N2S·HCl
    Purity:99.85%
    Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Molecular weight:320.88
  • Desvenlafaxine

    CAS:
    <p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>
    Formula:C16H25NO2
    Purity:99.46% - 99.81%
    Color and Shape:White Crystalline Powder
    Molecular weight:263.38
  • NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Formula:C20H24ClN3O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:357.88
  • Rimonabant hydrochloride

    CAS:
    <p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>
    Formula:C22H22Cl4N4O
    Purity:98.24% - 99.5%
    Color and Shape:Off-White To White Crystalline Powder
    Molecular weight:500.25
  • Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Formula:C20H22BrFN2O
    Purity:99.81%
    Color and Shape:White Crystalline Powder
    Molecular weight:405.304
  • PF-5190457

    CAS:
    PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
    Formula:C29H32N6OS
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:512.67
  • Ketanserin

    CAS:
    Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.
    Formula:C22H22FN3O3
    Purity:99.19% - 99.73%
    Color and Shape:Solid
    Molecular weight:395.43
  • Indusatumab

    CAS:
    <p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>
    Purity:> 95% - > 95%
    Color and Shape:Liquid
    Molecular weight:145.18 kDa
  • Anamorelin

    CAS:
    <p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>
    Formula:C31H42N6O3
    Purity:99.35% - 99.94%
    Color and Shape:Solid
    Molecular weight:546.7
  • Tripelennamine hydrochloride

    CAS:
    Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
    Formula:C16H21N3·HCl
    Purity:99.54% - 99.81%
    Color and Shape:White Solid
    Molecular weight:291.82
  • PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C31H30FN5O4
    Purity:97.19% - 99.56%
    Color and Shape:Solid
    Molecular weight:555.6
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.
    Formula:C11H9BrO
    Purity:98.51%
    Color and Shape:White To Off-White Powder
    Molecular weight:237.09
  • Cisapride

    CAS:
    Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.
    Formula:C23H29ClFN3O4
    Purity:99.77%
    Color and Shape:White To Slightly Biege Powder Solid
    Molecular weight:465.95
  • Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Formula:C19H21N·HCl
    Purity:98.54% - 99.98%
    Color and Shape:Solid
    Molecular weight:299.84
  • Urocortin (rat) acetate


    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Purity:97.76%
    Color and Shape:Soild
  • Nylidrin hydrochloride

    CAS:
    Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.
    Formula:C19H26ClNO2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:335.87
  • Terlipressin Acetate

    CAS:
    Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).
    Formula:C56H82N16O19S2
    Purity:98.50% - 99.69%
    Color and Shape:Solid
    Molecular weight:1347.5
  • Sonepcizumab

    CAS:
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Purity:SDS-PAGE:95% SEC-HPLC:98.90%
    Color and Shape:Liquid
    Molecular weight:146.43 kDa
  • Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purity:98.55%
    Color and Shape:Yellowish White Crystalline Powder
    Molecular weight:431.55
  • Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Formula:C18H26ClN3O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:367.87
  • Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Formula:C17H28ClNO2
    Purity:97.32% - 99.86%
    Color and Shape:White Crystalline Powder
    Molecular weight:313.86
  • Erenumab

    CAS:
    <p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>
    Purity:99.43% (SEC-HPLC) - > 95%
    Color and Shape:Liquid
    Molecular weight:146.2 kDa
  • Talastine

    CAS:
    Talastine is an antihistamine compound that can induce an allergic rash.
    Formula:C19H21N3O
    Purity:99.44% - 99.84%
    Color and Shape:Solid
    Molecular weight:307.39
  • Methyldopa

    CAS:
    Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or
    Formula:C10H13NO4
    Purity:98.95% - 99.86%
    Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Molecular weight:211.21
  • Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842
  • Rebamipide

    CAS:
    Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.
    Formula:C19H15ClN2O4
    Purity:99.48% - 99.61%
    Color and Shape:White Powder
    Molecular weight:370.79
  • Fluoxetine hydrochloride

    CAS:
    Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.
    Formula:C17H19ClF3NO
    Purity:99.6% - 99.98%
    Color and Shape:White To Off-White Crystalline Solid White To Off-White Powder
    Molecular weight:345.787
  • Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purity:99.16% - 99.86%
    Color and Shape:Solid
    Molecular weight:266.55
  • Sergliflozin A

    CAS:
    Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.
    Formula:C20H24O7
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:376.4
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:508.56
  • ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Formula:C20H25ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:388.89
  • CD80-IN-3

    CAS:
    <p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>
    Formula:C17H10FN3O3
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:323.28
  • CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purity:98% - 99.08%
    Color and Shape:Solid
    Molecular weight:416.86
  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Formula:C19H25F3N2O6
    Purity:99.92% - 99.94%
    Color and Shape:White Crystalline Powder
    Molecular weight:434.41
  • Silodosin

    CAS:
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Formula:C25H32F3N3O4
    Purity:99.282% - 99.76%
    Color and Shape:Colorless To Pink Solid
    Molecular weight:495.53
  • Metaproterenol hemisulfate

    CAS:
    Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
    Formula:C11H17NO3·5H2O4S
    Purity:98.53% - 99.74%
    Color and Shape:Solid
    Molecular weight:260.3
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Formula:C21H24ClNO
    Purity:99.77% - >99.99%
    Color and Shape:White To Slightly Yellowish Crystalline Solid
    Molecular weight:341.88
  • Urapidil hydrochloride

    CAS:
    Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
    Formula:C20H29N5O3·HCl
    Purity:99.58%
    Color and Shape:White Or Off-White Crystalline Powder
    Molecular weight:423.94
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Formula:C21H25N3O2S
    Purity:99.14% - 99.63%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:383.51
  • JNJ-18038683

    CAS:
    JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.
    Formula:C26H28ClN3O7
    Purity:97.29%
    Color and Shape:Solid
    Molecular weight:529.97
  • PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Formula:C25H37Cl2N3O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:482.49
  • Acetophenazine dimaleate

    CAS:
    Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.
    Formula:C31H37N3O10S
    Purity:99.39% - 99.48%
    Color and Shape:Solid
    Molecular weight:643.71
  • Naftopidil

    CAS:
    Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-
    Formula:C24H28N2O3
    Purity:99.60% - 99.97%
    Color and Shape:White Crystalline Powder
    Molecular weight:392.49
  • Ifenprodil

    CAS:
    Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.
    Formula:C21H27NO2
    Purity:99.58%
    Color and Shape:White Crystalline Powder
    Molecular weight:325.44
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Formula:C18H25ClN4O
    Purity:99.88% - 99.93%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:348.87
  • Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:231.65
  • Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:367.5
  • Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Formula:C9H15ClNO5P
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:283.65
  • NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Formula:C27H31Cl2N3O3
    Purity:99.33%
    Color and Shape:Soild
    Molecular weight:516.46
  • Levosulpiride

    CAS:
    Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43
  • Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Formula:C17H18F3NO
    Purity:99.07% - 99.28%
    Color and Shape:Solid
    Molecular weight:309.33
  • Astressin acetate


    <p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>
    Formula:C163H273N49O44
    Purity:96.87%
    Color and Shape:Solid
    Molecular weight:3623.21
  • Diphenylpyraline hydrochloride

    CAS:
    Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
    Formula:C19H23NO·HCl
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:317.85
  • Chlorprothixene hydrochloride

    CAS:
    Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
    Formula:C18H18ClNS·HCl
    Purity:99.76%
    Color and Shape:White Powder
    Molecular weight:352.32
  • Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>
    Formula:C28H30N2O8
    Purity:99.7% - >99.99%
    Color and Shape:Powder
    Molecular weight:522.55
  • Olanzapine

    CAS:
    Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
    Formula:C17H20N4S
    Purity:99.86% - ≥95%
    Color and Shape:Yellowish Crystalline Powder
    Molecular weight:312.43
  • CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Formula:C15H18Cl2N4O
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:341.24
  • Trazodone hydrochloride

    CAS:
    <p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>
    Formula:C19H23Cl2N5O
    Purity:99.5% - 99.52%
    Color and Shape:Solid
    Molecular weight:408.33
  • MK-0249 FA


    MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.
    Formula:C24H26F3N3O4
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:477.48
  • Antazoline hydrochloride

    CAS:
    Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous
    Formula:C17H19N3·HCl
    Purity:98% - 99.53%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:301.82
  • Solabegron

    CAS:
    <p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>
    Formula:C23H23ClN2O3
    Purity:97.89%
    Color and Shape:Solid
    Molecular weight:410.89
  • Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39
  • YNT-185

    CAS:
    YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
    Formula:C33H37N5O5S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:615.74
  • Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Formula:C26H35NO7
    Purity:98.53% - 99.43%
    Color and Shape:Coa
    Molecular weight:473.57
  • KGA-2727

    CAS:
    KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.
    Formula:C26H40N4O8
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:536.62
  • (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purity:97.82%
    Color and Shape:Soild
    Molecular weight:195.19
  • Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purity:99.85% - >99.99%
    Color and Shape:White Powder
    Molecular weight:300.25
  • Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36
  • Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Formula:C21H28N2O5
    Purity:99.61%
    Color and Shape:5 1 (Ntp 1992)
    Molecular weight:388.46
  • AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29
  • Phenothiazine

    CAS:
    Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.
    Formula:C12H9NS
    Purity:99.95%
    Color and Shape:Yellow Solid Pellets
    Molecular weight:199.27
  • Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28
  • ESI-05

    CAS:
    <p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>
    Formula:C16H18O2S
    Purity:97.22%
    Color and Shape:Solid
    Molecular weight:274.38
  • Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Formula:C17H22ClNO
    Purity:99.86%
    Color and Shape:White Solid
    Molecular weight:291.82
  • Duloxetine hydrochloride

    CAS:
    Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.
    Formula:C18H20ClNOS
    Purity:99.93% - >99.99%
    Color and Shape:White Or White Crystalline Powder
    Molecular weight:333.88
  • AB928

    CAS:
    AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
    Formula:C23H22N8O
    Purity:98.09% - >99.99%
    Color and Shape:Solid
    Molecular weight:426.47
  • LCKLSL hydrochloride


    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Formula:C30H58ClN7O8S
    Purity:98.02% - 99.31%
    Color and Shape:Solid
    Molecular weight:712.34
  • (R)-Elagolix

    CAS:
    (R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.
    Formula:C32H30F5N3O5
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:631.59
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Formula:C31H38N2O
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:454.65
  • Methoxamine hydrochloride

    CAS:
    Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
    Formula:C11H18ClNO3
    Purity:99.84% - >99.99%
    Color and Shape:Colorless Or White Plate-Like Crystals Or White Crystalline Powder Solid
    Molecular weight:247.719
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Formula:C15H24N2O4S·HCl
    Purity:99.4% - 99.77%
    Color and Shape:Solid
    Molecular weight:364.89
  • Filorexant

    CAS:
    Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).
    Formula:C24H25FN4O2
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:420.48
  • Levodropropizine

    CAS:
    Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
    Formula:C13H20N2O2
    Purity:99.87% - 99.93%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:236.31
  • Palonosetron hydrochloride

    CAS:
    Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.
    Formula:C19H24N2O·HCl
    Purity:99.84% - 99.92%
    Color and Shape:White Solid
    Molecular weight:332.87
  • Ro 10-5824 dihydrochloride

    CAS:
    Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).
    Formula:C17H22Cl2N4
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:353.29
  • Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Formula:C16H26ClNO3
    Purity:99.94% - ≥95%
    Color and Shape:Solid
    Molecular weight:315.84
  • Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Formula:C21H22CL2N4OS
    Purity:97.97% - 99.82%
    Color and Shape:Solid
    Molecular weight:449.4
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Formula:C26H27N5O2
    Purity:99.61%
    Color and Shape:Light Yellow Solid
    Molecular weight:441.52
  • Dopexamine hydrochloride

    CAS:
    Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.
    Formula:C22H34Cl2N2O2
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:429.42
  • Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96
  • Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Formula:C9H11NO3·HCl
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:217.65
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Formula:C11H16BrCl2N
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:313.06
  • Promazine hydrochloride

    CAS:
    Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
    Formula:C17H21ClN2S
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:320.88
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Formula:C18H29ClN2O4
    Purity:99.92% - >99.99%
    Color and Shape:White Or Slightly Off-White Crystalline Powder Solid
    Molecular weight:372.89
  • Pizotifen

    CAS:
    <p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>
    Formula:C19H21NS
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:295.44
  • Linaclotide

    CAS:
    Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.
    Formula:C59H79N15O21S6
    Purity:97.93% - 98.71%
    Color and Shape:Solid
    Molecular weight:1526.74
  • MP-A08

    CAS:
    MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.
    Formula:C27H25N3O4S2
    Purity:97.44%
    Color and Shape:Solid
    Molecular weight:519.64
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Formula:C15H20N2O2·HCl
    Purity:99.64% - 99.92%
    Color and Shape:Solid
    Molecular weight:296.79
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Formula:C21H24N4O2S
    Purity:99.64%
    Color and Shape:Light Yellow To Yellow Solid
    Molecular weight:396.51
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purity:99.4% - 99.97%
    Color and Shape:Solid
    Molecular weight:461.81
  • Olinciguat

    CAS:
    Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.
    Formula:C21H16F5N7O3
    Purity:99.33% - 99.71%
    Color and Shape:Solid
    Molecular weight:509.39
  • Roxatidine Acetate hydrochloride

    CAS:
    Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9
  • Monatepil 2maleate


    Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.
    Formula:C32H34FN3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:591.69